EA018064B1 - Способ лечения депрессии - Google Patents
Способ лечения депрессии Download PDFInfo
- Publication number
- EA018064B1 EA018064B1 EA201000280A EA201000280A EA018064B1 EA 018064 B1 EA018064 B1 EA 018064B1 EA 201000280 A EA201000280 A EA 201000280A EA 201000280 A EA201000280 A EA 201000280A EA 018064 B1 EA018064 B1 EA 018064B1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- escitalopram oxalate
- animals
- cariprazine
- treatment
- cariprazine hydrochloride
- Prior art date
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| PCT/US2008/072066 WO2009020897A1 (en) | 2007-08-03 | 2008-08-04 | Pharmaceutical compositions containing dopamine receptor ligands and methods of treatment using dopamine recptor ligands |
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Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI2317852T1 (sl) | 2008-07-16 | 2015-04-30 | Richter Gedeon Nyrt. | Farmacevtske formulacije, ki vsebujejo ligande dopaminskega receptorja |
| US20110117214A1 (en) * | 2009-11-16 | 2011-05-19 | Auspex Pharmaceuticals, Inc. | Cyclohexyl urea modulators of d2 receptors and/or d3 receptors |
| JP5860457B2 (ja) | 2010-06-18 | 2016-02-16 | アルトス・セラピューティクス・リミテッド・ライアビリティ・カンパニーＡｌｔｏｓ Ｔｈｅｒａｐｅｕｔｉｃｓ，Ｌｌｃ | Ｄ２アンタゴニスト、その合成方法および使用方法 |
| US8912197B2 (en) | 2012-08-20 | 2014-12-16 | Forest Laboratories Holdings Ltd. | Crystalline form of carbamoyl-cyclohexane derivatives |
| US11274087B2 (en) | 2016-07-08 | 2022-03-15 | Richter Gedeon Nyrt. | Industrial process for the preparation of cariprazine |
| HUP1700253A1 (hu) * | 2017-06-13 | 2019-01-28 | Richter Gedeon Nyrt | Szilárd orális gyógyszerkészítmények |
| GB2571696B (en) | 2017-10-09 | 2020-05-27 | Compass Pathways Ltd | Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced |
| US12459965B2 (en) | 2017-10-09 | 2025-11-04 | Compass Pathfinder Limited | Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use |
| US11547707B2 (en) | 2019-04-10 | 2023-01-10 | Richter Gedeon Nyrt. | Carbamoyl cyclohexane derivatives for treating autism spectrum disorder |
| HU231500B1 (hu) * | 2019-04-10 | 2024-04-28 | Richter Gedeon Nyrt | Karbamoil-ciklohexán származékok autizmus spektrum betegség kezelésére |
| WO2020212951A1 (en) | 2019-04-17 | 2020-10-22 | Compass Pathfinder Limited | Methods for treating anxiety disorders, headache disorders, and eating disorders with psilocybin |
| EP4422629A4 (en) * | 2021-10-28 | 2025-09-03 | Richter Gedeon Nyrt | TREATMENT OF MAJOR DEPRESSIVE DISORDER |
| JP2025500844A (ja) * | 2021-12-13 | 2025-01-15 | コンパス パスファインダー リミテッド | 治療抵抗性うつ病の治療に使用するためのサイロシビン及び補助的セロトニン再取り込み阻害剤 |
| CA3244202A1 (en) * | 2022-03-17 | 2023-09-21 | Mapi Pharma Ltd | DEPOSIT SYSTEMS INCLUDING CARIPRAZINE OR SALTS THEREOF |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US7030122B2 (en) * | 2002-04-12 | 2006-04-18 | Sepracor Inc. | 1,4-disubstituted piperazine ligands for neurotransmitter receptors |
| US20060229297A1 (en) * | 2003-08-04 | 2006-10-12 | Richter Gedeon Vegyeszeti Gyar Rt. | (THIO) Carbamoyl-cyclohexane derivatives as D3/D2 receptor antagonists |
