MX2012003220A - Formulaciones farmaceuticas que comprenden 9-cis-retinil esteres en un vehiculo de lipido. - Google Patents

Formulaciones farmaceuticas que comprenden 9-cis-retinil esteres en un vehiculo de lipido.

Info

Publication number
MX2012003220A
MX2012003220A MX2012003220A MX2012003220A MX2012003220A MX 2012003220 A MX2012003220 A MX 2012003220A MX 2012003220 A MX2012003220 A MX 2012003220A MX 2012003220 A MX2012003220 A MX 2012003220A MX 2012003220 A MX2012003220 A MX 2012003220A
Authority
MX
Mexico
Prior art keywords
cis
pharmaceutical formulations
lipid vehicle
retinyl esters
retinyl
Prior art date
Application number
MX2012003220A
Other languages
English (en)
Inventor
Ronald Erwin Boch
Original Assignee
Quadra Logic Tech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Quadra Logic Tech Inc filed Critical Quadra Logic Tech Inc
Publication of MX2012003220A publication Critical patent/MX2012003220A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/045Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/07Retinol compounds, e.g. vitamin A
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00Preparations for use in therapy

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dispersion Chemistry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Nutrition Science (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Non-Alcoholic Beverages (AREA)

Abstract

Se describen formulaciones farmacéuticas que comprenden 9-cis-retinil ésteres en un vehículo de lípido como terapias de reemplazo de retinoide para tratar degeneraciones retinales en seres humanos.
MX2012003220A 2009-09-15 2009-09-30 Formulaciones farmaceuticas que comprenden 9-cis-retinil esteres en un vehiculo de lipido. MX2012003220A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24274109P 2009-09-15 2009-09-15
PCT/US2009/059126 WO2011034551A2 (en) 2009-09-15 2009-09-30 Pharmaceutical formulations comprising 9-cis-retinyl esters in a lipid vehicle

Publications (1)

Publication Number Publication Date
MX2012003220A true MX2012003220A (es) 2012-08-03

Family

ID=43242391

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012003220A MX2012003220A (es) 2009-09-15 2009-09-30 Formulaciones farmaceuticas que comprenden 9-cis-retinil esteres en un vehiculo de lipido.

Country Status (14)

Country Link
US (3) US20120178806A1 (es)
JP (2) JP5663025B2 (es)
KR (1) KR101710505B1 (es)
CN (1) CN102612375B (es)
AR (1) AR076184A1 (es)
AU (1) AU2009352678B2 (es)
BR (1) BR112012005905A2 (es)
CA (1) CA2774168C (es)
HK (1) HK1170158A1 (es)
IN (1) IN2012DN02466A (es)
MX (1) MX2012003220A (es)
MY (1) MY174082A (es)
RU (1) RU2546005C2 (es)
WO (1) WO2011034551A2 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112012005905A2 (pt) 2009-09-15 2020-02-18 Qlt Inc. Formulação farmacêutica, método para tratar a amaurose congênita de leber em um indivíduo humano, e, método para tratar um indivíduo
US9173856B2 (en) * 2010-04-19 2015-11-03 Qlt Inc. Therapeutic regimen and methods for treating or ameliorating visual disorders associated with an endogenous retinoid deficiency
KR102029657B1 (ko) * 2011-06-08 2019-10-08 닛토덴코 가부시키가이샤 표적 약물 전달체 및 siRNA 활성을 증가시키는 화합물
BR112014021602A2 (pt) 2012-03-01 2021-06-08 Quadra Logic Tech Inc uso, kit e derivado de retinal sintético para melhorar a função visual em distúrbios visuais associados com a deficiência de produção endógena de retinóide
EP3317372B1 (en) 2015-06-30 2018-10-17 Unilever NV Composition containing vegetable oil, caramel and phenolic compounds
MY194096A (en) * 2016-04-28 2022-11-11 Spark Therapeutics Inc Relative potency assay for viral vector encoding isomerhydrolases
HUE064808T2 (hu) 2016-11-17 2024-04-28 Univ Of Debrecen Prekurzor vegyületek az A5-vitamin útvonal retinoidjainak elõállítására és azok alkalmazása
CN116056691A (zh) * 2020-06-09 2023-05-02 典晶生物医药科技(苏州)有限公司 使用每日低剂量的类视黄醇化合物治疗视觉障碍的方法

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Also Published As

Publication number Publication date
WO2011034551A2 (en) 2011-03-24
CN102612375B (zh) 2016-01-27
IN2012DN02466A (es) 2015-08-21
BR112012005905A2 (pt) 2020-02-18
US20120178806A1 (en) 2012-07-12
US20190183835A1 (en) 2019-06-20
HK1170158A1 (zh) 2013-02-22
CA2774168A1 (en) 2011-03-24
AU2009352678A1 (en) 2012-04-05
AR076184A1 (es) 2011-05-26
US20170007565A1 (en) 2017-01-12
KR20120064707A (ko) 2012-06-19
WO2011034551A3 (en) 2011-12-15
RU2546005C2 (ru) 2015-04-10
KR101710505B1 (ko) 2017-02-27
JP2013504617A (ja) 2013-02-07
CN102612375A (zh) 2012-07-25
US10736865B2 (en) 2020-08-11
JP2014185185A (ja) 2014-10-02
RU2012114791A (ru) 2013-10-27
MY174082A (en) 2020-03-09
JP5663025B2 (ja) 2015-02-04
AU2009352678B2 (en) 2015-05-21
US10130606B2 (en) 2018-11-20
CA2774168C (en) 2021-02-23

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