EA200700109A1 - Способы лечения офтальмологических состояний (варианты) - Google Patents

Способы лечения офтальмологических состояний (варианты)

Info

Publication number
EA200700109A1
EA200700109A1 EA200700109A EA200700109A EA200700109A1 EA 200700109 A1 EA200700109 A1 EA 200700109A1 EA 200700109 A EA200700109 A EA 200700109A EA 200700109 A EA200700109 A EA 200700109A EA 200700109 A1 EA200700109 A1 EA 200700109A1
Authority
EA
Eurasian Patent Office
Prior art keywords
treatment
methods
compounds
options
derivatives
Prior art date
Application number
EA200700109A
Other languages
English (en)
Other versions
EA011864B1 (ru
Inventor
Кеннет Уиддер
Джэй Личтер
Натан Л. Мэйта
Original Assignee
Сирион Терапьютикс, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34981643&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200700109(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Сирион Терапьютикс, Инк. filed Critical Сирион Терапьютикс, Инк.
Publication of EA200700109A1 publication Critical patent/EA200700109A1/ru
Publication of EA011864B1 publication Critical patent/EA011864B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N2800/00—Detection or diagnosis of diseases
    • G01N2800/16—Ophthalmology
    • G01N2800/164—Retinal disorders, e.g. retinopathy

Abstract

Соединения, которые вызывают обратимую ночную ("куриную") слепоту, можно использовать для лечения офтальмологических состояний, ассоциированных с избыточным продуцированием ненужных продуктов, которые аккумулируются в процессе зрительного цикла. Мы описываем способы и композиции с применением таких соединений и их производных для лечения, например, макулярных дегенераций (дегенераций жёлтого пята) или дистрофий или для ослабления симптомов, обусловленных такими состояниями. Такие соединения и их производные можно использовать в качестве самостоятельного терапевтического агента или в комбинации с другими агентами или методами лечения.
EA200700109A 2004-06-23 2005-06-06 Применение 4-гидроксифенилретинамида и 4-метоксифенилретинамида для лечения офтальмологических состояний EA011864B1 (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US58229304P 2004-06-23 2004-06-23
US62969504P 2004-11-19 2004-11-19
US66090405P 2005-03-11 2005-03-11
US67240505P 2005-04-18 2005-04-18
PCT/US2005/020080 WO2006007314A1 (en) 2004-06-23 2005-06-06 Methods and compositions for treating ophthalmic conditions with retinyl derivatives

Publications (2)

Publication Number Publication Date
EA200700109A1 true EA200700109A1 (ru) 2007-10-26
EA011864B1 EA011864B1 (ru) 2009-06-30

Family

ID=34981643

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200700109A EA011864B1 (ru) 2004-06-23 2005-06-06 Применение 4-гидроксифенилретинамида и 4-метоксифенилретинамида для лечения офтальмологических состояний

Country Status (27)

Country Link
US (3) US8314152B2 (ru)
EP (3) EP1768657B1 (ru)
JP (1) JP4855396B2 (ru)
KR (1) KR100862930B1 (ru)
AR (1) AR049929A1 (ru)
AT (1) ATE404188T1 (ru)
AU (1) AU2005262558B8 (ru)
BR (1) BRPI0512569A (ru)
CA (1) CA2569691C (ru)
CY (1) CY1110435T1 (ru)
DE (1) DE602005008970D1 (ru)
DK (1) DK1768657T3 (ru)
EA (1) EA011864B1 (ru)
ES (1) ES2313368T3 (ru)
GE (1) GEP20084520B (ru)
HK (1) HK1107671A1 (ru)
IL (1) IL179872A (ru)
LV (1) LV13564B (ru)
MX (1) MXPA06014978A (ru)
NO (1) NO20070408L (ru)
NZ (1) NZ551955A (ru)
PL (1) PL1768657T3 (ru)
PT (1) PT1768657E (ru)
SG (1) SG140607A1 (ru)
SI (1) SI1768657T1 (ru)
TW (1) TWI396532B (ru)
WO (1) WO2006007314A1 (ru)

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DE602005008970D1 (de) 2008-09-25
PL1768657T3 (pl) 2009-01-30
ATE404188T1 (de) 2008-08-15
TWI396532B (zh) 2013-05-21
US20100298443A1 (en) 2010-11-25
CA2569691C (en) 2010-08-17
EA011864B1 (ru) 2009-06-30
BRPI0512569A (pt) 2008-03-25
IL179872A0 (en) 2007-05-15
GEP20084520B (en) 2008-10-27
IL179872A (en) 2013-01-31
JP2008504257A (ja) 2008-02-14
EP2025336A1 (en) 2009-02-18
CA2569691A1 (en) 2006-01-19
JP4855396B2 (ja) 2012-01-18
AU2005262558A1 (en) 2006-01-19
PT1768657E (pt) 2008-11-25
AU2005262558B8 (en) 2008-04-10
EP2277516A1 (en) 2011-01-26
WO2006007314A1 (en) 2006-01-19
EP1768657B1 (en) 2008-08-13
LV13564B (en) 2008-02-20
NZ551955A (en) 2010-08-27
AR049929A1 (es) 2006-09-13
AU2005262558B2 (en) 2008-03-20
HK1107671A1 (en) 2008-04-11
US8314152B2 (en) 2012-11-20
SG140607A1 (en) 2008-03-28
CY1110435T1 (el) 2015-04-29
KR100862930B1 (ko) 2008-10-13
ES2313368T3 (es) 2009-03-01
NO20070408L (no) 2007-03-20
KR20070074541A (ko) 2007-07-12
US20110294891A1 (en) 2011-12-01
MXPA06014978A (es) 2007-04-25
DK1768657T3 (da) 2008-12-01
US8410168B2 (en) 2013-04-02
TW200612891A (en) 2006-05-01
US20060167088A1 (en) 2006-07-27
SI1768657T1 (sl) 2009-02-28
EP1768657A1 (en) 2007-04-04

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