| US20070042014A1 (en) * | 2003-09-04 | 2007-02-22 | H. Lundbeck A/S | Combination of a serotonin reuptake inhibitor and loxapine |
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| GB8814057D0 (en) * | 1988-06-14 | 1988-07-20 | Lundbeck & Co As H | New enantiomers & their isolation |
| ZA977967B (en) * | 1996-09-23 | 1999-03-04 | Lilly Co Eli | Combination therapy for treatment of psychoses |
| US6960577B2 (en) * | 1998-05-22 | 2005-11-01 | Eli Lilly And Company | Combination therapy for treatment of refractory depression |
| US6556540B1 (en) * | 1998-05-29 | 2003-04-29 | Paradyne Corporation | System and method for non-intrusive measurement of service quality in a communications network |
| SK287140B6 (sk) * | 1999-10-25 | 2010-01-07 | H. Lundbeck A/S | Spôsob prípravy citalopramu a medziprodukt na jeho výrobu |
| UA77650C2 (en) * | 1999-12-06 | 2007-01-15 | Lundbeck & Co As H | Use of serotonin reuptake inhibitor in combination with deramcyclane |
| US20040198809A1 (en) * | 2001-05-01 | 2004-10-07 | Connie Sanchez | Use of enantiomeric pure escitalopram |
| DE60312874T2 (de) * | 2002-06-20 | 2008-01-17 | H. Lundbeck A/S | Kombinationstherapie mit verwendung eines serotonin-wiederaufnahmehemmers |
| HUP0500170A3 (en) * | 2005-02-03 | 2007-11-28 | Richter Gedeon Nyrt | Piperazine derivatives, process for producing them and pharmaceutical compositions containing them |
| TW200812993A (en) * | 2006-05-02 | 2008-03-16 | Lundbeck & Co As H | New uses of escitalopram |
| HU230748B1 (hu) * | 2007-05-11 | 2018-02-28 | Richter Gedeon Nyrt | Új piperazin só és előállítási eljárása |
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| US7030122B2 (en) * | 2002-04-12 | 2006-04-18 | Sepracor Inc. | 1,4-disubstituted piperazine ligands for neurotransmitter receptors |
| US20060229297A1 (en) * | 2003-08-04 | 2006-10-12 | Richter Gedeon Vegyeszeti Gyar Rt. | (THIO) Carbamoyl-cyclohexane derivatives as D3/D2 receptor antagonists |
| US20070042014A1 (en) * | 2003-09-04 | 2007-02-22 | H. Lundbeck A/S | Combination of a serotonin reuptake inhibitor and loxapine |
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| US20120028991A1 (en) | 2012-02-02 |
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| EP2185155A1 (en) | 2010-05-19 |
| KR101612563B1 (ko) | 2016-04-14 |
| HK1144784A1 (en) | 2011-03-11 |
| HUE036004T2 (hu) | 2018-06-28 |
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| CN101815519A (zh) | 2010-08-25 |
| NO2185155T3 (enExample) | 2018-03-03 |
| SI2185155T1 (en) | 2018-02-28 |
| ES2653852T3 (es) | 2018-02-09 |
| US20090036468A1 (en) | 2009-02-05 |
| JP5460594B2 (ja) | 2014-04-02 |
| HRP20171908T1 (hr) | 2018-01-26 |
| LT2185155T (lt) | 2017-12-11 |
| WO2009020897A1 (en) | 2009-02-12 |
| EP2185155A4 (en) | 2012-04-25 |
| EA201000280A1 (ru) | 2010-08-30 |
| EP2185155B1 (en) | 2017-10-04 |
| PT2185155T (pt) | 2018-01-04 |
| DK2185155T3 (en) | 2018-01-02 |
| CY1119828T1 (el) | 2018-06-27 |
| JP2010535790A (ja) | 2010-11-25 |
| AU2008283989B2 (en) | 2013-12-05 |
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