ES2061247T3 - Imidazo (4,5-c) piridinas con actividad antagonista del paf. - Google Patents
Imidazo (4,5-c) piridinas con actividad antagonista del paf.Info
- Publication number
- ES2061247T3 ES2061247T3 ES91909431T ES91909431T ES2061247T3 ES 2061247 T3 ES2061247 T3 ES 2061247T3 ES 91909431 T ES91909431 T ES 91909431T ES 91909431 T ES91909431 T ES 91909431T ES 2061247 T3 ES2061247 T3 ES 2061247T3
- Authority
- ES
- Spain
- Prior art keywords
- paf
- imidazo
- piridinas
- antagonist activity
- leucotrene
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 239000005557 antagonist Substances 0.000 title 1
- HVAUUPRFYPCOCA-AREMUKBSSA-N 2-O-acetyl-1-O-hexadecyl-sn-glycero-3-phosphocholine Chemical compound CCCCCCCCCCCCCCCCOC[C@@H](OC(C)=O)COP([O-])(=O)OCC[N+](C)(C)C HVAUUPRFYPCOCA-AREMUKBSSA-N 0.000 abstract 2
- 108010003541 Platelet Activating Factor Proteins 0.000 abstract 2
- 206010008190 Cerebrovascular accident Diseases 0.000 abstract 1
- 208000018522 Gastrointestinal disease Diseases 0.000 abstract 1
- 201000004681 Psoriasis Diseases 0.000 abstract 1
- 208000006011 Stroke Diseases 0.000 abstract 1
- 206010003246 arthritis Diseases 0.000 abstract 1
- 208000006673 asthma Diseases 0.000 abstract 1
- 208000010125 myocardial infarction Diseases 0.000 abstract 1
- 230000035939 shock Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Rheumatology (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US52119990A | 1990-05-09 | 1990-05-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2061247T3 true ES2061247T3 (es) | 1994-12-01 |
Family
ID=24075786
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES91909431T Expired - Lifetime ES2061247T3 (es) | 1990-05-09 | 1991-05-01 | Imidazo (4,5-c) piridinas con actividad antagonista del paf. |
Country Status (28)
| Country | Link |
|---|---|
| EP (1) | EP0533695B1 (en, 2012) |
| JP (1) | JPH0678340B2 (en, 2012) |
| CN (1) | CN1057839A (en, 2012) |
| AP (1) | AP224A (en, 2012) |
| AT (1) | ATE112567T1 (en, 2012) |
| AU (1) | AU642265B2 (en, 2012) |
| BG (1) | BG97059A (en, 2012) |
| BR (1) | BR9106433A (en, 2012) |
| CA (1) | CA2080476A1 (en, 2012) |
| DE (1) | DE69104481T2 (en, 2012) |
| DK (1) | DK0533695T3 (en, 2012) |
| ES (1) | ES2061247T3 (en, 2012) |
| FI (1) | FI925053A0 (en, 2012) |
| GT (1) | GT199100031A (en, 2012) |
| HU (1) | HUT62894A (en, 2012) |
| IE (1) | IE911553A1 (en, 2012) |
| IL (1) | IL98075A0 (en, 2012) |
| MA (1) | MA22151A1 (en, 2012) |
| MY (1) | MY105512A (en, 2012) |
| NO (1) | NO924290D0 (en, 2012) |
| NZ (1) | NZ238089A (en, 2012) |
| PE (1) | PE26691A1 (en, 2012) |
| PT (1) | PT97616A (en, 2012) |
| RO (1) | RO109450B1 (en, 2012) |
| TW (1) | TW205549B (en, 2012) |
| WO (1) | WO1991017163A1 (en, 2012) |
| YU (1) | YU81191A (en, 2012) |
| ZA (1) | ZA913497B (en, 2012) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9102997D0 (en) * | 1991-02-13 | 1991-03-27 | Pfizer Ltd | Therapeutic agents |
| AU5016793A (en) * | 1992-08-20 | 1994-03-15 | Cytomed, Inc | Dual functional anti-inflammatory and immunosuppressive agents |
| US6372770B1 (en) | 1994-10-12 | 2002-04-16 | Euro-Celtique, S.A. | Benzoxazoles |
| CN1308622A (zh) * | 1998-05-12 | 2001-08-15 | 美国家用产品公司 | 用于治疗胰岛素抗性和高血糖的联苯基氧代－乙酸 |
| US6232322B1 (en) | 1998-05-12 | 2001-05-15 | American Home Products Corporation | Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia |
| US6310081B1 (en) | 1999-05-10 | 2001-10-30 | American Home Products Corporation | Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia |
| GB0302094D0 (en) | 2003-01-29 | 2003-02-26 | Pharmagene Lab Ltd | EP4 receptor antagonists |
| GB0324269D0 (en) | 2003-10-16 | 2003-11-19 | Pharmagene Lab Ltd | EP4 receptor antagonists |
| JP2016537398A (ja) * | 2013-09-13 | 2016-12-01 | コーテンドー エービー（ピーユービーエル）Ｃｏｒｔｅｎｄｏ Ａｂ（Ｐｕｂｌ） | 新規なチトクロムｐ４５０阻害剤及びこれらの使用方法 |
| CN105348182B (zh) * | 2014-08-24 | 2018-04-13 | 复旦大学 | 2‑烷氧基苯甲酰芳胺类化合物及其药物用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES8401486A1 (es) * | 1981-11-10 | 1983-12-01 | Wellcome Found | Un procedimiento para la preparacion de nuevos derivados de imidazo (4,5-c)piridina. |
| GB8804439D0 (en) * | 1988-02-25 | 1988-03-23 | Pfizer Ltd | Dihydropyridines |
| GB8822170D0 (en) * | 1988-09-21 | 1988-10-26 | Pfizer Ltd | Therapeutic agents |
-
1991
- 1991-05-01 FI FI925053A patent/FI925053A0/fi not_active Application Discontinuation
- 1991-05-01 BR BR919106433A patent/BR9106433A/pt not_active Application Discontinuation
