ES2653852T3 - Composiciones farmacéuticas que contienen ligandos del receptor de dopamina y procedimientos de tratamiento usando ligandos del receptor de dopamina - Google Patents
Composiciones farmacéuticas que contienen ligandos del receptor de dopamina y procedimientos de tratamiento usando ligandos del receptor de dopamina Download PDFInfo
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- ES2653852T3 ES2653852T3 ES08782602.0T ES08782602T ES2653852T3 ES 2653852 T3 ES2653852 T3 ES 2653852T3 ES 08782602 T ES08782602 T ES 08782602T ES 2653852 T3 ES2653852 T3 ES 2653852T3
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- treatment
- cariprazine
- animals
- escitalopram oxalate
- cariprazine hydrochloride
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Classifications
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- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| PCT/US2008/072066 WO2009020897A1 (en) | 2007-08-03 | 2008-08-04 | Pharmaceutical compositions containing dopamine receptor ligands and methods of treatment using dopamine recptor ligands |
Publications (1)
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| ES2653852T3 true ES2653852T3 (es) | 2018-02-09 |
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| SI2317852T1 (sl) | 2008-07-16 | 2015-04-30 | Richter Gedeon Nyrt. | Farmacevtske formulacije, ki vsebujejo ligande dopaminskega receptorja |
| US20110117214A1 (en) * | 2009-11-16 | 2011-05-19 | Auspex Pharmaceuticals, Inc. | Cyclohexyl urea modulators of d2 receptors and/or d3 receptors |
| JP5860457B2 (ja) | 2010-06-18 | 2016-02-16 | アルトス・セラピューティクス・リミテッド・ライアビリティ・カンパニーＡｌｔｏｓ Ｔｈｅｒａｐｅｕｔｉｃｓ，Ｌｌｃ | Ｄ２アンタゴニスト、その合成方法および使用方法 |
| US8912197B2 (en) | 2012-08-20 | 2014-12-16 | Forest Laboratories Holdings Ltd. | Crystalline form of carbamoyl-cyclohexane derivatives |
| US11274087B2 (en) | 2016-07-08 | 2022-03-15 | Richter Gedeon Nyrt. | Industrial process for the preparation of cariprazine |
| HUP1700253A1 (hu) * | 2017-06-13 | 2019-01-28 | Richter Gedeon Nyrt | Szilárd orális gyógyszerkészítmények |
| GB2571696B (en) | 2017-10-09 | 2020-05-27 | Compass Pathways Ltd | Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced |
| US12459965B2 (en) | 2017-10-09 | 2025-11-04 | Compass Pathfinder Limited | Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use |
| US11547707B2 (en) | 2019-04-10 | 2023-01-10 | Richter Gedeon Nyrt. | Carbamoyl cyclohexane derivatives for treating autism spectrum disorder |
| HU231500B1 (hu) * | 2019-04-10 | 2024-04-28 | Richter Gedeon Nyrt | Karbamoil-ciklohexán származékok autizmus spektrum betegség kezelésére |
| WO2020212951A1 (en) | 2019-04-17 | 2020-10-22 | Compass Pathfinder Limited | Methods for treating anxiety disorders, headache disorders, and eating disorders with psilocybin |
| EP4422629A4 (en) * | 2021-10-28 | 2025-09-03 | Richter Gedeon Nyrt | TREATMENT OF MAJOR DEPRESSIVE DISORDER |
| JP2025500844A (ja) * | 2021-12-13 | 2025-01-15 | コンパス パスファインダー リミテッド | 治療抵抗性うつ病の治療に使用するためのサイロシビン及び補助的セロトニン再取り込み阻害剤 |
| CA3244202A1 (en) * | 2022-03-17 | 2023-09-21 | Mapi Pharma Ltd | DEPOSIT SYSTEMS INCLUDING CARIPRAZINE OR SALTS THEREOF |
