CA2695519A1 - Pharmaceutical compositions containing dopamine receptor ligands and methods of treatment using dopamine receptor ligands - Google Patents
Pharmaceutical compositions containing dopamine receptor ligands and methods of treatment using dopamine receptor ligands Download PDFInfo
- Publication number
- CA2695519A1 CA2695519A1 CA2695519A CA2695519A CA2695519A1 CA 2695519 A1 CA2695519 A1 CA 2695519A1 CA 2695519 A CA2695519 A CA 2695519A CA 2695519 A CA2695519 A CA 2695519A CA 2695519 A1 CA2695519 A1 CA 2695519A1
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- Prior art keywords
- disorder
- escitalopram
- serotonin reuptake
- selective serotonin
- pharmaceutically acceptable
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- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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Landscapes
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| PCT/US2008/072066 WO2009020897A1 (en) | 2007-08-03 | 2008-08-04 | Pharmaceutical compositions containing dopamine receptor ligands and methods of treatment using dopamine recptor ligands |
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| US20110117214A1 (en) * | 2009-11-16 | 2011-05-19 | Auspex Pharmaceuticals, Inc. | Cyclohexyl urea modulators of d2 receptors and/or d3 receptors |
| ES2612471T3 (es) * | 2010-06-18 | 2017-05-17 | Altos Therapeutics, LLC | Antagonistas D2, métodos de síntesis y métodos de uso |
| US8912197B2 (en) | 2012-08-20 | 2014-12-16 | Forest Laboratories Holdings Ltd. | Crystalline form of carbamoyl-cyclohexane derivatives |
| US11274087B2 (en) | 2016-07-08 | 2022-03-15 | Richter Gedeon Nyrt. | Industrial process for the preparation of cariprazine |
| HUP1700253A1 (hu) * | 2017-06-13 | 2019-01-28 | Richter Gedeon Nyrt | Szilárd orális gyógyszerkészítmények |
| GB2571696B (en) | 2017-10-09 | 2020-05-27 | Compass Pathways Ltd | Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced |
| US12459965B2 (en) | 2017-10-09 | 2025-11-04 | Compass Pathfinder Limited | Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use |
| HU231500B1 (hu) | 2019-04-10 | 2024-04-28 | Richter Gedeon Nyrt | Karbamoil-ciklohexán származékok autizmus spektrum betegség kezelésére |
| US11547707B2 (en) | 2019-04-10 | 2023-01-10 | Richter Gedeon Nyrt. | Carbamoyl cyclohexane derivatives for treating autism spectrum disorder |
| US12377112B2 (en) | 2019-04-17 | 2025-08-05 | Compass Pathfinder Limited | Methods of treating neurocognitive disorders, chronic pain and reducing inflammation |
| JP2024537491A (ja) * | 2021-10-28 | 2024-10-10 | アッヴィ・インコーポレイテッド | 大うつ病性障害の治療 |
| JP2025500844A (ja) * | 2021-12-13 | 2025-01-15 | コンパス パスファインダー リミテッド | 治療抵抗性うつ病の治療に使用するためのサイロシビン及び補助的セロトニン再取り込み阻害剤 |
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| GB8814057D0 (en) * | 1988-06-14 | 1988-07-20 | Lundbeck & Co As H | New enantiomers & their isolation |
| ZA977967B (en) * | 1996-09-23 | 1999-03-04 | Lilly Co Eli | Combination therapy for treatment of psychoses |
| US6960577B2 (en) * | 1998-05-22 | 2005-11-01 | Eli Lilly And Company | Combination therapy for treatment of refractory depression |
| US6556540B1 (en) * | 1998-05-29 | 2003-04-29 | Paradyne Corporation | System and method for non-intrusive measurement of service quality in a communications network |
| DK1298124T3 (da) * | 1999-10-25 | 2007-07-09 | Lundbeck & Co As H | Fremgangsmåde til fremstilling af citalopram |
| UA77650C2 (en) * | 1999-12-06 | 2007-01-15 | Lundbeck & Co As H | Use of serotonin reuptake inhibitor in combination with deramcyclane |
| CZ20033267A3 (en) * | 2001-05-01 | 2004-06-16 | H. Lundbeck A/S | The use of enantiomeric pure escitalopram |
