EE04780B1 - Aminoalküül-asendatud bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja selle valmistamismeetod - Google Patents

Aminoalküül-asendatud bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja selle valmistamismeetod

Info

Publication number
EE04780B1
EE04780B1 EEP200100639A EEP200100639A EE04780B1 EE 04780 B1 EE04780 B1 EE 04780B1 EE P200100639 A EEP200100639 A EE P200100639A EE P200100639 A EEP200100639 A EE P200100639A EE 04780 B1 EE04780 B1 EE 04780B1
Authority
EE
Estonia
Prior art keywords
preparation
benzofuran
aminoalkyl
pharmaceutical composition
benzopyran derivatives
Prior art date
Application number
EEP200100639A
Other languages
English (en)
Inventor
Van Emelen Kristof
Frans Leopold De Bruyn Marcel
Original Assignee
Janssen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.
Publication of EE200100639A publication Critical patent/EE200100639A/et
Publication of EE04780B1 publication Critical patent/EE04780B1/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyrane Compounds (AREA)
EEP200100639A 1999-06-02 2000-05-23 Aminoalküül-asendatud bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja selle valmistamismeetod EE04780B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP99201747 1999-06-02
PCT/EP2000/004746 WO2000075136A1 (en) 1999-06-02 2000-05-23 Aminoalkyl substituted (benzodioxan, benzofuran or benzopyran) derivatives

Publications (2)

Publication Number Publication Date
EE200100639A EE200100639A (et) 2003-02-17
EE04780B1 true EE04780B1 (et) 2007-02-15

Family

ID=8240260

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100639A EE04780B1 (et) 1999-06-02 2000-05-23 Aminoalküül-asendatud bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja selle valmistamismeetod

Country Status (33)

Country Link
US (2) US6864273B1 (et)
EP (1) EP1187829B1 (et)
JP (1) JP2003501427A (et)
KR (1) KR100699512B1 (et)
CN (1) CN1150191C (et)
AR (1) AR033334A1 (et)
AT (1) ATE256125T1 (et)
AU (1) AU773773B2 (et)
BG (1) BG65269B1 (et)
BR (1) BR0011237A (et)
CA (1) CA2374902C (et)
CZ (1) CZ20014177A3 (et)
DE (1) DE60007124T2 (et)
DK (1) DK1187829T3 (et)
EA (1) EA004645B1 (et)
EE (1) EE04780B1 (et)
ES (1) ES2212774T3 (et)
HR (1) HRP20010868A2 (et)
HU (1) HUP0201404A3 (et)
IL (2) IL146840A0 (et)
MX (1) MXPA01012330A (et)
MY (1) MY120618A (et)
NO (1) NO319953B1 (et)
NZ (1) NZ514993A (et)
PL (1) PL198552B1 (et)
PT (1) PT1187829E (et)
SI (1) SI1187829T1 (et)
SK (1) SK285619B6 (et)
TR (1) TR200103430T2 (et)
TW (1) TWI289559B (et)
UA (1) UA73122C2 (et)
WO (1) WO2000075136A1 (et)
ZA (1) ZA200109860B (et)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CZ20014167A3 (cs) 1999-06-02 2002-06-12 Janssen Pharmaceutica N. V. Pyrrolidinylem, piperidinylem nebo homopiperidinylem substituované deriváty benzodioxanu, benzofuranu nebo benzopyranu
JO2352B1 (en) 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Compounds for the treatment of non-adaptation of the bottom of the uterus
JO2654B1 (en) 2000-09-04 2012-06-17 شركة جانسين فارماسوتيكا ان. في Multiple aryl caroxa amides are useful as lipid - lowering agents
JO2409B1 (en) 2000-11-21 2007-06-17 شركة جانسين فارماسوتيكا ان. في Second-phenyl carboxy amides are useful as lipid-lowering agents
AU2003236326B2 (en) * 2002-04-08 2008-02-28 Zeria Pharmaceutical Co., Ltd. A Therapeutic Agent for Impaired Gastric Accommodation
CA2597616A1 (en) 2005-02-17 2006-08-24 Wyeth Cycloalkylfused indole, benzothiophene, benzofuran and indene derivatives
EA027324B1 (ru) 2011-11-11 2017-07-31 Пфайзер Инк. 2-тиопиримидиноны
PE20180503A1 (es) 2015-05-05 2018-03-09 Pfizer 2-tiopirimidinonas

