BG104705A - Заместен 1,2,4-триазоло/3,4-а/пиридазин - Google Patents
Заместен 1,2,4-триазоло/3,4-а/пиридазин Download PDFInfo
- Publication number
- BG104705A BG104705A BG104705A BG10470500A BG104705A BG 104705 A BG104705 A BG 104705A BG 104705 A BG104705 A BG 104705A BG 10470500 A BG10470500 A BG 10470500A BG 104705 A BG104705 A BG 104705A
- Authority
- BG
- Bulgaria
- Prior art keywords
- compound
- triazolo
- phthalazine
- methylisoxazol
- methyloxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9803992.8A GB9803992D0 (en) | 1998-02-25 | 1998-02-25 | Therapeutic agents |
| PCT/GB1998/001307 WO1998050385A1 (en) | 1997-05-08 | 1998-05-06 | SUBSTITUTED 1,2,4-TRIAZOLO[3,4-a]PHTHALAZINE DERIVATIVES AS GABA ALPHA 5 LIGANDS |
| GBGB9824896.6A GB9824896D0 (en) | 1998-11-12 | 1998-11-12 | Therapeutic compound |
| PCT/GB1999/000485 WO1999043677A1 (en) | 1998-02-25 | 1999-02-17 | SUBSTITUTED 1,2,4-TRIAZOLO[3,4-a]PYRIDAZINE |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG104705A true BG104705A (bg) | 2001-04-30 |
Family
ID=27269184
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG104705A BG104705A (bg) | 1998-02-25 | 2000-08-22 | Заместен 1,2,4-триазоло/3,4-а/пиридазин |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP1070066A1 (ru) |
| JP (1) | JP2002504554A (ru) |
| CN (1) | CN1291194A (ru) |
| AU (1) | AU746719B2 (ru) |
| BG (1) | BG104705A (ru) |
| CA (1) | CA2317416A1 (ru) |
| EA (1) | EA002824B1 (ru) |
| HR (1) | HRP20000555A2 (ru) |
| HU (1) | HUP0100647A3 (ru) |
| NZ (1) | NZ505695A (ru) |
| PL (1) | PL341975A1 (ru) |
| SK (1) | SK12772000A3 (ru) |
| TR (1) | TR200002469T2 (ru) |
| WO (1) | WO1999043677A1 (ru) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9821179D0 (en) * | 1998-09-30 | 1998-11-25 | Merck Sharp & Dohme | Therapeutic use |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PH21834A (en) * | 1982-01-18 | 1988-03-17 | Lepetit Spa | New 6-substituted-s-triazolo(3,4-a)phthalazine derivatives |
| WO1998004560A1 (en) * | 1996-07-25 | 1998-02-05 | Merck Sharp & Dohme Limited | SUBSTITUTED TRIAZOLO PYRIDAZINE DERIVATIVES AS INVERSE AGONISTS OF THE GABAAα5 RECEPTOR SUBTYPE |
| CA2288789C (en) * | 1997-05-08 | 2009-07-21 | Merck Sharp & Dohme Limited | Substituted 1,2,4-triazolo[3,4-a]phthalazine derivatives as gaba alpha 5 ligands |
-
1999
- 1999-02-17 SK SK1277-2000A patent/SK12772000A3/sk unknown
- 1999-02-17 EP EP99905069A patent/EP1070066A1/en not_active Withdrawn
- 1999-02-17 CN CN99803190A patent/CN1291194A/zh active Pending
- 1999-02-17 EA EA200000878A patent/EA002824B1/ru not_active IP Right Cessation
- 1999-02-17 PL PL99341975A patent/PL341975A1/xx not_active Application Discontinuation
- 1999-02-17 WO PCT/GB1999/000485 patent/WO1999043677A1/en not_active Application Discontinuation
- 1999-02-17 AU AU25368/99A patent/AU746719B2/en not_active Ceased
- 1999-02-17 TR TR2000/02469T patent/TR200002469T2/xx unknown
- 1999-02-17 JP JP2000533432A patent/JP2002504554A/ja not_active Withdrawn
- 1999-02-17 HU HU0100647A patent/HUP0100647A3/hu unknown
- 1999-02-17 NZ NZ505695A patent/NZ505695A/en unknown
- 1999-02-17 CA CA002317416A patent/CA2317416A1/en not_active Abandoned
-
2000
- 2000-08-22 BG BG104705A patent/BG104705A/bg unknown
- 2000-08-25 HR HR20000555A patent/HRP20000555A2/hr not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO1999043677A1 (en) | 1999-09-02 |
| CA2317416A1 (en) | 1999-09-02 |
| HUP0100647A3 (en) | 2003-03-28 |
| CN1291194A (zh) | 2001-04-11 |
| JP2002504554A (ja) | 2002-02-12 |
| AU746719B2 (en) | 2002-05-02 |
| HRP20000555A2 (en) | 2001-08-31 |
| EA200000878A1 (ru) | 2001-02-26 |
| TR200002469T2 (tr) | 2000-12-21 |
| NZ505695A (en) | 2002-03-01 |
| EA002824B1 (ru) | 2002-10-31 |
| HUP0100647A2 (hu) | 2001-09-28 |
| SK12772000A3 (sk) | 2001-03-12 |
| AU2536899A (en) | 1999-09-15 |
| EP1070066A1 (en) | 2001-01-24 |
| PL341975A1 (en) | 2001-05-07 |
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