ES2262893T3 - Derivados de imidazo-piridina para su uso en el tratamiento de infeccion virica por herpes. - Google Patents

Derivados de imidazo-piridina para su uso en el tratamiento de infeccion virica por herpes.

Info

Publication number
ES2262893T3
ES2262893T3 ES02800844T ES02800844T ES2262893T3 ES 2262893 T3 ES2262893 T3 ES 2262893T3 ES 02800844 T ES02800844 T ES 02800844T ES 02800844 T ES02800844 T ES 02800844T ES 2262893 T3 ES2262893 T3 ES 2262893T3
Authority
ES
Spain
Prior art keywords
formula
compound
group
het
cycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES02800844T
Other languages
English (en)
Spanish (es)
Inventor
Kristjan GlaxoSmithKline GUDMUNDSSON
Brian A. GlaxoSmithKline JOHNS
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Corp
Original Assignee
SmithKline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Corp filed Critical SmithKline Beecham Corp
Application granted granted Critical
Publication of ES2262893T3 publication Critical patent/ES2262893T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biotechnology (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ES02800844T 2001-10-05 2002-09-23 Derivados de imidazo-piridina para su uso en el tratamiento de infeccion virica por herpes. Expired - Lifetime ES2262893T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32770501P 2001-10-05 2001-10-05
US327705P 2001-10-05

Publications (1)

Publication Number Publication Date
ES2262893T3 true ES2262893T3 (es) 2006-12-01

Family

ID=23277681

Family Applications (1)

Application Number Title Priority Date Filing Date
ES02800844T Expired - Lifetime ES2262893T3 (es) 2001-10-05 2002-09-23 Derivados de imidazo-piridina para su uso en el tratamiento de infeccion virica por herpes.

Country Status (7)

Country Link
US (2) US7244740B2 (enExample)
EP (1) EP1432712B1 (enExample)
JP (1) JP2005508955A (enExample)
AT (1) ATE326466T1 (enExample)
DE (1) DE60211539T2 (enExample)
ES (1) ES2262893T3 (enExample)
WO (1) WO2003031446A1 (enExample)

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UA103319C2 (en) 2008-05-06 2013-10-10 Глаксосмитклайн Ллк Thiazole- and oxazole-benzene sulfonamide compounds
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US8088771B2 (en) 2008-07-28 2012-01-03 Gilead Sciences, Inc. Cycloalkylidene and heterocycloalkylidene inhibitor compounds
US8283357B2 (en) 2009-06-08 2012-10-09 Gilead Sciences, Inc. Cycloalkylcarbamate benzamide aniline HDAC inhibitor compounds
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AU2010311511B2 (en) 2009-10-30 2014-07-17 Janssen Pharmaceutica Nv Imidazo[1,2-b]pyridazine derivatives and their use as PDE10 inhibitors
AR080754A1 (es) 2010-03-09 2012-05-09 Janssen Pharmaceutica Nv Derivados de imidazo (1,2-a) pirazina y su uso como inhibidores de pde10
MX344600B (es) 2011-06-27 2016-12-20 Janssen Pharmaceutica Nv Derivados de 1-aril-4-metil-[1,2,4]triazolo[4,3-a]quinoxalina.
AU2013283426B2 (en) 2012-06-26 2018-02-22 Janssen Pharmaceutica Nv Combinations comprising PDE 2 inhibitors such as 1-aryl-4-methyl- [1,2,4] triazolo [4,3-a] quinoxaline compounds and PDE 10 inhibitors for use in the treatment of neurological or metabolic disorders
CN104411314B (zh) 2012-07-09 2017-10-20 詹森药业有限公司 磷酸二酯酶10的抑制剂
SG11201907095UA (en) * 2017-02-01 2019-08-27 Aucentra Therapeutics Pty Ltd DERIVATIVES OF N-CYCLOALKYL/HETEROCYCLOALKYL-4-(IMIDAZO [1,2-a]PYRIDINE)PYRIMIDIN-2-AMINE AS THERAPEUTIC AGENTS
CN120829428A (zh) * 2024-04-18 2025-10-24 中国医学科学院药物研究所 咪唑并吡啶衍生物及其用途

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Also Published As

Publication number Publication date
DE60211539T2 (de) 2006-09-21
JP2005508955A (ja) 2005-04-07
EP1432712B1 (en) 2006-05-17
ATE326466T1 (de) 2006-06-15
US7244740B2 (en) 2007-07-17
EP1432712A1 (en) 2004-06-30
US20040248917A1 (en) 2004-12-09
DE60211539D1 (de) 2006-06-22
US20080139594A1 (en) 2008-06-12
WO2003031446A1 (en) 2003-04-17

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