FR2744451B1 - Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutique - Google Patents
Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutiqueInfo
- Publication number
- FR2744451B1 FR2744451B1 FR9601220A FR9601220A FR2744451B1 FR 2744451 B1 FR2744451 B1 FR 2744451B1 FR 9601220 A FR9601220 A FR 9601220A FR 9601220 A FR9601220 A FR 9601220A FR 2744451 B1 FR2744451 B1 FR 2744451B1
- Authority
- FR
- France
- Prior art keywords
- pyrimidinones
- imidazolidinones
- diazepin
- ones
- novel
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9601220A FR2744451B1 (fr) | 1996-02-01 | 1996-02-01 | Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutique |
PCT/FR1997/000179 WO1997028157A1 (fr) | 1996-02-01 | 1997-01-30 | Nouveaux derives de la piperidine substitues en position 4 par un groupe imidazolidin-2-on-1-yl-ethyl, tetrahydropyrimidin-2-on-1-yl-ethyl, et 1,3-dia-zepin-2-on-1-yl-ethyl, et leurs applications comme antagonistes des recepteurs alpha-2 adrenergiques |
AU16061/97A AU1606197A (en) | 1996-02-01 | 1997-01-30 | Novel piperidine derivatives 4-substituted by an imidazolidin-2-on-1-yl-ethyl, tetrahydropyrimidin-2-on-1-yl-ethyl and 1,3-diazepin-2-on-1-yl-ethyl group, and use thereof as alpha2-adrenergic receptor antagonists |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9601220A FR2744451B1 (fr) | 1996-02-01 | 1996-02-01 | Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2744451A1 FR2744451A1 (fr) | 1997-08-08 |
FR2744451B1 true FR2744451B1 (fr) | 1998-04-24 |
Family
ID=9488732
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR9601220A Expired - Fee Related FR2744451B1 (fr) | 1996-02-01 | 1996-02-01 | Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutique |
Country Status (3)
Country | Link |
---|---|
AU (1) | AU1606197A (fr) |
FR (1) | FR2744451B1 (fr) |
WO (1) | WO1997028157A1 (fr) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6133277A (en) * | 1997-12-05 | 2000-10-17 | Janssen Pharmaceutica N.V. | (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties |
FR2789681A1 (fr) * | 1999-02-12 | 2000-08-18 | Pf Medicament | Nouveaux derives du 8-[(1,4)-benzodioxane-2-ylmethyl]-8- azabicyclo[3,2]octane-3-alkyl urees ou imidazolidinones, leur procede de preparation et leurs applications en therapeutique pour traiter les maladies neurodegeneratives |
NZ514993A (en) | 1999-06-02 | 2003-05-30 | Janssen Pharmaceutica Nv | Aminoalkyl substituted (benzodioxan, benzofuran or benzopyran) derivatives |
AU777601B2 (en) * | 1999-06-02 | 2004-10-21 | Janssen Pharmaceutica N.V. | Pyrrolidinyl, piperidinyl or homopiperidinyl substituted (benzodioxan, benzofuran or benzopyran) derivatives |
AU2004202768B2 (en) * | 1999-12-30 | 2007-04-05 | Les Laboratoires Servier | New linear or cyclic ureas, a process for their preparation and pharmaceutical compositions containing them |
FR2803298A1 (fr) * | 1999-12-30 | 2001-07-06 | Adir | Nouvelles urees lineaires ou cycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
JO2352B1 (en) | 2000-06-22 | 2006-12-12 | جانسين فارماسيوتيكا ان. في | Compounds for the treatment of non-adaptation of the bottom of the uterus |
WO2004064865A1 (fr) * | 2003-01-17 | 2004-08-05 | Takeda Pharmaceutical Company Limited | Agent protecteur des muscles du squelette |
TWI457122B (zh) * | 2007-07-20 | 2014-10-21 | Orion Corp | 作為用於治療周邊和中央神經系統疾病之alpha2C拮抗劑的2,3-二氫苯並[1,4]戴奧辛-2-基甲基衍生物 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2852945A1 (de) * | 1978-12-07 | 1980-06-26 | Boehringer Sohn Ingelheim | Benzodioxanyl-hydroxyaethylpiperidyl- imidazolidinone, verfahren zu ihrer herstellung und diese enthaltende arzneimittel |
IL59619A0 (en) * | 1979-03-28 | 1980-06-30 | Pfizer | Phthalazine derivatives,their preparation and pharmaceutical compositions containing them |
JPS61215389A (ja) * | 1985-03-20 | 1986-09-25 | Kyowa Hakko Kogyo Co Ltd | キナゾリン誘導体およびそれを含有する強心剤 |
NZ221485A (en) * | 1986-08-28 | 1991-04-26 | Merck & Co Inc | Hexahydroarylquinolizine derivatives and pharmaceutical compositions |
JPH05505612A (ja) * | 1991-03-01 | 1993-08-19 | ハー・ルンドベック・アクティーゼルスカブ | 高血圧症及び末梢血管疾患の治療法 |
JPH09165385A (ja) * | 1994-08-26 | 1997-06-24 | Kyowa Hakko Kogyo Co Ltd | キナゾリン誘導体 |
-
1996
- 1996-02-01 FR FR9601220A patent/FR2744451B1/fr not_active Expired - Fee Related
-
1997
- 1997-01-30 WO PCT/FR1997/000179 patent/WO1997028157A1/fr active Application Filing
- 1997-01-30 AU AU16061/97A patent/AU1606197A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
WO1997028157A1 (fr) | 1997-08-07 |
AU1606197A (en) | 1997-08-22 |
FR2744451A1 (fr) | 1997-08-08 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
FR2671083B1 (fr) | Nouvelles 4-(4-imidazolyl) piperidines substituees en 1, leur preparation ainsi que leurs applications therapeutiques. | |
FR2751966B1 (fr) | Nouveaux derives 1,2-diarylindoles, leurs procedes de preparation, et leurs utilisations en therapeutique | |
FR2671352B1 (fr) | Nouveaux copolymeres cationiques, de nouvelles emulsions et leur application. | |
FR2667317B1 (fr) | Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique. | |
FR2681325B1 (fr) | Derives de l'aminomethyl-4 piperidine, leur preparation et leur application en therapeutique. | |
FR2769311B1 (fr) | Nouveaux derives 3,4-diarylthiazolin-2-one ou -2-thione, leurs procedes de preparation et leurs utilisations en therapeutique | |
FR2753449B1 (fr) | Nouveaux derives 3,4-diaryloxazolone, leurs procedes de preparation, et leurs utilisations en therapeutique | |
FR2659323B1 (fr) | Derives de 4-(aminomethyl) piperidine, leur preparation et leur application en therapeutique. | |
FR2744451B1 (fr) | Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutique | |
FR2757860B1 (fr) | Composes organoselenies cycliques, leur preparation et leurs utilisations, notamment therapeutiques | |
FR2771093B1 (fr) | Derives d'imidazole, leur preparation et leur application en therapeutique | |
MA22981A1 (fr) | Derives de piperidine, leur preparation et leur application en therapeutique. | |
FR2758329B1 (fr) | Derives d'imidazole-4-butane boronique, leur preparation et leur utilisation en therapeutique | |
FR2779429B1 (fr) | Derives d'oxindole, leurs preparations et leurs applications en therapeutique | |
FR2751647B1 (fr) | Derives de benzimidazole, leurs preparations et leurs applications en therapeutique | |
FR2772378B1 (fr) | Derives d'imidazole, leur preparation et leur application en therapeutique | |
DE68906245D1 (de) | Therapeutisches mittel gegen aids. | |
FR2765874B1 (fr) | Derives de 6-pyrrolidin-2-ylpyrindines, leur preparation et leur application en therapeutique | |
FR2725989B1 (fr) | Nouvelles 2-(1-(omega-phenoxyalcoylpiperidin-4-yl) aminomethylene)-2h-benzofuran-3-ones substituees, leur preparation et leur application en therapeutique | |
FR2724382B1 (fr) | Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique | |
FR2681320B1 (fr) | Derives de n-(4,7dimethoxyindan-2-yl)-1-(phenylcarbonyl)-n-propyl-piperidine-4-methanamine, leur preparation et leur application en therapeutique. | |
MA22143A1 (fr) | Derives de 1,5 benzothiazepinone, leurs preparations et leur application | |
FR2735469B1 (fr) | N2-(arylsulfonyl)-l-arginylpiperidin-2-carboxylates, leur preparation et leur application en therapeutique | |
FR2740776B1 (fr) | Polyurethannes, leur preparation et leurs utilisations | |
FR2777566B1 (fr) | Derives d'azacycloalcanes, leur preparation et leur application en therapeutique |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |