ES8506727A1 - Procedimiento para la obtencion de compuestos del acido 7b -acilamido-3-cefem-4-carboxilico - Google Patents

Procedimiento para la obtencion de compuestos del acido 7b -acilamido-3-cefem-4-carboxilico

Info

Publication number
ES8506727A1
ES8506727A1 ES535195A ES535195A ES8506727A1 ES 8506727 A1 ES8506727 A1 ES 8506727A1 ES 535195 A ES535195 A ES 535195A ES 535195 A ES535195 A ES 535195A ES 8506727 A1 ES8506727 A1 ES 8506727A1
Authority
ES
Spain
Prior art keywords
group
formula
preparation
application
pharmaceutical compositions
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES535195A
Other languages
English (en)
Other versions
ES535195A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of ES8506727A1 publication Critical patent/ES8506727A1/es
Publication of ES535195A0 publication Critical patent/ES535195A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/08—1,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/568—Four-membered rings

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE COMPUESTOS DEL ACIDO 7 BBB-ACILAMIDO-3-CEFEM-4-CARBOXILICO, DE FORMULA GENERAL (I), EN LA QUE M ES 0, 1 O 2; R1 SIGNIFICA HIDROGENO, ALQUILO INFERIOR O ALQUENILO INFERIOR; R2 SIGNIFICA UN GRUPO HIDROXI O MERCAPTO LIBRE; R3 SIGNIFICA CARBOXI O CARBOXI PROTEGIDO; R4 SIGNIFICA HIDROGENO; R5 SIGNIFICA UN RESTO ORGANICO QUE ESTA ENLAZADO CON UN ATOMO DE CARBONO AL GRUPO SULFONILO; Y R6 REPRESENTA UN RESTO HETEROCICLICO, SUS ESTEREOISOMEROS, SUS HIDRATOS Y SUS SALES FARMACEUTICAMENTE ACEPTABLES.CONSISTE EN SULFONIZAR MEDIANTE REACCION CON UN AGENTE DE SULFONILIZACION, INTRODUCTOR DEL RESTO R5-SULFONILO DE UN ACIDO SULFONICO DE FORMULA (II), UN COMPUESTO DE FORMULA GENERAL (III).DE APLICACION EN PREPARADOS FARMACEUTICOS.
ES535195A 1982-04-27 1984-08-16 Procedimiento para la obtencion de compuestos del acido 7b -acilamido-3-cefem-4-carboxilico Granted ES535195A0 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH256882 1982-04-27
CH650482 1982-11-09

Publications (2)

Publication Number Publication Date
ES8506727A1 true ES8506727A1 (es) 1985-08-01
ES535195A0 ES535195A0 (es) 1985-08-01

Family

ID=25690804

Family Applications (2)

Application Number Title Priority Date Filing Date
ES521824A Expired ES8504818A1 (es) 1982-04-27 1983-04-25 Procedimiento para la obtencion de compuestos del acido 7-acilamido-3-cefem-4-carboxilico.
ES535195A Granted ES535195A0 (es) 1982-04-27 1984-08-16 Procedimiento para la obtencion de compuestos del acido 7b -acilamido-3-cefem-4-carboxilico

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES521824A Expired ES8504818A1 (es) 1982-04-27 1983-04-25 Procedimiento para la obtencion de compuestos del acido 7-acilamido-3-cefem-4-carboxilico.

Country Status (12)

Country Link
EP (1) EP0092830A3 (es)
AU (1) AU1395183A (es)
DD (1) DD207720A5 (es)
DK (1) DK185383A (es)
ES (2) ES8504818A1 (es)
FI (1) FI831381L (es)
GB (1) GB2118942B (es)
GR (1) GR78190B (es)
HU (1) HU188459B (es)
IL (1) IL68477A0 (es)
NO (1) NO831470L (es)
PT (1) PT76597B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004111012A1 (ja) 2003-06-12 2004-12-23 Chugai Seiyaku Kabushiki Kaisha イミダゾリジン誘導体
JP5625614B2 (ja) 2010-08-20 2014-11-19 セイコーエプソン株式会社 光フィルター、光フィルターモジュール、分光測定器および光機器

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3270000A (en) * 1962-10-29 1966-08-30 Squibb & Sons Inc Protected amino acid derivatives of 7-aminocephalosporanic acid
DE2724073A1 (de) * 1976-06-03 1977-12-22 Fujisawa Pharmaceutical Co 3,7-disubstituierte 3-cephem-4- carbonsaeuren und sie enthaltende pharmazeutische zubereitungen

Also Published As

Publication number Publication date
GB2118942A (en) 1983-11-09
AU1395183A (en) 1983-11-03
HU188459B (en) 1986-04-28
FI831381L (fi) 1983-10-28
ES521824A0 (es) 1985-05-01
NO831470L (no) 1983-10-28
PT76597A (en) 1983-05-01
EP0092830A2 (de) 1983-11-02
GB8311222D0 (en) 1983-06-02
IL68477A0 (en) 1983-07-31
ES535195A0 (es) 1985-08-01
GR78190B (es) 1984-09-26
FI831381A0 (fi) 1983-04-22
GB2118942B (en) 1985-07-24
EP0092830A3 (de) 1984-12-27
ES8504818A1 (es) 1985-05-01
DK185383D0 (da) 1983-04-26
DD207720A5 (de) 1984-03-14
DK185383A (da) 1983-10-28
PT76597B (en) 1986-03-12

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