ES8401095A1 - Procedimiento para la preparacion de 11 -cloro-15-esteroides. - Google Patents
Procedimiento para la preparacion de 11 -cloro-15-esteroides.Info
- Publication number
- ES8401095A1 ES8401095A1 ES520206A ES520206A ES8401095A1 ES 8401095 A1 ES8401095 A1 ES 8401095A1 ES 520206 A ES520206 A ES 520206A ES 520206 A ES520206 A ES 520206A ES 8401095 A1 ES8401095 A1 ES 8401095A1
- Authority
- ES
- Spain
- Prior art keywords
- steroids
- oxo
- preparation
- group
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 238000002360 preparation method Methods 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical group [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 239000003433 contraceptive agent Substances 0.000 abstract 1
- 230000002254 contraceptive effect Effects 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 230000007062 hydrolysis Effects 0.000 abstract 1
- 238000006460 hydrolysis reaction Methods 0.000 abstract 1
- 239000000583 progesterone congener Substances 0.000 abstract 1
- 239000002994 raw material Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0059—Estrane derivatives substituted in position 17 by a keto group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
- C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
- C07J1/0096—Alkynyl derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J21/005—Ketals
- C07J21/006—Ketals at position 3
-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P33/00—Preparation of steroids
- C12P33/12—Acting on D ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Microbiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Engineering & Computer Science (AREA)
- Genetics & Genomics (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19823214690 DE3214690A1 (de) | 1982-04-16 | 1982-04-16 | 11ss-chlor-(delta)(pfeil hoch)1(pfeil hoch)(pfeil hoch)5(pfeil hoch)-steroide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES520206A0 ES520206A0 (es) | 1983-12-01 |
| ES8401095A1 true ES8401095A1 (es) | 1983-12-01 |
Family
ID=6161448
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES520206A Expired ES8401095A1 (es) | 1982-04-16 | 1983-03-01 | Procedimiento para la preparacion de 11 -cloro-15-esteroides. |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US4464365A (en, 2012) |
| EP (1) | EP0092174B1 (en, 2012) |
| JP (1) | JPS58188898A (en, 2012) |
| AT (1) | ATE18408T1 (en, 2012) |
| AU (1) | AU555285B2 (en, 2012) |
| CA (1) | CA1244004A (en, 2012) |
| DD (1) | DD209636A5 (en, 2012) |
| DE (2) | DE3214690A1 (en, 2012) |
| DK (2) | DK166089C (en, 2012) |
| ES (1) | ES8401095A1 (en, 2012) |
| GR (1) | GR78213B (en, 2012) |
| HU (1) | HU186686B (en, 2012) |
| IE (1) | IE54751B1 (en, 2012) |
| ZA (1) | ZA832674B (en, 2012) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4232521A1 (de) * | 1992-09-22 | 1994-03-24 | Schering Ag | Gestagen wirksame 4,5;11,12-Estradiene, Verfahren zu ihrer Herstellung, diese Estradiene enthaltende Arzneimittel sowie deren Verwendung zur Herstellung von Arzneimitteln |
| DE10104327A1 (de) * | 2001-01-24 | 2002-07-25 | Schering Ag | 11beta-Halogensteroide, deren Herstellung und Verwendung zur Herstellung von Arzneimitteln sowie 11beta-Halogensteroide enthaltende pharmazeutische Präparate |
| EP2354150A1 (en) * | 2010-02-09 | 2011-08-10 | Laboratoire Theramex | Process for the preparation of gestodene |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3665021A (en) * | 1966-07-29 | 1972-05-23 | Glaxo Lab Ltd | 9alpha-unsubstituted-11beta-chloro-l9 nos-steroids |
| US3933799A (en) * | 1969-01-29 | 1976-01-20 | Glaxo Laboratories Limited | 11β-Halo-9,12-unsubstituted-C19 -steroids |
| NL7209299A (en) * | 1972-07-01 | 1974-01-03 | Delta-4-3-oxo-11-beta-halo steroids - with hormonal activity | |
| US4081537A (en) * | 1975-10-10 | 1978-03-28 | Schering Aktiengesellschaft | Δ15 -Steroids and pharmaceutical compositions thereof |
-
1982
- 1982-04-16 DE DE19823214690 patent/DE3214690A1/de not_active Withdrawn
-
1983
- 1983-02-25 DK DK092183A patent/DK166089C/da active
- 1983-03-01 ES ES520206A patent/ES8401095A1/es not_active Expired
- 1983-03-16 AU AU12488/83A patent/AU555285B2/en not_active Ceased
- 1983-04-06 IE IE765/83A patent/IE54751B1/en not_active IP Right Cessation
- 1983-04-13 JP JP58063806A patent/JPS58188898A/ja active Granted
- 1983-04-14 DE DE8383103605T patent/DE3362381D1/de not_active Expired
- 1983-04-14 DD DD83249872A patent/DD209636A5/de not_active IP Right Cessation
- 1983-04-14 EP EP83103605A patent/EP0092174B1/de not_active Expired
- 1983-04-14 GR GR71090A patent/GR78213B/el unknown
- 1983-04-14 AT AT83103605T patent/ATE18408T1/de not_active IP Right Cessation
- 1983-04-15 HU HU831328A patent/HU186686B/hu not_active IP Right Cessation
- 1983-04-15 CA CA000426011A patent/CA1244004A/en not_active Expired
- 1983-04-15 ZA ZA832674A patent/ZA832674B/xx unknown
- 1983-04-18 US US06/485,800 patent/US4464365A/en not_active Expired - Fee Related
-
1991
- 1991-11-25 DK DK191591A patent/DK165879C/da active
Also Published As
| Publication number | Publication date |
|---|---|
| AU555285B2 (en) | 1986-09-18 |
| IE830765L (en) | 1983-10-16 |
| JPH0358359B2 (en, 2012) | 1991-09-05 |
| DE3362381D1 (en) | 1986-04-10 |
| EP0092174B1 (de) | 1986-03-05 |
| DK191591A (da) | 1991-11-25 |
| JPS58188898A (ja) | 1983-11-04 |
| ZA832674B (en) | 1983-12-28 |
| HU186686B (en) | 1985-09-30 |
| DK166089B (da) | 1993-03-08 |
| ATE18408T1 (de) | 1986-03-15 |
| ES520206A0 (es) | 1983-12-01 |
| DE3214690A1 (de) | 1983-10-27 |
| DK191591D0 (da) | 1991-11-25 |
| DK165879C (da) | 1993-06-21 |
| GR78213B (en, 2012) | 1984-09-26 |
| EP0092174A1 (de) | 1983-10-26 |
| AU1248883A (en) | 1983-10-20 |
| DK92183D0 (da) | 1983-02-25 |
| US4464365A (en) | 1984-08-07 |
| DK165879B (da) | 1993-02-01 |
| DD209636A5 (de) | 1984-05-16 |
| DK92183A (da) | 1983-10-17 |
| CA1244004A (en) | 1988-11-01 |
| DK166089C (da) | 1993-08-02 |
| IE54751B1 (en) | 1990-01-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19971001 |