ES8401497A1 - Un procedimiento para la preparacion de nuevos derivados de 3-amino-pregn-5-eno. - Google Patents

Un procedimiento para la preparacion de nuevos derivados de 3-amino-pregn-5-eno.

Info

Publication number
ES8401497A1
ES8401497A1 ES516825A ES516825A ES8401497A1 ES 8401497 A1 ES8401497 A1 ES 8401497A1 ES 516825 A ES516825 A ES 516825A ES 516825 A ES516825 A ES 516825A ES 8401497 A1 ES8401497 A1 ES 8401497A1
Authority
ES
Spain
Prior art keywords
radical
formula
amino
bab
pregn
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES516825A
Other languages
English (en)
Spanish (es)
Other versions
ES516825A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Publication of ES516825A0 publication Critical patent/ES516825A0/es
Publication of ES8401497A1 publication Critical patent/ES8401497A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Steroid Compounds (AREA)
ES516825A 1981-10-27 1982-10-26 Un procedimiento para la preparacion de nuevos derivados de 3-amino-pregn-5-eno. Expired ES8401497A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8120135A FR2515188A1 (fr) 1981-10-27 1981-10-27 Nouveaux derives du 3-amino-pregn-5-ene, leurs sels, procede de preparation, application a titre de medicaments et compositions les renfermant

Publications (2)

Publication Number Publication Date
ES516825A0 ES516825A0 (es) 1983-12-01
ES8401497A1 true ES8401497A1 (es) 1983-12-01

Family

ID=9263427

Family Applications (2)

Application Number Title Priority Date Filing Date
ES516825A Expired ES8401497A1 (es) 1981-10-27 1982-10-26 Un procedimiento para la preparacion de nuevos derivados de 3-amino-pregn-5-eno.
ES524922A Granted ES524922A0 (es) 1981-10-27 1983-08-12 Un procedimiento para la preparacion de nuevos derivados de 3-amino-pregn-5-eno

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES524922A Granted ES524922A0 (es) 1981-10-27 1983-08-12 Un procedimiento para la preparacion de nuevos derivados de 3-amino-pregn-5-eno

Country Status (19)

Country Link
US (1) US4444767A (OSRAM)
JP (1) JPS5883700A (OSRAM)
AT (1) AT387023B (OSRAM)
BE (1) BE894805A (OSRAM)
CA (1) CA1193247A (OSRAM)
CH (1) CH655936A5 (OSRAM)
DE (1) DE3239823C2 (OSRAM)
DK (1) DK160561C (OSRAM)
ES (2) ES8401497A1 (OSRAM)
FR (1) FR2515188A1 (OSRAM)
GB (1) GB2110212B (OSRAM)
HU (1) HU186983B (OSRAM)
IE (1) IE54278B1 (OSRAM)
IT (1) IT1158025B (OSRAM)
LU (1) LU84439A1 (OSRAM)
NL (1) NL8204159A (OSRAM)
PT (1) PT75756B (OSRAM)
SE (1) SE456423B (OSRAM)
ZA (1) ZA827745B (OSRAM)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4842862A (en) * 1986-07-03 1989-06-27 International Minerals & Chemical Corp. Immunostimulating agents
US5504074A (en) * 1993-08-06 1996-04-02 Children's Medical Center Corporation Estrogenic compounds as anti-angiogenic agents
US6908910B2 (en) * 1993-08-06 2005-06-21 The Children's Medical Center Corporation Estrogenic compounds as anti-mitotic agents
US20040214807A1 (en) * 1993-08-06 2004-10-28 D'amato Robert J. Estrogenic compounds as anti-mitotic agents
US5571933A (en) * 1994-11-17 1996-11-05 Duquesne University Of The Holy Ghost Derivatives of estra 1,3,5(10)triene-17-one, 3-amino compounds and their use
US6346510B1 (en) * 1995-10-23 2002-02-12 The Children's Medical Center Corporation Therapeutic antiangiogenic endostatin compositions
US7087592B1 (en) 1999-08-23 2006-08-08 Entre Med, Inc. Compositions comprising purified 2-methoxyestradiol and methods of producing same
US6995278B2 (en) * 2000-08-18 2006-02-07 Entre Med, Inc. Antiangiogenic agents
US20050192258A1 (en) * 2000-08-18 2005-09-01 Agoston Gregory E. Antiangiogenic agents
US7135581B2 (en) * 2000-08-18 2006-11-14 Entremed, Inc. Antiangiogenic agents
CA2527074A1 (en) * 2003-05-28 2005-04-07 Entremed, Inc. Antiangiogenic agents
US20070004689A1 (en) * 2004-03-12 2007-01-04 Agoston Gregory E Antiangiogenic agents
EP1756139A4 (en) 2004-03-12 2009-07-29 Entremed Inc ANTI-ANGIOGENIC AGENTS
JP2008521822A (ja) * 2004-11-29 2008-06-26 エントレメッド インコーポレイテッド 抗血管形成剤を投与する方法、およびそれを用いて疾病を治療する方法
US20070185069A1 (en) * 2005-11-14 2007-08-09 Plum Stacy M Anti-angiogenic activity of 2-methoxyestradiol in combination with anti-cancer agents
US20070176403A1 (en) * 2006-02-01 2007-08-02 Dennis Calderone Air adjustable seat
US8399440B2 (en) * 2006-03-20 2013-03-19 Entremed, Inc. Disease modifying anti-arthritic activity of 2-methoxyestradiol
US20080234243A1 (en) * 2007-01-31 2008-09-25 Lavallee Theresa M Method of treating amyloidosis mediated diseases
WO2015171489A1 (en) * 2014-05-05 2015-11-12 Apicore Us Llc Methods of making netupitant and intermediates thereof

