EE200300396A - Epotilooni derivaatide kasutamine refraktaarsete kasvajate raviks - Google Patents

Epotilooni derivaatide kasutamine refraktaarsete kasvajate raviks

Info

Publication number
EE200300396A
EE200300396A EEP200300396A EEP200300396A EE200300396A EE 200300396 A EE200300396 A EE 200300396A EE P200300396 A EEP200300396 A EE P200300396A EE P200300396 A EEP200300396 A EE P200300396A EE 200300396 A EE200300396 A EE 200300396A
Authority
EE
Estonia
Prior art keywords
treatment
epothilone derivatives
refractory tumors
tumors
refractory
Prior art date
Application number
EEP200300396A
Other languages
English (en)
Estonian (et)
Inventor
Y. F. Lee Francis
Original Assignee
Bristol-Myers Squibb Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23028846&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EE200300396(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol-Myers Squibb Company filed Critical Bristol-Myers Squibb Company
Publication of EE200300396A publication Critical patent/EE200300396A/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
EEP200300396A 2001-02-20 2002-02-06 Epotilooni derivaatide kasutamine refraktaarsete kasvajate raviks EE200300396A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26983601P 2001-02-20 2001-02-20
PCT/US2002/004255 WO2002066038A1 (fr) 2001-02-20 2002-02-06 Traitement de tumeurs refractaires a l'aide de derives d'epothilone

Publications (1)

Publication Number Publication Date
EE200300396A true EE200300396A (et) 2003-12-15

Family

ID=23028846

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300396A EE200300396A (et) 2001-02-20 2002-02-06 Epotilooni derivaatide kasutamine refraktaarsete kasvajate raviks

Country Status (18)

Country Link
US (2) US6686380B2 (fr)
EP (1) EP1385529A4 (fr)
JP (1) JP2004522774A (fr)
KR (1) KR20040025895A (fr)
CN (1) CN1774253A (fr)
BG (1) BG108075A (fr)
BR (1) BR0207487A (fr)
CA (1) CA2438610A1 (fr)
EE (1) EE200300396A (fr)
HU (1) HUP0303175A2 (fr)
IL (1) IL156988A0 (fr)
IS (1) IS6918A (fr)
MX (1) MXPA03007394A (fr)
NO (1) NO20033684L (fr)
PL (1) PL363362A1 (fr)
RU (1) RU2003128311A (fr)
WO (1) WO2002066038A1 (fr)
ZA (1) ZA200306173B (fr)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
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JP4579351B2 (ja) 1996-12-03 2010-11-10 スローン−ケッタリング インスティトュート フォア キャンサー リサーチ エポチロンの合成とその中間体及びその類似物並びにその使用
US6204388B1 (en) * 1996-12-03 2001-03-20 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
US6605599B1 (en) 1997-07-08 2003-08-12 Bristol-Myers Squibb Company Epothilone derivatives
US6780620B1 (en) * 1998-12-23 2004-08-24 Bristol-Myers Squibb Company Microbial transformation method for the preparation of an epothilone
US20020058286A1 (en) * 1999-02-24 2002-05-16 Danishefsky Samuel J. Synthesis of epothilones, intermediates thereto and analogues thereof
JP2004521122A (ja) 2001-01-25 2004-07-15 ブリストル−マイヤーズ　スクイブ　カンパニー エポチロン類似体の非経口製剤
CZ305799B6 (cs) * 2001-03-14 2016-03-23 Bristol-Myers Squibb Company Kombinace analogů epothilonu a chemoterapeutických činidel pro léčení proliferačních nemocí
TW200403994A (en) * 2002-04-04 2004-03-16 Bristol Myers Squibb Co Oral administration of EPOTHILONES
TW200400191A (en) * 2002-05-15 2004-01-01 Bristol Myers Squibb Co Pharmaceutical compositions and methods of using C-21 modified epothilone derivatives
EP1506203B1 (fr) 2002-08-23 2007-01-03 Sloan-Kettering Institute For Cancer Research Synthese d'epothilones, leurs intermediaires, leurs analogues et leurs utilisations
US7649006B2 (en) 2002-08-23 2010-01-19 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
US6921769B2 (en) 2002-08-23 2005-07-26 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
WO2004032866A2 (fr) 2002-10-09 2004-04-22 Kosan Biosciences, Inc. Preparations therapeutiques
TW200503738A (en) * 2003-07-16 2005-02-01 Tzu Chi Buddhist General Hospital Method for extracting antineoplastic components from bupleurum scorzonerifolium
US20050171167A1 (en) * 2003-11-04 2005-08-04 Haby Thomas A. Process and formulation containing epothilones and analogs thereof
US20090004277A1 (en) * 2004-05-18 2009-01-01 Franchini Miriam K Nanoparticle dispersion containing lactam compound
WO2006017761A2 (fr) * 2004-08-05 2006-02-16 Emory University Analogues d'epothilone en tant qu'agents therapeutiques
US20060134214A1 (en) * 2004-11-18 2006-06-22 Ismat Ullah Enteric coated bead comprising epothilone or epothilone analog, and preparation and administration thereof
ATE397442T1 (de) 2004-11-18 2008-06-15 Bristol Myers Squibb Co Magensaftresistent beschichtetes pellet mit ixabepilon
AU2006336468B2 (en) 2005-02-11 2012-04-12 University Of Southern California Method of expressing proteins with disulfide bridges
EP2029156A4 (fr) 2006-05-01 2010-07-21 Univ Southern California Polythérapie pour traiter le cancer
US8463852B2 (en) * 2006-10-06 2013-06-11 Oracle International Corporation Groupware portlets for integrating a portal with groupware systems
WO2010056901A2 (fr) 2008-11-13 2010-05-20 University Of Southern California Procédé d'expression de protéines avec ponts disulfure avec des rendements et une activité améliorés
EP2571525A4 (fr) 2010-05-18 2016-04-27 Cerulean Pharma Inc Compositions et procédés de traitement de maladies auto-immunes et autres
EP4087545A1 (fr) 2020-01-10 2022-11-16 R-Pharm US Operating LLC Compositions d'ixabépilone

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CZ305799B6 (cs) 2001-03-14 2016-03-23 Bristol-Myers Squibb Company Kombinace analogů epothilonu a chemoterapeutických činidel pro léčení proliferačních nemocí
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Also Published As

Publication number Publication date
RU2003128311A (ru) 2005-03-10
JP2004522774A (ja) 2004-07-29
CN1774253A (zh) 2006-05-17
IS6918A (is) 2003-08-18
IL156988A0 (en) 2004-02-08
PL363362A1 (en) 2004-11-15
US6686380B2 (en) 2004-02-03
HUP0303175A2 (hu) 2003-12-29
BG108075A (bg) 2005-04-30
USRE41393E1 (en) 2010-06-22
EP1385529A4 (fr) 2007-05-09
EP1385529A1 (fr) 2004-02-04
BR0207487A (pt) 2004-08-10
WO2002066038A1 (fr) 2002-08-29
ZA200306173B (en) 2004-11-23
NO20033684D0 (no) 2003-08-19
MXPA03007394A (es) 2003-12-04
NO20033684L (no) 2003-10-13
CA2438610A1 (fr) 2002-08-29
US20020165258A1 (en) 2002-11-07
KR20040025895A (ko) 2004-03-26

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