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3910930A (en) 1973-01-04 1975-10-07 Janssen Pharmaceutica Nv 1-{55 1-{8 2-(1,4-Benzodioxan-2-yl)-2-hydroxyethyl{9 -4-piperidyl{56 -2-benzimidazolinones
US3929801A (en) 1973-11-20 1975-12-30 Janssen Pharmaceutica Nv 2-Benzimidazolinones
GR71865B (et) 1978-03-20 1983-07-07 Ciba Geigy
DE2852945A1 (de) 1978-12-07 1980-06-26 Boehringer Sohn Ingelheim Benzodioxanyl-hydroxyaethylpiperidyl- imidazolidinone, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
US4329348A (en) 1979-02-26 1982-05-11 Ciba-Geigy Corporation N-Oxacyclic-alkylpiperidines as psychostimulants
DE3124366A1 (de) 1981-06-20 1982-12-30 Hoechst Ag, 6000 Frankfurt N-oxacyclyl-alkylpiperidin-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und deren verwendung
FR2533584B1 (fr) 1982-09-28 1986-03-21 Pasteur Institut Procede de detection du pouvoir mutagene de substances, susceptibles d'induire la deterioration d'adn cellulaires, mettant en jeu la production d'une reponse sos
DE3901814A1 (de) 1988-07-28 1990-02-01 Bayer Ag Substituierte aminomethylzetraline sowie ihre heterocyclischen analoga
DE4140540A1 (de) 1991-12-09 1993-06-17 Bayer Ag Neue azaheterocyclylmethyl-chromane
SI9300097B (en) * 1992-02-27 2001-12-31 Janssen Pharmaceutica Nv (benzodioxan, benzofuran or benzopyran) alkylamino) alkyl substituted guanidines
DE4319038A1 (de) 1993-06-08 1994-12-15 Bayer Ag Verwendung von teilweise bekannten substituierten Chromanen als Arzneimittel, neue Wirkstoffe und Verfahren zu ihrer Herstellung
PL181385B1 (pl) 1993-08-19 2001-07-31 Janssen Pharmaceutica Nv Nowe pochodne dihydrobenzopiranu o wlasciwosciach naczyniozwezajacych, kompozycja farmaceutyczna i sposób wytwarzania pochodnych dihydrobenzopiranu PL PL PL PL PL PL
US5541199A (en) 1995-06-02 1996-07-30 American Home Products Corporation Chroman-2-ylmethylamino derivatives
FR2744451B1 (fr) 1996-02-01 1998-04-24 Pf Medicament Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutique
US6133277A (en) * 1997-12-05 2000-10-17 Janssen Pharmaceutica N.V. (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties
CZ20014167A3 (cs) 1999-06-02 2002-06-12 Janssen Pharmaceutica N. V. Pyrrolidinylem, piperidinylem nebo homopiperidinylem substituované deriváty benzodioxanu, benzofuranu nebo benzopyranu
JO2352B1 (en) 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Compounds for the treatment of non-adaptation of the bottom of the uterus

Also Published As

Publication number Publication date
AR033334A1 (es) 2003-12-17
AU5525600A (en) 2000-12-28
BG65269B1 (bg) 2007-11-30
EP1187829B1 (en) 2003-12-10
EP1187829A1 (en) 2002-03-20
US20050096378A1 (en) 2005-05-05
ES2212774T3 (es) 2004-08-01
MXPA01012330A (es) 2002-07-30
BR0011237A (pt) 2002-03-05
BG106156A (en) 2002-05-31
IL146840A0 (en) 2002-07-25
AU773773B2 (en) 2004-06-03
UA73122C2 (en) 2005-06-15
ZA200109860B (en) 2003-05-28
IL146840A (en) 2006-12-10
ATE256125T1 (de) 2003-12-15
PL352112A1 (en) 2003-07-28
CA2374902A1 (en) 2000-12-14
NZ514993A (en) 2003-05-30
CZ20014177A3 (cs) 2002-05-15
DE60007124D1 (de) 2004-01-22
EA004645B1 (ru) 2004-06-24
TWI289559B (en) 2007-11-11
US7273862B2 (en) 2007-09-25
KR20010110806A (ko) 2001-12-13
CA2374902C (en) 2009-09-15
PL198552B1 (pl) 2008-06-30
EA200101236A1 (ru) 2002-08-29
EE200100639A (et) 2003-02-17
JP2003501427A (ja) 2003-01-14
KR100699512B1 (ko) 2007-03-26
SK285619B6 (sk) 2007-05-03
CN1150191C (zh) 2004-05-19
SI1187829T1 (en) 2004-04-30
TR200103430T2 (tr) 2002-06-21
WO2000075136A1 (en) 2000-12-14
US6864273B1 (en) 2005-03-08
MY120618A (en) 2005-11-30
SK17032001A3 (sk) 2002-07-02
DK1187829T3 (da) 2004-04-13
CN1353707A (zh) 2002-06-12
PT1187829E (pt) 2004-04-30
HUP0201404A3 (en) 2005-02-28
HUP0201404A2 (en) 2002-08-28
HRP20010868A2 (en) 2003-04-30
NO20015903D0 (no) 2001-12-03
NO319953B1 (no) 2005-10-03
DE60007124T2 (de) 2004-09-23
NO20015903L (no) 2001-12-03

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Legal Events

Date Code Title Description
KB4A Valid patent at the end of a year

Effective date: 20071231

KB4A Valid patent at the end of a year

Effective date: 20081231

MM4A Lapsed by not paying the annual fees

Effective date: 20100523