ES451449A1 - Un procedimiento para la preparacion de nuevos derivados delacido 6-(d-2-acilamido-2-fenilacetamido)penicilanico. - Google Patents

Un procedimiento para la preparacion de nuevos derivados delacido 6-(d-2-acilamido-2-fenilacetamido)penicilanico.

Info

Publication number
ES451449A1
ES451449A1 ES451449A ES451449A ES451449A1 ES 451449 A1 ES451449 A1 ES 451449A1 ES 451449 A ES451449 A ES 451449A ES 451449 A ES451449 A ES 451449A ES 451449 A1 ES451449 A1 ES 451449A1
Authority
ES
Spain
Prior art keywords
nhz
gram
hooc
formula
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES451449A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Tanabe Seiyaku Co Ltd
Original Assignee
Tanabe Seiyaku Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tanabe Seiyaku Co Ltd filed Critical Tanabe Seiyaku Co Ltd
Publication of ES451449A1 publication Critical patent/ES451449A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/46—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Un procedimiento para la preparación de nuevos derivados del ácido de 6-(D-2-amino-2-fenilacetamido) penicilánico de fórmula: **(Fórmula)** donde R1 es hidrógeno o hidroxi; R2 es un grupo de fórmula: -COCH(NH2)-CH2COR3 o -COCH2-CH(NH2)-COR3; y R3 está seleccionado del grupo formado por hidroxi, alquilamino inferior, di-alquilamino inferior, aloxi inferior e hidroxi alquilamino inferior; o alternativamente R3 es amino cuando R1 es hidroxi, o una sal farmacéuticamente aceptable del mismo, que comprende las etapas de condensar un compuesto de ácido 6-(D-2-amino-2-fenilacetamido)-penicilánico.
ES451449A 1975-09-12 1976-09-10 Un procedimiento para la preparacion de nuevos derivados delacido 6-(d-2-acilamido-2-fenilacetamido)penicilanico. Expired ES451449A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB37525/75A GB1533413A (en) 1975-09-12 1975-09-12 Penicillins

Publications (1)

Publication Number Publication Date
ES451449A1 true ES451449A1 (es) 1978-01-16

Family

ID=10397137

Family Applications (1)

Application Number Title Priority Date Filing Date
ES451449A Expired ES451449A1 (es) 1975-09-12 1976-09-10 Un procedimiento para la preparacion de nuevos derivados delacido 6-(d-2-acilamido-2-fenilacetamido)penicilanico.

Country Status (14)

Country Link
JP (3) JPS5236689A (es)
AR (1) AR220887A1 (es)
AT (1) AT344904B (es)
CH (1) CH622798A5 (es)
CS (1) CS202564B2 (es)
EG (1) EG12522A (es)
ES (1) ES451449A1 (es)
GB (1) GB1533413A (es)
HU (1) HU171688B (es)
MX (1) MX3970E (es)
PH (1) PH13848A (es)
PL (1) PL110862B1 (es)
PT (1) PT65575B (es)
SU (1) SU633482A3 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4839044B2 (ja) * 2005-08-30 2011-12-14 富士機工株式会社 シフトレバーのレンジ位置表示装置
CN104059087B (zh) * 2014-07-08 2016-02-17 湖南尔康制药股份有限公司 一种阿扑西林的合成方法
CN113999251A (zh) * 2021-11-12 2022-02-01 海南海灵化学制药有限公司 一种阿扑西林钠的合成方法

Also Published As

Publication number Publication date
MX3970E (es) 1981-10-20
GB1533413A (en) 1978-11-22
AR220887A1 (es) 1980-12-15
EG12522A (en) 1981-06-30
JPS6052125B2 (ja) 1985-11-18
CS202564B2 (en) 1981-01-30
PT65575A (en) 1976-10-01
PT65575B (en) 1978-03-28
JPS5443519B2 (es) 1979-12-20
SU633482A3 (ru) 1978-11-15
PL110862B1 (en) 1980-08-30
JPS58116418A (ja) 1983-07-11
CH622798A5 (en) 1981-04-30
PL192334A1 (pl) 1979-02-12
AT344904B (de) 1978-08-25
HU171688B (hu) 1978-02-28
JPS5236689A (en) 1977-03-22
PH13848A (en) 1980-10-22
ATA640476A (de) 1977-12-15
JPS5332125A (en) 1978-03-27

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