EA201370219A1 - Противогипертоническая фармацевтическая композиция - Google Patents

Противогипертоническая фармацевтическая композиция

Info

Publication number
EA201370219A1
EA201370219A1 EA201370219A EA201370219A EA201370219A1 EA 201370219 A1 EA201370219 A1 EA 201370219A1 EA 201370219 A EA201370219 A EA 201370219A EA 201370219 A EA201370219 A EA 201370219A EA 201370219 A1 EA201370219 A1 EA 201370219A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pharmaceutical composition
hypertonic pharmaceutical
solvate
hydrate
pharmaceutically acceptable
Prior art date
Application number
EA201370219A
Other languages
English (en)
Other versions
EA024096B1 (ru
Inventor
Сынь Хо Кхим
Чи Хан Кхим
Кхюн Сань Ю
Ин Чин Чан
Сан Коо Схин
Со Хюн Ёон
Чоо Ёун Чхо
Тхэ Ын Кхим
Со Чонь И
Соо Хыи Пхаик
Ён Ха Чхи
Чоо Хан Лее
Кхюн Ван Нам
Че Хак Кхим
Original Assignee
Борюн Фармасьютикал Ко., Лтд.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47006840&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201370219(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Борюн Фармасьютикал Ко., Лтд. filed Critical Борюн Фармасьютикал Ко., Лтд.
Publication of EA201370219A1 publication Critical patent/EA201370219A1/ru
Publication of EA024096B1 publication Critical patent/EA024096B1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/44221,4-Dihydropyridines, e.g. nifedipine, nicardipine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)

Abstract

Настоящее изобретение предусматривает противогипертоническую фармацевтическую композицию, содержащую фимасартан, его фармацевтически приемлемую соль, его сольват или его гидрат в качестве блокатора рецепторов ангиотензина II и амлодипин, его изомер, его фармацевтически приемлемую соль, его сольват или его гидрат в качестве блокатора кальциевых каналов.
EA201370219A 2011-04-12 2011-08-08 Противогипертоническая фармацевтическая композиция EA024096B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR20110033856 2011-04-12
PCT/KR2011/005754 WO2012141385A1 (en) 2011-04-12 2011-08-08 Antihypertensive pharmaceutical composition

Publications (2)

Publication Number Publication Date
EA201370219A1 true EA201370219A1 (ru) 2014-02-28
EA024096B1 EA024096B1 (ru) 2016-08-31

Family

ID=47006840

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201370219A EA024096B1 (ru) 2011-04-12 2011-08-08 Противогипертоническая фармацевтическая композиция

Country Status (20)

Country Link
US (1) US8765776B2 (ru)
JP (1) JP5782178B2 (ru)
AU (1) AU2011365756B2 (ru)
BR (1) BR112013025222B8 (ru)
CA (1) CA2832758C (ru)
CL (1) CL2013002905A1 (ru)
CO (1) CO6821940A2 (ru)
CR (1) CR20130526A (ru)
EA (1) EA024096B1 (ru)
EC (1) ECSP13012962A (ru)
GT (1) GT201300241A (ru)
MA (1) MA35107B1 (ru)
MX (1) MX341450B (ru)
MY (1) MY160432A (ru)
NI (1) NI201300106A (ru)
PE (1) PE20141049A1 (ru)
SG (1) SG194162A1 (ru)
UA (1) UA110244C2 (ru)
WO (1) WO2012141385A1 (ru)
ZA (1) ZA201307593B (ru)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA024096B1 (ru) 2011-04-12 2016-08-31 Борюн Фармасьютикал Ко., Лтд. Противогипертоническая фармацевтическая композиция
KR101490329B1 (ko) * 2012-10-12 2015-02-04 보령제약 주식회사 피마살탄 포타슘염의 일수화물 결정, 그 제조방법, 및 그를 포함하는 약제학적 조성물
KR20140096514A (ko) * 2013-01-28 2014-08-06 보령제약 주식회사 암 예방 또는 치료용 조성물
AU2014230182B2 (en) * 2013-03-14 2016-12-22 Boryung Pharmaceutical Co., Ltd. Pharmaceutical combination drug
KR20150041223A (ko) * 2013-10-04 2015-04-16 보령제약 주식회사 피마살탄을 포함하는 허혈성 뇌질환 예방 또는 치료용 약학적 조성물
CN105395552A (zh) * 2014-09-05 2016-03-16 南京华威医药科技开发有限公司 一种含非马沙坦及其盐的固体制剂
KR101545268B1 (ko) * 2015-02-05 2015-08-20 보령제약 주식회사 정제 및 이의 제조방법
WO2017091041A1 (ko) * 2015-11-26 2017-06-01 보령제약 주식회사 피마살탄의 신규 염
US11452690B1 (en) 2021-01-27 2022-09-27 ECI Pharmaceuticals, LLC Oral liquid compositions comprising amlodipine besylate and methods of using the same
CN112704667A (zh) * 2021-02-24 2021-04-27 施慧达药业集团(吉林)有限公司 含苯磺酸左氨氯地平水合物的组合物及其制备方法

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK161312C (da) 1982-03-11 1991-12-09 Pfizer Analogifremgangsmaade til fremstilling af 2-aminoalkoxymethyl-4-phenyl-6-methyl-1,4-dihydropyridin-3,5-dicarboxylsyreestere eller syreadditionssalte deraf samt phthalimidoderivater til anvendelse som udgangsmateriale ved fremgangsmaaden
CA1334092C (en) 1986-07-11 1995-01-24 David John Carini Angiotensin ii receptor blocking imidazoles
EP0733366B1 (en) 1988-01-07 1998-04-01 E.I. Du Pont De Nemours And Company Pharmaceutical compositions comprising angiotensin II receptor blocking imidazoles and diuretics
KR100300566B1 (ko) 1994-09-17 2001-11-22 조생현 피리미디논유도체와그의제조방법및용도
KR19990081093A (ko) * 1998-04-25 1999-11-15 조생현 피리미디논 화합물, 이를 함유하는 약제학적 조성물 및 이의제조방법
SK285863B6 (sk) * 1998-07-10 2007-10-04 Novartis Ag Kombinovaná farmaceutická kompozícia obsahujúca AT1-antagonistu valsartan a amlodipín
FR2783422A1 (fr) 1998-09-21 2000-03-24 Sanofi Sa Composition pharmaceutique contenant un antagoniste des recepteurs at1 de l'angiotensine ii et un antiagregant plaquettaire
KR100617953B1 (ko) 2000-03-23 2006-08-30 보령제약 주식회사 피리미디논 화합물 및 이의 염의 제조방법
AU2001292386B2 (en) * 2001-09-21 2006-06-22 Boryung Pharmaceutical Co., Ltd. Method for preparing pyrimidinone compound and pharmaceutically acceptable salts thereof
KR100521980B1 (ko) 2002-10-10 2005-10-17 보령제약 주식회사 피리미디논 화합물 및 이의 염의 삼수화물의 제조 방법
BRPI0612674B8 (pt) * 2005-06-27 2021-05-25 Daiichi Sankyo Co Ltd preparação farmacêutica, uso de um antagonista do receptor de angiotensina ii e um bloqueador do canal de cálcio
KR100888131B1 (ko) * 2006-10-10 2009-03-11 한올제약주식회사 시간차 투약 원리를 이용한 심혈관계 질환 치료용 복합제제
KR20100048137A (ko) 2008-10-30 2010-05-11 현대약품 주식회사 혈압 강하용 약학 조성물
KR101058284B1 (ko) 2010-01-22 2011-08-22 보령제약 주식회사 2-(2-n-부틸-4-히드록시-6-메틸-피리미딘-5-일)-N,N-디메틸아세트아미드의 신규한 제조방법
EA024096B1 (ru) 2011-04-12 2016-08-31 Борюн Фармасьютикал Ко., Лтд. Противогипертоническая фармацевтическая композиция

Also Published As

Publication number Publication date
CL2013002905A1 (es) 2014-04-11
JP5782178B2 (ja) 2015-09-24
BR112013025222A2 (pt) 2016-12-27
US20120264772A1 (en) 2012-10-18
US8765776B2 (en) 2014-07-01
PE20141049A1 (es) 2014-09-05
NI201300106A (es) 2014-05-05
MA35107B1 (fr) 2014-05-02
AU2011365756B2 (en) 2015-07-30
CO6821940A2 (es) 2013-12-31
GT201300241A (es) 2015-08-13
CR20130526A (es) 2014-03-11
UA110244C2 (en) 2015-12-10
JP2014510785A (ja) 2014-05-01
EA024096B1 (ru) 2016-08-31
WO2012141385A1 (en) 2012-10-18
MX341450B (es) 2016-08-19
CA2832758A1 (en) 2012-10-18
MX2013011879A (es) 2014-03-31
ZA201307593B (en) 2015-04-29
MY160432A (en) 2017-03-15
SG194162A1 (en) 2013-11-29
ECSP13012962A (es) 2013-11-29
BR112013025222B8 (pt) 2020-05-05
CA2832758C (en) 2015-12-15
AU2011365756A1 (en) 2013-10-31
BR112013025222B1 (pt) 2020-03-17

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MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ MD