EA200600400A1 - Новая композиция, содержащая росиглитазон и другое противодиабетическое средство - Google Patents
Новая композиция, содержащая росиглитазон и другое противодиабетическое средствоInfo
- Publication number
- EA200600400A1 EA200600400A1 EA200600400A EA200600400A EA200600400A1 EA 200600400 A1 EA200600400 A1 EA 200600400A1 EA 200600400 A EA200600400 A EA 200600400A EA 200600400 A EA200600400 A EA 200600400A EA 200600400 A1 EA200600400 A1 EA 200600400A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- diabetic
- composition containing
- new composition
- containing rosiglitazone
- rosiglitazone
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
Abstract
Пероральная лекарственная форма, включающая эродируемое ядро, которое содержит росиглитазон или его фармацевтически приемлемую соль или сольват и другое противодиабетическое средство, при этом ядро имеет покрытие с одним или несколькими отверстиями, характеризующееся тем, что покрытие является эродируемым в заданных условиях рН; способ получения такой лекарственной формы и применение такой лекарственной формы в медицине.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0318824.0A GB0318824D0 (en) | 2003-08-11 | 2003-08-11 | Novel composition |
PCT/EP2004/008970 WO2005013956A1 (en) | 2003-08-11 | 2004-08-09 | Novel composition comprising rosiglitazone and another antidiabetic agent |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200600400A1 true EA200600400A1 (ru) | 2006-08-25 |
EA011550B1 EA011550B1 (ru) | 2009-04-28 |
Family
ID=27840010
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200600400A EA011550B1 (ru) | 2003-08-11 | 2004-08-09 | Композиция росиглитазона и метформина |
EA200800966A EA200800966A1 (ru) | 2003-08-11 | 2004-08-09 | Новая композиция, содержащая росиглитазон и другое противодиабетическое средство |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200800966A EA200800966A1 (ru) | 2003-08-11 | 2004-08-09 | Новая композиция, содержащая росиглитазон и другое противодиабетическое средство |
Country Status (37)
Country | Link |
---|---|
US (1) | US20080206336A1 (ru) |
EP (1) | EP1663191B1 (ru) |
JP (1) | JP4714147B2 (ru) |
KR (1) | KR20060071396A (ru) |
CN (2) | CN102397551A (ru) |
AP (1) | AP2006003489A0 (ru) |
AR (1) | AR045230A1 (ru) |
AT (1) | ATE455542T1 (ru) |
AU (1) | AU2004262933B2 (ru) |
BR (1) | BRPI0413419A (ru) |
CA (1) | CA2534480A1 (ru) |
CY (1) | CY1109923T1 (ru) |
DE (1) | DE602004025257D1 (ru) |
DK (1) | DK1663191T3 (ru) |
EA (2) | EA011550B1 (ru) |
EC (1) | ECSP066338A (ru) |
ES (1) | ES2339554T3 (ru) |
GB (1) | GB0318824D0 (ru) |
HK (1) | HK1092051A1 (ru) |
HR (1) | HRP20100160T1 (ru) |
IL (1) | IL173177A0 (ru) |
IS (1) | IS2745B (ru) |
MA (1) | MA27996A1 (ru) |
MX (1) | MXPA06001629A (ru) |
MY (1) | MY151053A (ru) |
NO (1) | NO20061161L (ru) |
NZ (1) | NZ544632A (ru) |
OA (1) | OA13233A (ru) |
PE (1) | PE20050357A1 (ru) |
PL (1) | PL1663191T3 (ru) |
PT (1) | PT1663191E (ru) |
SG (1) | SG165178A1 (ru) |
SI (1) | SI1663191T1 (ru) |
TW (1) | TW200517146A (ru) |
UA (1) | UA82537C2 (ru) |
UY (1) | UY28461A1 (ru) |
WO (1) | WO2005013956A1 (ru) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY125516A (en) * | 1999-11-16 | 2006-08-30 | Smithkline Beecham Plc | Novel composition based on thiazolidinedione and metformin and use |
GB0203296D0 (en) * | 2002-02-12 | 2002-03-27 | Glaxo Group Ltd | Novel composition |
US8637512B2 (en) | 2002-07-29 | 2014-01-28 | Glaxo Group Limited | Formulations and method of treatment |
WO2005051325A2 (en) * | 2003-11-25 | 2005-06-09 | Sb Pharmco Puerto Rico Inc. | Carvedilol compositions methods of treatment and delivery |
WO2010009433A1 (en) * | 2008-07-18 | 2010-01-21 | Valeant Pharmaceuticals International | Modified release formulation and methods of use |
US20100323016A1 (en) * | 2008-07-18 | 2010-12-23 | Biljana Nadjsombati | Modified release formulation and methods of use |
US20100323015A1 (en) * | 2008-07-18 | 2010-12-23 | Biljana Nadjsombati | Modified release formulation and methods of use |
WO2011161521A1 (en) * | 2010-06-21 | 2011-12-29 | Lupin Limited | Compositions comprising metformin and rosiglitazone |
CN103153288B (zh) * | 2010-07-09 | 2017-02-15 | 詹姆斯·特林卡·格林 | 用于包括瑞格列净的短半衰期药物的组合立即/延迟释放递送系统 |
CN102727459A (zh) * | 2011-04-15 | 2012-10-17 | 江苏豪森医药集团有限公司 | 一种具有第一和第二活性药物的制剂 |
Family Cites Families (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3845770A (en) * | 1972-06-05 | 1974-11-05 | Alza Corp | Osmatic dispensing device for releasing beneficial agent |
GB8820353D0 (en) * | 1988-08-26 | 1988-09-28 | Staniforth J N | Controlled release tablet |
US5952509A (en) * | 1996-06-27 | 1999-09-14 | Takeda Chemical Industries, Ltd. | Production of benzaldehyde compounds |
GB9619757D0 (en) * | 1996-09-21 | 1996-11-06 | Knoll Ag | Chemical process |
US20020004515A1 (en) * | 1997-06-18 | 2002-01-10 | Smith Stephen Alistair | Treatment of diabetes with thiazolidinedione and metformin |
US20010049380A1 (en) * | 1997-06-18 | 2001-12-06 | Smith Stephen Alistair | Treatment of diabetes with thiazolidinedione and sulphonylurea |
US20020006939A1 (en) * | 1997-10-13 | 2002-01-17 | Smithkline Beecham P.L.C. | Use of thiazolidinediones for the treatment of hyperglycaemia |
EP1067910B1 (en) * | 1998-04-03 | 2004-05-26 | Egalet A/S | Controlled release composition |
US6099862A (en) * | 1998-08-31 | 2000-08-08 | Andrx Corporation | Oral dosage form for the controlled release of a biguanide and sulfonylurea |
UA67802C2 (ru) * | 1998-10-23 | 2004-07-15 | Пфайзер Рісьоч Енд Дівелепмент Компані, Н.В./С.А. | ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ ДЛЯ ПЕРОРАЛЬНОГО ПРИМЕНЕНИЯ С КОНТРОЛИРУЕМЫМ ВЫСВОБОЖДЕНИЕМ ИНГИБИТОРА цГМФ ФДЭ-5 (ВАРИАНТЫ), СПОСОБ ЕЕ ПОЛУЧЕНИЯ И СПОСОБ ЛЕЧЕНИЯ ЭРЕКТИЛЬНОЙ ДИСФУНКЦИИ |
ES2256927T3 (es) * | 1998-11-10 | 2006-07-16 | THE PROCTER & GAMBLE COMPANY | Composiciones blanqueantes. |
US20040081697A1 (en) * | 1998-11-12 | 2004-04-29 | Smithkline Beecham P.L.C. | Pharmaceutical composition for modified release of an insulin sensitiser and another antidiabetic agent |
EP1813273A1 (en) * | 1998-11-12 | 2007-08-01 | Smithkline Beecham Plc | Pharmaceutical composition for modified release of an insulin sensitiser and another antidiabetic agent |
US20030153607A1 (en) * | 1998-11-12 | 2003-08-14 | Smithkline Beecham P.L.C. | Novel composition and use |
US20040102486A1 (en) * | 1998-11-12 | 2004-05-27 | Smithkline Beecham Corporation | Novel method of treatment |
AU1403501A (en) * | 1999-11-16 | 2001-05-30 | Smithkline Beecham Plc | Novel composition and use |
CA2407713A1 (en) * | 2000-05-01 | 2001-11-08 | Aeropharm Technology, Inc. | A core formulation |
GB0027471D0 (en) * | 2000-11-08 | 2000-12-27 | Smithkline Beecham Plc | Processes |
GB0120835D0 (en) * | 2001-08-28 | 2001-10-17 | Smithkline Beecham Plc | Process |
