JPS5332125A - Bacteriostatic pharmaceutical composition - Google Patents

Bacteriostatic pharmaceutical composition

Info

Publication number
JPS5332125A
JPS5332125A JP4400877A JP4400877A JPS5332125A JP S5332125 A JPS5332125 A JP S5332125A JP 4400877 A JP4400877 A JP 4400877A JP 4400877 A JP4400877 A JP 4400877A JP S5332125 A JPS5332125 A JP S5332125A
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
bacteriostatic
bacteriostatic pharmaceutical
penicillanic acid
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP4400877A
Other languages
Japanese (ja)
Other versions
JPS6052125B2 (en
Inventor
Mitsutaka Kawazu
Kokichi Azuma
Masahiko Seto
Riichi Miyagishima
Totaro Yamaguchi
Satoshi Oshima
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Tanabe Seiyaku Co Ltd
Original Assignee
Tanabe Seiyaku Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tanabe Seiyaku Co Ltd filed Critical Tanabe Seiyaku Co Ltd
Publication of JPS5332125A publication Critical patent/JPS5332125A/en
Publication of JPS6052125B2 publication Critical patent/JPS6052125B2/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/46—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

PURPOSE: A penicillanic acid derivative I]R1 is H, OH: R2 is acyl II or III (R3 is OH, lower alkylamino, di-lower-alkyl amino, lower alkoxy, hydroxysubstituted alkyl; when R1 is OH, R3 may be amino)]; e.g. 6-[D-2-(D-2amino-3-N-methylcarbamoyl-propionamide)-2-p-hydroxypehnyl acetamide] penicillanic acid.
COPYRIGHT: (C)1978,JPO&Japio
JP52044008A 1975-09-12 1977-04-15 Antibacterial pharmaceutical composition Expired JPS6052125B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB37525/75A GB1533413A (en) 1975-09-12 1975-09-12 Penicillins
GB37525 1981-12-11

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP51104509A Division JPS5236689A (en) 1975-09-12 1976-08-31 Novel synthetic penicillins and their preparation process

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP57170795A Division JPS58116418A (en) 1975-09-12 1982-09-28 Antimicrobial pharmaceutical composition

Publications (2)

Publication Number Publication Date
JPS5332125A true JPS5332125A (en) 1978-03-27
JPS6052125B2 JPS6052125B2 (en) 1985-11-18

Family

ID=10397137

Family Applications (3)

Application Number Title Priority Date Filing Date
JP51104509A Granted JPS5236689A (en) 1975-09-12 1976-08-31 Novel synthetic penicillins and their preparation process
JP52044008A Expired JPS6052125B2 (en) 1975-09-12 1977-04-15 Antibacterial pharmaceutical composition
JP57170795A Pending JPS58116418A (en) 1975-09-12 1982-09-28 Antimicrobial pharmaceutical composition

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP51104509A Granted JPS5236689A (en) 1975-09-12 1976-08-31 Novel synthetic penicillins and their preparation process

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP57170795A Pending JPS58116418A (en) 1975-09-12 1982-09-28 Antimicrobial pharmaceutical composition

Country Status (14)

Country Link
JP (3) JPS5236689A (en)
AR (1) AR220887A1 (en)
AT (1) AT344904B (en)
CH (1) CH622798A5 (en)
CS (1) CS202564B2 (en)
EG (1) EG12522A (en)
ES (1) ES451449A1 (en)
GB (1) GB1533413A (en)
HU (1) HU171688B (en)
MX (1) MX3970E (en)
PH (1) PH13848A (en)
PL (1) PL110862B1 (en)
PT (1) PT65575B (en)
SU (1) SU633482A3 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4839044B2 (en) * 2005-08-30 2011-12-14 富士機工株式会社 Shift lever range position display device
CN104059087B (en) * 2014-07-08 2016-02-17 湖南尔康制药股份有限公司 A kind of synthetic method of aspoxicillin
CN113999251A (en) * 2021-11-12 2022-02-01 海南海灵化学制药有限公司 Synthetic method of aspoxicillin sodium

Also Published As

Publication number Publication date
ES451449A1 (en) 1978-01-16
MX3970E (en) 1981-10-20
GB1533413A (en) 1978-11-22
AR220887A1 (en) 1980-12-15
EG12522A (en) 1981-06-30
JPS6052125B2 (en) 1985-11-18
CS202564B2 (en) 1981-01-30
PT65575A (en) 1976-10-01
PT65575B (en) 1978-03-28
JPS5443519B2 (en) 1979-12-20
SU633482A3 (en) 1978-11-15
PL110862B1 (en) 1980-08-30
JPS58116418A (en) 1983-07-11
CH622798A5 (en) 1981-04-30
PL192334A1 (en) 1979-02-12
AT344904B (en) 1978-08-25
HU171688B (en) 1978-02-28
JPS5236689A (en) 1977-03-22
PH13848A (en) 1980-10-22
ATA640476A (en) 1977-12-15

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