EE9800264A - Taksoidid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid - Google Patents

Taksoidid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid

Info

Publication number
EE9800264A
EE9800264A EE9800264A EE9800264A EE9800264A EE 9800264 A EE9800264 A EE 9800264A EE 9800264 A EE9800264 A EE 9800264A EE 9800264 A EE9800264 A EE 9800264A EE 9800264 A EE9800264 A EE 9800264A
Authority
EE
Estonia
Prior art keywords
taxoids
preparation
pharmaceutical compositions
compositions containing
pharmaceutical
Prior art date
Application number
EE9800264A
Other languages
English (en)
Other versions
EE03611B1 (et
Inventor
Bouchard Herv
Bourzat Jean-Dominique
Commer�on Alain
Original Assignee
Rh�Ne-Poulenc Rorer S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rh�Ne-Poulenc Rorer S.A. filed Critical Rh�Ne-Poulenc Rorer S.A.
Publication of EE9800264A publication Critical patent/EE9800264A/et
Publication of EE03611B1 publication Critical patent/EE03611B1/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/04Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/041,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/061,3-Oxazines; Hydrogenated 1,3-oxazines not condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
EE9800264A 1996-03-06 1997-03-05 Taksoidid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid EE03611B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9602804A FR2745814B1 (fr) 1996-03-06 1996-03-06 Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent
PCT/FR1997/000386 WO1997032869A1 (fr) 1996-03-06 1997-03-05 Taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number Publication Date
EE9800264A true EE9800264A (et) 1999-02-15
EE03611B1 EE03611B1 (et) 2002-02-15

Family

ID=9489910

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9800264A EE03611B1 (et) 1996-03-06 1997-03-05 Taksoidid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid

Country Status (34)

Country Link
US (1) US6160135A (et)
EP (1) EP0885208B1 (et)
JP (1) JP2000506158A (et)
KR (1) KR19990087398A (et)
CN (1) CN1210525A (et)
AP (1) AP1023A (et)
AT (1) ATE204266T1 (et)
AU (1) AU715228B2 (et)
BG (1) BG63693B1 (et)
BR (1) BR9707887A (et)
CA (1) CA2248195A1 (et)
CZ (1) CZ283498A3 (et)
DE (1) DE69706146T2 (et)
DK (1) DK0885208T3 (et)
EA (1) EA001516B1 (et)
EE (1) EE03611B1 (et)
ES (1) ES2161446T3 (et)
FR (1) FR2745814B1 (et)
GE (1) GEP20012517B (et)
GR (1) GR3036410T3 (et)
HU (1) HUP9902425A3 (et)
IL (1) IL125998A (et)
IS (1) IS4809A (et)
NO (1) NO983472D0 (et)
NZ (1) NZ331040A (et)
OA (1) OA10855A (et)
PL (1) PL328691A1 (et)
PT (1) PT885208E (et)
SK (1) SK121598A3 (et)
TR (1) TR199801732T2 (et)
TW (1) TW474928B (et)
WO (1) WO1997032869A1 (et)
YU (1) YU38398A (et)
ZA (1) ZA971746B (et)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5973160A (en) 1992-12-23 1999-10-26 Poss; Michael A. Methods for the preparation of novel sidechain-bearing taxanes
MA23823A1 (fr) 1995-03-27 1996-10-01 Aventis Pharma Sa Nouveaux taxoides, leur preparation et les compositions qui les contiennent
US6372780B2 (en) 1995-03-27 2002-04-16 Aventis Pharma S.A. Methods of treating cell lines expressing multidrug resistance P-glycoprotein
KR100551945B1 (ko) * 1997-12-19 2006-02-20 가부시키가이샤 야쿠루트 혼샤 택산 유도체
EP1020188A1 (en) * 1999-01-13 2000-07-19 Aventis Pharma S.A. New use of taxoid derivatives
CO5280224A1 (es) * 2000-02-02 2003-05-30 Univ Florida State Res Found Taxanos sustituidos con ester en c7, utiles como agentes antitumorales y composiciones farmaceuticas que los contienen
HUP0200759A3 (en) 2000-02-02 2002-10-28 Univ Florida State Res Found C10 carbonate substituted taxanes as antitumor agents and pharmaceutical compositions containing them and their use
FR2859996B1 (fr) * 2003-09-19 2006-02-03 Aventis Pharma Sa Solvat acetonique du dimethoxy docetaxel et son procede de preparation
PE20060014A1 (es) 2004-03-05 2006-02-18 Univ Florida State Res Found Taxanos con sustituyentes lactiloxilo en el c7
US20110118473A1 (en) * 2007-08-22 2011-05-19 6570763 Canada Inc. Process for converting 9-dihydro-13acetylbaccatin iii paclitaxel and docetaxel
FR2926551A1 (fr) * 2008-01-17 2009-07-24 Aventis Pharma Sa Formes cristallines du dimethoxy docetaxel et leurs procedes de preparation
MY164086A (en) 2009-10-29 2017-11-30 Aventis Pharma Sa Novel antitumoral use of cabazitaxel
CN104650012A (zh) * 2013-11-22 2015-05-27 天士力控股集团有限公司 一种紫杉烷类化合物

