ES2843952T3 - Composiciones para tratar el insomnio - Google Patents
Composiciones para tratar el insomnio Download PDFInfo
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- ES2843952T3 ES2843952T3 ES15851934T ES15851934T ES2843952T3 ES 2843952 T3 ES2843952 T3 ES 2843952T3 ES 15851934 T ES15851934 T ES 15851934T ES 15851934 T ES15851934 T ES 15851934T ES 2843952 T3 ES2843952 T3 ES 2843952T3
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
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- A—HUMAN NECESSITIES
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
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- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
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- Inorganic Chemistry (AREA)
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- Medicinal Preparation (AREA)
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Applications Claiming Priority (2)
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| US201462067443P | 2014-10-23 | 2014-10-23 | |
| PCT/JP2015/080304 WO2016063995A1 (en) | 2014-10-23 | 2015-10-21 | Compositions and methods for treating insomnia |
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| ES2843952T3 true ES2843952T3 (es) | 2021-07-21 |
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| ES15851934T Active ES2843952T3 (es) | 2014-10-23 | 2015-10-21 | Composiciones para tratar el insomnio |
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| SG10202007759RA (en) | 2014-10-23 | 2020-09-29 | Eisai R&D Man Co Ltd | Compositions and methods for treating insomnia |
| IL291791B2 (en) * | 2016-05-12 | 2025-09-01 | Eisai R&D Man Co Ltd | Methods for treating sleep timing disorders |
| CA3032233C (en) | 2016-08-10 | 2021-09-14 | F. Hoffmann-La Roche Ag | Pharmaceutical compositions comprising akt protein kinase inhibitors |
| CN115710250A (zh) | 2017-08-01 | 2023-02-24 | 博健制药有限责任公司 | 一种食欲素受体拮抗剂的晶型及其制备方法和用途 |
| CA3119728A1 (en) | 2018-11-21 | 2020-05-28 | Tremeau Pharmaceuticals, Inc. | Purified forms of rofecoxib, methods of manufacture and use |
| JP2022538170A (ja) * | 2019-06-26 | 2022-08-31 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 睡眠問題の治療のためのレンボレキサント |
| US20220305012A1 (en) * | 2019-06-26 | 2022-09-29 | Eisai R&D Management Co., Ltd. | Lemborexant for treating sleep issues |
| WO2020263253A1 (en) * | 2019-06-26 | 2020-12-30 | Moline Margaret | Lemborexant for treating sleep issues |
| CN114502167A (zh) * | 2019-09-13 | 2022-05-13 | 卫材R&D管理有限公司 | 用于治疗失眠的药物组合物 |
| US20220339143A1 (en) * | 2019-09-13 | 2022-10-27 | Takeda Pharmaceutical Company Limited | Tak-925 for use in treating narcolepsy |
| KR20220119065A (ko) | 2019-12-20 | 2022-08-26 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 불면증 치료를 위한 렘보렉산트의 용도 |
| TW202140014A (zh) | 2020-01-16 | 2021-11-01 | 日商衛材R&D企管股份有限公司 | 萊博雷生的原料藥及含有其的醫藥組成物 |
| EP4138822A1 (en) | 2020-04-19 | 2023-03-01 | Idorsia Pharmaceuticals Ltd | Medical use of daridorexant |
| CN111450076A (zh) * | 2020-05-25 | 2020-07-28 | 安徽省逸欣铭医药科技有限公司 | 一种Lemborexant软胶囊组合物及其制备方法 |
| WO2024064897A1 (en) | 2022-09-23 | 2024-03-28 | Eisai R&D Management Co., Ltd. | Methods of reducing neurodegeneration associated with neurodegenerative diseases |
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| EP1998774A1 (en) | 2006-03-15 | 2008-12-10 | Actelion Pharmaceuticals Ltd. | Tetrahydroisoquinoline derivatives to enhance memory function |
| WO2007129188A1 (en) | 2006-05-10 | 2007-11-15 | Pfizer Japan Inc. | Cyclopropanecarboxamide compound |
| BRPI0716532A2 (pt) | 2006-09-11 | 2013-09-24 | Glaxo Group Ltd | compostos azabicÍclios como inidores de reabsorÇço de monoaminas |
| CL2007002809A1 (es) | 2006-09-29 | 2008-04-18 | Actelion Pharmaceuticals Ltd | Compuestos derivados de 3-aza biciclo [3.1.0]hexano; y su uso en el tratamiento de enfermedades tales como desordenes psicoticos y de ansiedad, desordenes del sueno, uso y abuso de sustancias psicoactivas, demencia y deterioro de funciones cognitivas |
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| PE20091010A1 (es) | 2007-10-10 | 2009-08-08 | Actelion Pharmaceuticals Ltd | Derivados de tetrahidroquinolina |
| EP2537282B1 (en) * | 2010-02-15 | 2015-09-16 | Koninklijke Philips N.V. | Mitigation of control channel interference |
| SI2626350T1 (sl) * | 2010-09-22 | 2015-09-30 | Eisai R&D Management Co., Ltd. | Spojina ciklopropana |
| US20120165339A1 (en) | 2010-12-22 | 2012-06-28 | Eisai R&D Management Co., Ltd. | Cyclopropane derivatives |
| SG10202007759RA (en) | 2014-10-23 | 2020-09-29 | Eisai R&D Man Co Ltd | Compositions and methods for treating insomnia |
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| EP3209298A4 (en) | 2018-06-20 |
| RU2703297C2 (ru) | 2019-10-16 |
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| US11026944B2 (en) | 2021-06-08 |
| US20200268754A1 (en) | 2020-08-27 |
| IL251759B (en) | 2021-01-31 |
| WO2016063995A1 (en) | 2016-04-28 |
| CN107810006B (zh) | 2021-03-30 |
| US20170252342A1 (en) | 2017-09-07 |
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| SG10202007759RA (en) | 2020-09-29 |
| RU2017112308A (ru) | 2018-11-26 |
| CA2964504A1 (en) | 2016-04-28 |
| KR20170068478A (ko) | 2017-06-19 |
| MX376164B (es) | 2025-03-07 |
| SG11201703064WA (en) | 2017-05-30 |
| AU2015336463A1 (en) | 2017-05-04 |
| MX2017004950A (es) | 2018-01-16 |
| CA2964504C (en) | 2022-08-23 |
| KR102444608B1 (ko) | 2022-09-20 |
| EP3209298B1 (en) | 2020-12-02 |
| JP2017531683A (ja) | 2017-10-26 |
| US20190201399A1 (en) | 2019-07-04 |
| CN107810006A (zh) | 2018-03-16 |
| EP3209298A1 (en) | 2017-08-30 |
| US10702529B2 (en) | 2020-07-07 |
| IL251759A0 (en) | 2017-06-29 |
| AU2015336463B2 (en) | 2020-06-18 |
| US10188652B2 (en) | 2019-01-29 |
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