ES2653852T3 - Composiciones farmacéuticas que contienen ligandos del receptor de dopamina y procedimientos de tratamiento usando ligandos del receptor de dopamina - Google Patents
Composiciones farmacéuticas que contienen ligandos del receptor de dopamina y procedimientos de tratamiento usando ligandos del receptor de dopamina Download PDFInfo
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- ES2653852T3 ES2653852T3 ES08782602.0T ES08782602T ES2653852T3 ES 2653852 T3 ES2653852 T3 ES 2653852T3 ES 08782602 T ES08782602 T ES 08782602T ES 2653852 T3 ES2653852 T3 ES 2653852T3
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- treatment
- cariprazine
- animals
- escitalopram oxalate
- cariprazine hydrochloride
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Classifications
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Epidemiology (AREA)
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- Psychology (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Otolaryngology (AREA)
- Addiction (AREA)
- Pregnancy & Childbirth (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US95369407P | 2007-08-03 | 2007-08-03 | |
| US953694P | 2007-08-03 | ||
| PCT/US2008/072066 WO2009020897A1 (en) | 2007-08-03 | 2008-08-04 | Pharmaceutical compositions containing dopamine receptor ligands and methods of treatment using dopamine recptor ligands |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2653852T3 true ES2653852T3 (es) | 2018-02-09 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| ES08782602.0T Active ES2653852T3 (es) | 2007-08-03 | 2008-08-04 | Composiciones farmacéuticas que contienen ligandos del receptor de dopamina y procedimientos de tratamiento usando ligandos del receptor de dopamina |
Country Status (20)
| Country | Link |
|---|---|
| US (3) | US20090036468A1 (OSRAM) |
| EP (1) | EP2185155B1 (OSRAM) |
| JP (1) | JP5460594B2 (OSRAM) |
| KR (1) | KR101612563B1 (OSRAM) |
| CN (1) | CN101815519B (OSRAM) |
| AU (1) | AU2008283989B2 (OSRAM) |
| CA (1) | CA2695519A1 (OSRAM) |
| CY (1) | CY1119828T1 (OSRAM) |
| DK (1) | DK2185155T3 (OSRAM) |
| EA (1) | EA018064B1 (OSRAM) |
| ES (1) | ES2653852T3 (OSRAM) |
| HR (1) | HRP20171908T1 (OSRAM) |
| HU (1) | HUE036004T2 (OSRAM) |
| LT (1) | LT2185155T (OSRAM) |
| MY (1) | MY157192A (OSRAM) |
| NO (1) | NO2185155T3 (OSRAM) |
| PL (1) | PL2185155T3 (OSRAM) |
| PT (1) | PT2185155T (OSRAM) |
| SI (1) | SI2185155T1 (OSRAM) |
| WO (1) | WO2009020897A1 (OSRAM) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
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| NZ590852A (en) | 2008-07-16 | 2013-03-28 | Richter Gedeon Nyrt | Pharmaceutical formulations containing dopamine receptor ligands trans-1{ 4-[2-[4-(2,3-dichlorophenyl)-piperizin-1-yl]-ethyl]-cyclohexyl} -3,3-dimethyl-urea also known as cariprazine |
| US20110117214A1 (en) * | 2009-11-16 | 2011-05-19 | Auspex Pharmaceuticals, Inc. | Cyclohexyl urea modulators of d2 receptors and/or d3 receptors |
| HUE031556T2 (en) * | 2010-06-18 | 2017-07-28 | Altos Therapeutics Llc | D2 antagonists, methods of synthesis and methods of use |
| WO2014031162A1 (en) | 2012-08-20 | 2014-02-27 | Forest Laboratories Holdings Limited | Crystalline form of carbamoyl-cyclohexane derivatives |
| US11274087B2 (en) | 2016-07-08 | 2022-03-15 | Richter Gedeon Nyrt. | Industrial process for the preparation of cariprazine |
| HUP1700253A1 (hu) * | 2017-06-13 | 2019-01-28 | Richter Gedeon Nyrt | Szilárd orális gyógyszerkészítmények |
| US12459965B2 (en) | 2017-10-09 | 2025-11-04 | Compass Pathfinder Limited | Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use |
| GB2571696B (en) | 2017-10-09 | 2020-05-27 | Compass Pathways Ltd | Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced |
| HU231500B1 (hu) * | 2019-04-10 | 2024-04-28 | Richter Gedeon Nyrt | Karbamoil-ciklohexán származékok autizmus spektrum betegség kezelésére |
| US11547707B2 (en) | 2019-04-10 | 2023-01-10 | Richter Gedeon Nyrt. | Carbamoyl cyclohexane derivatives for treating autism spectrum disorder |
| AU2020258086A1 (en) | 2019-04-17 | 2021-11-11 | Compass Pathfinder Limited | Methods of treating neurocognitive disorders, chronic pain and reducing inflammation |
| US20230149392A1 (en) * | 2021-10-28 | 2023-05-18 | Abbvie Inc. | Treatment of major depressive disorder |
| JP2025500844A (ja) * | 2021-12-13 | 2025-01-15 | コンパス パスファインダー リミテッド | 治療抵抗性うつ病の治療に使用するためのサイロシビン及び補助的セロトニン再取り込み阻害剤 |
| CN119136804A (zh) * | 2022-03-17 | 2024-12-13 | Mapi医药公司 | 包含卡利拉嗪或其盐的储库系统 |
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| GB8814057D0 (en) * | 1988-06-14 | 1988-07-20 | Lundbeck & Co As H | New enantiomers & their isolation |
| ZA977967B (en) * | 1996-09-23 | 1999-03-04 | Lilly Co Eli | Combination therapy for treatment of psychoses |
| US6960577B2 (en) * | 1998-05-22 | 2005-11-01 | Eli Lilly And Company | Combination therapy for treatment of refractory depression |
| US6556540B1 (en) * | 1998-05-29 | 2003-04-29 | Paradyne Corporation | System and method for non-intrusive measurement of service quality in a communications network |
| HRP20020344B1 (hr) * | 1999-10-25 | 2010-10-31 | H. Lundbeck A/S | Način priprave citaloprama |
| UA77650C2 (en) * | 1999-12-06 | 2007-01-15 | Lundbeck & Co As H | Use of serotonin reuptake inhibitor in combination with deramcyclane |
| YU85303A (sh) * | 2001-05-01 | 2006-05-25 | H. Lundbeck A/S | Upotreba enantiomerno čistog escitaloprama |
| US7030122B2 (en) * | 2002-04-12 | 2006-04-18 | Sepracor Inc. | 1,4-disubstituted piperazine ligands for neurotransmitter receptors |
| DE60312874T2 (de) * | 2002-06-20 | 2008-01-17 | H. Lundbeck A/S | Kombinationstherapie mit verwendung eines serotonin-wiederaufnahmehemmers |
| HU227534B1 (en) * | 2003-08-04 | 2011-08-29 | Richter Gedeon Nyrt | (thio)carbamoyl-cyclohexane derivatives, process for producing them and pharmaceutical compositions containing them |
| US20070042014A1 (en) * | 2003-09-04 | 2007-02-22 | H. Lundbeck A/S | Combination of a serotonin reuptake inhibitor and loxapine |
| HUP0500170A3 (en) * | 2005-02-03 | 2007-11-28 | Richter Gedeon Nyrt | Piperazine derivatives, process for producing them and pharmaceutical compositions containing them |
| TW200812993A (en) * | 2006-05-02 | 2008-03-16 | Lundbeck & Co As H | New uses of escitalopram |
| HU230748B1 (hu) * | 2007-05-11 | 2018-02-28 | Richter Gedeon Nyrt | Új piperazin só és előállítási eljárása |
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- 2008-08-04 SI SI200831900T patent/SI2185155T1/en unknown
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2010
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2011
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2017
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Also Published As
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|---|---|
| WO2009020897A1 (en) | 2009-02-12 |
| US20110015208A1 (en) | 2011-01-20 |
| SI2185155T1 (en) | 2018-02-28 |
| EP2185155A4 (en) | 2012-04-25 |
| EP2185155A1 (en) | 2010-05-19 |
| DK2185155T3 (en) | 2018-01-02 |
| HUE036004T2 (hu) | 2018-06-28 |
| EA201000280A1 (ru) | 2010-08-30 |
| NO2185155T3 (OSRAM) | 2018-03-03 |
| MY157192A (en) | 2016-05-13 |
| PT2185155T (pt) | 2018-01-04 |
| PL2185155T3 (pl) | 2018-03-30 |
| JP2010535790A (ja) | 2010-11-25 |
| CN101815519B (zh) | 2013-08-21 |
| EP2185155B1 (en) | 2017-10-04 |
| US20120028991A1 (en) | 2012-02-02 |
| US20090036468A1 (en) | 2009-02-05 |
| HK1144784A1 (en) | 2011-03-11 |
| LT2185155T (lt) | 2017-12-11 |
| AU2008283989B2 (en) | 2013-12-05 |
| CY1119828T1 (el) | 2018-06-27 |
| KR20100059830A (ko) | 2010-06-04 |
| EA018064B1 (ru) | 2013-05-30 |
| HRP20171908T1 (hr) | 2018-01-26 |
| JP5460594B2 (ja) | 2014-04-02 |
| AU2008283989A1 (en) | 2009-02-12 |
| CA2695519A1 (en) | 2009-02-12 |
| CN101815519A (zh) | 2010-08-25 |
| KR101612563B1 (ko) | 2016-04-14 |
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