EA200702386A1 - Твердая фармацевтическая композиция для продолжительного высвобождения 1-(2,3,4-триметоксибензил)пиперазина и способ ее получения - Google Patents
Твердая фармацевтическая композиция для продолжительного высвобождения 1-(2,3,4-триметоксибензил)пиперазина и способ ее полученияInfo
- Publication number
- EA200702386A1 EA200702386A1 EA200702386A EA200702386A EA200702386A1 EA 200702386 A1 EA200702386 A1 EA 200702386A1 EA 200702386 A EA200702386 A EA 200702386A EA 200702386 A EA200702386 A EA 200702386A EA 200702386 A1 EA200702386 A1 EA 200702386A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- piperazine
- pharmaceutical composition
- solid pharmaceutical
- trimetoxibenzyl
- exemption
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
Abstract
Твердая фармацевтическая композиция продолжительного высвобождения, которая включает активный ингредиент 1-(2,3,4-триметоксибензил)пиперазин или фармацевтически приемлемую соль 1-(2,3,4-триметоксибензил)пиперазина, в комбинации по крайней мере с одним полиэтиленоксидом и по крайней мере одним смазывающим агентом и одним или более фармацевтически приемлемыми наполнителями.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0504997A FR2885807B1 (fr) | 2005-05-18 | 2005-05-18 | Composition pharmaceutique solide a liberation prolongee de 1-(2,3,4-trimethoxybenzyl) piperazine, et procede de preparation |
PCT/FR2006/050128 WO2006123073A1 (fr) | 2005-05-18 | 2006-02-13 | Composition pharmaceutique solide a liberation prolongee de 1-(2,3,4-trimethoxybenzyl)piperazine, et procede de preparation. |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200702386A1 true EA200702386A1 (ru) | 2008-04-28 |
EA013645B1 EA013645B1 (ru) | 2010-06-30 |
Family
ID=35583424
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200702386A EA013645B1 (ru) | 2005-05-18 | 2006-02-13 | Твердая фармацевтическая композиция с пролонгированным высвобождением 1-(2,3,4-триметоксибензил)пиперазина и способ ее получения |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP1881831A1 (ru) |
EA (1) | EA013645B1 (ru) |
FR (1) | FR2885807B1 (ru) |
UA (1) | UA89408C2 (ru) |
WO (1) | WO2006123073A1 (ru) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0815602A2 (pt) * | 2007-08-08 | 2015-03-03 | Usv Ltd | Composições de liberação prolongada de trimetazidina e processo para a preparação das mesmas |
EP2200591A2 (en) * | 2007-09-11 | 2010-06-30 | Ranbaxy Laboratories Limited | Controlled release pharmaceutical dosage forms of trimetazidine |
JP2012515757A (ja) * | 2009-01-20 | 2012-07-12 | マイクロ ラブス リミテッド | トリメタジジンの放出調節固形薬剤組成物及びその製造方法 |
TR201001902A2 (tr) * | 2010-03-12 | 2011-04-21 | Ali̇ Rai̇f İlaç Sanayi̇ Ve Ti̇caret A.Ş. | Uzatılmış salınımlı trimetazidin tablet |
PL2394644T3 (pl) * | 2010-05-04 | 2014-11-28 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Preparat trimetazydyny o różnych profilach uwalniania |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2717687B1 (fr) * | 1994-03-24 | 1996-06-14 | Adir | Compositions pharmaceutiques permettant la libération prolongée de trimétazidine après administration par voie orale. |
FR2802424B1 (fr) * | 1999-12-17 | 2002-02-15 | Adir | Comprime matriciel permettant la liberation prolongee de trimetazidine apres administration par voie orale |
DE60042972D1 (de) * | 2000-10-05 | 2009-10-29 | Usv Ltd | Trimetazidine enthaltendes Arzneimittel mit verzögerter Wirkstoffabgabe und Verfahren zur Herstellung |
FR2818549B1 (fr) * | 2000-12-26 | 2003-02-07 | Servier Lab | Composition pharmaceutique solide thermoformable pour la liberation controlee de trimetazidine |
HUP0500382A3 (en) * | 2001-11-21 | 2008-03-28 | Themis Lab Private Ltd | Sustained release pharmaceutical compositions containing microbeads of trimetazidine dihydrochloride and process for producing them |
-
2005
- 2005-05-18 FR FR0504997A patent/FR2885807B1/fr active Active
-
2006
- 2006-02-13 EP EP06709507A patent/EP1881831A1/fr not_active Withdrawn
- 2006-02-13 UA UAA200714180A patent/UA89408C2/ru unknown
- 2006-02-13 WO PCT/FR2006/050128 patent/WO2006123073A1/fr not_active Application Discontinuation
- 2006-02-13 EA EA200702386A patent/EA013645B1/ru not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
FR2885807B1 (fr) | 2008-05-16 |
FR2885807A1 (fr) | 2006-11-24 |
EP1881831A1 (fr) | 2008-01-30 |
EA013645B1 (ru) | 2010-06-30 |
WO2006123073A1 (fr) | 2006-11-23 |
UA89408C2 (ru) | 2010-01-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |