EA200870093A1 - Применение производных бензоконденсированного гетероциклического сульфамида для лечения ожирения - Google Patents

Применение производных бензоконденсированного гетероциклического сульфамида для лечения ожирения

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Publication number
EA200870093A1
EA200870093A1 EA200870093A EA200870093A EA200870093A1 EA 200870093 A1 EA200870093 A1 EA 200870093A1 EA 200870093 A EA200870093 A EA 200870093A EA 200870093 A EA200870093 A EA 200870093A EA 200870093 A1 EA200870093 A1 EA 200870093A1
Authority
EA
Eurasian Patent Office
Prior art keywords
derivatives
obesity
benzen
treatment
application
Prior art date
Application number
EA200870093A
Other languages
English (en)
Other versions
EA016560B1 (ru
Inventor
Вирджиния Л. Смит-Свинтоски
Аллен Б. Рейтц
Original Assignee
Янссен Фармацевтика Н.В.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Янссен Фармацевтика Н.В. filed Critical Янссен Фармацевтика Н.В.
Publication of EA200870093A1 publication Critical patent/EA200870093A1/ru
Publication of EA016560B1 publication Critical patent/EA016560B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrane Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)

Abstract

Настоящее изобретение относится к способу лечения ожирения, стимулирования потери массы тела и/или снижения аппетита, который включает введение нуждающемуся в этом субъекту терапевтически эффективного количества одного или нескольких новых производных бензоконденсированного гетероциклического сульфамида формулы (I), представленных в настоящем описании изобретения.
EA200870093A 2005-12-19 2006-12-19 Способ лечения ожирения, стимулирования потери массы тела и снижения аппетита с использованием производных бензоконденсированного гетероциклического сульфамида EA016560B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US75149905P 2005-12-19 2005-12-19
US11/611,938 US8492431B2 (en) 2005-12-19 2006-12-18 Use of benzo-fused heterocycle sulfamide derivatives for the treatment of obesity
PCT/US2006/048681 WO2007075833A2 (en) 2005-12-19 2006-12-19 Use of benzo-fused heterocycle sulfamide derivatives for the treatment of obesity

Publications (2)

Publication Number Publication Date
EA200870093A1 true EA200870093A1 (ru) 2009-02-27
EA016560B1 EA016560B1 (ru) 2012-05-30

Family

ID=37992995

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200870093A EA016560B1 (ru) 2005-12-19 2006-12-19 Способ лечения ожирения, стимулирования потери массы тела и снижения аппетита с использованием производных бензоконденсированного гетероциклического сульфамида

Country Status (31)

Country Link
US (1) US8492431B2 (ru)
EP (1) EP1968574B9 (ru)
JP (1) JP5190378B2 (ru)
KR (1) KR101363308B1 (ru)
CN (1) CN101365442B (ru)
AR (1) AR058389A1 (ru)
AT (1) ATE519484T1 (ru)
AU (1) AU2006331637B2 (ru)
BR (1) BRPI0620019A2 (ru)
CA (1) CA2634093C (ru)
CR (1) CR10164A (ru)
CY (1) CY1112357T1 (ru)
DK (1) DK1968574T3 (ru)
EA (1) EA016560B1 (ru)
ES (1) ES2369761T3 (ru)
HK (1) HK1124540A1 (ru)
HR (1) HRP20110726T2 (ru)
IL (1) IL192107A (ru)
ME (1) ME01344B (ru)
MY (1) MY145823A (ru)
NO (1) NO20083006L (ru)
NZ (1) NZ568960A (ru)
PE (1) PE20070813A1 (ru)
PL (1) PL1968574T3 (ru)
PT (1) PT1968574E (ru)
RS (1) RS52044B (ru)
SI (1) SI1968574T1 (ru)
SV (1) SV2008002952A (ru)
UY (1) UY30033A1 (ru)
WO (1) WO2007075833A2 (ru)
ZA (1) ZA200806279B (ru)

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US8497298B2 (en) 2005-12-19 2013-07-30 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
AU2007253814A1 (en) 2006-05-19 2007-11-29 Janssen Pharmaceutica N.V. Co-therapy for the treatment of epilepsy
US20090247616A1 (en) * 2008-03-26 2009-10-01 Smith-Swintosky Virginia L Use of benzo-fused heterocyle sulfamide derivatives for the treatment of anxiety
CA2722978A1 (en) 2008-04-29 2009-11-05 Nsab, Filial Af Neurosearch Sweden Ab, Sverige Modulators of dopamine neurotransmission
DK2271638T3 (da) * 2008-04-29 2011-11-28 Nsab Af Neurosearch Sweden Ab Modulatorer af dopaminneurotransmission
JP2011519839A (ja) * 2008-04-29 2011-07-14 エヌエスエイビー、フィリアル アヴ ノイロサーチ スウェーデン エービー、スヴェーリエ ドーパミン神経伝達のモジュレーター
EA018567B1 (ru) 2008-06-23 2013-08-30 Янссен Фармацевтика Нв Кристаллическая форма (2s)-(-)-n-(6-хлор-2,3-дигидробензо[1,4]диоксин-2-илметил)сульфамида
US8815939B2 (en) * 2008-07-22 2014-08-26 Janssen Pharmaceutica Nv Substituted sulfamide derivatives
WO2013049021A1 (en) 2011-09-29 2013-04-04 Janssen Pharmaceutica Nv Process for the preparation of sulfamide derivatives
WO2013045681A1 (en) 2011-09-29 2013-04-04 Janssen Pharmaceutica Nv Improved process for the preparation of sulfamide derivatives

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AU2006331637B2 (en) 2013-01-10
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UY30033A1 (es) 2007-03-30
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