ES8100268A1 - Procedimiento para la preparacion de agentes antiglaucomicos - Google Patents

Procedimiento para la preparacion de agentes antiglaucomicos

Info

Publication number
ES8100268A1
ES8100268A1 ES487642A ES487642A ES8100268A1 ES 8100268 A1 ES8100268 A1 ES 8100268A1 ES 487642 A ES487642 A ES 487642A ES 487642 A ES487642 A ES 487642A ES 8100268 A1 ES8100268 A1 ES 8100268A1
Authority
ES
Spain
Prior art keywords
hydrogen
image
carbostyril
glaucoma
lower alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES487642A
Other languages
English (en)
Spanish (es)
Other versions
ES487642A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Otsuka Pharmaceutical Co Ltd
Original Assignee
Otsuka Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26345304&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES8100268(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from JP54010108A external-priority patent/JPS5951927B2/ja
Priority claimed from JP54070361A external-priority patent/JPS5951928B2/ja
Application filed by Otsuka Pharmaceutical Co Ltd filed Critical Otsuka Pharmaceutical Co Ltd
Publication of ES8100268A1 publication Critical patent/ES8100268A1/es
Publication of ES487642A0 publication Critical patent/ES487642A0/es
Granted legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES487642A 1979-01-30 1980-01-11 Procedimiento para la preparacion de agentes antiglaucomicos Granted ES487642A0 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP54010108A JPS5951927B2 (ja) 1979-01-30 1979-01-30 緑内障治療剤
JP54070361A JPS5951928B2 (ja) 1979-06-04 1979-06-04 緑内障治療剤

Publications (2)

Publication Number Publication Date
ES8100268A1 true ES8100268A1 (es) 1980-11-01
ES487642A0 ES487642A0 (es) 1980-11-01

Family

ID=26345304

Family Applications (1)

Application Number Title Priority Date Filing Date
ES487642A Granted ES487642A0 (es) 1979-01-30 1980-01-11 Procedimiento para la preparacion de agentes antiglaucomicos

Country Status (15)

Country Link
US (1) US4309432A (US06373033-20020416-M00035.png)
AT (1) AT371340B (US06373033-20020416-M00035.png)
AU (1) AU518814B2 (US06373033-20020416-M00035.png)
CA (1) CA1139669A (US06373033-20020416-M00035.png)
CH (1) CH646057A5 (US06373033-20020416-M00035.png)
DE (1) DE3001011C2 (US06373033-20020416-M00035.png)
DK (1) DK11580A (US06373033-20020416-M00035.png)
ES (1) ES487642A0 (US06373033-20020416-M00035.png)
FI (1) FI800089A (US06373033-20020416-M00035.png)
FR (1) FR2447721A1 (US06373033-20020416-M00035.png)
GB (1) GB2042338B (US06373033-20020416-M00035.png)
IT (1) IT1141662B (US06373033-20020416-M00035.png)
NL (1) NL191575C (US06373033-20020416-M00035.png)
NO (1) NO800059L (US06373033-20020416-M00035.png)
SE (1) SE451069B (US06373033-20020416-M00035.png)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0056420A1 (en) * 1981-01-15 1982-07-28 Schering Corporation Ophthalmic gel
FR2539413A1 (fr) * 1983-01-17 1984-07-20 Pos Lab Carbostyriloximinopropanolamines utiles comme medicaments et procede pour leur preparation
US4921862A (en) * 1986-05-29 1990-05-01 Syntex (U.S.A.) Inc. Carbostyril derivatives as combined thromboxane synthetase and cyclic-amp phosphodiesterase inhibitors
US4792561A (en) * 1986-05-29 1988-12-20 Syntex (U.S.A.) Inc. Carbostyril derivatives as combined thromboxane synthetase and cyclic-AMP phosphodiesterase inhibitors
DK391189A (da) * 1988-08-10 1990-02-11 Otsuka Pharma Co Ltd Carbostyrilderivater
US5198448A (en) * 1988-08-10 1993-03-30 Otsuka Pharmaceutical Company, Limited Cardiotonics
ES2075082T3 (es) * 1989-03-28 1995-10-01 Nisshin Flour Milling Co Derivados de isoquinolina para el tratamiento del glaucoma o hipertension ocular.
FR2676740B1 (fr) * 1991-05-23 1993-11-05 Roussel Uclaf Nouveaux derives sterouides du pregna-4,9(11),17(20)-trie-3-one, leur preparation, leur application a la preparation de composes sterouides de type pregna-4,9(11),16-triene-3,20-dione et nouveaux intermediaires.
US5629345A (en) * 1993-07-23 1997-05-13 Vide Pharmaceuticals Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure
US5965620A (en) * 1993-07-23 1999-10-12 Vide Pharmaceuticals Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure
US5776482A (en) * 1996-03-29 1998-07-07 University Of Iowa Research Foundation Tetrahydroquinoline analogues for use in glaucoma treatment
MY116782A (en) 1997-12-22 2004-03-31 Otsuka Pharma Co Ltd Water-soluble eye drop
CN101578051A (zh) * 2006-12-06 2009-11-11 美国硼砂公司 动物饲料组合物

