PT2461686E - Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1 - Google Patents

Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1 Download PDF

Info

Publication number
PT2461686E
PT2461686E PT108071754T PT10807175T PT2461686E PT 2461686 E PT2461686 E PT 2461686E PT 108071754 T PT108071754 T PT 108071754T PT 10807175 T PT10807175 T PT 10807175T PT 2461686 E PT2461686 E PT 2461686E
Authority
PT
Portugal
Prior art keywords
oxopyrimidinone
fluoro
substituted
carboxamide derivatives
carboxamide
Prior art date
Application number
PT108071754T
Other languages
English (en)
Portuguese (pt)
Inventor
Chenglin Yao
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT2461686(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of PT2461686E publication Critical patent/PT2461686E/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT108071754T 2009-08-07 2010-08-05 Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1 PT2461686E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23224509P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
PT2461686E true PT2461686E (pt) 2015-11-18

Family

ID=43535294

Family Applications (1)

Application Number Title Priority Date Filing Date
PT108071754T PT2461686E (pt) 2009-08-07 2010-08-05 Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1

Country Status (26)

Country Link
US (2) US8552020B2 (enExample)
EP (1) EP2461686B1 (enExample)
JP (1) JP5735510B2 (enExample)
KR (1) KR101792284B1 (enExample)
CN (1) CN102497781B (enExample)
BR (1) BR112012002757B1 (enExample)
CA (1) CA2769656C (enExample)
CL (1) CL2012000312A1 (enExample)
CO (1) CO6491115A2 (enExample)
CR (1) CR20120032A (enExample)
DK (1) DK2461686T3 (enExample)
EA (1) EA020910B1 (enExample)
EC (1) ECSP12011652A (enExample)
ES (1) ES2552097T3 (enExample)
HU (1) HUE027390T2 (enExample)
IL (1) IL217950A (enExample)
IN (1) IN2012DN00369A (enExample)
MX (1) MX2012001617A (enExample)
NI (1) NI201200021A (enExample)
NZ (1) NZ597483A (enExample)
PE (1) PE20120692A1 (enExample)
PL (1) PL2461686T3 (enExample)
PT (1) PT2461686E (enExample)
UA (1) UA107671C2 (enExample)
WO (1) WO2011017545A1 (enExample)
ZA (1) ZA201200813B (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
JP5784603B2 (ja) * 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー N1−スルホニル−5−フルオロピリミジノン誘導体
AU2010279377B2 (en) 2009-08-07 2014-07-03 Dow Agrosciences Llc Pesticidal compositions
WO2014105821A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
CN104902757B (zh) * 2012-12-28 2019-01-08 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物
JP6258969B2 (ja) 2012-12-28 2018-01-10 アダマ・マクテシム・リミテッド N−(置換)−5−フルオロ−4−イミノ−3−メチル−2−オキソ−3,4−ジヒドロピリミジン−1(2h)−カルボキサミド誘導体
CN112094262A (zh) 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
CR20160344A (es) 2013-12-31 2016-12-19 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas para el control fúngico en cereales
UA129860C2 (uk) 2013-12-31 2025-08-27 Адама Махтешім Лтд. 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання
IL271950B2 (en) 2017-07-17 2024-06-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
CA3118729A1 (en) 2018-11-05 2020-05-14 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
US12466796B2 (en) 2019-09-23 2025-11-11 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound
WO2021115926A1 (en) * 2019-12-10 2021-06-17 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of peanut plants by phytopathogenic microorganisms

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enExample) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
JPS60123486A (ja) * 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンsおよびその製法
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (de) 1988-03-09 1994-08-15 Ciba Geigy Ag Mittel zum schutz von pflanzen gegen krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ[5,4−d]ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
EP0836602B1 (en) * 1995-07-05 2002-01-30 E.I. Du Pont De Nemours And Company Fungicidal pyrimidinones
DE69712331T2 (de) 1996-03-11 2002-11-28 Syngenta Participations Ag, Basel Pyrimidin-4-on derivate als pestizidesmittel
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
US20080269238A1 (en) * 2004-04-01 2008-10-30 Takeda Pharmaceutical Company Limited Thiazolopyrimidine Derivative
US20080004253A1 (en) * 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
EP2562166B1 (en) * 2008-01-22 2015-08-19 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
EP2317851B1 (en) * 2008-08-01 2014-01-15 Dow AgroSciences LLC Use of 5-fluorocytosine as a fungicide
PL2389375T3 (pl) * 2009-01-23 2015-11-30 Euro Celtique Sa Pochodne kwasu hydroksamowego
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
JP5784603B2 (ja) * 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー N1−スルホニル−5−フルオロピリミジノン誘導体

Also Published As

Publication number Publication date
US20110034492A1 (en) 2011-02-10
IL217950A0 (en) 2012-03-29
HUE027390T2 (en) 2016-10-28
BR112012002757B1 (pt) 2020-10-06
ES2552097T3 (es) 2015-11-25
EP2461686A4 (en) 2013-02-13
UA107671C2 (en) 2015-02-10
HK1171915A1 (en) 2013-04-12
PL2461686T3 (pl) 2016-04-29
CN102497781B (zh) 2014-12-10
CN102497781A (zh) 2012-06-13
AU2010279409A1 (en) 2012-02-02
EA020910B1 (ru) 2015-02-27
WO2011017545A1 (en) 2011-02-10
IL217950A (en) 2015-04-30
CO6491115A2 (es) 2012-07-31
PE20120692A1 (es) 2012-06-08
NI201200021A (es) 2012-05-22
IN2012DN00369A (enExample) 2015-08-21
JP2013501727A (ja) 2013-01-17
EP2461686B1 (en) 2015-10-07
CR20120032A (es) 2012-03-22
US8552020B2 (en) 2013-10-08
NZ597483A (en) 2014-02-28
KR101792284B1 (ko) 2017-10-31
EP2461686A1 (en) 2012-06-13
US20140011824A1 (en) 2014-01-09
ZA201200813B (en) 2013-05-29
BR112012002757A2 (pt) 2019-12-17
CL2012000312A1 (es) 2012-10-05
DK2461686T3 (en) 2016-01-18
EA201270256A1 (ru) 2012-07-30
KR20120052281A (ko) 2012-05-23
ECSP12011652A (es) 2012-03-30
CA2769656A1 (en) 2011-02-10
CA2769656C (en) 2018-05-15
MX2012001617A (es) 2012-04-11
US9000002B2 (en) 2015-04-07
JP5735510B2 (ja) 2015-06-17

Similar Documents

Publication Publication Date Title
IL217950A0 (en) N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
IL219087A0 (en) Benzimidazole-imidazole derivatives
IL217956A0 (en) N1-sulfonyl-5-fluoropyrimidinone derivatives
IL217953A0 (en) 5-fluoropyrimidinone derivatives
IL216007A0 (en) Isoxazole-pyridine derivatives
IL215109A0 (en) Isoxazole-pyridazine derivatives
ZA201305992B (en) 5-fluoro-2-oxopyrimidine-1(2h)-carboxylate derivatives
IL214941A0 (en) Isoxazole-pyrazole derivatives
IL217952A0 (en) N1-acyl-5-fluoropyrimidinone derivatives
IL213927A0 (en) Deoxyactagardine derivatives
ZA201105780B (en) Pyridazinone derivatives
IL216761A0 (en) Pyrazinooxazepine derivatives
ZA201105781B (en) Pyridazinone derivatives
ZA201104279B (en) Tetrahydronaphthalen-2-ol derivatives
GB0912499D0 (en) Indopyl-pyridone derivatives