ES2398348T3 - Sistema de administración de fármacos controlada por retención gástrica - Google Patents
Sistema de administración de fármacos controlada por retención gástrica Download PDFInfo
- Publication number
- ES2398348T3 ES2398348T3 ES10165807T ES10165807T ES2398348T3 ES 2398348 T3 ES2398348 T3 ES 2398348T3 ES 10165807 T ES10165807 T ES 10165807T ES 10165807 T ES10165807 T ES 10165807T ES 2398348 T3 ES2398348 T3 ES 2398348T3
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- Prior art keywords
- baclofen
- core
- controlled
- drug delivery
- release
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- Expired - Lifetime
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- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0065—Forms with gastric retention, e.g. floating on gastric juice, adhering to gastric mucosa, expanding to prevent passage through the pylorus
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
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-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- Health & Medical Sciences (AREA)
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- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nutrition Science (AREA)
- Neurology (AREA)
- Physiology (AREA)
- Neurosurgery (AREA)
- Urology & Nephrology (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| INMU06122001 | 2001-07-04 | ||
| IN612MU2001 | 2001-07-04 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2398348T3 true ES2398348T3 (es) | 2013-03-15 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES10165807T Expired - Lifetime ES2398348T3 (es) | 2001-07-04 | 2002-07-04 | Sistema de administración de fármacos controlada por retención gástrica |
Country Status (17)
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|---|---|
| US (2) | US7776345B2 (https=) |
| EP (2) | EP1411901B1 (https=) |
| JP (2) | JP4994570B2 (https=) |
| KR (1) | KR20040018394A (https=) |
| CN (1) | CN1520286B (https=) |
| AT (1) | ATE477795T1 (https=) |
| AU (1) | AU2002355686B2 (https=) |
| BR (1) | BR0211317A (https=) |
| CA (1) | CA2452738C (https=) |
| DE (1) | DE60237372D1 (https=) |
| ES (1) | ES2398348T3 (https=) |
| HU (1) | HUP0500795A3 (https=) |
| MX (1) | MXPA03012041A (https=) |
| PL (1) | PL370793A1 (https=) |
| RU (1) | RU2325152C2 (https=) |
| WO (1) | WO2003011255A1 (https=) |
| ZA (1) | ZA200400799B (https=) |
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-
2002
- 2002-07-04 MX MXPA03012041A patent/MXPA03012041A/es active IP Right Grant
- 2002-07-04 CA CA2452738A patent/CA2452738C/en not_active Expired - Fee Related
- 2002-07-04 AT AT02751608T patent/ATE477795T1/de not_active IP Right Cessation
- 2002-07-04 DE DE60237372T patent/DE60237372D1/de not_active Expired - Lifetime
- 2002-07-04 BR BR0211317-1A patent/BR0211317A/pt not_active Application Discontinuation
- 2002-07-04 US US10/482,770 patent/US7776345B2/en active Active
- 2002-07-04 AU AU2002355686A patent/AU2002355686B2/en not_active Ceased
- 2002-07-04 EP EP02751608A patent/EP1411901B1/en not_active Expired - Lifetime
- 2002-07-04 PL PL02370793A patent/PL370793A1/xx unknown
- 2002-07-04 CN CN028128575A patent/CN1520286B/zh not_active Expired - Lifetime
- 2002-07-04 RU RU2003138075/15A patent/RU2325152C2/ru not_active IP Right Cessation
- 2002-07-04 ES ES10165807T patent/ES2398348T3/es not_active Expired - Lifetime
- 2002-07-04 JP JP2003516487A patent/JP4994570B2/ja not_active Expired - Fee Related
- 2002-07-04 KR KR10-2003-7016967A patent/KR20040018394A/ko not_active Ceased
- 2002-07-04 WO PCT/IN2002/000144 patent/WO2003011255A1/en not_active Ceased
- 2002-07-04 EP EP10165807A patent/EP2238975B1/en not_active Expired - Lifetime
- 2002-07-04 HU HU0500795A patent/HUP0500795A3/hu unknown
-
2004
- 2004-01-30 ZA ZA2004/00799A patent/ZA200400799B/en unknown
-
2009
- 2009-12-11 JP JP2009281402A patent/JP2010090161A/ja active Pending
-
2010
- 2010-08-13 US US12/856,097 patent/US8012496B2/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| EP1411901B1 (en) | 2010-08-18 |
| CA2452738C (en) | 2011-06-14 |
| US7776345B2 (en) | 2010-08-17 |
| MXPA03012041A (es) | 2004-03-26 |
| KR20040018394A (ko) | 2004-03-03 |
| CN1520286B (zh) | 2010-12-01 |
| JP2010090161A (ja) | 2010-04-22 |
| ATE477795T1 (de) | 2010-09-15 |
| CA2452738A1 (en) | 2003-02-13 |
| EP2238975B1 (en) | 2012-12-05 |
| US8012496B2 (en) | 2011-09-06 |
| JP4994570B2 (ja) | 2012-08-08 |
| US20040180088A1 (en) | 2004-09-16 |
| ZA200400799B (en) | 2005-07-27 |
| PL370793A1 (en) | 2005-05-30 |
| WO2003011255A1 (en) | 2003-02-13 |
| AU2002355686B2 (en) | 2007-11-29 |
| RU2003138075A (ru) | 2005-06-10 |
| BR0211317A (pt) | 2004-12-14 |
| EP2238975A1 (en) | 2010-10-13 |
| RU2325152C2 (ru) | 2008-05-27 |
| HUP0500795A2 (en) | 2007-02-28 |
| DE60237372D1 (de) | 2010-09-30 |
| EP1411901A1 (en) | 2004-04-28 |
| HUP0500795A3 (en) | 2008-04-28 |
| US20100305208A1 (en) | 2010-12-02 |
| JP2004538301A (ja) | 2004-12-24 |
| CN1520286A (zh) | 2004-08-11 |
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