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| GB8814057D0 (en) * | 1988-06-14 | 1988-07-20 | Lundbeck & Co As H | New enantiomers & their isolation |
| ZA977967B (en) * | 1996-09-23 | 1999-03-04 | Lilly Co Eli | Combination therapy for treatment of psychoses |
| US6960577B2 (en) * | 1998-05-22 | 2005-11-01 | Eli Lilly And Company | Combination therapy for treatment of refractory depression |
| US6556540B1 (en) * | 1998-05-29 | 2003-04-29 | Paradyne Corporation | System and method for non-intrusive measurement of service quality in a communications network |
| SK287140B6 (sk) * | 1999-10-25 | 2010-01-07 | H. Lundbeck A/S | Spôsob prípravy citalopramu a medziprodukt na jeho výrobu |
| UA77650C2 (en) * | 1999-12-06 | 2007-01-15 | Lundbeck & Co As H | Use of serotonin reuptake inhibitor in combination with deramcyclane |
| US20040198809A1 (en) * | 2001-05-01 | 2004-10-07 | Connie Sanchez | Use of enantiomeric pure escitalopram |
| WO2003086393A1 (en) * | 2002-04-12 | 2003-10-23 | Sepracor, Inc. | 3-aza- and 1,4-diaza-bicyclo[4.3.0]nonanes, and methods of use thereof |
| DE60312874T2 (de) * | 2002-06-20 | 2008-01-17 | H. Lundbeck A/S | Kombinationstherapie mit verwendung eines serotonin-wiederaufnahmehemmers |
| HU227534B1 (en) * | 2003-08-04 | 2011-08-29 | Richter Gedeon Nyrt | (thio)carbamoyl-cyclohexane derivatives, process for producing them and pharmaceutical compositions containing them |
| EA200600531A1 (ru) * | 2003-09-04 | 2006-08-25 | Х. Лундбекк А/С | Сочетание ингибитора обратного захвата серотонина и локсапина |
| HUP0500170A3 (en) * | 2005-02-03 | 2007-11-28 | Richter Gedeon Nyrt | Piperazine derivatives, process for producing them and pharmaceutical compositions containing them |
| TW200812993A (en) * | 2006-05-02 | 2008-03-16 | Lundbeck & Co As H | New uses of escitalopram |
| HU230748B1 (hu) * | 2007-05-11 | 2018-02-28 | Richter Gedeon Nyrt | Új piperazin só és előállítási eljárása |
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Also Published As
| Publication number | Publication date |
|---|---|
| PL2185155T3 (pl) | 2018-03-30 |
| CN101815519B (zh) | 2013-08-21 |
| US20110015208A1 (en) | 2011-01-20 |
| AU2008283989A1 (en) | 2009-02-12 |
| US20120028991A1 (en) | 2012-02-02 |
| KR20100059830A (ko) | 2010-06-04 |
| CA2695519A1 (en) | 2009-02-12 |
| EP2185155A1 (en) | 2010-05-19 |
| KR101612563B1 (ko) | 2016-04-14 |
| HK1144784A1 (en) | 2011-03-11 |
| HUE036004T2 (hu) | 2018-06-28 |
| MY157192A (en) | 2016-05-13 |
| CN101815519A (zh) | 2010-08-25 |
| NO2185155T3 (enExample) | 2018-03-03 |
| SI2185155T1 (en) | 2018-02-28 |
| EA018064B1 (ru) | 2013-05-30 |
| US20090036468A1 (en) | 2009-02-05 |
| JP5460594B2 (ja) | 2014-04-02 |
| HRP20171908T1 (hr) | 2018-01-26 |
| LT2185155T (lt) | 2017-12-11 |
| WO2009020897A1 (en) | 2009-02-12 |
| EP2185155A4 (en) | 2012-04-25 |
| EA201000280A1 (ru) | 2010-08-30 |
| EP2185155B1 (en) | 2017-10-04 |
| PT2185155T (pt) | 2018-01-04 |
| DK2185155T3 (en) | 2018-01-02 |
| CY1119828T1 (el) | 2018-06-27 |
| JP2010535790A (ja) | 2010-11-25 |
| AU2008283989B2 (en) | 2013-12-05 |
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