ES546061A0 - Un procedimiento para preparar un derivado de uridina - Google Patents

Un procedimiento para preparar un derivado de uridina

Info

Publication number
ES546061A0
ES546061A0 ES546061A ES546061A ES546061A0 ES 546061 A0 ES546061 A0 ES 546061A0 ES 546061 A ES546061 A ES 546061A ES 546061 A ES546061 A ES 546061A ES 546061 A0 ES546061 A0 ES 546061A0
Authority
ES
Spain
Prior art keywords
uridine
derivative
preparing
procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES546061A
Other languages
English (en)
Other versions
ES8607982A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Taiho Pharmaceutical Co Ltd
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP58091190A external-priority patent/JPS59216899A/ja
Priority claimed from JP58170149A external-priority patent/JPS6061593A/ja
Priority claimed from JP58170147A external-priority patent/JPS6061591A/ja
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Publication of ES546061A0 publication Critical patent/ES546061A0/es
Publication of ES8607982A1 publication Critical patent/ES8607982A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES546061A 1983-05-23 1985-08-09 Un procedimiento para preparar un derivado de uridina Expired ES8607982A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP58091190A JPS59216899A (ja) 1983-05-23 1983-05-23 2′―デオキシ―5―トリフルオロメチルウリジン誘導体及びそれを含む抗腫瘍剤
JP58170149A JPS6061593A (ja) 1983-09-14 1983-09-14 2’−デオキシ−5−トリフルオロメチルウリジン誘導体及びそれを含む抗腫瘍剤
JP58170147A JPS6061591A (ja) 1983-09-14 1983-09-14 2′―デオキシ―5―フルオロウリジン誘導体及びそれを含む抗腫瘍剤

Publications (2)

Publication Number Publication Date
ES546061A0 true ES546061A0 (es) 1986-06-01
ES8607982A1 ES8607982A1 (es) 1986-06-01

Family

ID=27306680

Family Applications (4)

Application Number Title Priority Date Filing Date
ES532716A Expired ES8606382A1 (es) 1983-05-23 1984-05-23 Un procedimiento para preparar un derivado de uridina 2'-desoxi-5-sustituido
ES546060A Expired ES8706715A1 (es) 1983-05-23 1985-08-09 Un procedimiento para preparar un derivado de uridina.
ES546061A Expired ES8607982A1 (es) 1983-05-23 1985-08-09 Un procedimiento para preparar un derivado de uridina
ES85546062A Expired ES8606381A1 (es) 1983-05-23 1985-08-09 Un procedimiento para preparar un derivado de uridina.

Family Applications Before (2)

Application Number Title Priority Date Filing Date
ES532716A Expired ES8606382A1 (es) 1983-05-23 1984-05-23 Un procedimiento para preparar un derivado de uridina 2'-desoxi-5-sustituido
ES546060A Expired ES8706715A1 (es) 1983-05-23 1985-08-09 Un procedimiento para preparar un derivado de uridina.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES85546062A Expired ES8606381A1 (es) 1983-05-23 1985-08-09 Un procedimiento para preparar un derivado de uridina.

Country Status (7)

Country Link
US (1) US4886877A (es)
EP (1) EP0129984B1 (es)
KR (1) KR860001865B1 (es)
AU (1) AU548712B2 (es)
CA (1) CA1227794A (es)
DE (1) DE3469533D1 (es)
ES (4) ES8606382A1 (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5250673A (en) * 1983-05-23 1993-10-05 Taiho Pharmaceutical Company, Ltd. 2'-deoxy-5-substituted uridine derivatives
US4864021A (en) * 1984-10-30 1989-09-05 Otsuka Pharmaceutical Co., Ltd. 5-fluorouracil derivatives
DE3588036T2 (de) * 1984-10-30 1995-11-16 Otsuka Pharma Co Ltd 5-Fluoruracilderivate.
WO1987000435A1 (fr) * 1985-07-22 1987-01-29 Teijin Limited Medicament antiviral
ES2058073T3 (es) * 1986-04-30 1994-11-01 Otsuka Pharma Co Ltd Derivados de 5-fluorouracilo.
DK363987A (da) * 1986-08-08 1988-02-09 Hoffmann La Roche Pyrimidinderivater
AU610913B2 (en) * 1987-07-31 1991-05-30 Taiho Pharmaceutical Co., Ltd. 2'-deoxy-5-fluorouridine derivatives
US4992534A (en) * 1987-08-12 1991-02-12 Otsuka Pharmaceutical Co., Ltd. 3'-O-,5'-O-derivatives of 2'-deoxy-5-fluorouridine
EP0517262A1 (en) * 1991-06-07 1992-12-09 MITSUI TOATSU CHEMICALS, Inc. Trifluorothymidine derivatives, process for producing the same and anti-cancer agent containing the same
FI935444A (fi) * 1992-12-07 1994-06-08 Mitsui Toatsu Chemicals 3'-O-propargyyli-trifluoritymidiinin tioesterijohdannaiset, menetelmä niiden valmistamiseksi ja niiden käyttö syövänvastaisena aineena
JP4110347B2 (ja) * 1999-11-05 2008-07-02 大鵬薬品工業株式会社 抗hiv剤
US7160537B2 (en) * 2003-12-15 2007-01-09 Siemens Medical Solutions Usa, Inc. Method for preparing radiolabeled thymidine having low chromophoric byproducts
US20050131224A1 (en) * 2003-12-15 2005-06-16 Cti Pet Systems, Inc. Method for preparing radiolabeled thymidine

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2658672A1 (de) * 1976-12-23 1978-06-29 Robugen Gmbh Neue nucleosid-verbindungen und verfahren zu ihrer herstellung
US4210638A (en) * 1978-03-17 1980-07-01 Pcr, Inc. Antiviral composition and method of treating virus diseases
GB2016921B (en) * 1978-03-27 1982-08-18 Taiho Pharmaceutical Co Ltd Anti cancer compositions containing uracil derivatives
JPS5924999B2 (ja) * 1978-06-10 1984-06-13 富山化学工業株式会社 新規な5−フルオロ−2′−デオキシ−β−ウリジン誘導体の製造法
DE3105111A1 (de) * 1980-02-15 1981-12-24 Funai Yakuhin Kogyo K.K., Osaka "2 -desoxy-3',5-di-o-alkylcarbonyl-5-fluoruridin-derivate, verfahren zu ihrer herstellung, ihre verwendung zur behandlung von tumoren und antitumormittel"
JP3834939B2 (ja) * 1997-06-12 2006-10-18 松下電工株式会社 照明装置

Also Published As

Publication number Publication date
ES546060A0 (es) 1987-06-16
AU2846784A (en) 1984-11-29
ES8606381A1 (es) 1986-04-01
CA1227794A (en) 1987-10-06
ES8607982A1 (es) 1986-06-01
ES546062A0 (es) 1986-04-01
EP0129984A1 (en) 1985-01-02
ES532716A0 (es) 1986-04-01
AU548712B2 (en) 1986-01-02
KR840009104A (ko) 1984-12-24
EP0129984B1 (en) 1988-03-02
US4886877A (en) 1989-12-12
ES8606382A1 (es) 1986-04-01
DE3469533D1 (en) 1988-04-07
KR860001865B1 (ko) 1986-10-24
ES8706715A1 (es) 1987-06-16

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