ES2336911T3 - Trans-9,10-dehidroepotilonas c y d, sus analogos y procedimientos de preparacion. - Google Patents
Trans-9,10-dehidroepotilonas c y d, sus analogos y procedimientos de preparacion. Download PDFInfo
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- ES2336911T3 ES2336911T3 ES03768730T ES03768730T ES2336911T3 ES 2336911 T3 ES2336911 T3 ES 2336911T3 ES 03768730 T ES03768730 T ES 03768730T ES 03768730 T ES03768730 T ES 03768730T ES 2336911 T3 ES2336911 T3 ES 2336911T3
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- WRIKHQLVHPKCJU-UHFFFAOYSA-N sodium bis(trimethylsilyl)amide Chemical compound C[Si](C)(C)N([Na])[Si](C)(C)C WRIKHQLVHPKCJU-UHFFFAOYSA-N 0.000 description 22
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
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| US42535202P | 2002-11-07 | 2002-11-07 | |
| US425352P | 2002-11-07 | ||
| US47374303P | 2003-05-27 | 2003-05-27 | |
| US473743P | 2003-05-27 |
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| ES2336911T3 true ES2336911T3 (es) | 2010-04-19 |
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| ES09012671T Expired - Lifetime ES2436296T3 (es) | 2002-11-07 | 2003-11-07 | Trans-9,10-dehidroepotilona C y trans-9,10-dehidroepotilona D, sus análogos y procedimientos de fabricación de las mismas |
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| ES09012671T Expired - Lifetime ES2436296T3 (es) | 2002-11-07 | 2003-11-07 | Trans-9,10-dehidroepotilona C y trans-9,10-dehidroepotilona D, sus análogos y procedimientos de fabricación de las mismas |
Country Status (14)
| Country | Link |
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| US (2) | US20040152708A1 (OSRAM) |
| EP (3) | EP2135867B1 (OSRAM) |
| JP (3) | JP4641941B2 (OSRAM) |
| KR (2) | KR100996996B1 (OSRAM) |
| AT (1) | ATE452888T1 (OSRAM) |
| AU (1) | AU2003291337B2 (OSRAM) |
| CA (1) | CA2505368C (OSRAM) |
| CY (1) | CY1110295T1 (OSRAM) |
| DE (1) | DE60330703D1 (OSRAM) |
| DK (1) | DK1562941T3 (OSRAM) |
| ES (2) | ES2336911T3 (OSRAM) |
| PT (1) | PT1562941E (OSRAM) |
| SI (1) | SI1562941T1 (OSRAM) |
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| EP0977563B1 (en) | 1996-12-03 | 2005-10-12 | Sloan-Kettering Institute For Cancer Research | Synthesis of epothilones, intermediates thereto, analogues and uses thereof |
| US8618085B2 (en) * | 2000-04-28 | 2013-12-31 | Koasn Biosciences Incorporated | Therapeutic formulations of desoxyepothilones |
| US7649006B2 (en) | 2002-08-23 | 2010-01-19 | Sloan-Kettering Institute For Cancer Research | Synthesis of epothilones, intermediates thereto and analogues thereof |
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2003
- 2003-11-07 KR KR1020107000780A patent/KR100996996B1/ko not_active Expired - Fee Related
- 2003-11-07 EP EP09012671.5A patent/EP2135867B1/en not_active Expired - Lifetime
- 2003-11-07 EP EP09012860A patent/EP2135868A1/en not_active Withdrawn
- 2003-11-07 ES ES03768730T patent/ES2336911T3/es not_active Expired - Lifetime
- 2003-11-07 SI SI200331732T patent/SI1562941T1/sl unknown
- 2003-11-07 AT AT03768730T patent/ATE452888T1/de active
- 2003-11-07 DK DK03768730.8T patent/DK1562941T3/da active
- 2003-11-07 US US10/703,404 patent/US20040152708A1/en not_active Abandoned
- 2003-11-07 ES ES09012671T patent/ES2436296T3/es not_active Expired - Lifetime
- 2003-11-07 PT PT03768730T patent/PT1562941E/pt unknown
- 2003-11-07 WO PCT/US2003/035411 patent/WO2004043954A2/en not_active Ceased
- 2003-11-07 CA CA2505368A patent/CA2505368C/en not_active Expired - Fee Related
- 2003-11-07 DE DE60330703T patent/DE60330703D1/de not_active Expired - Lifetime
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- 2003-11-07 JP JP2005507102A patent/JP4641941B2/ja not_active Expired - Fee Related
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- 2008-07-11 US US12/172,174 patent/US20090186927A1/en not_active Abandoned
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| EP2135867B1 (en) | 2013-09-25 |
| PT1562941E (pt) | 2010-01-25 |
| CA2505368C (en) | 2011-09-20 |
| JP2011006480A (ja) | 2011-01-13 |
| ES2436296T3 (es) | 2013-12-30 |
| WO2004043954A3 (en) | 2004-11-18 |
| EP2135867A1 (en) | 2009-12-23 |
| SI1562941T1 (sl) | 2010-05-31 |
| DE60330703D1 (de) | 2010-02-04 |
| KR100996996B1 (ko) | 2010-11-25 |
| AU2003291337B2 (en) | 2010-09-09 |
| AU2003291337A1 (en) | 2004-06-03 |
| CA2505368A1 (en) | 2004-05-27 |
| JP5679757B2 (ja) | 2015-03-04 |
| JP2013213054A (ja) | 2013-10-17 |
| KR100966667B1 (ko) | 2010-06-29 |
| EP2135868A1 (en) | 2009-12-23 |
| JP4641941B2 (ja) | 2011-03-02 |
| EP1562941A2 (en) | 2005-08-17 |
| ATE452888T1 (de) | 2010-01-15 |
| JP2006510743A (ja) | 2006-03-30 |
| KR20100018075A (ko) | 2010-02-16 |
| KR20050084959A (ko) | 2005-08-29 |
| WO2004043954A2 (en) | 2004-05-27 |
| US20040152708A1 (en) | 2004-08-05 |
| DK1562941T3 (da) | 2010-04-19 |
| EP1562941B1 (en) | 2009-12-23 |
| US20090186927A1 (en) | 2009-07-23 |
| CY1110295T1 (el) | 2015-01-14 |
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