DK3046901T3 - Sammensætninger til behandling af forhøjet blodtryk og/eller fibrose - Google Patents
Sammensætninger til behandling af forhøjet blodtryk og/eller fibrose Download PDFInfo
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- DK3046901T3 DK3046901T3 DK14845373.1T DK14845373T DK3046901T3 DK 3046901 T3 DK3046901 T3 DK 3046901T3 DK 14845373 T DK14845373 T DK 14845373T DK 3046901 T3 DK3046901 T3 DK 3046901T3
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- fibrosis
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- C07C235/34—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/09—Geometrical isomers
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Claims (14)
1. Forbindelse med formlen
eller et farmaceutisk acceptabelt salt deraf.
2. Forbindelse ifølge krav 1, hvor forbindelsen er med formlen
(VB0004), eller et farmaceutisk acceptabelt salt deraf.
3. Farmaceutisk sammensætning omfattende en forbindelse, en stereoisomer eller et farmaceutisk acceptabelt salt deraf ifølge krav 1 eller krav 2 og en farmaceutisk acceptabel excipiens.
4. Forbindelse eller en stereoisomer eller et farmaceutisk acceptabelt salt deraf ifølge krav 1 eller krav 2 til anvendelse i terapeutisk behandling af forhøjet blodtryk eller let forhøjet blodtryk.
5. Forbindelse eller en stereoisomer eller et farmaceutisk acceptabelt salt deraf ifølge krav 1 eller krav 2 til anvendelse i profylaktisk behandling af fibrose.
6. Forbindelse eller en stereoisomer eller et farmaceutisk acceptabelt salt deraf ifølge krav 1 eller krav 2 til anvendelse i terapeutisk behandling af fibrose.
7. Forbindelse eller en stereoisomer eller et farmaceutisk acceptabelt salt deraf ifølge krav 1 eller krav 2 til anvendelse i terapeutisk behandling af forhøjet blodtryk og fibrose.
8. Forbindelse eller en stereoisomer eller et farmaceutisk acceptabelt salt deraf ifølge krav 1 eller krav 2 til anvendelse i behandling af let forhøjet blodtryk og fibrose.
9. Forbindelse eller en stereoisomer eller et farmaceutisk acceptabelt salt deraf ifølge et hvilket som helst af kravene 5 til 8, hvor fibrosen er myokardiefibrose eller nyrefibrose.
10. Forbindelse eller en stereoisomer eller et farmaceutisk acceptabelt salt deraf ifølge et hvilket som helst af kravene 5 til 8, hvor fibrosen er myokardiefibrose og nyrefibrose.
11. Farmaceutisk sammensætning ifølge krav 3 til anvendelse i terapeutisk behandling af forhøjet blodtryk eller let forhøjet blodtryk.
12. Farmaceutisk sammensætning ifølge krav 3 til anvendelse i profylaktisk behandling af fibrose.
13. Farmaceutisk sammensætning ifølge krav 3 til anvendelse i terapeutisk behandling af fibrose.
14. Farmaceutisk sammensætning ifølge krav 3 til anvendelse i terapeutisk behandling af forhøjet blodtryk og fibrose eller let forhøjet blodtryk og fibrose.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2013903573A AU2013903573A0 (en) | 2013-09-17 | Compositions for the treatment of hypertension and/or fibrosis | |
| PCT/AU2014/000923 WO2015039173A1 (en) | 2013-09-17 | 2014-09-17 | Compositions for the treatment of hypertension and/or fibrosis |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK3046901T3 true DK3046901T3 (da) | 2018-01-02 |
Family
ID=52687998
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK14845373.1T DK3046901T3 (da) | 2013-09-17 | 2014-09-17 | Sammensætninger til behandling af forhøjet blodtryk og/eller fibrose |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US9458093B2 (da) |
| EP (1) | EP3046901B1 (da) |
| JP (1) | JP6122548B2 (da) |
| KR (1) | KR101736416B1 (da) |
| CN (1) | CN105683152B (da) |
| AP (1) | AP2016009079A0 (da) |
| AU (1) | AU2014324078B2 (da) |
| BR (1) | BR112016005601B1 (da) |
| CA (1) | CA2924356C (da) |
| DK (1) | DK3046901T3 (da) |
| ES (1) | ES2655455T3 (da) |
| IL (1) | IL244621A (da) |
| MX (1) | MX368865B (da) |
| MY (1) | MY172557A (da) |
| NO (1) | NO3046901T3 (da) |
| NZ (1) | NZ717927A (da) |
| PH (1) | PH12016500497B1 (da) |
| PL (1) | PL3046901T3 (da) |
| RU (1) | RU2635564C2 (da) |
| SG (1) | SG11201601642WA (da) |
| UA (1) | UA118111C2 (da) |
| WO (1) | WO2015039173A1 (da) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3284981B2 (ja) | 1998-11-02 | 2002-05-27 | 株式会社デンソー | 車両用交流発電機およびそのステータの製造方法 |
| US9956166B2 (en) | 2013-09-18 | 2018-05-01 | Sorrento Therapeutics, Inc. | Methods for administration and methods for treating cardiovascular diseases with resiniferatoxin |
| JP6734294B2 (ja) * | 2015-03-18 | 2020-08-05 | ヴェクタス バイオシステムズ リミテッド | 線維症及び線維症に関連する状態の処置のための組成物 |
| JP6716598B2 (ja) * | 2015-03-18 | 2020-07-01 | ヴェクタス バイオシステムズ リミテッド | 腎臓及び／又は肝臓疾患を治療するための組成物 |
| WO2017049343A1 (en) | 2015-09-22 | 2017-03-30 | Vectus Biosystems Limited | Synthesis of terphenyl compounds |
| CN109562096A (zh) * | 2016-04-13 | 2019-04-02 | 内布拉斯加大学董事会 | 施用树脂毒素的方法和用树脂毒素治疗心血管疾病的方法 |
| WO2018018091A1 (en) | 2016-07-28 | 2018-02-01 | Vectus Biosystems Limited | Compositions for the treatment of pulmonary fibrosis |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2694288B1 (fr) * | 1992-06-30 | 1994-09-09 | Rhone Poulenc Agrochimie | Phenylbenzamides fongicides et procédés pour les préparer. |
| MXPA06014462A (es) * | 2004-06-11 | 2007-05-23 | Vectus Biosystems Ltd | Composiciones y metodos para tratamiento de enfermedades cardiovasculares. |
| RU2466738C2 (ru) * | 2005-12-09 | 2012-11-20 | Вектас Байосистемз Лимитед | Фрагменты vip и способы их применения |
| US20120088737A2 (en) | 2009-10-02 | 2012-04-12 | Ajinomoto Co., Inc | Novel acyl guanidine derivatives |
| US9630935B2 (en) * | 2013-09-17 | 2017-04-25 | Vectus Biosystems Limited | Compositions for the treatment of hypertension and/or fibrosis |
-
2014
- 2014-09-17 AP AP2016009079A patent/AP2016009079A0/xx unknown
- 2014-09-17 ES ES14845373.1T patent/ES2655455T3/es active Active
- 2014-09-17 MX MX2016003371A patent/MX368865B/es active IP Right Grant
- 2014-09-17 DK DK14845373.1T patent/DK3046901T3/da active
- 2014-09-17 KR KR1020167008664A patent/KR101736416B1/ko active Active
- 2014-09-17 SG SG11201601642WA patent/SG11201601642WA/en unknown
- 2014-09-17 JP JP2016515425A patent/JP6122548B2/ja active Active
- 2014-09-17 NO NO14845373A patent/NO3046901T3/no unknown
- 2014-09-17 NZ NZ717927A patent/NZ717927A/en unknown
- 2014-09-17 BR BR112016005601-9A patent/BR112016005601B1/pt active IP Right Grant
- 2014-09-17 CN CN201480050979.1A patent/CN105683152B/zh active Active
- 2014-09-17 MY MYPI2016000482A patent/MY172557A/en unknown
- 2014-09-17 US US15/022,278 patent/US9458093B2/en active Active
- 2014-09-17 CA CA2924356A patent/CA2924356C/en active Active
- 2014-09-17 UA UAA201602267A patent/UA118111C2/uk unknown
- 2014-09-17 WO PCT/AU2014/000923 patent/WO2015039173A1/en not_active Ceased
- 2014-09-17 RU RU2016112257A patent/RU2635564C2/ru active
- 2014-09-17 AU AU2014324078A patent/AU2014324078B2/en active Active
- 2014-09-17 PL PL14845373T patent/PL3046901T3/pl unknown
- 2014-09-17 EP EP14845373.1A patent/EP3046901B1/en active Active
-
2016
- 2016-03-14 PH PH12016500497A patent/PH12016500497B1/en unknown
- 2016-03-16 IL IL244621A patent/IL244621A/en active IP Right Grant
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