EA020910B1 - Производные n1-замещенного 5-фтор-2-оксопиримидинон-1(2h)-карбоксамида и их применение в качестве фунгицидов - Google Patents

Производные n1-замещенного 5-фтор-2-оксопиримидинон-1(2h)-карбоксамида и их применение в качестве фунгицидов Download PDF

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Publication number
EA020910B1
EA020910B1 EA201270256A EA201270256A EA020910B1 EA 020910 B1 EA020910 B1 EA 020910B1 EA 201270256 A EA201270256 A EA 201270256A EA 201270256 A EA201270256 A EA 201270256A EA 020910 B1 EA020910 B1 EA 020910B1
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EA
Eurasian Patent Office
Prior art keywords
compounds
herbicides
insecticides
alkyl
plant
Prior art date
Application number
EA201270256A
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English (en)
Russian (ru)
Other versions
EA201270256A1 (ru
Inventor
Тимоти Бебель
Кристи Брайан
Бет Лорсбах
Тимоти Мартин
В. Оуэн
Марк Побанс
Скотт Торнберг
Джеффри Вебстер
Чэнлинь Яо
Original Assignee
ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA020910(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи filed Critical ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи
Publication of EA201270256A1 publication Critical patent/EA201270256A1/ru
Publication of EA020910B1 publication Critical patent/EA020910B1/ru

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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EA201270256A 2009-08-07 2010-08-05 Производные n1-замещенного 5-фтор-2-оксопиримидинон-1(2h)-карбоксамида и их применение в качестве фунгицидов EA020910B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23224509P 2009-08-07 2009-08-07
PCT/US2010/044588 WO2011017545A1 (en) 2009-08-07 2010-08-05 N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives

Publications (2)

Publication Number Publication Date
EA201270256A1 EA201270256A1 (ru) 2012-07-30
EA020910B1 true EA020910B1 (ru) 2015-02-27

Family

ID=43535294

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201270256A EA020910B1 (ru) 2009-08-07 2010-08-05 Производные n1-замещенного 5-фтор-2-оксопиримидинон-1(2h)-карбоксамида и их применение в качестве фунгицидов

Country Status (26)

Country Link
US (2) US8552020B2 (enExample)
EP (1) EP2461686B1 (enExample)
JP (1) JP5735510B2 (enExample)
KR (1) KR101792284B1 (enExample)
CN (1) CN102497781B (enExample)
BR (1) BR112012002757B1 (enExample)
CA (1) CA2769656C (enExample)
CL (1) CL2012000312A1 (enExample)
CO (1) CO6491115A2 (enExample)
CR (1) CR20120032A (enExample)
DK (1) DK2461686T3 (enExample)
EA (1) EA020910B1 (enExample)
EC (1) ECSP12011652A (enExample)
ES (1) ES2552097T3 (enExample)
HU (1) HUE027390T2 (enExample)
IL (1) IL217950A (enExample)
IN (1) IN2012DN00369A (enExample)
MX (1) MX2012001617A (enExample)
NI (1) NI201200021A (enExample)
NZ (1) NZ597483A (enExample)
PE (1) PE20120692A1 (enExample)
PL (1) PL2461686T3 (enExample)
PT (1) PT2461686E (enExample)
UA (1) UA107671C2 (enExample)
WO (1) WO2011017545A1 (enExample)
ZA (1) ZA201200813B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2656101C2 (ru) * 2012-12-28 2018-05-31 Адама Мактешим Лтд. Производные 1-(замещенный бензоил)-5-фтор-4-имино-3-метил-3,4-дигидропиримидин-2(1h)-она

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
US8674109B2 (en) 2009-08-07 2014-03-18 Dow Agrosciences, Llc. Pesticidal compositions
AU2010279411B2 (en) * 2009-08-07 2014-10-23 Adama Makhteshim Ltd. N1-sulfonyl-5-fluoropyrimidinone derivatives
HUE047711T2 (hu) 2012-12-28 2020-05-28 Adama Makhteshim Ltd N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok
RU2015131149A (ru) * 2012-12-28 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные
CA2894553C (en) 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
EA030030B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
EP3097096A4 (en) 2013-12-31 2017-10-11 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
CR20210270A (es) 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
TWI808347B (zh) 2019-09-23 2023-07-11 以色列商亞當馬赫特希姆有限公司 用於製備5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2(1h)-酮及該化合物的衍生物之方法
BR112022011245A2 (pt) * 2019-12-10 2022-09-06 Syngenta Crop Protection Ag Métodos de controle ou prevenção de infestação de plantas de amendoim por microrganismos fitopatogênicos
MX2022011088A (es) 2020-03-09 2022-09-29 Adama Makhteshim Ltd Procedimiento para preparar 5-fluoro-4-imino-3-metil-1-(tolueno-4- sulfonil)-3,4-dihidro-1h-pirimidin-2-ona.

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Publication number Priority date Publication date Assignee Title
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US6066638A (en) * 1995-07-05 2000-05-23 E. I. Du Pont De Nemours And Company Fungicidal pyrimidinones
WO2010047866A2 (en) * 2008-08-01 2010-04-29 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide

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US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enExample) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
JPS60123486A (ja) 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンsおよびその製法
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ES2057172T3 (es) 1988-03-09 1994-10-16 Ciba Geigy Ag Agente para la proteccion de plantas contra enfermedades.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ[5,4−d]ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
IL125589A0 (en) 1996-03-11 1999-03-12 Novartis Ag Pyrimidin-4-one derivatives as pesticides
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
JPWO2005095419A1 (ja) * 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
US20080004253A1 (en) * 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
AR070228A1 (es) 2008-01-22 2010-03-25 Dow Agrosciences Llc Derivados de 5-fluoro pirimidina
ME02254B (me) * 2009-01-23 2015-12-31 Euro Celtique Sa Derivati hidroksamske kiseline
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
AU2010279411B2 (en) * 2009-08-07 2014-10-23 Adama Makhteshim Ltd. N1-sulfonyl-5-fluoropyrimidinone derivatives

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US6066638A (en) * 1995-07-05 2000-05-23 E. I. Du Pont De Nemours And Company Fungicidal pyrimidinones
WO2010047866A2 (en) * 2008-08-01 2010-04-29 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2656101C2 (ru) * 2012-12-28 2018-05-31 Адама Мактешим Лтд. Производные 1-(замещенный бензоил)-5-фтор-4-имино-3-метил-3,4-дигидропиримидин-2(1h)-она

Also Published As

Publication number Publication date
CA2769656C (en) 2018-05-15
PE20120692A1 (es) 2012-06-08
KR101792284B1 (ko) 2017-10-31
CN102497781A (zh) 2012-06-13
CR20120032A (es) 2012-03-22
US9000002B2 (en) 2015-04-07
PT2461686E (pt) 2015-11-18
DK2461686T3 (en) 2016-01-18
WO2011017545A1 (en) 2011-02-10
JP5735510B2 (ja) 2015-06-17
ES2552097T3 (es) 2015-11-25
EP2461686A4 (en) 2013-02-13
EP2461686A1 (en) 2012-06-13
ECSP12011652A (es) 2012-03-30
IN2012DN00369A (enExample) 2015-08-21
CA2769656A1 (en) 2011-02-10
US8552020B2 (en) 2013-10-08
MX2012001617A (es) 2012-04-11
IL217950A0 (en) 2012-03-29
BR112012002757B1 (pt) 2020-10-06
PL2461686T3 (pl) 2016-04-29
UA107671C2 (en) 2015-02-10
EA201270256A1 (ru) 2012-07-30
US20110034492A1 (en) 2011-02-10
KR20120052281A (ko) 2012-05-23
US20140011824A1 (en) 2014-01-09
NZ597483A (en) 2014-02-28
CN102497781B (zh) 2014-12-10
NI201200021A (es) 2012-05-22
AU2010279409A1 (en) 2012-02-02
JP2013501727A (ja) 2013-01-17
CL2012000312A1 (es) 2012-10-05
ZA201200813B (en) 2013-05-29
CO6491115A2 (es) 2012-07-31
IL217950A (en) 2015-04-30
BR112012002757A2 (pt) 2019-12-17
HK1171915A1 (en) 2013-04-12
HUE027390T2 (en) 2016-10-28
EP2461686B1 (en) 2015-10-07

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PC4A Registration of transfer of a eurasian patent by assignment
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

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