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5136060A (en) * 1989-11-14 1992-08-04 Florida State University Method for preparation of taxol using an oxazinone
WO1993002067A1 (fr) * 1991-07-17 1993-02-04 Nippon Steel Corporation Compose antitumoral nsc-lsc1 et son procede de production
CA2100808A1 (en) * 1992-10-01 1994-04-02 Vittorio Farina Deoxy paclitaxels
AU6367994A (en) * 1993-03-22 1994-10-11 Florida State University Taxanes having alkoxy, alkenoxy or aryloxy substituted side-chain and pharmaceutical compositions containing same
FR2711369B1 (fr) * 1993-10-20 1995-11-17 Rhone Poulenc Rorer Sa Nouveaux taxoïdes, leur préparation et les compositions qui les contiennent.
RO116549B1 (ro) * 1994-07-26 2001-03-30 Indena Spa Derivati de taxan, procedeu pentru prepararea acestora, intermediar pentru prepararea acestora si compozitie farmaceutica care ii contine
US6201140B1 (en) * 1994-07-28 2001-03-13 Bristol-Myers Squibb Company 7-0-ethers of taxane derivatives

Also Published As

Publication number Publication date
US6160135A (en) 2000-12-12
NO983472L (no) 1998-07-28
AU715228B2 (en) 2000-01-20
AP9801335A0 (en) 1998-09-30
DK0885208T3 (da) 2001-10-15
GEP20012517B (en) 2001-08-27
EA001516B1 (ru) 2001-04-23
FR2745814A1 (fr) 1997-09-12
ZA971746B (en) 1997-09-16
PL328691A1 (en) 1999-02-15
EP0885208B1 (fr) 2001-08-16
KR19990087398A (ko) 1999-12-27
CN1210525A (zh) 1999-03-10
PT885208E (pt) 2001-11-30
BR9707887A (pt) 1999-09-21
WO1997032869A1 (fr) 1997-09-12
DE69706146D1 (de) 2001-09-20
HUP9902425A2 (hu) 2001-04-28
BG63693B1 (bg) 2002-09-30
IL125998A (en) 2002-02-10
GR3036410T3 (en) 2001-11-30
AP1023A (en) 2001-11-16
EP0885208A1 (fr) 1998-12-23
YU38398A (sh) 1999-07-28
BG102753A (en) 1999-09-30
NO983472D0 (no) 1998-07-28
HUP9902425A3 (en) 2001-08-28
IS4809A (is) 1998-07-24
DE69706146T2 (de) 2002-05-02
FR2745814B1 (fr) 1998-04-03
ATE204266T1 (de) 2001-09-15
TR199801732T2 (xx) 1998-12-21
IL125998A0 (en) 1999-04-11
EE03611B1 (et) 2002-02-15
ES2161446T3 (es) 2001-12-01
AU2030297A (en) 1997-09-22
CZ283498A3 (cs) 1999-01-13
OA10855A (fr) 2003-02-05
TW474928B (en) 2002-02-01
JP2000506158A (ja) 2000-05-23
CA2248195A1 (fr) 1997-09-12
SK121598A3 (en) 1999-01-11
NZ331040A (en) 2000-02-28
EA199800795A1 (ru) 1999-02-25

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Effective date: 20020305