ES2687780T3 - Inhibidor de la actividad heparanasa - Google Patents
Inhibidor de la actividad heparanasa Download PDFInfo
- Publication number
- ES2687780T3 ES2687780T3 ES10820611.1T ES10820611T ES2687780T3 ES 2687780 T3 ES2687780 T3 ES 2687780T3 ES 10820611 T ES10820611 T ES 10820611T ES 2687780 T3 ES2687780 T3 ES 2687780T3
- Authority
- ES
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- Prior art keywords
- pigmentation
- heparan sulfate
- sulfate
- normal
- skin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Landscapes
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- Cosmetics (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pyrrole Compounds (AREA)
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| US11787783B2 (en) | 2016-12-13 | 2023-10-17 | Beta Therapeutics Pty Ltd | Heparanase inhibitors and use thereof |
| RU2019121873A (ru) | 2016-12-13 | 2021-01-15 | БЕТА ТЕРАПЬЮТИКС ПиТиУай ЛТД | Ингибиторы гепараназы и их применение |
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| CN110740729B (zh) | 2017-06-13 | 2023-05-16 | 国立研究开发法人国立癌症研究中心 | 致癌抑制剂 |
| US20220202964A1 (en) * | 2019-04-24 | 2022-06-30 | University Of Florida Research Foundation, Incorporated | Heparanase compounds and methods of use |
| WO2022131182A1 (ja) | 2020-12-15 | 2022-06-23 | 株式会社 資生堂 | 表皮幹細胞増加促進剤 |
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| US4049650A (en) | 1976-10-18 | 1977-09-20 | Morton-Norwich Products, Inc. | 1-[[[5-(Substituted phenyl)-2-oxazolyl]methylene]amino]-2,4-imidazolidinediones |
| US4593038A (en) * | 1985-04-03 | 1986-06-03 | Burzynski Stanislaw R | Topical use of 3-phenylacetylamino-2,6-piperidinedione for treatment of skin wrinkles and hyperpigmentation |
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-
2010
- 2010-09-29 CN CN2010800438641A patent/CN102655863B/zh active Active
- 2010-09-29 US US13/261,244 patent/US8609075B2/en active Active
- 2010-09-29 RU RU2012117797/15A patent/RU2503454C1/ru not_active IP Right Cessation
- 2010-09-29 EP EP10820611.1A patent/EP2484359B1/en active Active
- 2010-09-29 WO PCT/JP2010/066998 patent/WO2011040496A1/ja active Application Filing
- 2010-09-29 KR KR1020127004685A patent/KR101431348B1/ko active Active
- 2010-09-29 ES ES10820611.1T patent/ES2687780T3/es active Active
- 2010-09-29 IN IN2632DEN2012 patent/IN2012DN02632A/en unknown
- 2010-09-29 JP JP2011534288A patent/JP5593323B2/ja active Active
- 2010-09-29 BR BR112012007090-8A patent/BR112012007090A2/pt not_active Application Discontinuation
- 2010-09-30 TW TW099133410A patent/TWI461221B/zh active
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Also Published As
| Publication number | Publication date |
|---|---|
| CN102655863A (zh) | 2012-09-05 |
| US20140080878A1 (en) | 2014-03-20 |
| KR20120060205A (ko) | 2012-06-11 |
| EP2484359A4 (en) | 2015-07-08 |
| JPWO2011040496A1 (ja) | 2013-02-28 |
| TWI461221B (zh) | 2014-11-21 |
| US20120183481A1 (en) | 2012-07-19 |
| IN2012DN02632A (forum.php) | 2015-09-04 |
| WO2011040496A1 (ja) | 2011-04-07 |
| EP2484359A1 (en) | 2012-08-08 |
| AU2010301641A1 (en) | 2012-03-22 |
| JP5593323B2 (ja) | 2014-09-24 |
| JP2014111640A (ja) | 2014-06-19 |
| KR101431348B1 (ko) | 2014-08-19 |
| RU2503454C1 (ru) | 2014-01-10 |
| EP2484359B1 (en) | 2018-07-25 |
| US8901160B2 (en) | 2014-12-02 |
| TW201117832A (en) | 2011-06-01 |
| RU2012117797A (ru) | 2013-11-10 |
| BR112012007090A2 (pt) | 2018-06-05 |
| US8609075B2 (en) | 2013-12-17 |
| CN102655863B (zh) | 2013-11-20 |
| HK1171390A1 (en) | 2013-03-28 |
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