GB0127805D0 (en) * | 2001-11-20 | 2002-01-09 | Smithkline Beecham Plc | Pharmaceutical composition |
MY139719A (en) * | 2002-02-12 | 2009-10-30 | Glaxo Group Ltd | Oral dosage form for controlled drug release |
GB0203296D0 (en) * | 2002-02-12 | 2002-03-27 | Glaxo Group Ltd | Novel composition |
US7785627B2 (en) * | 2002-09-20 | 2010-08-31 | Watson Pharmaceuticals, Inc. | Pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative |
-
2003
- 2003-08-11 GB GBGB0318824.0A patent/GB0318824D0/en not_active Ceased
-
2004
- 2004-08-09 JP JP2006522974A patent/JP4714147B2/ja not_active Expired - Fee Related
- 2004-08-09 EP EP04741403A patent/EP1663191B1/en active Active
- 2004-08-09 MY MYPI20043234 patent/MY151053A/en unknown
- 2004-08-09 PE PE2004000771A patent/PE20050357A1/es not_active Application Discontinuation
- 2004-08-09 MX MXPA06001629A patent/MXPA06001629A/es active IP Right Grant
- 2004-08-09 PT PT04741403T patent/PT1663191E/pt unknown
- 2004-08-09 SI SI200431376T patent/SI1663191T1/sl unknown
- 2004-08-09 DE DE602004025257T patent/DE602004025257D1/de active Active
- 2004-08-09 US US10/567,803 patent/US20080206336A1/en not_active Abandoned
- 2004-08-09 AR ARP040102846A patent/AR045230A1/es not_active Application Discontinuation
- 2004-08-09 EA EA200600400A patent/EA011550B1/ru not_active IP Right Cessation
- 2004-08-09 AP AP2006003489A patent/AP2006003489A0/xx unknown
- 2004-08-09 KR KR1020067002884A patent/KR20060071396A/ko not_active Application Discontinuation
- 2004-08-09 SG SG200901679-1A patent/SG165178A1/en unknown
- 2004-08-09 CA CA002534480A patent/CA2534480A1/en not_active Abandoned
- 2004-08-09 UY UY28461A patent/UY28461A1/es not_active Application Discontinuation
- 2004-08-09 ES ES04741403T patent/ES2339554T3/es active Active
- 2004-08-09 AU AU2004262933A patent/AU2004262933B2/en not_active Ceased
- 2004-08-09 CN CN2011103143770A patent/CN102397551A/zh active Pending
- 2004-08-09 OA OA1200600045A patent/OA13233A/en unknown
- 2004-08-09 AT AT04741403T patent/ATE455542T1/de active
- 2004-08-09 WO PCT/EP2004/008970 patent/WO2005013956A1/en active Application Filing
- 2004-08-09 EA EA200800966A patent/EA200800966A1/ru unknown
- 2004-08-09 CN CN2004800232304A patent/CN1835741B/zh not_active Expired - Fee Related
- 2004-08-09 NZ NZ544632A patent/NZ544632A/en not_active IP Right Cessation
- 2004-08-09 PL PL04741403T patent/PL1663191T3/pl unknown
- 2004-08-09 BR BRPI0413419-2A patent/BRPI0413419A/pt not_active IP Right Cessation
- 2004-08-09 DK DK04741403.2T patent/DK1663191T3/da active
- 2004-08-09 TW TW093123804A patent/TW200517146A/zh unknown
- 2004-09-08 UA UAA200601353A patent/UA82537C2/ru unknown
-
2006
- 2006-01-16 IL IL173177A patent/IL173177A0/en unknown
- 2006-01-31 EC EC2006006338A patent/ECSP066338A/es unknown
- 2006-02-17 MA MA28817A patent/MA27996A1/fr unknown
- 2006-03-02 IS IS8337A patent/IS2745B/is unknown
- 2006-03-10 NO NO20061161A patent/NO20061161L/no not_active Application Discontinuation
- 2006-11-15 HK HK06112571.6A patent/HK1092051A1/xx not_active IP Right Cessation
-
2010
- 2010-03-18 HR HR20100160T patent/HRP20100160T1/hr unknown
- 2010-03-22 CY CY20101100261T patent/CY1109923T1/el unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC1A | Registration of transfer to a eurasian application by force of assignment | ||
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |