ES2715844T3 - Formulaciones farmacéuticas que comprenden antagonistas de CCR3 - Google Patents

Formulaciones farmacéuticas que comprenden antagonistas de CCR3 Download PDF

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Publication number
ES2715844T3
ES2715844T3 ES13714618T ES13714618T ES2715844T3 ES 2715844 T3 ES2715844 T3 ES 2715844T3 ES 13714618 T ES13714618 T ES 13714618T ES 13714618 T ES13714618 T ES 13714618T ES 2715844 T3 ES2715844 T3 ES 2715844T3
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Spain
Prior art keywords
pharmaceutical composition
diluent
composition according
disintegrant
lubricant
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Application number
ES13714618T
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English (en)
Spanish (es)
Inventor
Alfred Fetscher
Jochen Matthias Scher
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Alkahest Inc
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Alkahest Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49292482&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES2715844(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alkahest Inc filed Critical Alkahest Inc
Application granted granted Critical
Publication of ES2715844T3 publication Critical patent/ES2715844T3/es
Active legal-status Critical Current
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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
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    • A61K9/2004Excipients; Inactive ingredients
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    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
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    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • A61K9/2022Organic macromolecular compounds
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    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
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    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
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    • A61K9/2853Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
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    • AHUMAN NECESSITIES
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Pulmonology (AREA)
  • Inorganic Chemistry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Neurology (AREA)
  • Urology & Nephrology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Transplantation (AREA)
  • Otolaryngology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES13714618T 2012-04-04 2013-04-02 Formulaciones farmacéuticas que comprenden antagonistas de CCR3 Active ES2715844T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12163078 2012-04-04
PCT/EP2013/056867 WO2013149987A1 (en) 2012-04-04 2013-04-02 Pharmaceutical formulations comprising ccr3 antagonists

Publications (1)

Publication Number Publication Date
ES2715844T3 true ES2715844T3 (es) 2019-06-06

Family

ID=49292482

Family Applications (2)

Application Number Title Priority Date Filing Date
ES18213458T Active ES2898179T3 (es) 2012-04-04 2013-04-02 Formulaciones farmacéuticas que comprenden antagonistas de CCR3
ES13714618T Active ES2715844T3 (es) 2012-04-04 2013-04-02 Formulaciones farmacéuticas que comprenden antagonistas de CCR3

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES18213458T Active ES2898179T3 (es) 2012-04-04 2013-04-02 Formulaciones farmacéuticas que comprenden antagonistas de CCR3

Country Status (31)

Country Link
US (3) US10213421B2 (instruction)
EP (3) EP3524230B1 (instruction)
JP (4) JP6320990B2 (instruction)
KR (2) KR102338465B1 (instruction)
CN (1) CN104203213A (instruction)
AR (1) AR090596A1 (instruction)
AU (1) AU2013245028B2 (instruction)
BR (1) BR112014024479A8 (instruction)
CA (1) CA2869058C (instruction)
CL (1) CL2014002524A1 (instruction)
CY (1) CY1121137T1 (instruction)
DK (2) DK2833864T3 (instruction)
EA (1) EA027627B1 (instruction)
ES (2) ES2898179T3 (instruction)
HR (1) HRP20190069T1 (instruction)
HU (2) HUE041519T2 (instruction)
IL (1) IL234299A (instruction)
IN (1) IN2014DN07082A (instruction)
LT (1) LT2833864T (instruction)
MX (1) MX358307B (instruction)
NZ (1) NZ628993A (instruction)
PH (1) PH12014502241A1 (instruction)
PL (2) PL3524230T3 (instruction)
PT (2) PT2833864T (instruction)
RS (1) RS58360B1 (instruction)
SI (1) SI2833864T1 (instruction)
SM (1) SMT201900121T1 (instruction)
TR (1) TR201821285T4 (instruction)
TW (1) TW201400115A (instruction)
UY (1) UY34730A (instruction)
WO (1) WO2013149987A1 (instruction)

Families Citing this family (12)

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Publication number Priority date Publication date Assignee Title
US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
US8680280B2 (en) 2012-04-02 2014-03-25 Boehringer Ingelheim International Gmbh Process for the manufacturing of CRR inhibitors
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
MX394341B (es) * 2017-04-05 2025-03-24 Alkahest Inc Metodos y composiciones para tratar deterioros asociados con el envejecimiento usando inhibidores de ccr3
JP7179755B2 (ja) 2017-04-05 2022-11-29 アルカヘスト インコーポレイテッド Ccr3阻害剤を使用した網膜関連疾患を治療するための方法および組成物
SG11202002437VA (en) * 2017-10-13 2020-04-29 Alkahest Inc Methods and compositions for treating pruritus, xerosis, and associated disease using ccr3-inhibitors
MX2020011114A (es) 2018-05-15 2021-01-29 Alkahest Inc Tratamiento de enfermedades asociadas con el envejecimiento con moduladores de la leucotrieno a4 hidrolasa.
BR112021004938A2 (pt) * 2018-09-26 2021-06-01 Alkahest, Inc. métodos e composições para tratamento de danos associados com o envelhecimento usando inibidores de ccr3
EP4206153A4 (en) 2020-08-27 2024-05-15 Agc Inc. ALKALI-FREE GLASS AND PLATE GLASS
US11957671B2 (en) 2021-11-01 2024-04-16 Alkahest, Inc. Benzodioxane modulators of leukotriene A4 hydrolase (LTA4H) for prevention and treatment of aging-associated diseases

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