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS48103590A (US06373033-20020416-M00035.png) * 1972-04-13 1973-12-25
US3910924A (en) * 1972-04-13 1975-10-07 Otsuka Pharma Co Ltd 3,4-Dihydrocarbostyril derivatives and a process for preparing the same
AR207554A1 (es) * 1972-12-02 1976-10-15 Otsuka Pharma Co Ltd Procedimiento para producir derivados de 3-alquil-5-((3,4-dihidro-5-carbostiril)oximetil)-oxazolidinona-(2)
JPS5239035B2 (US06373033-20020416-M00035.png) * 1972-12-14 1977-10-03
US3975391A (en) * 1973-12-26 1976-08-17 Otsuka Pharmaceutical Company Limited 5-[1-Hydroxy-2-(substituted-amino)]ethyl-8-hydroxy-3,4-dihydrocarbostyril derivatives
AU467612B2 (en) * 1973-07-31 1975-12-04 Novel organophosphorous pesticide
JPS5082218A (US06373033-20020416-M00035.png) * 1973-11-10 1975-07-03
US3994901A (en) * 1974-06-13 1976-11-30 Otsuka Pharmaceutical Company Limited 5-[1-Hydroxy-2-(substituted-amino)]alkyl-8-hydroxy-3,4-dihydrocarbostyril derivatives
US4081447A (en) * 1975-04-09 1978-03-28 Abbott Laboratories 5-[2-Hydroxy-3-(3,4-dimethoxy phenethylamino)]-propoxy-3,4-dihydro carbostyril and pharmaceutically acceptable salts thereof
CH619453A5 (US06373033-20020416-M00035.png) * 1976-03-17 1980-09-30 Otsuka Pharma Co Ltd
US4210753A (en) * 1976-03-17 1980-07-01 Otsuka Pharmaceutical Co., Ltd. Carbostyril compounds
GB1574665A (en) * 1976-05-08 1980-09-10 Otsuka Pharma Co Ltd 3,4-dihydrocarbostyril derivatives and process for preparing the same
JPS552631A (en) * 1978-06-19 1980-01-10 Otsuka Pharmaceut Co Ltd 3,4-dihydrocarbostyril derivative
JPS5513241A (en) * 1978-07-14 1980-01-30 Otsuka Pharmaceut Co Ltd Remedy for glaucoma

Also Published As

Publication number Publication date
NO800059L (no) 1980-07-31
ATA14480A (de) 1982-11-15
CA1139669A (en) 1983-01-18
US4309432A (en) 1982-01-05
AT371340B (de) 1983-06-27
NL8000211A (nl) 1980-08-01
GB2042338A (en) 1980-09-24
GB2042338B (en) 1983-11-30
NL191575B (nl) 1995-06-01
CH646057A5 (de) 1984-11-15
FI800089A (fi) 1980-07-31
NL191575C (nl) 1995-10-03
IT1141662B (it) 1986-10-08
AU518814B2 (en) 1981-10-22
IT8005106A0 (it) 1980-01-09
FR2447721A1 (fr) 1980-08-29
FR2447721B1 (US06373033-20020416-M00035.png) 1983-03-11
ES487642A0 (es) 1980-11-01
DE3001011C2 (de) 1986-02-06
AU5426579A (en) 1980-08-07
DE3001011A1 (de) 1980-08-28
SE8000245L (sv) 1980-07-31
DK11580A (da) 1980-07-31
SE451069B (sv) 1987-08-31

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Legal Events

Date Code Title Description
RL1A Appeal rendered by the court

Free format text: 19951214

RL1A Appeal rendered by the court

Free format text: 19951214