EA201591874A1 - Замещенные производные оксопиридина и их применение для лечения сердечно-сосудистых заболеваний - Google Patents

Замещенные производные оксопиридина и их применение для лечения сердечно-сосудистых заболеваний

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EA201591874A1
EA201591874A1 EA201591874A EA201591874A EA201591874A1 EA 201591874 A1 EA201591874 A1 EA 201591874A1 EA 201591874 A EA201591874 A EA 201591874A EA 201591874 A EA201591874 A EA 201591874A EA 201591874 A1 EA201591874 A1 EA 201591874A1
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cardiovascular diseases
treatment
diseases
application
well
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EA201591874A
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EA028034B9 (ru
EA028034B1 (ru
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Зузаннэ Рёриг
Александр Хиллиш
Юлия Штрассбургер
Штефан Хайтмайер
Мартина Виктория Шмидт
Карл-Хайнц Шлеммер
Адриан Терстееген
Анья Бухмюллер
Кристоф Гердес
Мартина Шэфер
Том Кинцель
Хенрик Теллер
Хартмут Широк
Юрген Клар
Элоиза Хименес Нунес
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Байер Фарма Акциенгезельшафт
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Publication of EA201591874A1 publication Critical patent/EA201591874A1/ru
Publication of EA028034B1 publication Critical patent/EA028034B1/ru
Publication of EA028034B9 publication Critical patent/EA028034B9/ru

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Abstract

Изобретение касается замещенных производных оксопиридина формулы, в которой Rозначает группу формулы, причем * означает место присоединения к оксопиридиновому кольцу, Rозначает бром, хлор, фтор, метил, дифторметил, трифторметил, метокси, дифторметокси или трифторметокси, Rозначает бром, хлор, фтор, циано, нитро, гидрокси, метил, дифторметил, трифторметил, метокси, этокси, дифторметокси, трифторметокси, этинил, 3,3,3-трифторпроп-1-ин-1-ил или циклопропил, и способа их получения, а также их применения для приготовления лекарственных средств для лечения и/или профилактики заболеваний, в частности сердечно-сосудистых заболеваний, предпочтительно тромботических или тромбоэмболических заболеваний, а также опухолей, как и офтальмологических заболеваний.
EA201591874A 2013-03-28 2014-03-27 Замещенные производные оксопиридина и их применение для лечения сердечно-сосудистых заболеваний EA028034B9 (ru)

Applications Claiming Priority (3)

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EP13161588 2013-03-28
EP13190944 2013-10-30
PCT/EP2014/056135 WO2014154794A1 (de) 2013-03-28 2014-03-27 Substituierte oxopyridin-derivate und ihre verwendung bei der behandlung von herz-kreislauf-erkrankungen

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EA201591874A1 true EA201591874A1 (ru) 2016-04-29
EA028034B1 EA028034B1 (ru) 2017-09-29
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