DK562888A - Aminomethyl-oxooxazolidinyl-cycloalkylbenzenderivater, fremstilling deraf, praeparater indeholdende disse og deres anvendelse som antibakterielle midler - Google Patents
Aminomethyl-oxooxazolidinyl-cycloalkylbenzenderivater, fremstilling deraf, praeparater indeholdende disse og deres anvendelse som antibakterielle midlerInfo
- Publication number
- DK562888A DK562888A DK562888A DK562888A DK562888A DK 562888 A DK562888 A DK 562888A DK 562888 A DK562888 A DK 562888A DK 562888 A DK562888 A DK 562888A DK 562888 A DK562888 A DK 562888A
- Authority
- DK
- Denmark
- Prior art keywords
- oxooxazolidinyl
- antibacterials
- aminomethyl
- preparing
- preparations containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/106,358 US4801600A (en) | 1987-10-09 | 1987-10-09 | Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents |
Publications (2)
Publication Number | Publication Date |
---|---|
DK562888D0 DK562888D0 (da) | 1988-10-07 |
DK562888A true DK562888A (da) | 1989-04-10 |
Family
ID=22310972
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK562888A DK562888A (da) | 1987-10-09 | 1988-10-07 | Aminomethyl-oxooxazolidinyl-cycloalkylbenzenderivater, fremstilling deraf, praeparater indeholdende disse og deres anvendelse som antibakterielle midler |
Country Status (16)
Country | Link |
---|---|
US (1) | US4801600A (fi) |
EP (1) | EP0311090A1 (fi) |
JP (1) | JPH01132569A (fi) |
KR (1) | KR890006632A (fi) |
AU (1) | AU613669B2 (fi) |
CA (1) | CA1322001C (fi) |
DK (1) | DK562888A (fi) |
FI (1) | FI884610A (fi) |
HU (1) | HU202216B (fi) |
IL (1) | IL87972A (fi) |
MY (1) | MY103618A (fi) |
NO (1) | NO172890C (fi) |
NZ (1) | NZ226493A (fi) |
PT (1) | PT88713B (fi) |
SU (1) | SU1616518A3 (fi) |
ZA (1) | ZA887550B (fi) |
Families Citing this family (49)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4985429A (en) * | 1987-10-09 | 1991-01-15 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents |
US4942183A (en) * | 1987-10-16 | 1990-07-17 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents |
US4977173A (en) * | 1987-10-21 | 1990-12-11 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl ethenylbenzene derivatives useful as antibacterial agents |
US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
ATE201870T1 (de) * | 1988-09-15 | 2001-06-15 | Upjohn Co | 3-(stickstoff substituierte)phenyl-5-beta- amidomethyloxazoliden-2-one |
US5164510A (en) * | 1988-09-15 | 1992-11-17 | The Upjohn Company | 5'Indolinyl-5β-amidomethyloxazolidin-2-ones |
US5225565A (en) * | 1988-09-15 | 1993-07-06 | The Upjohn Company | Antibacterial 3-(fused-ring substituted)phenyl-5β-amidomethyloxazolidin-2-ones |
US5182403A (en) * | 1988-09-15 | 1993-01-26 | The Upjohn Company | Substituted 3(5'indazolyl) oxazolidin-2-ones |
US5231188A (en) * | 1989-11-17 | 1993-07-27 | The Upjohn Company | Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents |
SI9111010B (sl) * | 1990-06-07 | 2005-02-28 | Astrazeneca Ab | 3,5-disubstituirani indolni derivati kot "5-HT1-podobni" receptorski agonisti |
JP2669579B2 (ja) * | 1991-10-23 | 1997-10-29 | エーザイ株式会社 | オキサゾリドン誘導体 |
DE69216251T2 (de) * | 1991-11-01 | 1997-05-15 | Pharmacia & Upjohn Co., Kalamazoo, Mich. | Substituierte aryl- und heteroaryl-phenyloxazolidinone |
SK283420B6 (sk) * | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
NZ257031A (en) * | 1992-12-08 | 1996-07-26 | Upjohn Co | Tropone substituted phenyloxazolidinone derivatives and anti-bacterial medicaments thereof |
US5688792A (en) * | 1994-08-16 | 1997-11-18 | Pharmacia & Upjohn Company | Substituted oxazine and thiazine oxazolidinone antimicrobials |
KR100312903B1 (ko) * | 1993-11-22 | 2002-02-28 | 로렌스 티. 마이젠헬더 | 치환된-하이드록시아세틸피페라진페닐옥사졸리디논의에스테르 |
DE4425612A1 (de) * | 1994-07-20 | 1996-04-04 | Bayer Ag | 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone |
DE4425609A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | Benzofuranyl- und Benzothienyloxazolidinone |
DE4425613A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | 5-gliedrige Heteroaryl-oxazolidinone |
DE19514313A1 (de) | 1994-08-03 | 1996-02-08 | Bayer Ag | Benzoxazolyl- und Benzothiazolyloxazolidinone |
KR100392216B1 (ko) * | 1994-11-15 | 2003-10-17 | 파마시아 앤드 업존 캄파니 | 이환상옥사진및티아진옥사졸리디논항세균물질 |
RU2154645C2 (ru) * | 1995-02-03 | 2000-08-20 | Фармация Энд Апджон Компани | Фенилоксазолидиноны, замещенные в кольце гетероароматическими кольцами, в качестве антимикробных агентов |
HRP960159A2 (en) * | 1995-04-21 | 1997-08-31 | Bayer Ag | Benzocyclopentane oxazolidinones containing heteroatoms |
ATE204874T1 (de) * | 1995-05-11 | 2001-09-15 | Upjohn Co | Spirocyclische und bicyclische diazinyl- und carbazinyloxazolidinone |
MX9703040A (es) * | 1995-09-12 | 1997-07-31 | Upjohn Co | Antimicrobianos de feniloxazolidinona. |
DE19601265A1 (de) * | 1996-01-16 | 1997-07-17 | Bayer Ag | 2-Oxo- und 2-Thio-1,2-dihydrochinolinyl-oxazolidinone |
DE19601264A1 (de) * | 1996-01-16 | 1997-07-17 | Bayer Ag | Pyrido-annellierte Thienyl- und Furanyl-Oxazolidinone |
DE19601627A1 (de) * | 1996-01-18 | 1997-07-24 | Bayer Ag | Heteroatomhaltige Cyclopentanopyridyl-Oxazolidinone |
DE19604223A1 (de) * | 1996-02-06 | 1997-08-07 | Bayer Ag | Neue substituierte Oxazolidinone |
HRP970049A2 (en) * | 1996-02-06 | 1998-04-30 | Bayer Ag | New heteroaryl oxazolidinones |
MY116093A (en) * | 1996-02-26 | 2003-11-28 | Upjohn Co | Azolyl piperazinyl phenyl oxazolidinone antimicrobials |
KR20010031953A (ko) * | 1997-11-12 | 2001-04-16 | 로렌스 티. 마이젠헬더 | 옥사졸리디논 유도체 및 제약 조성물 |
DE19802235A1 (de) * | 1998-01-22 | 1999-07-29 | Bayer Ag | Mit tricyclischen Indolen substituierte Oxazolidinone |
BR9907183A (pt) * | 1998-01-23 | 2003-06-10 | Versicor Inc | Colet neas combinatórias de oxazolidinona, composições e processos de preparação |
JP2002535680A (ja) | 1999-01-27 | 2002-10-22 | ファルマシア・アンド・アップジョン・カンパニー | 延長因子p活性モジュレーターのアッセイ方法 |
DK1181288T3 (da) * | 1999-05-27 | 2003-11-17 | Upjohn Co | Bicycliske oxazolidinoner som antibakterielle midler |
US6444813B2 (en) * | 2000-02-02 | 2002-09-03 | Pharmacia & Upjohn Company | Linezolid-crystal form II |
WO2002006278A1 (en) | 2000-07-17 | 2002-01-24 | Ranbaxy Laboratories Limited | Oxazolidinone derivatives as antimicrobials |
PE20020689A1 (es) * | 2000-11-17 | 2002-08-03 | Upjohn Co | Oxazolidinonas con un heterociclo de 6 o 7 miembros unidos con enlace anular al benceno |
EP1349853B1 (en) | 2000-12-21 | 2006-03-08 | Pharmacia & Upjohn Company LLC | Antimicrobial quinolone derivatives and use of the same to treat bacterial infections |
EP1409464A4 (en) * | 2001-07-16 | 2005-11-02 | Ranbaxy Lab Ltd | OXAZOLIDINONE DERIVATIVES AS POTENTIAL ANTIMICROBIALS |
US6956040B2 (en) | 2001-07-16 | 2005-10-18 | Ranbaxy Laboratories Limited | Oxazolidinone piperazinyl derivatives as potential antimicrobials |
CN1662240A (zh) * | 2002-05-15 | 2005-08-31 | 兰贝克赛实验室有限公司 | 苯基噁唑烷酮衍生物 |
EP1542696A4 (en) * | 2002-07-29 | 2006-08-02 | Ranbaxy Lab Ltd | OXAZOLIDINONE DERIVATIVES AS ANTIMICROBIAL AGENTS |
WO2004069244A1 (en) * | 2003-02-07 | 2004-08-19 | Warner-Lambert Company Llc | Oxazolidinone derivatives n-substituted by a bicyclic ring, for use as antibacterial agents |
EP1620433A1 (en) * | 2003-04-07 | 2006-02-01 | Ranbaxy Laboratories, Ltd. | Oxazolidinone derivatives as antimicrobials |
CA2602073A1 (en) * | 2005-02-24 | 2006-08-31 | Teva Pharmaceutical Industries Ltd. | Processes for the preparation of linezolid intermediate |
WO2008143649A2 (en) * | 2006-12-04 | 2008-11-27 | Dr. Reddy's Laboratories Limited | Novel oxazolidinone compounds as antiinfective agents |
CA2712613C (en) * | 2008-03-26 | 2017-02-28 | Global Alliance For Tb Drug Development | Bicyclic nitroimidazoles covalently linked to substituted phenyl oxazolidinones |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US29607A (en) * | 1860-08-14 | Portable scaffold | ||
GB1222708A (en) * | 1968-10-22 | 1971-02-17 | Delalande Sa | Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation |
USRE29607E (en) | 1969-03-18 | 1978-04-11 | Delalande S. A. | Derivatives of 5-hydroxymethyl-3-substituted-2-oxazolidinones, process of preparation thereof and therapeutic application |
LU80081A1 (fr) * | 1977-08-26 | 1979-05-15 | Delalande Sa | Nouvelles hydroxymethyl-5 oxazolidinones-2,leur procede de preparation et leur application therapeutique |
US4128654A (en) * | 1978-02-10 | 1978-12-05 | E. I. Du Pont De Nemours And Company | 5-Halomethyl-3-phenyl-2-oxazolidinones |
CA1171865A (en) * | 1980-06-04 | 1984-07-31 | Alain Lacour | N-aryl azolone derivatives, the process for preparing the same and their application in therapeutics |
US4340606A (en) * | 1980-10-23 | 1982-07-20 | E. I. Du Pont De Nemours And Company | 3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents |
FR2500450A1 (fr) * | 1981-02-25 | 1982-08-27 | Delalande Sa | Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique |
US4461773A (en) * | 1982-09-15 | 1984-07-24 | E. I. Dupont De Nemours And Company | P-Oxooxazolidinylbenzene compounds as antibacterial agents |
ES533097A0 (es) * | 1983-06-07 | 1985-08-01 | Du Pont | Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno. |
US4705799A (en) * | 1983-06-07 | 1987-11-10 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents |
CA1260948A (en) * | 1984-12-05 | 1989-09-26 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents |
-
1987
- 1987-10-09 US US07/106,358 patent/US4801600A/en not_active Expired - Lifetime
-
1988
- 1988-10-04 CA CA000579301A patent/CA1322001C/en not_active Expired - Fee Related
- 1988-10-06 SU SU884356653A patent/SU1616518A3/ru active
- 1988-10-06 AU AU23507/88A patent/AU613669B2/en not_active Ceased
- 1988-10-07 FI FI884610A patent/FI884610A/fi not_active Application Discontinuation
- 1988-10-07 HU HU885214A patent/HU202216B/hu not_active IP Right Cessation
- 1988-10-07 JP JP63252207A patent/JPH01132569A/ja active Pending
- 1988-10-07 MY MYPI88001123A patent/MY103618A/en unknown
- 1988-10-07 ZA ZA887550A patent/ZA887550B/xx unknown
- 1988-10-07 PT PT88713A patent/PT88713B/pt not_active IP Right Cessation
- 1988-10-07 NZ NZ226493A patent/NZ226493A/xx unknown
- 1988-10-07 KR KR1019880013071A patent/KR890006632A/ko not_active Application Discontinuation
- 1988-10-07 EP EP88116621A patent/EP0311090A1/en not_active Withdrawn
- 1988-10-07 DK DK562888A patent/DK562888A/da not_active Application Discontinuation
- 1988-10-07 NO NO884467A patent/NO172890C/no unknown
- 1988-10-07 IL IL87972A patent/IL87972A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
MY103618A (en) | 1993-08-28 |
DK562888D0 (da) | 1988-10-07 |
JPH01132569A (ja) | 1989-05-25 |
SU1616518A3 (ru) | 1990-12-23 |
PT88713B (pt) | 1992-12-31 |
