EA200000878A1 - ЗАМЕЩЕННЫЙ 1,2,4-ТРИАЗОЛО[3,4-а]ПИРИДАЗИН - Google Patents
ЗАМЕЩЕННЫЙ 1,2,4-ТРИАЗОЛО[3,4-а]ПИРИДАЗИНInfo
- Publication number
- EA200000878A1 EA200000878A1 EA200000878A EA200000878A EA200000878A1 EA 200000878 A1 EA200000878 A1 EA 200000878A1 EA 200000878 A EA200000878 A EA 200000878A EA 200000878 A EA200000878 A EA 200000878A EA 200000878 A1 EA200000878 A1 EA 200000878A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- triazolo
- pyridazine
- substitute
- therapy
- derivative
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Описывается производное замещенного триазолопиридазина, его использование в терапии для повышения умственной способности, содержащие его композиции и способы его получения.Международная заявка была опубликована вместе с отчетом о международном поиске.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9803992.8A GB9803992D0 (en) | 1998-02-25 | 1998-02-25 | Therapeutic agents |
PCT/GB1998/001307 WO1998050385A1 (en) | 1997-05-08 | 1998-05-06 | SUBSTITUTED 1,2,4-TRIAZOLO[3,4-a]PHTHALAZINE DERIVATIVES AS GABA ALPHA 5 LIGANDS |
GBGB9824896.6A GB9824896D0 (en) | 1998-11-12 | 1998-11-12 | Therapeutic compound |
PCT/GB1999/000485 WO1999043677A1 (en) | 1998-02-25 | 1999-02-17 | SUBSTITUTED 1,2,4-TRIAZOLO[3,4-a]PYRIDAZINE |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200000878A1 true EA200000878A1 (ru) | 2001-02-26 |
EA002824B1 EA002824B1 (ru) | 2002-10-31 |
Family
ID=27269184
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200000878A EA002824B1 (ru) | 1998-02-25 | 1999-02-17 | ЗАМЕЩЕННЫЙ 1,2,4-ТРИАЗОЛО[3,4-а]ПИРИДАЗИН |
Country Status (14)
Country | Link |
---|---|
EP (1) | EP1070066A1 (ru) |
JP (1) | JP2002504554A (ru) |
CN (1) | CN1291194A (ru) |
AU (1) | AU746719B2 (ru) |
BG (1) | BG104705A (ru) |
CA (1) | CA2317416A1 (ru) |
EA (1) | EA002824B1 (ru) |
HR (1) | HRP20000555A2 (ru) |
HU (1) | HUP0100647A3 (ru) |
NZ (1) | NZ505695A (ru) |
PL (1) | PL341975A1 (ru) |
SK (1) | SK12772000A3 (ru) |
TR (1) | TR200002469T2 (ru) |
WO (1) | WO1999043677A1 (ru) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9821179D0 (en) * | 1998-09-30 | 1998-11-25 | Merck Sharp & Dohme | Therapeutic use |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PH21834A (en) * | 1982-01-18 | 1988-03-17 | Lepetit Spa | New 6-substituted-s-triazolo(3,4-a)phthalazine derivatives |
AU724076B2 (en) * | 1996-07-25 | 2000-09-14 | Merck Sharp & Dohme Limited | Substituted triazolo pyridazine derivatives as inverse agonists of the GABAAalpha5 receptor subtype |
AU732455C (en) * | 1997-05-08 | 2002-09-05 | Merck Sharp & Dohme Limited | Substituted 1,2,4-triazolo{3,4-a}phthalazine derivatives as gaba alpha 5 ligands |
-
1999
- 1999-02-17 HU HU0100647A patent/HUP0100647A3/hu unknown
- 1999-02-17 NZ NZ505695A patent/NZ505695A/en unknown
- 1999-02-17 WO PCT/GB1999/000485 patent/WO1999043677A1/en not_active Application Discontinuation
- 1999-02-17 SK SK1277-2000A patent/SK12772000A3/sk unknown
- 1999-02-17 PL PL99341975A patent/PL341975A1/xx not_active Application Discontinuation
- 1999-02-17 AU AU25368/99A patent/AU746719B2/en not_active Ceased
- 1999-02-17 EP EP99905069A patent/EP1070066A1/en not_active Withdrawn
- 1999-02-17 JP JP2000533432A patent/JP2002504554A/ja not_active Withdrawn
- 1999-02-17 CN CN99803190A patent/CN1291194A/zh active Pending
- 1999-02-17 CA CA002317416A patent/CA2317416A1/en not_active Abandoned
- 1999-02-17 EA EA200000878A patent/EA002824B1/ru not_active IP Right Cessation
- 1999-02-17 TR TR2000/02469T patent/TR200002469T2/xx unknown
-
2000
- 2000-08-22 BG BG104705A patent/BG104705A/bg unknown
- 2000-08-25 HR HR20000555A patent/HRP20000555A2/hr not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
HUP0100647A2 (hu) | 2001-09-28 |
EA002824B1 (ru) | 2002-10-31 |
EP1070066A1 (en) | 2001-01-24 |
AU2536899A (en) | 1999-09-15 |
HUP0100647A3 (en) | 2003-03-28 |
NZ505695A (en) | 2002-03-01 |
HRP20000555A2 (en) | 2001-08-31 |
CA2317416A1 (en) | 1999-09-02 |
PL341975A1 (en) | 2001-05-07 |
SK12772000A3 (sk) | 2001-03-12 |
AU746719B2 (en) | 2002-05-02 |
BG104705A (bg) | 2001-04-30 |
CN1291194A (zh) | 2001-04-11 |
TR200002469T2 (tr) | 2000-12-21 |
WO1999043677A1 (en) | 1999-09-02 |
JP2002504554A (ja) | 2002-02-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |