EE03611B1 - Taksoidid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid - Google Patents

Taksoidid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid

Info

Publication number
EE03611B1
EE03611B1 EE9800264A EE9800264A EE03611B1 EE 03611 B1 EE03611 B1 EE 03611B1 EE 9800264 A EE9800264 A EE 9800264A EE 9800264 A EE9800264 A EE 9800264A EE 03611 B1 EE03611 B1 EE 03611B1
Authority
EE
Estonia
Prior art keywords
taxoids
preparation
pharmaceutical compositions
compositions containing
pharmaceutical
Prior art date
Application number
EE9800264A
Other languages
English (en)
Estonian (et)
Other versions
EE9800264A (et
Inventor
Bouchard Herv
Bourzat Jean-Dominique
Commer�on Alain
Original Assignee
Rh�Ne-Poulenc Rorer S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rh�Ne-Poulenc Rorer S.A. filed Critical Rh�Ne-Poulenc Rorer S.A.
Publication of EE9800264A publication Critical patent/EE9800264A/xx
Publication of EE03611B1 publication Critical patent/EE03611B1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/04Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/041,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/061,3-Oxazines; Hydrogenated 1,3-oxazines not condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
EE9800264A 1996-03-06 1997-03-05 Taksoidid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid EE03611B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9602804A FR2745814B1 (fr) 1996-03-06 1996-03-06 Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent
PCT/FR1997/000386 WO1997032869A1 (fr) 1996-03-06 1997-03-05 Taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number Publication Date
EE9800264A EE9800264A (et) 1999-02-15
EE03611B1 true EE03611B1 (et) 2002-02-15

Family

ID=9489910

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9800264A EE03611B1 (et) 1996-03-06 1997-03-05 Taksoidid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid

Country Status (34)

Country Link
US (1) US6160135A (xx)
EP (1) EP0885208B1 (xx)
JP (1) JP2000506158A (xx)
KR (1) KR19990087398A (xx)
CN (1) CN1210525A (xx)
AP (1) AP1023A (xx)
AT (1) ATE204266T1 (xx)
AU (1) AU715228B2 (xx)
BG (1) BG63693B1 (xx)
BR (1) BR9707887A (xx)
CA (1) CA2248195A1 (xx)
CZ (1) CZ283498A3 (xx)
DE (1) DE69706146T2 (xx)
DK (1) DK0885208T3 (xx)
EA (1) EA001516B1 (xx)
EE (1) EE03611B1 (xx)
ES (1) ES2161446T3 (xx)
FR (1) FR2745814B1 (xx)
GE (1) GEP20012517B (xx)
GR (1) GR3036410T3 (xx)
HU (1) HUP9902425A3 (xx)
IL (1) IL125998A (xx)
IS (1) IS4809A (xx)
NO (1) NO983472D0 (xx)
NZ (1) NZ331040A (xx)
OA (1) OA10855A (xx)
PL (1) PL328691A1 (xx)
PT (1) PT885208E (xx)
SK (1) SK121598A3 (xx)
TR (1) TR199801732T2 (xx)
TW (1) TW474928B (xx)
WO (1) WO1997032869A1 (xx)
YU (1) YU38398A (xx)
ZA (1) ZA971746B (xx)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5973160A (en) 1992-12-23 1999-10-26 Poss; Michael A. Methods for the preparation of novel sidechain-bearing taxanes
US6372780B2 (en) 1995-03-27 2002-04-16 Aventis Pharma S.A. Methods of treating cell lines expressing multidrug resistance P-glycoprotein
MA23823A1 (fr) 1995-03-27 1996-10-01 Aventis Pharma Sa Nouveaux taxoides, leur preparation et les compositions qui les contiennent
CN1221539C (zh) * 1997-12-19 2005-10-05 株式会社益力多本社 紫杉烷衍生物
EP1020188A1 (en) * 1999-01-13 2000-07-19 Aventis Pharma S.A. New use of taxoid derivatives
AR030188A1 (es) * 2000-02-02 2003-08-13 Univ Florida State Res Found Compuestos de taxano sustituidos con esteres en el c7; composiciones farmaceuticas que los contienen y proceso para tratar un sujeto mamifero que sufre de una condicion que responde a los taxanos
CN1186340C (zh) 2000-02-02 2005-01-26 佛罗里达州立大学研究基金有限公司 用作抗肿瘤剂的c10碳酸酯取代的紫杉烷
FR2859996B1 (fr) * 2003-09-19 2006-02-03 Aventis Pharma Sa Solvat acetonique du dimethoxy docetaxel et son procede de preparation
CN1960721A (zh) 2004-03-05 2007-05-09 佛罗里达州立大学研究基金有限公司 C7乳酰氧基取代的紫杉烷类
AU2008288651A1 (en) * 2007-08-22 2009-02-26 6570763 Canada Inc. Process for converting 9-dihydro-13-acetylbaccatin III into docetaxel or paclitaxel
FR2926551A1 (fr) * 2008-01-17 2009-07-24 Aventis Pharma Sa Formes cristallines du dimethoxy docetaxel et leurs procedes de preparation
PE20121429A1 (es) 2009-10-29 2012-11-06 Aventis Pharma Sa Nuevo uso antitumoral de cabazitaxel
CN104650012A (zh) * 2013-11-22 2015-05-27 天士力控股集团有限公司 一种紫杉烷类化合物

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5136060A (en) * 1989-11-14 1992-08-04 Florida State University Method for preparation of taxol using an oxazinone
EP0555485A4 (en) * 1991-07-17 1993-11-03 Nippon Steel Corporation Antitumor compound nsc-lsc1 and production thereof
CA2100808A1 (en) * 1992-10-01 1994-04-02 Vittorio Farina Deoxy paclitaxels
DE69434373T2 (de) * 1993-03-22 2006-03-09 Florida State University, Tallahassee Beta-laktame zur Herstellung von Taxanen mit Furyl oder Thienyl substituierter Seitenkette
FR2711369B1 (fr) * 1993-10-20 1995-11-17 Rhone Poulenc Rorer Sa Nouveaux taxoïdes, leur préparation et les compositions qui les contiennent.
RO115875B1 (ro) * 1994-07-26 2000-07-28 Indena Spa Derivati de taxan, procedeu pentru prepararea acestora, intermediar pentru prepararea acestora si compozitie farmaceutica care ii contine
US6201140B1 (en) * 1994-07-28 2001-03-13 Bristol-Myers Squibb Company 7-0-ethers of taxane derivatives

Also Published As

Publication number Publication date
CN1210525A (zh) 1999-03-10
NZ331040A (en) 2000-02-28
FR2745814B1 (fr) 1998-04-03
US6160135A (en) 2000-12-12
KR19990087398A (ko) 1999-12-27
TW474928B (en) 2002-02-01
CA2248195A1 (fr) 1997-09-12
PT885208E (pt) 2001-11-30
EA001516B1 (ru) 2001-04-23
YU38398A (sh) 1999-07-28
FR2745814A1 (fr) 1997-09-12
IL125998A0 (en) 1999-04-11
GEP20012517B (en) 2001-08-27
ATE204266T1 (de) 2001-09-15
BR9707887A (pt) 1999-09-21
EP0885208B1 (fr) 2001-08-16
BG63693B1 (bg) 2002-09-30
TR199801732T2 (xx) 1998-12-21
ES2161446T3 (es) 2001-12-01
EA199800795A1 (ru) 1999-02-25
GR3036410T3 (en) 2001-11-30
AU2030297A (en) 1997-09-22
DK0885208T3 (da) 2001-10-15
DE69706146T2 (de) 2002-05-02
BG102753A (en) 1999-09-30
NO983472L (no) 1998-07-28
AP1023A (en) 2001-11-16
OA10855A (fr) 2003-02-05
PL328691A1 (en) 1999-02-15
DE69706146D1 (de) 2001-09-20
ZA971746B (en) 1997-09-16
HUP9902425A3 (en) 2001-08-28
HUP9902425A2 (hu) 2001-04-28
AP9801335A0 (en) 1998-09-30
WO1997032869A1 (fr) 1997-09-12
AU715228B2 (en) 2000-01-20
EP0885208A1 (fr) 1998-12-23
CZ283498A3 (cs) 1999-01-13
SK121598A3 (en) 1999-01-11
JP2000506158A (ja) 2000-05-23
EE9800264A (et) 1999-02-15
NO983472D0 (no) 1998-07-28
IS4809A (is) 1998-07-24
IL125998A (en) 2002-02-10

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Legal Events

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MM4A Lapsed by not paying the annual fees

Effective date: 20020305