EA012433B1 - Многовалентные vla-4 антагонисты, содержащие полимерные фрагменты - Google Patents

Многовалентные vla-4 антагонисты, содержащие полимерные фрагменты Download PDF

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Publication number
EA012433B1
EA012433B1 EA200700212A EA200700212A EA012433B1 EA 012433 B1 EA012433 B1 EA 012433B1 EA 200700212 A EA200700212 A EA 200700212A EA 200700212 A EA200700212 A EA 200700212A EA 012433 B1 EA012433 B1 EA 012433B1
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EA
Eurasian Patent Office
Prior art keywords
substituted
group
alkyl
alkylene
aryl
Prior art date
Application number
EA200700212A
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English (en)
Russian (ru)
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EA200700212A1 (ru
Inventor
Андрей В. Конради
Майкл А. Плисс
Кристофер М. Семко
Теодор Йеднок
Дженифер Л. Смит
Original Assignee
Элан Фармасьютикалз, Инк.
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Application filed by Элан Фармасьютикалз, Инк. filed Critical Элан Фармасьютикалз, Инк.
Publication of EA200700212A1 publication Critical patent/EA200700212A1/ru
Publication of EA012433B1 publication Critical patent/EA012433B1/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
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EA200700212A 2004-07-08 2005-07-08 Многовалентные vla-4 антагонисты, содержащие полимерные фрагменты EA012433B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US58697504P 2004-07-08 2004-07-08
PCT/US2005/024369 WO2006010054A2 (en) 2004-07-08 2005-07-08 Multivalent vla-4 antagonists comprising polyethylene glycol moieties

Publications (2)

Publication Number Publication Date
EA200700212A1 EA200700212A1 (ru) 2007-08-31
EA012433B1 true EA012433B1 (ru) 2009-10-30

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US (4) US7794700B2 (US07794700-20100914-C00077.png)
EP (4) EP2258400A3 (US07794700-20100914-C00077.png)
JP (1) JP2008505927A (US07794700-20100914-C00077.png)
KR (1) KR101273614B1 (US07794700-20100914-C00077.png)
CN (1) CN101035563B (US07794700-20100914-C00077.png)
AR (1) AR050425A1 (US07794700-20100914-C00077.png)
AU (1) AU2005265316B2 (US07794700-20100914-C00077.png)
BR (1) BRPI0513143A (US07794700-20100914-C00077.png)
CA (1) CA2573245C (US07794700-20100914-C00077.png)
EA (1) EA012433B1 (US07794700-20100914-C00077.png)
EC (1) ECSP077231A (US07794700-20100914-C00077.png)
HK (1) HK1111674A1 (US07794700-20100914-C00077.png)
IL (1) IL180558A0 (US07794700-20100914-C00077.png)
MA (1) MA28786B1 (US07794700-20100914-C00077.png)
MX (1) MX2007000228A (US07794700-20100914-C00077.png)
NO (1) NO20070216L (US07794700-20100914-C00077.png)
NZ (1) NZ588839A (US07794700-20100914-C00077.png)
TW (1) TWI418346B (US07794700-20100914-C00077.png)
WO (1) WO2006010054A2 (US07794700-20100914-C00077.png)
ZA (1) ZA200700238B (US07794700-20100914-C00077.png)

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