- 1991-05-01 RO RO92-01395A patent/RO109450B1/ro unknown
- 1991-05-01 EP EP91909431A patent/EP0533695B1/en not_active Expired - Lifetime
- 1991-05-01 DE DE69104481T patent/DE69104481T2/de not_active Expired - Fee Related
- 1991-05-01 AT AT91909431T patent/ATE112567T1/de not_active IP Right Cessation
- 1991-05-01 DK DK91909431.8T patent/DK0533695T3/da active
- 1991-05-01 AU AU78671/91A patent/AU642265B2/en not_active Ceased
- 1991-05-01 JP JP3509156A patent/JPH0678340B2/ja not_active Expired - Fee Related
- 1991-05-01 CA CA002080476A patent/CA2080476A1/en not_active Abandoned
- 1991-05-01 ES ES91909431T patent/ES2061247T3/es not_active Expired - Lifetime
- 1991-05-01 HU HU923496A patent/HUT62894A/hu unknown
- 1991-05-01 WO PCT/US1991/002997 patent/WO1991017163A1/en active IP Right Grant
- 1991-05-07 IL IL98075A patent/IL98075A0/xx unknown
- 1991-05-08 TW TW080103606A patent/TW205549B/zh active
- 1991-05-08 MA MA22421A patent/MA22151A1/fr unknown
- 1991-05-08 AP APAP/P/1991/000259A patent/AP224A/en active
- 1991-05-08 NZ NZ238089A patent/NZ238089A/en unknown
- 1991-05-08 ZA ZA913497A patent/ZA913497B/xx unknown
- 1991-05-08 IE IE155391A patent/IE911553A1/en unknown
- 1991-05-08 MY MYPI91000776A patent/MY105512A/en unknown
- 1991-05-08 PE PE1991185432A patent/PE26691A1/es unknown
- 1991-05-08 CN CN91103959A patent/CN1057839A/zh active Pending
- 1991-05-09 PT PT97616A patent/PT97616A/pt not_active Application Discontinuation
- 1991-05-09 GT GT199100031A patent/GT199100031A/es unknown
- 1991-05-09 YU YU81191A patent/YU81191A/sh unknown
-
1992
- 1992-11-06 NO NO924290A patent/NO924290D0/no unknown
- 1992-11-06 BG BG097059A patent/BG97059A/bg unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| MX9203018A (es) | Fluoroalcoxibencilamino-derivados de heterociclos nitrogenados. | |
| DK326588D0 (da) | Cyclosporiner | |
| ES2138977T3 (es) | Agonistas muscarinicos. | |
| ES2195125T3 (es) | Nucleosidos l monociclicos, analogos, y empleos de los mismos. | |
| ES2061247T3 (es) | Imidazo (4,5-c) piridinas con actividad antagonista del paf. | |
| ES2184794T3 (es) | Profarmacos de morfolina como antagonistas de receptores de taquicininas. | |
| ES2128544T3 (es) | Pirrolopirimidinas como antagonistas del crf. | |
| ES2141133T3 (es) | Morfolina y tiomorfolina como antagonistas de receptores de taquiquininas. | |
| ES2162061T3 (es) | Derivados de piperidina como antagonistas de la neuroquinina. | |
| RU94002482A (ru) | Пятичленные гетероциклы, смесь их изомеров или отдельные изомеры и их соли | |
| ES2058306T3 (es) | Tetralinas substituidas, cromanos y compuestos relacionados en el tratamiento del asma, artritis y enfermedades relacionadas. | |
| ES2181995T3 (es) | Derivados de bencimidazol y uso como antagonistas del factor de liberacion de la corticotropina. | |
| CO4480024A1 (es) | Nuevos benzopiranos y otros antagonistas de b4(ltb4) leuco- triena fusionada con benzo | |
| IT1200657B (it) | Benzammidi sostituite farmacologicamente attive utili per il trattamento della emesi da chemioterapia | |
| ES2169150T3 (es) | Compuestos a base de dihidrobenzofurano y compuestos relacionados utiles como agentes anti-inflamatorios. | |
| CA1236699A (en) | RANKINE CYCLE ENERGY PLANT USING ENHANCED ORGANIC FLUID | |
| ES2062202T3 (es) | Derivado del indol. | |
| ES2063261T3 (es) | 1-(3-(heteroarilmetoxi)fenil) alcanoles sustituidos y compuestos relacionados en el tratamiento de asma, artritis y enfermedades relacionadas. | |
| IT1197713B (it) | Dicloro-derivati della serie del 16 alfa-metil pregnano,procedimento per la produzione,loro applicazione come medicamenti e composizioni che li contengono | |
| MX9300409A (es) | Hexahidroazepinonas y tetrahidrobenzoazepinonas sustituidas. | |
| ES539242A0 (es) | Maquina movil para excavar el balasto de las vias ferreas | |
| ES2062332T3 (es) | Benzoxazolonas antiinflamatorias. | |
| MX9305312A (es) | 2,4-diazepina aril-fusionada y hetaril-fusionada y agentes antiarritmicosde 2,4-diazocina. | |
| RU94014629A (ru) | Производные 4-хинолилдигидропиридина, смесь их изомеров или отдельные изомеры и их соли | |
| ES2152959T3 (es) | Utilizacion en perfumeria de isomeros opticamente activos del (e)-3,3-dimetil-5-(2,2,3-trimetil-3-ciclopenten-1-il)-4-penten-2-ol. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
Ref document number: 533695 Country of ref document: ES |