ES2000382A6 - Un procedimiento para la produccion de derivados de fenetilamina substituidos - Google Patents
Un procedimiento para la produccion de derivados de fenetilamina substituidosInfo
- Publication number
- ES2000382A6 ES2000382A6 ES8600685A ES8600685A ES2000382A6 ES 2000382 A6 ES2000382 A6 ES 2000382A6 ES 8600685 A ES8600685 A ES 8600685A ES 8600685 A ES8600685 A ES 8600685A ES 2000382 A6 ES2000382 A6 ES 2000382A6
- Authority
- ES
- Spain
- Prior art keywords
- formula
- reduced
- deriv
- phenethylamine
- aminopropyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- BHHGXPLMPWCGHP-UHFFFAOYSA-N Phenethylamine Chemical class NCCC1=CC=CC=C1 BHHGXPLMPWCGHP-UHFFFAOYSA-N 0.000 title abstract 5
- UHOVQNZJYSORNB-UHFFFAOYSA-N Benzene Chemical compound C1=CC=CC=C1 UHOVQNZJYSORNB-UHFFFAOYSA-N 0.000 abstract 3
- OKKJLVBELUTLKV-UHFFFAOYSA-N Methanol Chemical compound OC OKKJLVBELUTLKV-UHFFFAOYSA-N 0.000 abstract 3
- RTZKZFJDLAIYFH-UHFFFAOYSA-N Diethyl ether Chemical compound CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 abstract 2
- KDLHZDBZIXYQEI-UHFFFAOYSA-N Palladium Chemical compound [Pd] KDLHZDBZIXYQEI-UHFFFAOYSA-N 0.000 abstract 2
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 229940117803 phenethylamine Drugs 0.000 abstract 2
- XFFILAFLGDUMBF-UHFFFAOYSA-N 2-phenoxyacetaldehyde Chemical class O=CCOC1=CC=CC=C1 XFFILAFLGDUMBF-UHFFFAOYSA-N 0.000 abstract 1
- IORITYIZDHJCGT-SSDOTTSWSA-N 5-[(2r)-2-aminopropyl]-2-methoxybenzenesulfonamide Chemical compound COC1=CC=C(C[C@@H](C)N)C=C1S(N)(=O)=O IORITYIZDHJCGT-SSDOTTSWSA-N 0.000 abstract 1
- 239000012448 Lithium borohydride Substances 0.000 abstract 1
- 239000007868 Raney catalyst Substances 0.000 abstract 1
- NPXOKRUENSOPAO-UHFFFAOYSA-N Raney nickel Chemical compound [Al].[Ni] NPXOKRUENSOPAO-UHFFFAOYSA-N 0.000 abstract 1
- 229910000564 Raney nickel Inorganic materials 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 239000003054 catalyst Substances 0.000 abstract 1
- 230000003197 catalytic effect Effects 0.000 abstract 1
- 239000012442 inert solvent Substances 0.000 abstract 1
- 238000002955 isolation Methods 0.000 abstract 1
- 239000012280 lithium aluminium hydride Substances 0.000 abstract 1
- 229910052987 metal hydride Inorganic materials 0.000 abstract 1
- 150000004681 metal hydrides Chemical class 0.000 abstract 1
- MUMZUERVLWJKNR-UHFFFAOYSA-N oxoplatinum Chemical compound [Pt]=O MUMZUERVLWJKNR-UHFFFAOYSA-N 0.000 abstract 1
- 229910003446 platinum oxide Inorganic materials 0.000 abstract 1
- 239000012279 sodium borohydride Substances 0.000 abstract 1
- 229910000033 sodium borohydride Inorganic materials 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/37—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP60254326A JPS62114952A (ja) | 1985-11-13 | 1985-11-13 | 置換フエネチルアミン誘導体の製造法 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2000382A6 true ES2000382A6 (es) | 1988-02-16 |
Family
ID=17263445
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES8600685A Expired ES2000382A6 (es) | 1985-11-13 | 1986-07-29 | Un procedimiento para la produccion de derivados de fenetilamina substituidos |
Country Status (5)
Country | Link |
---|---|
JP (1) | JPS62114952A (enrdf_load_stackoverflow) |
KR (1) | KR940007746B1 (enrdf_load_stackoverflow) |
AT (1) | AT397960B (enrdf_load_stackoverflow) |
CA (1) | CA1282077C (enrdf_load_stackoverflow) |
ES (1) | ES2000382A6 (enrdf_load_stackoverflow) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2200699A1 (es) * | 2002-07-12 | 2004-03-01 | Ragactives Sl | Procedimiento para la separacion de r(-)- y s(+)-5-(2-((2-(2-etoxifenoxi)etil)amino)propil-2-metoxibenceno-sulfonamida. |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4971990A (en) * | 1988-02-19 | 1990-11-20 | Hokuriku Pharmaceutical Co., Ltd. | Phenoxyethylamine derivatives, for preparing the same and composition for exhibiting excellent α1 -blocking activity containing the same |
US5288759A (en) * | 1992-08-27 | 1994-02-22 | Alcon Laboratories, Inc. | Use of certain sulfamoyl-substituted phenethylamine derivatives to reverse drug-induced mydriasis |
TW536402B (en) | 1998-06-26 | 2003-06-11 | Yamanouchi Pharma Co Ltd | Pharmaceutical composition for the therapy of voiding dysfunction |
KR100525493B1 (ko) * | 2001-02-23 | 2005-11-02 | 연성정밀화학(주) | 설파모일 치환 페네틸아민 유도체의 제조 방법 |
CZ20013848A3 (cs) * | 2001-10-25 | 2003-05-14 | Léčiva, A.S. | Způsob výroby (R)-(-)-5-[2-[2-(2-ethoxyfenoxy)ethylamino]propyl]-2-methoxybenzensulfonamidu |
WO2004016582A1 (en) * | 2002-08-14 | 2004-02-26 | Natco Pharma Limited | An improved process for the preparation of tamsulosin hydrochloride |
KR100503639B1 (ko) | 2003-02-12 | 2005-07-26 | 보령제약 주식회사 | 탐술로신의 정제 방법 |
WO2005056521A1 (en) | 2003-12-09 | 2005-06-23 | Cj Corporation | Method of preparing optically pure phenethylamine derivatives |
SI21656A (sl) * | 2003-12-29 | 2005-06-30 | LEK farmacevtska družba d.d. | Priprava (R)-5-(2-(2-(2-etoksifenoksi) etilamino)-1-propil)-2-metoksibenzensulfonamida hidroklorida z visoko kemijsko čistoto |
SI21655A (sl) * | 2003-12-29 | 2005-06-30 | LEK farmacevtska dru�ba d.d. | Sinteza optično čistega (R)-5-(2-aminopropil)-2-metoksibenzensulfonamida |
CZ295583B6 (cs) * | 2004-02-05 | 2005-08-17 | Zentiva, A. S. | Způsob výroby (R)-(-)-5-(2-aminopropyl)-2-methoxybenzensulfonamidu |
EP1720830A1 (en) * | 2004-02-23 | 2006-11-15 | Cadila Healthcare Ltd. | Process for manufacturing optically pure (r) or (s)-5-(2-aminopropyl)-2-methoxybenzene sulfonamide |
WO2006004093A1 (ja) * | 2004-07-07 | 2006-01-12 | Hamari Chemicals, Ltd. | 光学活性フェニルプロピルアミン誘導体の製法 |
CN100545148C (zh) | 2004-08-16 | 2009-09-30 | 神隆新加坡私人有限公司 | 一种抗良性前列腺肥大药物坦索罗辛之合成方法 |
WO2007031823A1 (en) * | 2005-09-12 | 2007-03-22 | Aurobindo Pharma Limited | An improved process for preparing tamsulosin hydrochloride |
WO2008152653A2 (en) * | 2007-06-11 | 2008-12-18 | Matrix Laboratories Ltd | An improved process for the preparation of tamsulosin hydrochloride |
AU2010211725C1 (en) | 2009-02-04 | 2014-10-16 | Astellas Pharma Inc. | Pharmaceutical composition for oral administration |
EP2255793A1 (en) | 2009-05-28 | 2010-12-01 | Krka Tovarna Zdravil, D.D., Novo Mesto | Pharmaceutical composition comprising tamsulosin |
EP2475634B1 (en) * | 2009-09-12 | 2017-05-24 | Sandoz AG | Process for the preparation of indoline derivatives and their intermediates thereof |
DE202023102187U1 (de) | 2023-04-25 | 2023-05-02 | Nusrath Anjum | Auf Tamsulosin basierende Derivatformulierung |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1147342A (en) * | 1977-10-12 | 1983-05-31 | Kazuo Imai | Process of producing novel phenylethanolamine derivatives |
JPS56110665A (en) * | 1980-02-08 | 1981-09-01 | Yamanouchi Pharmaceut Co Ltd | Sulfamoyl-substituted phenetylamine derivative and its preparation |
US4558156A (en) * | 1980-02-08 | 1985-12-10 | Yamanouchi Pharmaceutical Co., Ltd. | Sulfamoyl-substituted phenethylamine derivatives |
-
1985
- 1985-11-13 JP JP60254326A patent/JPS62114952A/ja active Granted
-
1986
- 1986-07-07 KR KR1019860005460A patent/KR940007746B1/ko not_active Expired - Lifetime
- 1986-07-28 AT AT0203286A patent/AT397960B/de not_active IP Right Cessation
- 1986-07-29 ES ES8600685A patent/ES2000382A6/es not_active Expired
- 1986-07-31 CA CA000515041A patent/CA1282077C/en not_active Expired - Lifetime
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2200699A1 (es) * | 2002-07-12 | 2004-03-01 | Ragactives Sl | Procedimiento para la separacion de r(-)- y s(+)-5-(2-((2-(2-etoxifenoxi)etil)amino)propil-2-metoxibenceno-sulfonamida. |
WO2004006829A3 (es) * | 2002-07-12 | 2004-04-08 | Ragactives Sl | Procedimiento para la separación de r(-)- y s(+)-5-[2-[[2-(2-etoxifenoxi)etil]amino]propil-2-metoxibenceno-sulfonamida |
US7105698B2 (en) | 2002-07-12 | 2006-09-12 | Ragactives, S.L. | Process for the separation of R(-)-and S(+)-5-[2-[[2-(2-ethoxyphenoxy)ethyl]amino]propyl]-2- methoxybenzenesulfonamide |
Also Published As
Publication number | Publication date |
---|---|
AT397960B (de) | 1994-08-25 |
CA1282077C (en) | 1991-03-26 |
KR870004949A (ko) | 1987-06-02 |
KR940007746B1 (ko) | 1994-08-24 |
ATA203286A (de) | 1993-12-15 |
JPS62114952A (ja) | 1987-05-26 |
JPH0137391B2 (enrdf_load_stackoverflow) | 1989-08-07 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ES2000382A6 (es) | Un procedimiento para la produccion de derivados de fenetilamina substituidos | |
AU8829791A (en) | Process for the preparation of 1,3-propanediol | |
Kikukawa et al. | Reaction of diazonium salts with transition metals: XII. Palladium-catalyzed aryldestannylation of α-styrylstannanes by arenediazonium salts | |
YU46711B (sh) | Postupak za dobijanje novih tioksilozida | |
DE3562913D1 (en) | Process for the preparation of 4-acylamino-2-alkylaminophenyl ethers | |
HUT41779A (en) | Process for n-alkylating dihydro-lisergic acid | |
Rivera et al. | Ibuprofen and naproxen via organoboranes | |
ES8703408A1 (es) | Procedimiento para preparar un derivado de eter oximino-di- fenilico | |
Moriya et al. | Stereoselective Synthesis of (Z)-(1-Organo-1-alkenyl) boronic Esters by the Palladium-Catalyzed Cross-Coupling Reaction of (Z)-(1-Iodo-1-alkenyl) boronic Esters with Organozinc Reagents. | |
Banerjee et al. | Homogeneous reduction of aromatic nitrocompounds by a triphenylphosphine complex of palladium | |
KR860002959A (ko) | 제초제 중간화합물의 제법 | |
US4996324A (en) | Preparation of alkanols which are substituted in the 1 position by aromatic or heterocyclic radicals | |
US5107034A (en) | Method for producing 4-(2'-methoxyethyl)phenol | |
JPS5967237A (ja) | 2−メチル−4,5,6−トリアルコキシフエノ−ルの製造法 | |
DE3560108D1 (en) | Process for the preparation of 3-cyano-4-amino-acetophenones | |
JPS5671039A (en) | Preparation of cinnamic acid ester | |
JPS5824429B2 (ja) | エ−テルケツゴウオユウスル カゴウブツノ セイゾウホウ | |
JPH03215472A (ja) | 新規な4―置換―3,5―ジメチルピコリン酸化合物およびその製造方法 | |
JPS61291550A (ja) | 芳香族第二級アミノ化合物の製造法 | |
JPS5775947A (en) | Production of 2-(substituted phenoxy)phenylacetic acid | |
FR2405232A1 (fr) | Procede de preparation du citronellal et de ses homologues par hydrogenation du citral et de ses homologues | |
JPS5671069A (en) | Preparation of piperidine derivative | |
JPS6230741A (ja) | N−モノ置換p−フエニレンジアミンの製造法 | |
JPS5594368A (en) | Preparation of 1,3-dimethyl-4-(2,4-dichlorobenzoyl)-5- pyrazolyl4-toluenesulfonate | |
JPS5679661A (en) | Preparation of alpha-chlorohydrocinnamnitrile |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD1A | Patent lapsed |
Effective date: 20060731 |