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE663020A (OSRAM) *
US3374252A (en) * 1958-08-19 1968-03-19 Oletta Sa Pharmaceutical product obtained from plants of the genus holarrhena (apocynaceae)
US3244696A (en) * 1959-04-30 1966-04-05 Oletta Sa Extraction of alkaloids from plants of genus holarrhena
GB948485A (en) * 1959-04-30 1964-02-05 Oletta Sa New alkaloids and other new compounds from holarrhena species and processes for obtaining the same
DE1470219A1 (de) * 1961-06-02 1969-06-04 Biochemische Forschung Biofor Verfahren zum Herstellen von Adenin-Abkoemmlingen
BE672238A (OSRAM) * 1965-11-12 1966-03-01
BE687512A (OSRAM) * 1966-09-28 1967-03-01
FR7512M (OSRAM) * 1966-11-14 1969-12-15
BE701968A (OSRAM) * 1967-07-28 1968-01-02
GB1439605A (en) * 1972-07-14 1976-06-16 Akzo Nv 2beta-hydroxy-3-alpha-amino-steroids and derivatives thereof and the processes for their preparation
FR2463777A1 (fr) * 1979-08-17 1981-02-27 Roussel Uclaf Nouveaux derives du 5a-pregnan-20-ol, leur procede de preparation et leur application comme medicaments

Also Published As

Publication number Publication date
SE8204918L (sv) 1983-04-28
SE8204918D0 (sv) 1982-08-27
JPS5883700A (ja) 1983-05-19
GB2110212A (en) 1983-06-15
US4444767A (en) 1984-04-24
AT387023B (de) 1988-11-25
FR2515188B1 (OSRAM) 1984-09-28
ES8405035A1 (es) 1984-05-16
PT75756A (fr) 1982-11-01
ATA391282A (de) 1988-04-15
SE456423B (sv) 1988-10-03
DK160561B (da) 1991-03-25
DK160561C (da) 1991-09-09
DE3239823C2 (de) 1994-06-16
HU186983B (en) 1985-10-28
ZA827745B (en) 1983-11-30
CH655936A5 (fr) 1986-05-30
ES516825A0 (es) 1983-12-01
CA1193247A (fr) 1985-09-10
IE822581L (en) 1983-04-27
IE54278B1 (en) 1989-08-16
DK473182A (da) 1983-04-28
IT1158025B (it) 1987-02-18
DE3239823A1 (de) 1983-05-05
IT8249354A1 (it) 1984-04-25
GB2110212B (en) 1985-10-30
ES524922A0 (es) 1984-05-16
JPH0411559B2 (OSRAM) 1992-02-28
FR2515188A1 (fr) 1983-04-29
NL8204159A (nl) 1983-05-16
BE894805A (fr) 1983-04-26
LU84439A1 (fr) 1983-06-13
PT75756B (fr) 1985-11-20
IT8249354A0 (it) 1982-10-25

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19971001