| WO2003086393A1 (en) * | 2002-04-12 | 2003-10-23 | Sepracor, Inc. | 3-aza- and 1,4-diaza-bicyclo[4.3.0]nonanes, and methods of use thereof |
| AU2003240434A1 (en) * | 2002-06-20 | 2004-01-06 | H. Lundbeck A/S | Combination therapy wherein a serotinin reuptake inhibitor is used |
| HU227534B1 (en) * | 2003-08-04 | 2011-08-29 | Richter Gedeon Nyrt | (thio)carbamoyl-cyclohexane derivatives, process for producing them and pharmaceutical compositions containing them |
| ZA200601459B (en) * | 2003-09-04 | 2007-05-30 | Lundbeck & Co As H | The combination of a serotonin reuptake inhibitor and Loxapine |
| HUP0500170A3 (en) * | 2005-02-03 | 2007-11-28 | Richter Gedeon Nyrt | Piperazine derivatives, process for producing them and pharmaceutical compositions containing them |
| TW200812993A (en) * | 2006-05-02 | 2008-03-16 | Lundbeck & Co As H | New uses of escitalopram |
| HU230748B1 (hu) * | 2007-05-11 | 2018-02-28 | Richter Gedeon Nyrt | Új piperazin só és előállítási eljárása |
-
2008
- 2008-08-04 EP EP08782602.0A patent/EP2185155B1/en active Active
- 2008-08-04 WO PCT/US2008/072066 patent/WO2009020897A1/en not_active Ceased
- 2008-08-04 DK DK08782602.0T patent/DK2185155T3/en active
- 2008-08-04 HU HUE08782602A patent/HUE036004T2/hu unknown
- 2008-08-04 US US12/185,211 patent/US20090036468A1/en not_active Abandoned
- 2008-08-04 KR KR1020107004638A patent/KR101612563B1/ko active Active
- 2008-08-04 JP JP2010520238A patent/JP5460594B2/ja active Active
- 2008-08-04 PL PL08782602T patent/PL2185155T3/pl unknown
- 2008-08-04 PT PT87826020T patent/PT2185155T/pt unknown
- 2008-08-04 AU AU2008283989A patent/AU2008283989B2/en active Active
- 2008-08-04 NO NO08782602A patent/NO2185155T3/no unknown
- 2008-08-04 LT LTEP08782602.0T patent/LT2185155T/lt unknown
- 2008-08-04 EA EA201000280A patent/EA018064B1/ru unknown
- 2008-08-04 HR HRP20171908TT patent/HRP20171908T1/hr unknown
- 2008-08-04 ES ES08782602.0T patent/ES2653852T3/es active Active
- 2008-08-04 CA CA2695519A patent/CA2695519A1/en not_active Abandoned
- 2008-08-04 CN CN2008801062563A patent/CN101815519B/zh active Active
- 2008-08-04 MY MYPI2010000523A patent/MY157192A/en unknown
- 2008-08-04 SI SI200831900T patent/SI2185155T1/en unknown
-
2010
- 2010-09-27 US US12/890,752 patent/US20110015208A1/en not_active Abandoned
-
2011
- 2011-10-10 US US13/269,928 patent/US20120028991A1/en not_active Abandoned
-
2017
- 2017-12-07 CY CY20171101293T patent/CY1119828T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2653852T3 (es) | 2018-02-09 |
| PT2185155T (pt) | 2018-01-04 |
| US20110015208A1 (en) | 2011-01-20 |
| HUE036004T2 (hu) | 2018-06-28 |
| LT2185155T (lt) | 2017-12-11 |
| KR20100059830A (ko) | 2010-06-04 |
| EA201000280A1 (ru) | 2010-08-30 |
| EP2185155A1 (en) | 2010-05-19 |
| CY1119828T1 (el) | 2018-06-27 |
| EP2185155B1 (en) | 2017-10-04 |
| PL2185155T3 (pl) | 2018-03-30 |
| SI2185155T1 (en) | 2018-02-28 |
| HRP20171908T1 (hr) | 2018-01-26 |
| US20120028991A1 (en) | 2012-02-02 |
| NO2185155T3 (enExample) | 2018-03-03 |
| DK2185155T3 (en) | 2018-01-02 |
| EA018064B1 (ru) | 2013-05-30 |
| CN101815519A (zh) | 2010-08-25 |
| KR101612563B1 (ko) | 2016-04-14 |
| CN101815519B (zh) | 2013-08-21 |
| HK1144784A1 (en) | 2011-03-11 |
| US20090036468A1 (en) | 2009-02-05 |
| JP2010535790A (ja) | 2010-11-25 |
| AU2008283989B2 (en) | 2013-12-05 |
| AU2008283989A1 (en) | 2009-02-12 |
| MY157192A (en) | 2016-05-13 |
| JP5460594B2 (ja) | 2014-04-02 |
| WO2009020897A1 (en) | 2009-02-12 |
| EP2185155A4 (en) | 2012-04-25 |
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| Date | Code | Title | Description |
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| EEER | Examination request | ||
| FZDE | Discontinued |
Effective date: 20131101 |