ZA887550B (en) | 1990-06-27 |
EP0311090A1 (en) | 1989-04-12 |
IL87972A0 (en) | 1989-03-31 |
NO884467L (no) | 1989-04-10 |
US4801600A (en) | 1989-01-31 |
HU202216B (en) | 1991-02-28 |
NZ226493A (en) | 1990-09-26 |
FI884610A0 (fi) | 1988-10-07 |
NO884467D0 (no) | 1988-10-07 |
FI884610A (fi) | 1989-04-10 |
KR890006632A (ko) | 1989-06-14 |
CA1322001C (en) | 1993-09-07 |
NO172890C (no) | 1993-09-22 |
HUT53359A (en) | 1990-10-28 |
AU2350788A (en) | 1989-04-13 |
IL87972A (en) | 1993-05-13 |
AU613669B2 (en) | 1991-08-08 |
NO172890B (no) | 1993-06-14 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DK562888A (da) | Aminomethyl-oxooxazolidinyl-cycloalkylbenzenderivater, fremstilling deraf, praeparater indeholdende disse og deres anvendelse som antibakterielle midler | |
DK288184A (da) | 13alfa-alkylgonaner, deres fremstilling og farmaceutiske praeparater indeholdende disse | |
DK143588A (da) | Substituerede 9-amino-tetrahydroacridiner, deres fremstilling og anvendelse som laegemidler | |
NO870666L (no) | Substituerte thienoinidasolderivater, fremgangsmaate til deres fremstilling og farmasoeytiske tilberedninger inneholdende disse og deres anvendelse som magesyresekresjonshemmer | |
DK381985D0 (da) | 3-pyridylforbindelser, deres fremstilling og anvendelse som laegemiddel | |
DK81986A (da) | Pyridinylimidazolidinoner, deres fremstilling og anvendelse som herbicider | |
DK209188D0 (da) | Bifunktionelle proteiner, deres fremstilling og anvendelse som laegemiddel | |
DK166583C (da) | 1-pyrimidinyloxy-3-alkylamino-2-propanoler, deres fremstilling og farmaceutiske praeparater indeholdende disse | |
DK660788D0 (da) | 2,2-difluorcyklopropylethanderivater, fremgangsmaade til deres fremstilling og deres anvendelse som skadedyrsbekaempelsesmiddel | |
DK435588D0 (da) | Aralkylaminoalkoxyphenylderivater, fremgangsmaade til deres fremstilling og midler indeholdende disse | |
DK131887A (da) | 1,2,3,4-tetrahydro-3-carbamoyl-2-thioxo/oxo-5-pyrimidencarboxylsyre-derivater og deres anvendelse som laegemidler | |
DK366888A (da) | Castanosperminestre og -glykosider, deres fremstilling og anvendelse som laegemidler | |
DK384088A (da) | Substituerede benzimidazoler, deres fremstilling, praeparater indeholdende disse samt deres anvendelse som laegemidler | |
DK284688D0 (da) | Beta-lactam-forbindelser, deres fremstilling og anvendelse som laegemidler | |
DK548486D0 (da) | L-arylpyrazoler, deres fremstilling og anvendelse som herbicider | |
DK627684D0 (da) | 1,4-naphthoquinolinderivater, deres fremstilling og anvendelse som laegemiddel | |
DK10685A (da) | Sulfonylguanidinderivater, deres fremstilling og anvendelse som herbicider | |
DK501888A (da) | 6-mercaptopurin-derivater, deres fremstilling og anvendelse som laegemidler | |
DK37787D0 (da) | 2,3-dioxabicyclooe3,3,0aaoctan-derivater og deres anvendelse som laegemidler | |
NO903967L (no) | Dihydrocaffeinsyrederivater og farmasoeytiske preparater som inneholder disse. | |
DK223987D0 (da) | Pyridylthioacylanilider, deres fremstilling og anvendelse som herbicider | |
DK276690A (da) | Selenophenderivater, fremgangsmaade til deres fremstilling og terapeutiske praeparater indeholdende disse | |
DK447687A (da) | Urdamycin g og derivater deraf samt deres fremstilling og anvendelse | |
DK134988D0 (da) | Thiazolylderivater, deres fremstilling og anvendelse som herbicider | |
DK448086D0 (da) | Tetrahydroisoindolinoner, deres fremstilling og anvendelse som herbicider |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
AHB | Application shelved due to non-payment |