CA2964504C - Oral dosage form comprising a cyclopropanecarboxamide derivative for use in treating insomnia - Google Patents
Oral dosage form comprising a cyclopropanecarboxamide derivative for use in treating insomnia Download PDFInfo
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- CA2964504C CA2964504C CA2964504A CA2964504A CA2964504C CA 2964504 C CA2964504 C CA 2964504C CA 2964504 A CA2964504 A CA 2964504A CA 2964504 A CA2964504 A CA 2964504A CA 2964504 C CA2964504 C CA 2964504C
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| WO2017197160A1 (en) * | 2016-05-12 | 2017-11-16 | Eisai R&D Management Co., Ltd. | Methods of treating circadian rhythm sleep disorders |
| CN115350192B (zh) * | 2016-08-10 | 2025-05-13 | 豪夫迈·罗氏有限公司 | 包含Akt蛋白激酶抑制剂的药物组合物 |
| JP7179049B2 (ja) * | 2017-08-01 | 2022-11-28 | ベルゲン ファーマシューティカル、 エルエルシー | オレキシン受容体拮抗薬の結晶形及びその製造方法並びに用途 |
| CN113660934A (zh) | 2018-11-21 | 2021-11-16 | 特默罗制药股份有限公司 | 罗非昔布的纯化形式、制备方法和用途 |
| JP2022538170A (ja) * | 2019-06-26 | 2022-08-31 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 睡眠問題の治療のためのレンボレキサント |
| WO2020263253A1 (en) * | 2019-06-26 | 2020-12-30 | Moline Margaret | Lemborexant for treating sleep issues |
| CN114096251A (zh) * | 2019-06-26 | 2022-02-25 | 卫材R&D管理有限公司 | 用于治疗睡眠问题的莱博雷生 |
| CA3154321A1 (en) * | 2019-09-13 | 2021-03-18 | Takeda Pharmaceutical Company Limited | Tak-925 for use in treating narcolepsy |
| CN114502167A (zh) * | 2019-09-13 | 2022-05-13 | 卫材R&D管理有限公司 | 用于治疗失眠的药物组合物 |
| BR112022012246A2 (pt) | 2019-12-20 | 2022-08-30 | Eisai R&D Man Co Ltd | Uso de lemborexant para tratar insônia |
| US20230103250A1 (en) * | 2020-01-16 | 2023-03-30 | Eisai R&D Management Co., Ltd. | Drug substance of lemborexant and medicinal composition comprising same |
| US20230134935A1 (en) * | 2020-04-19 | 2023-05-04 | Idorsia Pharmaceuticals Ltd | Medical use of daridorexant |
| CN111450076A (zh) * | 2020-05-25 | 2020-07-28 | 安徽省逸欣铭医药科技有限公司 | 一种Lemborexant软胶囊组合物及其制备方法 |
| KR20250070087A (ko) | 2022-09-23 | 2025-05-20 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 신경변성 질병과 관련된 신경변성의 감소 방법 |
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| EA200970266A1 (ru) | 2006-09-11 | 2009-08-28 | Глэксо Груп Лимитед | Азабициклические соединения в качестве ингибиторов повторного поглощения моноаминов |
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| BRPI0817198A2 (pt) | 2007-09-21 | 2015-03-17 | Sanofi Aventis | (ciclopropilfenil)feniloxalamidas, método para a produção das mesmas, e uso das mesmas como um medicamento |
| PE20091010A1 (es) | 2007-10-10 | 2009-08-08 | Actelion Pharmaceuticals Ltd | Derivados de tetrahidroquinolina |
| KR101823339B1 (ko) * | 2010-02-15 | 2018-01-31 | 코닌클리케 필립스 엔.브이. | 제어 채널 간섭의 완화 |
| SI2626350T1 (sl) * | 2010-09-22 | 2015-09-30 | Eisai R&D Management Co., Ltd. | Spojina ciklopropana |
| US20120165339A1 (en) | 2010-12-22 | 2012-06-28 | Eisai R&D Management Co., Ltd. | Cyclopropane derivatives |
| JP6659681B2 (ja) | 2014-10-23 | 2020-03-04 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 不眠症を治療するための組成物および方法 |
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| WO2016063995A1 (en) | 2016-04-28 |
| ES2843952T3 (es) | 2021-07-21 |
| KR20170068478A (ko) | 2017-06-19 |
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| MX376164B (es) | 2025-03-07 |
| KR102444608B1 (ko) | 2022-09-20 |
| EP3209298A1 (en) | 2017-08-30 |
| EP3209298A4 (en) | 2018-06-20 |
| CA2964504A1 (en) | 2016-04-28 |
| US20200268754A1 (en) | 2020-08-27 |
| JP6659681B2 (ja) | 2020-03-04 |
| SG10202007759RA (en) | 2020-09-29 |
| CN107810006B (zh) | 2021-03-30 |
| US11026944B2 (en) | 2021-06-08 |
| IL251759A0 (en) | 2017-06-29 |
| US10188652B2 (en) | 2019-01-29 |
| BR112017007063A2 (pt) | 2018-02-14 |
| MX2017004950A (es) | 2018-01-16 |
| AU2015336463B2 (en) | 2020-06-18 |
| JP2017531683A (ja) | 2017-10-26 |
| RU2017112308A3 (enExample) | 2019-05-08 |
| SG11201703064WA (en) | 2017-05-30 |
| RU2703297C2 (ru) | 2019-10-16 |
| AU2015336463A1 (en) | 2017-05-04 |
| EP3209298B1 (en) | 2020-12-02 |
| US20170252342A1 (en) | 2017-09-07 |
| US10702529B2 (en) | 2020-07-07 |
| CN107810006A (zh) | 2018-03-16 |
| RU2017112308A (ru) | 2018-11-26 |
| IL251759B (en) | 2021-01-31 |
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