DK3080100T3 - Hæmmere af lysinspecifik demethylase-1 - Google Patents

Hæmmere af lysinspecifik demethylase-1 Download PDF

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Publication number
DK3080100T3
DK3080100T3 DK14868829.4T DK14868829T DK3080100T3 DK 3080100 T3 DK3080100 T3 DK 3080100T3 DK 14868829 T DK14868829 T DK 14868829T DK 3080100 T3 DK3080100 T3 DK 3080100T3
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lysine
inhibitors
specific demethylase
demethylase
specific
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DK14868829.4T
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Danish (da)
English (en)
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Young K Chen
Toufike Kanouni
Stephen W Kaldor
Jeffrey Alan Stafford
James Marvin Veal
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Celgene Quanticel Res Inc
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    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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    • C07D498/18Bridged systems
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  • Chemical & Material Sciences (AREA)
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  • General Chemical & Material Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Polyamides (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK14868829.4T 2013-12-11 2014-12-10 Hæmmere af lysinspecifik demethylase-1 DK3080100T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361914927P 2013-12-11 2013-12-11
PCT/US2014/069562 WO2015089192A1 (en) 2013-12-11 2014-12-10 Inhibitors of lysine specific demethylase-1

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Publication Number Publication Date
DK3080100T3 true DK3080100T3 (da) 2023-02-06

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US (3) US9944636B2 (enExample)
EP (2) EP4257591A3 (enExample)
JP (1) JP6430512B2 (enExample)
CA (2) CA2933480C (enExample)
DK (1) DK3080100T3 (enExample)
ES (1) ES2935746T3 (enExample)
FI (1) FI3080100T3 (enExample)
HR (1) HRP20230086T1 (enExample)
HU (1) HUE061252T2 (enExample)
LT (1) LT3080100T (enExample)
MX (2) MX376047B (enExample)
PL (1) PL3080100T3 (enExample)
PT (1) PT3080100T (enExample)
RS (1) RS63939B1 (enExample)
SI (1) SI3080100T1 (enExample)
SM (1) SMT202300014T1 (enExample)
WO (1) WO2015089192A1 (enExample)

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JP6430512B2 (ja) 2018-11-28
HRP20230086T1 (hr) 2023-03-31
US10385051B2 (en) 2019-08-20
CA3161836A1 (en) 2015-06-18
EP3080100A1 (en) 2016-10-19
LT3080100T (lt) 2023-02-27
MX2020010496A (es) 2020-10-28
PT3080100T (pt) 2023-01-19
JP2017502940A (ja) 2017-01-26
US20160304516A1 (en) 2016-10-20
US10131664B2 (en) 2018-11-20
MX376047B (es) 2025-03-07
ES2935746T3 (es) 2023-03-09
CA2933480C (en) 2022-08-23
CA2933480A1 (en) 2015-06-18
FI3080100T3 (fi) 2023-03-15
EP3080100B1 (en) 2022-11-30
US20180179204A1 (en) 2018-06-28
RS63939B1 (sr) 2023-02-28
WO2015089192A1 (en) 2015-06-18
EP3080100A4 (en) 2017-09-06
EP4257591A2 (en) 2023-10-11
PL3080100T3 (pl) 2023-03-06
US20190055242A1 (en) 2019-02-21
US9944636B2 (en) 2018-04-17
HUE061252T2 (hu) 2023-05-28
SI3080100T1 (sl) 2023-04-28
SMT202300014T1 (it) 2023-05-12
EP4257591A3 (en) 2023-11-22
MX2016007585A (es) 2016-12-16

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