EA200700217A1 - Фармацевтическая композиция в форме таблетки для нахождения в желудке, содержащая активное вещество - Google Patents

Фармацевтическая композиция в форме таблетки для нахождения в желудке, содержащая активное вещество

Info

Publication number
EA200700217A1
EA200700217A1 EA200700217A EA200700217A EA200700217A1 EA 200700217 A1 EA200700217 A1 EA 200700217A1 EA 200700217 A EA200700217 A EA 200700217A EA 200700217 A EA200700217 A EA 200700217A EA 200700217 A1 EA200700217 A1 EA 200700217A1
Authority
EA
Eurasian Patent Office
Prior art keywords
stomach
pharmaceutical composition
active substance
tablet
location
Prior art date
Application number
EA200700217A
Other languages
English (en)
Other versions
EA012981B1 (ru
Inventor
Жерар Ало
Эстелль Шуэн
Натали Дюфрен-Арокиассами
Original Assignee
Санофи-Авентис
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34950702&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200700217(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Санофи-Авентис filed Critical Санофи-Авентис
Publication of EA200700217A1 publication Critical patent/EA200700217A1/ru
Publication of EA012981B1 publication Critical patent/EA012981B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0065—Forms with gastric retention, e.g. floating on gastric juice, adhering to gastric mucosa, expanding to prevent passage through the pylorus
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat

Abstract

Фармацевтическая композиция в форме матричной таблетки для нахождения в желудке, содержащая активное вещество, отличающаяся тем, что через 15 мин с момента начала контактирования со средой, характерной для содержимого желудка, она увеличивается в объеме со степенью разбухания по меньшей мере 200%.
EA200700217A 2004-08-19 2005-08-17 Фармацевтическая композиция в форме таблетки для нахождения в желудке, содержащая активное вещество EA012981B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0408986A FR2874325B1 (fr) 2004-08-19 2004-08-19 Composition pharmaceutique sous forme de comprime a residence gastrique contenant de l'alfuzosine
PCT/FR2005/002092 WO2006021692A1 (fr) 2004-08-19 2005-08-17 Composition pharmaceutique sous forme de comprime a residence gastrique contenant un principe actif

Publications (2)

Publication Number Publication Date
EA200700217A1 true EA200700217A1 (ru) 2007-08-31
EA012981B1 EA012981B1 (ru) 2010-02-26

Family

ID=34950702

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200700217A EA012981B1 (ru) 2004-08-19 2005-08-17 Фармацевтическая композиция в форме таблетки для нахождения в желудке, содержащая активное вещество

Country Status (23)

Country Link
US (1) US20070190140A1 (ru)
EP (1) EP1781295A1 (ru)
JP (1) JP5048492B2 (ru)
KR (1) KR20070046124A (ru)
CN (1) CN101022808B (ru)
AR (1) AR050696A1 (ru)
AU (1) AU2005276307B2 (ru)
BR (1) BRPI0514532A (ru)
CA (1) CA2577361C (ru)
EA (1) EA012981B1 (ru)
FR (1) FR2874325B1 (ru)
HK (1) HK1112575A1 (ru)
IL (1) IL181150A0 (ru)
MA (1) MA28862B1 (ru)
MX (1) MX2007001957A (ru)
MY (1) MY145832A (ru)
NO (1) NO20071315L (ru)
NZ (1) NZ553673A (ru)
PE (1) PE20060639A1 (ru)
TW (1) TWI357329B (ru)
UY (1) UY29073A1 (ru)
WO (1) WO2006021692A1 (ru)
ZA (1) ZA200701443B (ru)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9205094B2 (en) 2006-12-22 2015-12-08 Ironwood Pharmaceuticals, Inc. Compositions comprising bile acid sequestrants for treating esophageal disorders
WO2008102235A1 (en) * 2007-02-20 2008-08-28 Aurobindo Pharma Limited Controlled release formulations of alfuzosin
JP2008280251A (ja) * 2007-05-08 2008-11-20 Shin Etsu Chem Co Ltd 多層錠及びその製造方法
CN102076215A (zh) 2008-06-30 2011-05-25 托卡根公司 5-氟胞嘧啶制剂及其用途
WO2011102506A1 (ja) * 2010-02-22 2011-08-25 第一三共株式会社 経口用徐放性固形製剤
US20130156720A1 (en) 2010-08-27 2013-06-20 Ironwood Pharmaceuticals, Inc. Compositions and methods for treating or preventing metabolic syndrome and related diseases and disorders
US10569071B2 (en) 2015-08-31 2020-02-25 Ethicon Llc Medicant eluting adjuncts and methods of using medicant eluting adjuncts
US10245034B2 (en) * 2015-08-31 2019-04-02 Ethicon Llc Inducing tissue adhesions using surgical adjuncts and medicants

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH630257A5 (en) * 1975-03-17 1982-06-15 Hoffmann La Roche Sustained release formulation
DE4036757A1 (de) * 1990-11-17 1992-05-21 Bayer Ag Antazida-zubereitung mit verlaengerter magenverweilzeit
IT1282650B1 (it) * 1996-02-19 1998-03-31 Jagotec Ag Compressa farmaceutica,caratterizzata da elevato aumento di volume a contatto con liquidi biologici
PT938318E (pt) * 1996-08-29 2001-10-30 Jagotec Ag Comprimido com libertacao controlada de cloridrato de alfuzosina
US6271278B1 (en) * 1997-05-13 2001-08-07 Purdue Research Foundation Hydrogel composites and superporous hydrogel composites having fast swelling, high mechanical strength, and superabsorbent properties
US6197340B1 (en) * 1998-05-28 2001-03-06 Medical Research Institute Controlled release lipoic acid
FR2784583B1 (fr) * 1998-10-16 2002-01-25 Synthelabo Composition pharmaceutique a residence gastrique et a liberation controlee
US6632451B2 (en) * 1999-06-04 2003-10-14 Dexcel Pharma Technologies Ltd. Delayed total release two pulse gastrointestinal drug delivery system
DE10014588A1 (de) * 2000-03-27 2001-10-04 Basf Ag Wirkstoffhaltige Schwimmformen enthaltend Polyvinylacetat und Polyvinylpyrrolidon, deren Verwendung und Herstellung
US6476006B2 (en) * 2000-06-23 2002-11-05 Teva Pharmaceutical Industries, Ltd. Composition and dosage form for delayed gastric release of alendronate and/or other bis-phosphonates
US7674480B2 (en) * 2000-06-23 2010-03-09 Teva Pharmaceutical Industries Ltd. Rapidly expanding composition for gastric retention and controlled release of therapeutic agents, and dosage forms including the composition
AU2001268722B8 (en) * 2000-06-23 2005-09-29 Teva Pharmaceutical Industries Ltd. Rapidly expanding composition for gastric retention and controlled release of therapeutic agents, and dosage forms including the composition
US6881424B1 (en) * 2000-09-05 2005-04-19 Mionix Corporation Highly acidic metalated organic acid
FR2820319B3 (fr) * 2001-02-08 2003-12-05 Ellipse Pharmaceuticals Procede de fabrication d'un comprime flottant incluant de l'alfuzosine et comprime obtenu
ATE477795T1 (de) * 2001-07-04 2010-09-15 Sun Pharma Advanced Res Co Ltd Magenretentionssystem mit kontrollierter arzneimittelfreisetzung
US20040219186A1 (en) * 2001-08-16 2004-11-04 Ayres James W. Expandable gastric retention device
US20030152622A1 (en) * 2001-10-25 2003-08-14 Jenny Louie-Helm Formulation of an erodible, gastric retentive oral diuretic
US20030215526A1 (en) * 2002-03-08 2003-11-20 Scott Stofik Stable formulations of angiotensin converting enzyme (ACE) inhibitors

Also Published As

Publication number Publication date
KR20070046124A (ko) 2007-05-02
CN101022808B (zh) 2013-05-29
AR050696A1 (es) 2006-11-15
WO2006021692A8 (fr) 2007-04-12
FR2874325A1 (fr) 2006-02-24
EA012981B1 (ru) 2010-02-26
US20070190140A1 (en) 2007-08-16
JP2008509973A (ja) 2008-04-03
FR2874325B1 (fr) 2006-10-20
TWI357329B (en) 2012-02-01
ZA200701443B (en) 2008-05-25
NZ553673A (en) 2010-10-29
EP1781295A1 (fr) 2007-05-09
CA2577361C (fr) 2013-10-01
AU2005276307A1 (en) 2006-03-02
WO2006021692A1 (fr) 2006-03-02
MY145832A (en) 2012-04-30
NO20071315L (no) 2007-03-09
CN101022808A (zh) 2007-08-22
IL181150A0 (en) 2007-07-04
CA2577361A1 (fr) 2006-03-02
BRPI0514532A (pt) 2008-06-17
JP5048492B2 (ja) 2012-10-17
TW200618802A (en) 2006-06-16
MX2007001957A (es) 2007-04-25
UY29073A1 (es) 2006-03-31
AU2005276307B2 (en) 2011-02-24
HK1112575A1 (en) 2008-09-12
PE20060639A1 (es) 2006-07-20
MA28862B1 (fr) 2007-09-03

Similar Documents

Publication Publication Date Title
EA200700217A1 (ru) Фармацевтическая композиция в форме таблетки для нахождения в желудке, содержащая активное вещество
BRPI0414000B8 (pt) composição farmacêutica sólida oral de liberação prolongada contendo tacrolimus na forma de uma dispersão sólida, forma de dosagem, e, uso da composição farmacêutica
CY1120377T1 (el) Στερεη φαρμακευτικη δοσολογικη φαρμακοτεχνικη μορφη που περιεχει λοπιναβιρη
MXPA05005527A (es) Forma de dosis de alergeno.
DK1781277T3 (da) Kombinationssammensætning, der omfatter Ibuprofen og Paracetamol
EA200702116A1 (ru) Фармацевтическая дозированная форма (варианты) с контролируемым высвобождением антигипергликемического средства в комбинации с производным тиазолидиндиона
IS8542A (is) Efni, lyfjasamsetningar og notkun á efnum til að framleiða lyf gegn efnaskiptaröskunum
DE60205749D1 (de) Oral anzuwendende arzneizusammensetzungen mit gesteuerter wirkstoffabgabe
RS50660B (sr) Dihidrotetrabenazini i farmaceutske kompozicije koje ih sadrže
PA8578301A1 (es) Composicion de tabletas de liberacion sostenida de pramipexol
MY147641A (en) Fast release paracetamol tablets
ATE354362T1 (de) Stabilisierte pharmazeutische zusammensetzung enthaltend einen amorphen wirkstoff
WO2006041878A3 (en) Primary examiner
GB2443793B (en) Product, method of manufacture and use
WO2005007137A3 (de) Ambroxolhaltige tabletten
TR201819108T4 (tr) Kontrollü salımlı matrisli farmasötik dozaj formülasyonu.
ZA200506992B (en) Fibrate tablet and method for the production thereof
MY149933A (en) Dosage form comprising an exine coating of sporopollenin or derivatized sporopollenin
WO2007016350A3 (en) Modified release tablet formulations with enhanced mechanical properties
BR0314787A (pt) Forma de dosagem de liberação modificada
EA200702386A1 (ru) Твердая фармацевтическая композиция для продолжительного высвобождения 1-(2,3,4-триметоксибензил)пиперазина и способ ее получения
RS51307B (sr) Farmaceutski sastav u obliku hidrogela za transdermalnu aplikaciju aktivnih materija
WO2009120844A3 (en) Pharmaceutical compositions comprising insulin sensitizer and insulin secretagogue
SV2006002224A (es) Composicion farmaceutica ref. bhco41368-sv
TR200701424T1 (tr) Suda çözünebilen katı dozaj formunda farmasötik bileşim.

Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU