DK2375898T3 - Hidtil ukendte herbicider - Google Patents

Hidtil ukendte herbicider Download PDF

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DK2375898T3
DK2375898T3 DK09765114.5T DK09765114T DK2375898T3 DK 2375898 T3 DK2375898 T3 DK 2375898T3 DK 09765114 T DK09765114 T DK 09765114T DK 2375898 T3 DK2375898 T3 DK 2375898T3
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formula
compound
pyridyl
methyl
pyrimidyl
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DK09765114.5T
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John Benjamin Taylor
Jeffrey Steven Wailes
Stephane André Marie Jeanmart
Mangala Govenkar
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Syngenta Participations Ag
Syngenta Ltd
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    • C07D261/08Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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Claims (19)

1. Forbindelse med formel I
(i) hvor G er hydrogen eller en/et landbrugsmæssigt acceptabel(t) metal, sulfoniumgruppe, ammoniumgruppe eller beskyttelsesgruppe (latentiating group); R1 er methyl, ethyl, n-propyl, isopropyl, cyclopropyl, halogenmethyl, halogenethyl, vinyl, ethynyl, halogen, Ci-C2alkoxy eller Ci-C2halogenalkoxy; R2 og R3 uafhængigt af hinanden er hydrogen, methyl, ethyl, n-propyl, isopropyl, cyclopropyl, halogenmethyl, halogenethyl, vinyl, propenyl, ethynyl, propynyl, halogen, Ci-C2alkoxy, Ci-C2halogenalkoxy, eventuelt substitueret aryl eller eventuelt substitueret heteroaryl; og hvor i R2 og R3, når de er til stede, de eventuelle substituenter på aryl er udvalgt uafhængigt blandt: halogen, nitro, cyano, rhodano, isothiocyanato, Ci-C6alkyl, Ci-C6halogenalkyl, Ci-C6alkoxy (Ci-C6) alkyl, C2-C6alkenyl, C2- C6halogenalkenyl, C2-C6alkynyl, C3-C7cycloalkyl (som selv eventuelt er substitueret med Ci-C6alkyl eller halogen), C5- 7cycloalkenyl (som selv eventuelt er substitueret med Ci~ C6alkyl eller halogen), hydroxy, Ci-Ci0alkoxy, Ci-Ci0alkoxy (Ci — Cio)alkoxy, tri (C1-C4) alkylsilyl (Ci-C6) alkoxy, Ci- C6alkoxycarbonyl (C1-C10) alkoxy, Ci-Ci0halogenalkoxy, aryl (Ci — C4)alkoxy (hvor arylgruppen eventuelt er substitueret med halogen eller Ci-C6alkyl) , C3-C7cycloalkyloxy (hvor cycloalkylgruppen eventuelt er substitueret med Ci-C6alkyl eller halogen) , C3-Cioalkenyloxy, C3-Cioalkynyloxy, mercapto, Ci-Cioalkylthio, Ci-Ciohalogenalkylthio, aryl (C1-C4) alkylthio, C3-Cvcycloalkylthio (hvor cycloalkylgruppen eventuelt er substitueret med Ci-C6alkyl eller halogen), tri (C1-C4) -alkylsilyl (C1-C6) alkylthio, arylthio, Ci-C6alkylsulfonyl, Ci-Cehalogenalkylsulfonyl, Ci-C6alkylsulfinyl, Ci- Cehalogenalkylsulfinyl, arylsulfonyl, tri (C1-C4) alkylsilyl, aryldi(C1-C4)alkylsilyl, Ci-C4alkyldiarylsilyl, triarylsilyl, Ci-Cioalkylcarbonyl, HO2C, Ci-Cioalkoxycarbonyl, aminocarbonyl, Ci-C6alkylaminocarbonyl, di (Ci-Cgalkyl)aminocarbonyl, N-(Ci-Csalkyl)-N-(Ci-C3alkoxy)aminocarbonyl, Ci-C6alkylcarbonyloxy, arylcarbonyloxy, di(Οι-Οε)alkylaminocarbonyloxy, aryl (som selv eventuelt er substitueret med Ci-C6alkyl eller halogen), heterocyclyl (som selv eventuelt er substitueret med Ci-C6alkyl eller halogen), aryloxy (hvor arylgruppen eventuelt er substitueret med Ci-Cgalkyl eller halogen), heterocyclyloxy (hvor heterocyclylgruppen eventuelt er substitueret med Ci~ Cgalkyl eller halogen), amino, Ci-Cgalkylamino, di(Ci— Cg) alkylamino, Ci-Cgalkylcarbonylamino, Λ/'-(Ci-Cg) alkylcarbonyl-N- (Ci~Cis) alkylamino eller arylcarbonyl (hvor arylgruppen eventuelt selv er substitueret med halogen eller Ci-Cgalkyl) ; eller to nabopositioner på et arylsystem er cykliseret til frembringelse af en 5-, 6- eller 7-leddet carbocyklisk eller heterocyklisk ring, som selv eventuelt er substitueret med halogen eller Ci-C6alkyl; og hvor i R2 og R3, når de er til stede, heteroarylgruppen eventuelt er substitueret med Ci-C4alkyl, Ci-C3halogenalkyl, Ci-Csalkoxy, Ci-C3halogenalkoxy, cyano, nitro, halogen, Ci- Csalkylthio, Ci-C3alkylsulfinyl eller Ci-C3alkylsulfonyl; R4 er methyl, ethyl, n-propyl, isopropyl, cyclopropyl, halogenmethyl, halogenethyl, vinyl, propenyl, ethynyl, propynyl, halogen, Ci-C2alkoxy eller Ci-C2halogenalkoxy; og R5, R6, R7, R8 og R9 uafhængigt er hydrogen, halogen, Ci-C6alkyl, Ci-C6halogenalkyl, Ci-C6alkoxy, Ci-Cehalogenalkoxy, C2~C6alkenyl, C2-Cehalogenalkenyl, C2-C6alkynyl, C3-C6alkenyloxy, C3- Cehalogenalkenyloxy, C3-C6alkynyloxy, C3-C6cycloalkyl, Ci- C6alkylthio, Ci-C6alkylsulfinyl, Ci-C6alkylsulfonyl, Ci~ Cgalkoxysulfonyl, Ci-Cghalogenalkoxysulfonyl, cyano, nitro, phenyl, phenyl substitueret med Ci-C4alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, cyano, nitro, halogen, Cg-Csalkylthio, Ci-C3alkylsulfinyl eller Ci-C3alkylsulfonyl, eller heteroaryl eller heteroaryl substitueret med Ci-C4alkyl, C2-Cshalogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, cyano, nitro, halogen, Ci-C3alkylthio, Ci-C3alkylsulfinyl eller C2-Csalkylsulfonyl; eller R6 og R7 eller R8 og R9 sammen med carbonatomerne, hvortil de er bundet, danner en eventuelt substitueret carbocyklisk ring eller en heterocyclylgruppe, der eventuelt er substitueret med Ci-C6alkyl eller Ci-Cehalogenalkyl; hvor en "carbocyklisk ring" betyder en cycloalkyl- eller cycloalkenylgruppe; og hvor, når de er til stede, de eventuelle substituenter på cycloalkyl eller cycloalkenyl er Ci-C3alkyl; eller R5 og R6 sammen danner en binding; og HetAr er en heteroarylgruppe eller en heteroarylgruppe substitueret med Ci-C4alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, C2-Cshalogenalkoxy, cyano, nitro, halogen, Ci-C3alkylthio, C2-Csalkylsulfinyl eller Ci-C3alkylsulfonyl; og hvor, når G er en beskyttelsesgruppe, G er udvalgt blandt grupperne phenylCi-Csalkyl (hvor phenylgruppen eventuelt er substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, C2-Cshalogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, C2- Csalkylsulfonyl, halogen, cyano eller med nitro), heteroarylCi-Csalkyl (hvor heteroarylgruppen eventuelt er substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, Ci-C3alkylsulfonyl, halogen, cyano eller med nitro) , C3-Csalkenyl, C3-Cshalogenalkenyl, C3- C8alkynyl, C (Xa) -Ra, C (Xb) -Xc-Rb, C (Xd) -N (Rc) -Rd, -S02-Re, P(Xe) (Rf)-Rg og CH2-Xf-Rh; hvor Xa, Xb, Xc, Xd, Xe og Xf uafhængigt af hinanden er oxygen eller svovl; og hvor Ra er H, Ci-Cisalkyl, C2-Cisalkenyl, C2-Cisalkynyl, C2- Ciohalogenalkyl, Ci-Ciocyanoalkyl, Ci-Cionitroalkyl, C2- Cioaminoalkyl, Ci-Csalkylamino (C1-C5) alkyl, C2-C8dialkylamino (C2-C5) alkyl, C3-C7cycloalkyl (C1-C5) alkyl, Ci-Csalkoxy (C1-C5) alkyl, C3-C5alkenyloxy (C1-C5) alkyl, Ci-C5alkylthio (C1-C5) alkyl, C2- C5alkylsulfinyl (C1-C5) alkyl, Ci-C5alkylsulfonyl (C1-C5) alkyl, C2-C8alkylidenaminoxy (C1-C5) alkyl, Ci-C5alkylcarbonyl (C1-C5) alkyl, Ci-C5alkoxycarbonyl (C1-C5) alkyl, aminocarbonyl (C1-C5) alkyl, C2- Csalkylaminocarbonyl (C1-C5) alkyl, C2-C8dialkylaminocarbonyl (C2- C5) alkyl, Ci-Csalkylcarbonylamino (C1-C5) alkyl, N- (Ci — C5) alkylcarbonyl-A/- (C1-C5) alkylamino (C1-C5) alkyl, C3- Cetrialkylsilyl (C1-C5) alkyl, phenyl (C1-C5) alkyl (hvor phenylgruppenen eventuelt er substitueret med Ci-C3alkyl, C2-Cshalogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, Ci-C3alkylsulfonyl, halogen, cyano eller med nitro), heteroaryl(C1-C5)alkyl (hvor heteroarylgruppen eventuelt er substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, C2-Csalkoxy, Ci-C3halogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, Ci-C3alkylsulfonyl, halogen, cyano eller med nitro), C2- Cshalogenalkenyl, C3-C8cycloalkyl; phenyl eller phenyl substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, C2-Cshalogenalkoxy, halogen, cyano eller nitro; eller heteroaryl eller heteroaryl substitueret med Ci-C3alkyl, Ci-Cshalogenalkyl, Ci-C3alkoxy, Ci-Cshalogenalkoxy, halogen, cyano eller nitro; Rb er Ci-Cigalkyl, C3-Ci8alkenyl, C3-Ci8alkynyl, C2- Ciohalogenalkyl, Ci-Ci0cyanoalkyl, Ci-Ci0nitroalkyl, C2- Cioaminoalkyl, Ci-Csalkylamino (C1-C5) alkyl, C2-C8dialkylamino (C2-C5) alkyl, C3-C7cycloalkyl (C1-C5) alkyl, Ci-C5alkoxy (C1-C5) alkyl, C3-C5alkenyloxy (C1-C5) alkyl, C3-C5alkynyloxy (C1-C5) alkyl, C2- C5alkylthio (C1-C5) alkyl, Ci-C5alkylsulf inyl (C1-C5) alkyl, C2- Csalkylsulfonyl (C1-C5) alkyl, C2-C8alkylidenaminoxy (C1-C5) alkyl, Ci-Csalkylcarbonyl (C1-C5) alkyl, Ci-Csalkoxycarbonyl (C1-C5) alkyl, aminocarbonyl (C1-C5) alkyl, Ci-Csalkylaminocarbonyl (C1-C5) alkyl, C2-C8dialkylaminocarbonyl (C1-C5) alkyl, C2- Csalkylcarbonylamino (C1-C5) alkyl, N- (C1-C5) alkylcarbonyl-iV- (C2-C5) alkylamino (C1-C5) alkyl, C3-C6trialkylsilyl (C1-C5) alkyl, phenyl(C1-C5)alkyl (hvor phenylgruppen eventuelt er substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, C2-Cshalogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, C2- Csalkylsulfonyl, halogen, cyano eller med nitro), heteroarylCi-Csalkyl (hvor heteroarylgruppen eventuelt er substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, Ci-C3alkylsulfonyl, halogen, cyano eller med nitro), C3-C5halogenalkenyl, C3-C8cycloalkyl; phenyl eller phenyl substitueret med Ci-C3alkyl, C2-Cshalogenalkyl, Ci-C3alkoxy, Ci-Cshalogenalkoxy, halogen, cyano eller nitro; eller heteroaryl eller heteroaryl substitueret med Ci-C3alkyl, CR-Cshalogenalkyl, CR-C3alkoxy, CR- Cshalogenalkoxy, halogen, cyano eller nitro; og Rc og Rd hver uafhængigt af hinanden er hydrogen, Ci-Cioalkyl, C3-Cioalkenyl, C3-Cioalkynyl, C2-Ciohalogenalkyl, CR- Ciocyanoalkyl, Ci-Cionitroalkyl, Ci-Cioaminoalkyl, CR- Csalkylamino (CR-C5) alkyl, C2-C8dialkylamino (C1-C5) alkyl, C3- Cvcycloalkyl (C1-C5) alkyl, CR-Csalkoxy (C1-C5) alkyl, C3- Csalkenyloxy (C1-C5) alkyl, C3-Csalkynyloxy (C1-C5) alkyl, CR- Csalkylthio (C1-C5) alkyl, CR-Csalkylsulfinyl (C1-C5) alkyl, CR- Csalkylsulfonyl (CR-C5) alkyl, C2-C8alkylidenaminoxy (C1-C5) alkyl, Ci-Csalkylcarbonyl (C1-C5) alkyl, Ci-Csalkoxycarbonyl (C1-C5) alkyl, aminocarbonyl (CR-C5) alkyl, Ci-Csalkylaminocarbonyl (C1-C5) alkyl, C2-C8dialkylaminocarbonyl (C1-C5) alkyl, CR- Csalkylcarbonylamino (C1-C5) alkyl, N- (C1-C5) alkylcarbonyl-ΙΊ- (C2— C5) alkylaminoalkyl, C3-C6trialkylsilyl (CR-C5) alkyl, phenyl (Ci — C5)alkyl (hvor phenylgruppen eventuelt er substitueret med CR-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, CR-Csalkylthio, CR-C3alkylsulfinyl, Ci-C3alkylsulfonyl, halogen, cyano eller med nitro), heteroaryl(CR-C5)alkyl (hvor heteroarylgruppen eventuelt er substitueret med CR-C3alkyl, CR-Cshalogenalkyl, Ci-C3alkoxy, CR-Cshalogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, CR-C3alkylsulfonyl, halogen, cyano eller med nitro), C2-Cshalogenalkenyl, Cs-Cscycloalkyl; phenyl eller phenyl substitueret med CR-C3alkyl, CR-Cshalogenalkyl, CR-Csalkoxy, CR-Cshalogenalkoxy, halogen, cyano eller nitro; heteroaryl eller heteroaryl substitueret med CR-C3alkyl, CR-Cshalogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, halogen, cyano eller nitro; heteroarylamino eller heteroarylamino substitueret med CR-C3alkyl, CR-Cshalogenalkyl, Ci-C3alkoxy, Ci-Cshalogenalkoxy, halogen, cyano eller nitro; diheteroarylamino eller diheteroarylamino substitueret med CR-C3alkyl, CR-Cshalogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, halogen, cyano eller nitro; phenylamino eller phenylamino substitueret med CR-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, halogen, cyano eller med nitro; diphenylamino eller diphenylamino substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, CR-C3alkoxy, Ci-Cshalogenalkoxy, halogen, cyano eller med nitro; eller C3-C7cycloalkylamino, diC3-C7cycloalkylamino eller C3- Cvcycloalkoxy ; eller Rc og Rd kan være forbundet til frembringelse af en 3-7-leddet ring, der eventuelt indeholder ét heteroatom, der er udvalgt blandt 0 eller S; og Re er Ci-Cioalkyl, C2-Cioalkenyl, C2-Cioalkynyl, CR-Ciohalogenalkyl, Ci-Ciocyanoalkyl, Ci-Cionitroalkyl, Ci- Cioaminoalkyl, Ci-Csalkylamino (C1-C5) alkyl, C2-C8dialkylamino (Ci — C5) alkyl, C3-C7cycloalkyl (C1-C5) alkyl, CR-Csalkoxy (C1-C5) alkyl, C3_C5alkenyloxy (C1-C5) alkyl, C3-Csalkynyloxy (C1-C5) alkyl, Ci-Csalkylthio (C1-C5) alkyl, Ci-Csalkylsulf inyl (C1-C5) alkyl, CR- Csalkylsulfonyl (C1-C5) alkyl, C2-C8alkylidenaminoxy (C1-C5) alkyl, Ci-C5alkylcarbonyl (C1-C5) alkyl, Ci-C5alkoxycarbonyl (C1-C5) alkyl, aminocarbonyl (C1-C5) alkyl, Ci-Csalkylaminocarbonyl (C1-C5) alkyl, C2-C8dialkylaminocarbonyl (C1-C5) alkyl, Ci- Csalkylcarbonylamino (C1-C5) alkyl, N- (C1-C5) alkylcarbonyl-N- (Ci — C5) alkylamino (C1-C5) alkyl, C3-C6trialkylsilyl (C1-C5) alkyl, phenyl(C1-C5)alkyl (hvor phenylgruppen eventuelt er substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Cg-Cshalogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, Ci~ Csalkylsulfonyl, halogen, cyano eller med nitro), heteroaryl(C1-C5)alkyl (hvor heteroarylgruppen eventuelt er substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-Cshalogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, Ci- Csalkylsulfonyl, halogen, cyano eller med nitro), C2- Cshalogenalkenyl, C3-Cscycloalkyl; phenyl eller phenyl substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci_ Cshalogenalkoxy, halogen, cyano eller nitro; heteroaryl eller heteroaryl substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-Csalkoxy, Ci-C3halogenalkoxy, halogen, cyano eller med nitro; heteroarylamino eller heteroarylamino substitueret med Ci-Csalkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, halogen, cyano eller med nitro; diheteroarylamino eller diheteroarylamino substitueret med Ci-C3alkyl, Ci- Cshalogenalkyl, Ci-C3alkoxy, Ci-Cshalogenalkoxy, halogen, cyano eller nitro; phenylamino eller phenylamino substitueret med Cg-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, halogen, cyano eller nitro; diphenylamino eller diphenylamino substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci- Cshalogenalkoxy, halogen, cyano eller nitro; eller C3- C7cycloalkylamino, diC3-C7cycloalkylamino, C3-C7cycloalkoxy, CR-Cioalkoxy, Ci-Ciohalogenalkoxy, Ci-Csalkylamino eller C2-Csdialkylamino ; Rf og Rg hver uafhængigt af hinanden er Ci-Cioalkyl, C2- Cioalkenyl, C2-Cioalkynyl, Ci-Cioalkoxy, Ci-Ciohalogenalkyl, CR-Ciocyanoalkyl, Ci-Cionitroalkyl, Ci-Cioaminoalkyl, CR- Csalkylamino (C1-C5) alkyl, C2-C8dialkylamino (C1-C5) alkyl, C3- C7cycloalkyl (C1-C5) alkyl, CR-Csalkoxy (C1-C5) alkyl. C3- Csalkenyloxy (C1-C5) alkyl, C3-Csalkynyloxy (C1-C5) alkyl, CR- Csalkylthio (C1-C5) alkyl, Ci-Csalkylsulf inyl (C1-C5) alkyl, CR- C5alkylsulfonyl (C1-C5) alkyl, C2-C8alkylidenaminoxy (C1-C5) alkyl, Ci-C5alkylcarbonyl (C1-C5) alkyl, Ci-C5alkoxycarbonyl (CR-C5) alkyl, aminocarbonyl (C1-C5) alkyl, Ci-Csalkylaminocarbonyl (C1-C5) alkyl, C2-C8dialkylaminocarbonyl (C1-C5) alkyl, CR- Csalkylcarbonylamino (C1-C5) alkyl, N- (C1-C5) alkylcarbonyl-iV- (C2-C5) alkylaminoalkyl, C3-C6trialkylsilyl (C1-C5) alkyl, phenyl (CR-C5)alkyl (hvor phenylgruppen eventuelt er substitueret med CR-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, CR-Csalkylthio, Ci-C3alkylsulfinyl, Ci-C3alkylsulfonyl, halogen, cyano eller med nitro), heteroaryl(CR-C5)alkyl (hvor heteroarylgruppen eventuelt er substitueret med CR-C3alkyl, CR-Cshalogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, Ci-C3alkylsulfonyl, halogen, cyano eller med nitro), C2-Cshalogenalkenyl, Cs-Cscycloalkyl; phenyl eller phenyl substitueret med CR-C3alkyl, CR-Cshalogenalkyl, CR-Csalkoxy, Ci-C3halogenalkoxy, halogen, cyano eller nitro; heteroaryl eller heteroaryl substitueret med CR-C3alkyl, Ci-Cshalogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, halogen, cyano eller med nitro; heteroarylamino eller heteroarylamino substitueret med CR-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, CR-Cshalogenalkoxy, halogen, cyano eller med nitro; diheteroarylamino eller diheteroarylamino substitueret med CR-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, halogen, cyano eller nitro; phenylamino eller phenylamino substitueret med CR-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-Cshalogenalkoxy, halogen, cyano eller nitro; diphenylamino eller diphenylamino substitueret med CR-C3alkyl, Ci~ Cshalogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, halogen, cyano eller nitro; eller C3-C7cycloalkylamino, diC3-C7cycloalkylamino, C3-C7cycloalkoxy, Ci-Ciohalogenalkoxy, Ci-Csalkylamino eller C2-C8dialkylamino; eller benzyloxy eller phenoxy, hvor benzyl- og phenylgrupperne selv kan være substitueret med Ci-C3alkyl, Ci-Cshalogenalkyl, Ci~C3alkoxy, Ci-C3halogenalkoxy, halogen, cyano eller nitro; og Rh er Ci-Cioalkyl, C3-Cioalkenyl, C3-Cioalkynyl, Ci- Ciohalogenalkyl, Ci-Ciocyanoalkyl, Ci-Cionitroalkyl, C2- Cioaminoalkyl, Ci-Csalkylamino (C1-C5) alkyl, C2-C8dialkylamino (Ci — C5) alkyl, C3-C7cycloalkyl (C1-C5) alkyl, Ci-Csalkoxy (C1-C5) alkyl, C3-C5alkenyloxy (C1-C5) alkyl, C3-C5alkynyloxy (C1-C5) alkyl, Cg-C5alkylthio (C1-C5) alkyl, Ci-C5alkylsulf inyl (C1-C5) alkyl, Cg- C5alkylsulfonyl (C1-C5) alkyl, C2-C8alkylidenaminoxy (C1-C5) alkyl, Ci-C5alkylcarbonyl (C1-C5) alkyl, Ci-C5alkoxycarbonyl (C1-C5) alkyl, aminocarbonyl (C1-C5) alkyl, Ci-Csalkylaminocarbonyl (C1-C5) alkyl, C2-C8dialkylaminocarbonyl (C1-C5) alkyl, Ci~ Csalkylcarbonylamino (C1-C5) alkyl, N- (C1-C5) alkylcarbonyl-iV- (Ci — C5) alkylamino (C1-C5) alkyl, C3-C6trialkylsilyl (C1-C5) alkyl, phenyl(C1-C5)alkyl (hvor phenylgruppen eventuelt er substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Cg-Cshalogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, Ci- Csalkylsulfonyl, halogen, cyano eller med nitro), heteroaryl(C1-C5)alkyl (hvor heteroarylgruppen eventuelt er substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-Cshalogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, Ci- Csalkylsulfonyl, halogen, cyano eller med nitro), phenoxy(Ci — C5)alkyl (hvor phenylgruppen eventuelt er substitueret med Ci-Csalkyl, Ci-C3halogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, Ci-Csalkylthio, Ci-C3alkylsulfinyl, Ci-C3alkylsulfonyl, halogen, cyano eller med nitro), heteroaryloxy (C1-C5) alkyl (hvor heteroarylgruppen eventuelt er substitueret med Ci-C3alkyl, Ci-Cshalogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, Ci-C3alkylthio, Ci-C3alkylsulfinyl, Ci-C3alkylsulfonyl, halogen, cyano eller med nitro), C3-C5halogenalkenyl, C3-C8cycloalkyl; phenyl eller phenyl substitueret med Ci-C3alkyl, Ci-C3halogenalkyl, Ci-Cgalkoxy, Ci-Cghalogenalkoxy, halogen eller med nitro; eller heteroaryl eller heteroaryl substitueret med Ci-C3alkyl, Ci- Cshalogenalkyl, Ci-C3alkoxy, Ci-C3halogenalkoxy, halogen, cyano eller med nitro; og hvor "aryl" betyder phenyl; hvor "heteroaryl" betyder en 6-leddet heteroarylring, der eventuelt er benzoanneleret; og hvor "heterocyclyl" betyder et ikke-aromatisk, monocyklisk eller bicyklisk ringsystem, der indeholder op til 7 atomer, herunder et eller to heteroatomer, der er udvalgt blandt 0, S og N.
2. Forbindelse ifølge krav 1, hvor "heteroaryl" betyder pyridyl, pyrimidinyl, pyridazinyl, quinolinyl, isoquinolinyl, cinnolinyl, phthalazinyl, quinazolinyl eller quinoxalinyl.
3. Forbindelse ifølge krav 1, hvor: "cycloalkyl" er cyclopropyl, cyclobutyl, cyclopentyl eller cyclohexyl; "cycloalkylalkyl" er cyclopropylmethyl; og "cycloalkenyl" er cyclopentenyl eller cyclohexenyl.
4. Forbindelse ifølge krav 1, hvor R1 er methyl, ethyl, n-propyl, vinyl, ethynyl, halogen, CR-C2alkoxy eller Ci-C2halogenalkoxy; R2 er methyl, halogen, Ci-C2alkoxy eller Ci-C2halogenalkoxy eller eventuelt substitueret phenyl; R3 er hydrogen; R4 er methyl, ethyl, n-propyl, vinyl, ethynyl eller methoxy; og R5, R6, R7, R8 og R9 uafhængigt er hydrogen, halogen, Ci-C4alkyl, Ci-C4halogenalkyl, Ci-C4alkoxy, Ci-C4halogenalkoxy, C2~C4alkenyl, C2-C4halogenalkenyl eller C2~C4alkynyl; eller R6 og R7 eller R8 og R9 sammen med carbonatomerne, hvortil de er bundet, danner en eventuelt substitueret carbocyklisk ring som defineret i krav 1 eller en eventuelt substitueret heterocyclylgruppe som defineret i krav 1; eller R5 og R6 sammen danner en binding; og HetAr er heteroarylgruppen eller heteroarylgruppen substitueret en til tre gange med fluor, chlor, brom, methyl, methoxy, cyano eller trifluormethyl.
5. Forbindelse ifølge krav 4, hvor R1 er methyl eller ethyl, R2 er methyl eller chlor, R3 er hydrogen, og R4 er methyl, ethyl eller methoxy, og R5, R6, R7, R8 og R9 er hydrogen, eller R5 og R6 sammen danner en binding; og HetAr er en 6-leddet heteroarylgruppe eller en 6-leddet heteroarylgruppe, der er substitueret en til tre gange med fluor, chlor, brom, methyl, methoxy, cyano eller trifluormethyl.
6. Forbindelse ifølge krav 1, 4 eller 5, hvor HetAr er pyridyl, pyrimidinyl, pyridazinyl, quinolinyl, isoquinolinyl, cinnolinyl, phthalazinyl, quinazolinyl eller quinoxalinyl, hvor disse ringe eventuelt er substitueret en eller to gange med fluor, chlor, brom, methyl, methoxy, cyano eller trifluormethyl.
7. Forbindelse ifølge krav 1, hvor, når G er en beskyttelsesgruppe, G er en gruppe -C (Xa)-Ra eller -C (Xb) -Xc-Rb, og betydningerne af Xa, Ra, Xb, Xc og Rb er som defineret i krav 1.
8. Forbindelse ifølge krav 1, hvor G er hydrogen.
9. Forbindelse ifølge krav 1, der er en af følgende forbindelser:
(T10),
(T13),
(T14),
(T15),
(T16),
(T17),
(Τ18)
(Τ22),
(Τ23),
(Τ24),
(Τ25),
(Τ26),
(Τ27),
(Τ28),
(Τ29),
(Τ30),
(Τ31)
(Τ32)
(Τ33),
(Τ34),
(T35),
(T36),
(T37),
(T38),
(T40),
(T41),
(T43),
(T 44),
(Τ45),
(Τ46),
(Τ47),
(Τ48),
(Τ50),
(Τ51),
(Τ52),
(Τ55),
(T57),
(T61),
(T65),
<T66),
(Τ67),
(Τ68).
(Τ69),
(Τ70),
(Τ71),
(Τ72),
(Τ73),
(Τ74),
(Τ76),
(Τ79),
(Τ80),
(Τ81),
(T85),
(T89),
(T90),
(T98),
(T101),
(T102),
(T103),
(Ρ4),
(PS),
(Ρ9),
(Ρ14), eller
(Ρ15).
10. Forbindelse ifølge krav 1, der er en forbindelse med strukturtype T-l:
T-1 hvor R5, R6, R7, R8 og R9 er H; og hvor HetAr er 2-pyridyl, 3-fluor-2-pyridyl, 4-fluor-2-pyridyl, 5-fluor-2-pyridyl, 6-fluor-2-pyridyl, 3-chlor-2-pyridyl, 4-chlor-2-pyridyl, 5-chlor-2-pyridyl, 6-chlor-2-pyridyl, 3- methyl-2-pyridyl, 4-methyl-2-pyridyl, 5-methyl-2-pyridyl, 6- methyl-2-pyridyl, 3-trifluormethyl-2-pyridyl, 4- trifluormethyl-2-pyridyl, 5-trifluormethyl-2-pyridyl, 6- trifluormethyl-2-pyridyl, 3-methoxy-2-pyridyl, 4-methoxy-2-pyridyl, 5-methoxy-2-pyridyl, 6-methoxy-2-pyridyl, 3-trifluormethoxy-2-pyridyl, 4-trifluormethoxy-2-pyridyl, 5- trifluormethoxy-2-pyridyl, 6-trifluormethoxy-2-pyridyl, 3- cyano-2-pyridyl, 4-cyano-2-pyridyl, 5-cyano-2-pyridyl, 6- cyano-2-pyridyl, 3-nitro-2-pyridyl, 4-nitro-2-pyridyl, 5- nitro-2-pyridyl, 6-nitro-2-pyridyl, 3-methansulfonyl-2- pyridyl, 4-methansulfonyl-2-pyridyl, 5-methansulfonyl-2- pyridyl, 6-methansulfonyl-2-pyridyl, 3-pyridyl, 2-fluor-3- pyridyl, 4-fluor-3-pyridyl, 5-fluor-3-pyridyl, 6-fluor-3- pyridyl, 2-chlor-3-pyridyl, 4-chlor-3-pyridyl, 5-chlor-3- pyridyl, 6-chlor-3-pyridyl, 2-brom-3-pyridyl, 4-brom-3-pyridyl, 5-brom-3-pyridyl, 6-brom-3-pyridyl, 2-methoxy-3-pyridyl, 4-methoxy-3-pyridyl, 5-methoxy-3-pyridyl, 6-methoxy- 3-pyridyl, 2-trifluormethoxy-3-pyridyl, 4-trifluormethoxy-3-pyridyl, 5-trifluormethoxy-3-pyridyl, 6-trifluormethoxy-3- pyridyl, 2-methyl-3-pyridyl, 4-methyl-3-pyridyl, 5-methyl-3-pyridyl, 6-methyl-3-pyridyl, 2-trifluormethyl-3-pyridyl, 4-trifluormethyl-3-pyridyl, 5-trifluormethyl-3-pyridyl, 6- trifluormethyl-3-pyridyl, 2-cyano-3-pyridyl, 4-cyano-3- pyridyl, 5-cyano-3-pyridyl, 6-cyano-3-pyridyl, 2-nitro-3- pyridyl, 4-nitro-3-pyridyl, 5-nitro-3-pyridyl, 6-nitro-3- pyridyl, 2-methansulfonyl-3-pyridyl, 4-methansulfonyl-3- pyridyl, 5-methansulfonyl-3-pyridyl, 6-methansulfonyl-3- pyridyl, 4-pyridyl, 2-fluor-4-pyridyl, 3-fluor-4-pyridyl, 2-chlor-4-pyridyl, 3-chlor-4-pyridyl, 2-brom-4-pyridyl, 3-brom- 4-pyridyl, 2-methoxy-4-pyridyl, 3-methoxy-4-pyridyl, 2-trifluormethoxy-4-pyridyl, 3-trifluormethoxy-4-pyridyl, 2- methyl-4-pyridyl, 3-methyl-4-pyridyl, 2-trifluormethyl-4-pyridyl, 3-trifluormethyl-4-pyridyl, 2-cyano-4-pyridyl, 3- cyano-4-pyridyl, 2-nitro-4-pyridyl, 3-nitro-4-pyridyl, 2- methansulfonyl-4-pyridyl, 3- methansulfonyl-4-pyridyl, 2-pyridazinyl, 4-fluor-2-pyridazinyl, 5-fluor-2-pyridazinyl, 6-fluor-2-pyridazinyl, 4-chlor-2-pyridazinyl, 5-chlor-2- pyridazinyl, 6-chlor-2-pyridazinyl, 4-brom-2-pyridazinyl, 5-brom-2-pyridazinyl, 6-brom-2-pyridazinyl, 4-methoxy-2- pyridazinyl, 5-methoxy-2-pyridazinyl, 6-methoxy-2-pyridazinyl, 4-trifluormethoxy-2-pyridazinyl, 5-trifluormethoxy-2- pyridazinyl, 6-trifluormethoxy-2-pyridazinyl, 4-methyl-2- pyridazinyl, 5-methyl-2-pyridazinyl, 6-methyl-2-pyridazinyl, 4- trifluormethyl-2-pyridazinyl, 5-trifluormethyl-2- pyridazinyl, 6-trifluormethyl-2-pyridazinyl, 4-cyano-2- pyridazinyl, 5-cyano-2-pyridazinyl, 6-cyano-2-pyridazinyl, 4-nitro-2-pyridazinyl, 5-nitro-2-pyridazinyl, 6-nitro-2- pyridazinyl, 4-methansulfonyl-2-pyridazinyl, 5-methansulfonyl- 2-pyridazinyl, 6-methansulfonyl-2-pyridazinyl, 3-pyridazinyl, 2-fluor-3-pyridazinyl, 5-fluor-3-pyridazinyl, 6-fluor-3- pyridazinyl, 2-chlor-3-pyridazinyl, 5-chlor-3-pyridazinyl, 6- chlor-3-pyridazinyl, 2-brom-3-pyridazinyl, 5-brom-3- pyridazinyl, 6-brom-3-pyridazinyl, 2-methoxy-3-pyridazinyl, 5-methoxy-3-pyridazinyl, 6-methoxy-3-pyridazinyl, 2- trifluormethoxy-3-pyridazinyl, 5-trifluormethoxy-3- pyridazinyl, 6-trifluormethoxy-3-pyridazinyl, 2-methyl-3- pyridazinyl, 5-methyl-3-pyridazinyl, 6-methyl-3-pyridazinyl, 2- trifluormethyl-3-pyridazinyl, 5-trifluormethyl-3- pyridazinyl, 6-trifluormethyl-3-pyridazinyl, 2-cyano-3- pyridazinyl, 5-cyano-3-pyridazinyl, 6-cyano-3-pyridazinyl, 2- nitro-3-pyridazinyl, 5-nitro-3-pyridazinyl, 6-nitro-3- pyridazinyl, 2-methansulfonyl-3-pyridazinyl, 5-methansulfonyl- 3- pyridazinyl, 6-methansulfonyl-3-pyridazinyl, 2-pyrimidyl, 4-fluor-2-pyrimidyl, 5-fluor-2-pyrimidyl, 4-chlor-2-pyrimidyl, 5- chlor-2-pyrimidyl, 4-brom-2-pyrimidyl, 5-brom-2-pyrimidyl, 4- methoxy-2-pyrimidyl, 5-methoxy-2-pyrimidyl, 4- trifluormethoxy-2-pyrimidyl, 5-trifluormethoxy-2-pyrimidyl, 4- methyl-2-pyrimidyl, 5-methyl-2-pyrimidyl, 4-trifluormethyl-2-pyrimidyl, 5-trifluormethyl-2-pyrimidyl, 4-cyano-2-pyrimidyl, 5- cyano-2-pyrimidyl, 4-nitro-2-pyrimidyl, 5-nitro-2-pyrimidyl, 4-methansulfonyl-2-pyrimidyl, 5-methansulfonyl-2-pyrimidyl, 4- pyrimidyl, 2-fluor-4-pyrimidyl, 5-fluor-4-pyrimidyl, 6-fluor-4-pyrimidyl, 2-chlor-4-pyrimidyl, 5-chlor-4-pyrimidyl, 6-chlor-4-pyrimidyl, 2-brom-4-pyrimidyl, 5-brom-4-pyrimidyl, 6-brom-4-pyrimidyl, 2-methoxy-4-pyrimidyl, 5-methoxy-4- pyrimidyl, 6-methoxy-4-pyrimidyl, 2-trifluormethoxy-4- pyrimidyl, 5-trifluormethoxy-4-pyrimidyl, 6-trifluormethoxy-4-pyrimidyl, 2-methyl-4-pyrimidyl, 5-methyl-4-pyrimidyl, 6-methyl-4-pyrimidyl, 2-trifluormethyl-4-pyrimidyl, 5- trifluormethyl-4-pyrimidyl, 6-trifluormethyl-4-pyrimidyl, 2-cyano-4-pyrimidyl, 5-cyano-4-pyrimidyl, 6-cyano-4-pyrimidyl, 2-nitro-4-pyrimidyl, 5-nitro-4-pyrimidyl, 6-nitro-4-pyrimidyl, 2-methansulfonyl-4-pyrimidyl, 5-methansulfonyl-4-pyrimidyl, 6- methansulfonyl-4-pyrimidyl, 5-pyrimidyl, 2-fluor-5-pyrimidyl, 4-fluor-5-pyrimidyl, 2-chlor-5-pyrimidyl, 4-chlor-5-pyrimidyl, 2-brom-5-pyrimidyl, 4-brom-5-pyrimidyl, 2-methoxy-5-pyrimidyl, 4- methoxy-5-pyrimidyl, 2-trifluormethoxy-5-pyrimidyl, 4- trifluormethoxy-5-pyrimidyl, 2-methyl-5-pyrimidyl, 4-methyl-5-pyrimidyl, 2-trifluormethyl-5-pyrimidyl, 4-trifluormethyl-5-pyrimidyl, 2-cyano-5-pyrimidyl, 4-cyano-5-pyrimidyl, 2-nitro- 5- pyrimidyl, 4-nitro-5-pyrimidyl, 2-methansulfonyl-5- pyrimidyl, 4-methansulfonyl-5-pyrimidyl, 2-pyrazinyl, 3-fluor- 2- pyrazinyl, 5-fluor-2-pyrazinyl, 6-fluor-2-pyrazinyl, 3-chlor-2-pyrazinyl, 5-chlor-2-pyrazinyl, 6-chlor-2-pyrazinyl, 3- brom-2-pyrazinyl, 5-brom-2-pyrazinyl, 6-brom-2-pyrazinyl, 3- methoxy-2-pyrazinyl, 5-methoxy-2-pyrazinyl, 6-methoxy-2- pyrazinyl, 3-trifluormethoxy-2-pyrazinyl, 5-trifluormethoxy-2-pyrazinyl, 6-trifluormethoxy-2-pyrazinyl, 3-methyl-2- pyrazinyl, 5-methyl-2-pyrazinyl, 6-methyl-2-pyrazinyl, 3-trifluormethyl-2-pyrazinyl, 5-trifluormethyl-2-pyrazinyl, 6-trifluormethyl-2-pyrazinyl, 3-cyano-2-pyrazinyl, 5-cyano-2-pyrazinyl, 6-cyano-2-pyrazinyl, 3-nitro-2-pyrazinyl, 5-nitro-2-pyrazinyl, 6-nitro-2-pyrazinyl, 3-methylsulfonat-2- pyrazinyl, 5-methylsulfonat-2-pyrazinyl eller 6- methylsulfonat-2-pyrazinyl; og hvor: R1, R2 og R4 er methyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er chlorid, og R3 er hydrogen; eller R1 og R2 er methyl, R4 er chlorid, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er bromid, og R3 er hydrogen; eller R1 er methyl, R2 er chlorid, R3 er hydrogen, og R4 er methoxy; eller R1 er methyl, R2 er bromid, R3 er hydrogen, og R4 er methoxy; eller R1 og R2 er methyl, R4 er ethenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er ethynyl, og R3 er hydrogen; eller R1 og R2 er methyl, R4 er ethynyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er phenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-f luorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-chlorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-trifluorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 4-f luorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 4-chlorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 4-trifluorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3,4-difluorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-f luor-4-chlorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-chlor-4-f luorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3,4-dichlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R2 og R4 er methyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er chlorid, og R3 er hydrogen; eller R1 er ethyl, R2 er methyl, R4 er chlorid, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er bromid, og R3 er hydrogen; eller R1 er ethyl, R2 er chlorid, R3 er hydrogen, og R4 er methoxy; eller R1 er ethyl, R2 er bromid, R3 er hydrogen, og R4 er methoxy; eller R1 er ethyl, R2 er methyl, R4 er ethenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er ethynyl, og R3 er hydrogen; eller R1 er ethyl, R2 er methyl, R4 er ethynyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er phenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-f luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-chlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-trif luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 4-f luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 4-chlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 4-trif luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3,4-difluorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-fluor-4-chlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-chlor-4-fluorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3,4-dichlorphenyl, og R3 er hydrogen; eller R1 og R4 er ethyl, R2 er methyl, og R3 er hydrogen.
11. Forbindelse ifølge krav 1, som er en forbindelse med strukturtype T-l:
T-1 hvor R5 er H, R6 er CH3, og R7, R8 og R9 er H; og hvor HetAr er 2-pyridyl, 3-fluor-2-pyridyl, 4-fluor-2-pyridyl, 5-fluor-2-pyridyl, 6-fluor-2-pyridyl, 3-chlor-2-pyridyl, 4-chlor-2-pyridyl, 5-chlor-2-pyridyl, 6-chlor-2-pyridyl, 3- methyl-2-pyridyl, 4-methyl-2-pyridyl, 5-methyl-2-pyridyl, 6- methyl-2-pyridyl, 3-trifluormethyl-2-pyridyl, 4- trifluormethyl-2-pyridyl, 5-trifluormethyl-2-pyridyl, 6- trifluormethyl-2-pyridyl, 3-methoxy-2-pyridyl, 4-methoxy-2-pyridyl, 5-methoxy-2-pyridyl, 6-methoxy-2-pyridyl, 3-trifluormethoxy-2-pyridyl, 4-trifluormethoxy-2-pyridyl, 5- trifluormethoxy-2-pyridyl, 6-trifluormethoxy-2-pyridyl, 3- cyano-2-pyridyl, 4-cyano-2-pyridyl, 5-cyano-2-pyridyl, 6- cyano-2-pyridyl, 3-nitro-2-pyridyl, 4-nitro-2-pyridyl, 5- nitro-2-pyridyl, 6-nitro-2-pyridyl, 3-methansulfonyl-2- pyridyl, 4-methansulfonyl-2-pyridyl, 5-methansulfonyl-2- pyridyl, 6-methansulfonyl-2-pyridyl, 3-pyridyl, 2-fluor-3- pyridyl, 4-fluor-3-pyridyl, 5-fluor-3-pyridyl, 6-fluor-3- pyridyl, 2-chlor-3-pyridyl, 4-chlor-3-pyridyl, 5-chlor-3- pyridyl, 6-chlor-3-pyridyl, 2-brom-3-pyridyl, 4-brom-3-pyridyl, 5-brom-3-pyridyl, 6-brom-3-pyridyl, 2-methoxy-3-pyridyl, 4-methoxy-3-pyridyl, 5-methoxy-3-pyridyl, 6-methoxy- 3-pyridyl, 2-trifluormethoxy-3-pyridyl, 4-trifluormethoxy-3-pyridyl, 5-trifluormethoxy-3-pyridyl, 6-trifluormethoxy-3-pyridyl, 2-methyl-3-pyridyl, 4-methyl-3-pyridyl, 5-methyl-3-pyridyl, 6-methyl-3-pyridyl, 2-trifluormethyl-3-pyridyl, 4-trifluormethyl-3-pyridyl, 5-trifluormethyl-3-pyridyl, 6- trifluormethyl-3-pyridyl, 2-cyano-3-pyridyl, 4-cyano-3- pyridyl, 5-cyano-3-pyridyl, 6-cyano-3-pyridyl, 2-nitro-3-pyridyl, 4-nitro-3-pyridyl, 5-nitro-3-pyridyl, 6-nitro-3-pyridyl, 2-methansulfonyl-3-pyridyl, 4-methansulfonyl-3-pyridyl, 5-methansulfonyl-3-pyridyl, 6-methansulfonyl-3-pyridyl, 4-pyridyl, 2-fluor-4-pyridyl, 3-fluor-4-pyridyl, 2-chlor-4-pyridyl, 3-chlor-4-pyridyl, 2-brom-4-pyridyl, 3-brom- 4-pyridyl, 2-methoxy-4-pyridyl, 3-methoxy-4-pyridyl, 2-trifluormethoxy-4-pyridyl, 3-trifluormethoxy-4-pyridyl, 2-methyl-4-pyridyl, 3-methyl-4-pyridyl, 2-trifluormethyl-4-pyridyl, 3-trifluormethyl-4-pyridyl, 2-cyano-4-pyridyl, 3-cyano-4-pyridyl, 2-nitro-4-pyridyl, 3-nitro-4-pyridyl, 2-methansulfonyl-4-pyridyl, 3- methansulfonyl-4-pyridyl, 2-pyridazinyl, 4-fluor-2-pyridazinyl, 5-fluor-2-pyridazinyl, 6-fluor-2-pyridazinyl, 4-chlor-2-pyridazinyl, 5-chlor-2-pyridazinyl, 6-chlor-2-pyridazinyl, 4-brom-2-pyridazinyl, 5-brom-2-pyridazinyl, 6-brom-2-pyridazinyl, 4-methoxy-2-pyridazinyl, 5-methoxy-2-pyridazinyl, 6-methoxy-2-pyridazinyl, 4-trifluormethoxy-2-pyridazinyl, 5-trifluormethoxy-2-pyridazinyl, 6-trifluormethoxy-2-pyridazinyl, 4-methyl-2-pyridazinyl, 5-methyl-2-pyridazinyl, 6-methyl-2-pyridazinyl, 4-trifluormethyl-2-pyridazinyl, 5-trifluormethyl-2-pyridazinyl, 6-trifluormethyl-2-pyridazinyl, 4-cyano-2-pyridazinyl, 5-cyano-2-pyridazinyl, 6-cyano-2-pyridazinyl, 4-nitro-2-pyridazinyl, 5-nitro-2-pyridazinyl, 6-nitro-2-pyridazinyl, 4-methansulfonyl-2-pyridazinyl, 5-methansulfonyl-2-pyridazinyl, 6-methansulfonyl-2-pyridazinyl, 3-pyridazinyl, 2-fluor-3-pyridazinyl, 5-fluor-3-pyridazinyl, 6-fluor-3-pyridazinyl, 2-chlor-3-pyridazinyl, 5-chlor-3-pyridazinyl, 6-chlor-3-pyridazinyl, 2-brom-3-pyridazinyl, 5-brom-3-pyridazinyl, 6-brom-3-pyridazinyl, 2-methoxy-3-pyridazinyl, 5-methoxy-3-pyridazinyl, 6-methoxy-3-pyridazinyl, 2-trifluormethoxy-3-pyridazinyl, 5-trifluormethoxy-3-pyridazinyl, 6-trifluormethoxy-3-pyridazinyl, 2-methyl-3-pyridazinyl, 5-methyl-3-pyridazinyl, 6-methyl-3-pyridazinyl, 2-trifluormethyl-3-pyridazinyl, 5-trifluormethyl-3-pyridazinyl, 6-trifluormethyl-3-pyridazinyl, 2-cyano-3-pyridazinyl, 5-cyano-3-pyridazinyl, 6-cyano-3-pyridazinyl, 2-nitro-3-pyridazinyl, 5-nitro-3-pyridazinyl, 6-nitro-3- pyridazinyl, 2-methansulfonyl-3-pyridazinyl, 5-methansulfonyl- 3- pyridazinyl, 6-methansulfonyl-3-pyridazinyl, 2-pyrimidyl, 4-fluor-2-pyrimidyl, 5-fluor-2-pyrimidyl, 4-chlor-2-pyrimidyl, 5-chlor-2-pyrimidyl, 4-brom-2-pyrimidyl, 5-brom-2-pyrimidyl, 4- methoxy-2-pyrimidyl, 5-methoxy-2-pyrimidyl, 4- trifluormethoxy-2-pyrimidyl, 5-trifluormethoxy-2-pyrimidyl, 4- methyl-2-pyrimidyl, 5-methyl-2-pyrimidyl, 4-trifluormethyl-2-pyrimidyl, 5-trifluormethyl-2-pyrimidyl, 4-cyano-2-pyrimidyl, 5- cyano-2-pyrimidyl, 4-nitro-2-pyrimidyl, 5-nitro-2-pyrimidyl, 4-methansulfonyl-2-pyrimidyl, 5-methansulfonyl-2-pyrimidyl, 4- pyrimidyl, 2-fluor-4-pyrimidyl, 5-fluor-4-pyrimidyl, 6-fluor-4-pyrimidyl, 2-chlor-4-pyrimidyl, 5-chlor-4-pyrimidyl, 6-chlor-4-pyrimidyl, 2-brom-4-pyrimidyl, 5-brom-4-pyrimidyl, 6-brom-4-pyrimidyl, 2-methoxy-4-pyrimidyl, 5-methoxy-4- pyrimidyl, 6-methoxy-4-pyrimidyl, 2-trifluormethoxy-4- pyrimidyl, 5-trifluormethoxy-4-pyrimidyl, 6-trifluormethoxy-4-pyrimidyl, 2-methyl-4-pyrimidyl, 5-methyl-4-pyrimidyl, 6-methyl-4-pyrimidyl, 2-trifluormethyl-4-pyrimidyl, 5- trifluormethyl-4-pyrimidyl, 6-trifluormethyl-4-pyrimidyl, 2-cyano-4-pyrimidyl, 5-cyano-4-pyrimidyl, 6-cyano-4-pyrimidyl, 2-nitro-4-pyrimidyl, 5-nitro-4-pyrimidyl, 6-nitro-4-pyrimidyl, 2-methansulfonyl-4-pyrimidyl, 5-methansulfonyl-4-pyrimidyl, 6- methansulfonyl-4-pyrimidyl, 5-pyrimidyl, 2-fluor-5-pyrimidyl, 4-fluor-5-pyrimidyl, 2-chlor-5-pyrimidyl, 4-chlor-5-pyrimidyl, 2-brom-5-pyrimidyl, 4-brom-5-pyrimidyl, 2-methoxy-5-pyrimidyl, 4- methoxy-5-pyrimidyl, 2-trifluormethoxy-5-pyrimidyl, 4- trifluormethoxy-5-pyrimidyl, 2-methyl-5-pyrimidyl, 4-methyl-5-pyrimidyl, 2-trifluormethyl-5-pyrimidyl, 4-trifluormethyl-5-pyrimidyl, 2-cyano-5-pyrimidyl, 4-cyano-5-pyrimidyl, 2-nitro- 5- pyrimidyl, 4-nitro-5-pyrimidyl, 2-methansulfonyl-5- pyrimidyl, 4-methansulfonyl-5-pyrimidyl, 2-pyrazinyl, 3-fluor- 2- pyrazinyl, 5-fluor-2-pyrazinyl, 6-fluor-2-pyrazinyl, 3-chlor-2-pyrazinyl, 5-chlor-2-pyrazinyl, 6-chlor-2-pyrazinyl, 3- brom-2-pyrazinyl, 5-brom-2-pyrazinyl, 6-brom-2-pyrazinyl, 3- methoxy-2-pyrazinyl, 5-methoxy-2-pyrazinyl, 6-methoxy-2- pyrazinyl, 3-trifluormethoxy-2-pyrazinyl, 5-trifluormethoxy-2-pyrazinyl, 6-trifluormethoxy-2-pyrazinyl, 3-methyl-2- pyrazinyl, 5-methyl-2-pyrazinyl, 6-methyl-2-pyrazinyl, 3- trifluormethyl-2-pyrazinyl, 5-trifluormethyl-2-pyrazinyl, 6- trifluormethyl-2-pyrazinyl, 3-cyano-2-pyrazinyl, 5-cyano-2- pyrazinyl, 6-cyano-2-pyrazinyl, 3-nitro-2-pyrazinyl, 5-nitro-2-pyrazinyl, 6-nitro-2-pyrazinyl, 3-methylsulfonat-2- pyrazinyl, 5-methylsulfonat-2-pyrazinyl eller 6- methylsulfonat-2-pyrazinyl; og hvor: R1, R2 og R4 er methyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er chlorid, og R3 er hydrogen; eller R1 og R2 er methyl, R4 er chlorid, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er bromid, og R3 er hydrogen; eller R1 er methyl, R2 er chlorid, R3 er hydrogen, og R4 er methoxy; eller R1 er methyl, R2 er bromid, R3 er hydrogen, og R4 er methoxy; eller R1 og R2 er methyl, R4 er ethenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er ethynyl, og R3 er hydrogen; eller R1 og R2 er methyl, R4 er ethynyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er phenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-f luorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-chlorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-trifluorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 4-f luorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 4-chlorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 4-trifluorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3,4-difluorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-f luor-4-chlorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-chlor-4-f luorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3,4-dichlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R2 og R4 er methyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er chlorid, og R3 er hydrogen; eller R1 er ethyl, R2 er methyl, R4 er chlorid, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er bromid, og R3 er hydrogen; eller R1 er ethyl, R2 er chlorid, R3 er hydrogen, og R4 er methoxy; eller R1 er ethyl, R2 er bromid, R3 er hydrogen, og R4 er methoxy; eller R1 er ethyl, R2 er methyl, R4 er ethenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er ethynyl, og R3 er hydrogen; eller R1 er ethyl, R2 er methyl, R4 er ethynyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er phenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-f luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-chlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-trif luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 4-f luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 4-chlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 4-trif luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3,4-difluorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-fluor-4-chlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-chlor-4-fluorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3,4-dichlorphenyl, og R3 er hydrogen; eller R1 og R4 er ethyl, R2 er methyl, og R3 er hydrogen.
12. Forbindelse ifølge krav 1, som er en forbindelse med strukturtype T-l:
T-1 hvor R5 er H, R6 og R7 er CH3, og R8 og R9 er H; og hvor HetAr er 2-pyridyl, 3-fluor-2-pyridyl, 4-fluor-2-pyridyl, 5-fluor-2-pyridyl, 6-fluor-2-pyridyl, 3-chlor-2-pyridyl, 4-chlor-2-pyridyl, 5-chlor-2-pyridyl, 6-chlor-2-pyridyl, 3- methyl-2-pyridyl, 4-methyl-2-pyridyl, 5-methyl-2-pyridyl, 6- methyl-2-pyridyl, 3-trifluormethyl-2-pyridyl, 4- trifluormethyl-2-pyridyl, 5-trifluormethyl-2-pyridyl, 6- trifluormethyl-2-pyridyl, 3-methoxy-2-pyridyl, 4-methoxy-2-pyridyl, 5-methoxy-2-pyridyl, 6-methoxy-2-pyridyl, 3-trifluormethoxy-2-pyridyl, 4-trifluormethoxy-2-pyridyl, 5- trifluormethoxy-2-pyridyl, 6-trifluormethoxy-2-pyridyl, 3- cyano-2-pyridyl, 4-cyano-2-pyridyl, 5-cyano-2-pyridyl, 6- cyano-2-pyridyl, 3-nitro-2-pyridyl, 4-nitro-2-pyridyl, 5- nitro-2-pyridyl, 6-nitro-2-pyridyl, 3-methansulfonyl-2- pyridyl, 4-methansulfonyl-2-pyridyl, 5-methansulfonyl-2- pyridyl, 6-methansulfonyl-2-pyridyl, 3-pyridyl, 2-fluor-3- pyridyl, 4-fluor-3-pyridyl, 5-fluor-3-pyridyl, 6-fluor-3- pyridyl, 2-chlor-3-pyridyl, 4-chlor-3-pyridyl, 5-chlor-3- pyridyl, 6-chlor-3-pyridyl, 2-brom-3-pyridyl, 4-brom-3-pyridyl, 5-brom-3-pyridyl, 6-brom-3-pyridyl, 2-methoxy-3-pyridyl, 4-methoxy-3-pyridyl, 5-methoxy-3-pyridyl, 6-methoxy- 3-pyridyl, 2-trifluormethoxy-3-pyridyl, 4-trifluormethoxy-3-pyridyl, 5-trifluormethoxy-3-pyridyl, 6-trifluormethoxy-3- pyridyl, 2-methyl-3-pyridyl, 4-methyl-3-pyridyl, 5-methyl-3-pyridyl, 6-methyl-3-pyridyl, 2-trifluormethyl-3-pyridyl, 4-trifluormethyl-3-pyridyl, 5-trifluormethyl-3-pyridyl, 6-trifluormethyl-3-pyridyl, 2-cyano-3-pyridyl, 4-cyano-3-pyridyl, 5-cyano-3-pyridyl, 6-cyano-3-pyridyl, 2-nitro-3-pyridyl, 4-nitro-3-pyridyl, 5-nitro-3-pyridyl, 6-nitro-3-pyridyl, 2-methansulfonyl-3-pyridyl, 4-methansulfonyl-3-pyridyl, 5-methansulfonyl-3-pyridyl, 6-methansulfonyl-3-pyridyl, 4-pyridyl, 2-fluor-4-pyridyl, 3-fluor-4-pyridyl, 2-chlor-4-pyridyl, 3-chlor-4-pyridyl, 2-brom-4-pyridyl, 3-brom- 4-pyridyl, 2-methoxy-4-pyridyl, 3-methoxy-4-pyridyl, 2-trifluormethoxy-4-pyridyl, 3-trifluormethoxy-4-pyridyl, 2-methyl-4-pyridyl, 3-methyl-4-pyridyl, 2-trifluormethyl-4-pyridyl, 3-trifluormethyl-4-pyridyl, 2-cyano-4-pyridyl, 3-cyano-4-pyridyl, 2-nitro-4-pyridyl, 3-nitro-4-pyridyl, 2-methansulfonyl-4-pyridyl, 3- methansulfonyl-4-pyridyl, 2-pyridazinyl, 4-fluor-2-pyridazinyl, 5-fluor-2-pyridazinyl, 6-fluor-2-pyridazinyl, 4-chlor-2-pyridazinyl, 5-chlor-2-pyridazinyl, 6-chlor-2-pyridazinyl, 4-brom-2-pyridazinyl, 5-brom-2-pyridazinyl, 6-brom-2-pyridazinyl, 4-methoxy-2-pyridazinyl, 5-methoxy-2-pyridazinyl, 6-methoxy-2-pyridazinyl, 4-trifluormethoxy-2-pyridazinyl, 5-trifluormethoxy-2-pyridazinyl, 6-trifluormethoxy-2-pyridazinyl, 4-methyl-2-pyridazinyl, 5-methyl-2-pyridazinyl, 6-methyl-2-pyridazinyl, 4-trifluormethyl-2-pyridazinyl, 5-trifluormethyl-2-pyridazinyl, 6-trifluormethyl-2-pyridazinyl, 4-cyano-2-pyridazinyl, 5-cyano-2-pyridazinyl, 6-cyano-2-pyridazinyl, 4-nitro-2-pyridazinyl, 5-nitro-2-pyridazinyl, 6-nitro-2-pyridazinyl, 4-methansulfonyl-2-pyridazinyl, 5-methansulfonyl-2-pyridazinyl, 6-methansulfonyl-2-pyridazinyl, 3-pyridazinyl, 2-fluor-3-pyridazinyl, 5-fluor-3-pyridazinyl, 6-fluor-3-pyridazinyl, 2-chlor-3-pyridazinyl, 5-chlor-3-pyridazinyl, 6-chlor-3-pyridazinyl, 2-brom-3-pyridazinyl, 5-brom-3-pyridazinyl, 6-brom-3-pyridazinyl, 2-methoxy-3-pyridazinyl, 5-methoxy-3-pyridazinyl, 6-methoxy-3-pyridazinyl, 2-trifluormethoxy-3-pyridazinyl, 5-trifluormethoxy-3-pyridazinyl, 6-trifluormethoxy-3-pyridazinyl, 2-methyl-3-pyridazinyl, 5-methyl-3-pyridazinyl, 6-methyl-3-pyridazinyl, 2- trifluormethyl-3-pyridazinyl, 5-trifluormethyl-3- pyridazinyl, 6-trifluormethyl-3-pyridazinyl, 2-cyano-3- pyridazinyl, 5-cyano-3-pyridazinyl, 6-cyano-3-pyridazinyl, 2- nitro-3-pyridazinyl, 5-nitro-3-pyridazinyl, 6-nitro-3- pyridazinyl, 2-methansulfonyl-3-pyridazinyl, 5-methansulfonyl- 3- pyridazinyl, 6-methansulfonyl-3-pyridazinyl, 2-pyrimidyl, 4-fluor-2-pyrimidyl, 5-fluor-2-pyrimidyl, 4-chlor-2-pyrimidyl, 5-chlor-2-pyrimidyl, 4-brom-2-pyrimidyl, 5-brom-2-pyrimidyl, 4- methoxy-2-pyrimidyl, 5-methoxy-2-pyrimidyl, 4- trifluormethoxy-2-pyrimidyl, 5-trifluormethoxy-2-pyrimidyl, 4- methyl-2-pyrimidyl, 5-methyl-2-pyrimidyl, 4-trifluormethyl-2-pyrimidyl, 5-trifluormethyl-2-pyrimidyl, 4-cyano-2-pyrimidyl, 5- cyano-2-pyrimidyl, 4-nitro-2-pyrimidyl, 5-nitro-2-pyrimidyl, 4-methansulfonyl-2-pyrimidyl, 5-methansulfonyl-2-pyrimidyl, 4- pyrimidyl, 2-fluor-4-pyrimidyl, 5-fluor-4-pyrimidyl, 6-fluor-4-pyrimidyl, 2-chlor-4-pyrimidyl, 5-chlor-4-pyrimidyl, 6-chlor-4-pyrimidyl, 2-brom-4-pyrimidyl, 5-brom-4-pyrimidyl, 6-brom-4-pyrimidyl, 2-methoxy-4-pyrimidyl, 5-methoxy-4- pyrimidyl, 6-methoxy-4-pyrimidyl, 2-trifluormethoxy-4- pyrimidyl, 5-trifluormethoxy-4-pyrimidyl, 6-trifluormethoxy-4-pyrimidyl, 2-methyl-4-pyrimidyl, 5-methyl-4-pyrimidyl, 6-methyl-4-pyrimidyl, 2-trifluormethyl-4-pyrimidyl, 5- trifluormethyl-4-pyrimidyl, 6-trifluormethyl-4-pyrimidyl, 2-cyano-4-pyrimidyl, 5-cyano-4-pyrimidyl, 6-cyano-4-pyrimidyl, 2-nitro-4-pyrimidyl, 5-nitro-4-pyrimidyl, 6-nitro-4-pyrimidyl, 2-methansulfonyl-4-pyrimidyl, 5-methansulfonyl-4-pyrimidyl, 6- methansulfonyl-4-pyrimidyl, 5-pyrimidyl, 2-fluor-5-pyrimidyl, 4-fluor-5-pyrimidyl, 2-chlor-5-pyrimidyl, 4-chlor-5-pyrimidyl, 2-brom-5-pyrimidyl, 4-brom-5-pyrimidyl, 2-methoxy-5-pyrimidyl, 4- methoxy-5-pyrimidyl, 2-trifluormethoxy-5-pyrimidyl, 4- trifluormethoxy-5-pyrimidyl, 2-methyl-5-pyrimidyl, 4-methyl-5-pyrimidyl, 2-trifluormethyl-5-pyrimidyl, 4-trifluormethyl-5-pyrimidyl, 2-cyano-5-pyrimidyl, 4-cyano-5-pyrimidyl, 2-nitro- 5- pyrimidyl, 4-nitro-5-pyrimidyl, 2-methansulfonyl-5- pyrimidyl, 4-methansulfonyl-5-pyrimidyl, 2-pyrazinyl, 3-fluor- 2- pyrazinyl, 5-fluor-2-pyrazinyl, 6-fluor-2-pyrazinyl, 3-chlor-2-pyrazinyl, 5-chlor-2-pyrazinyl, 6-chlor-2-pyrazinyl, 3- brom-2-pyrazinyl, 5-brom-2-pyrazinyl, 6-brom-2-pyrazinyl, 3- methoxy-2-pyrazinyl, 5-methoxy-2-pyrazinyl, 6-methoxy-2- pyrazinyl, 3-trifluormethoxy-2-pyrazinyl, 5-trifluormethoxy-2-pyrazinyl, 6-trifluormethoxy-2-pyrazinyl, 3-methyl-2- pyrazinyl, 5-methyl-2-pyrazinyl, 6-methyl-2-pyrazinyl, 3-trifluormethyl-2-pyrazinyl, 5-trifluormethyl-2-pyrazinyl, 6- trifluormethyl-2-pyrazinyl, 3-cyano-2-pyrazinyl, 5-cyano-2- pyrazinyl, 6-cyano-2-pyrazinyl, 3-nitro-2-pyrazinyl, 5-nitro-2-pyrazinyl, 6-nitro-2-pyrazinyl, 3-methylsulfonat-2- pyrazinyl, 5-methylsulfonat-2-pyrazinyl eller 6- methylsulfonat-2-pyrazinyl; og hvor: R1, R2 og R4 er methyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er chlorid, og R3 er hydrogen; eller R1 og R2 er methyl, R4 er chlorid, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er bromid, og R3 er hydrogen; eller R1 er methyl, R2 er chlorid, R3 er hydrogen, og R4 er methoxy; eller R1 er methyl, R2 er bromid, R3 er hydrogen, og R4 er methoxy; eller R1 og R2 er methyl, R4 er ethenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er ethynyl, og R3 er hydrogen; eller R1 og R2 er methyl, R4 er ethynyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er phenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-f luorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-chlorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-trifluorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 4-f luorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 4-chlorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 4-trifluorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3,4-difluorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-f luor-4-chlorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3-chlor-4-f luorphenyl, og R3 er hydrogen; eller R1 og R4 er methyl, R2 er 3,4-dichlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R2 og R4 er methyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er chlorid, og R3 er hydrogen; eller R1 er ethyl, R2 er methyl, R4 er chlorid, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er bromid, og R3 er hydrogen; eller R1 er ethyl, R2 er chlorid, R3 er hydrogen, og R4 er methoxy; eller R1 er ethyl, R2 er bromid, R3 er hydrogen, og R4 er methoxy; eller R1 er ethyl, R2 er methyl, R4 er ethenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er ethynyl, og R3 er hydrogen; eller R1 er ethyl, R2 er methyl, R4 er ethynyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er phenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-f luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-chlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-trif luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 4-f luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 4-chlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 4-trif luorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3,4-difluorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-fluor-4-chlorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3-chlor-4-fluorphenyl, og R3 er hydrogen; eller R1 er ethyl, R4 er methyl, R2 er 3,4-dichlorphenyl, og R3 er hydrogen; eller R1 og R4 er ethyl, R2 er methyl, og R3 er hydrogen.
13. Herbicidsammensætning, der foruden at omfatte formuleringsadjuvanser omfatter en herbicidt effektiv mængde af en forbindelse med formel I ifølge et hvilket som helst af kravene 1 til 8.
14. Herbicidsammensætning ifølge krav 13, der foruden at omfatte formuleringsadjuvanser omfatter en herbicidt effektiv mængde af forbindelsen med formel I, et yderligere herbicid og eventuelt en safener.
15. Herbicidsammensætning ifølge krav 13, der foruden at omfatte formuleringsadjuvanser omfatter en herbicidt effektiv mængde af forbindelsen med formel I, en safener og eventuelt et yderligere herbicid.
16. Fremgangsmåde til bekæmpelse af græsser og ukrudt i afgrøder af nytteplanter, hvilken fremgangsmåde omfatter påføring af en herbicidt effektiv mængde af en forbindelse med formel I ifølge et hvilket som helst af kravene 1 til 8 eller af en sammensætning, der omfatter en sådan forbindelse, på planterne eller voksestedet derfor.
17. Fremgangsmåde ifølge krav 16, der er en fremgangsmåde til bekæmpelse af græsser og ukrudt i afgrøder af nytteplanter, hvilken fremgangsmåde omfatter påføring af en herbicidt effektiv mængde af en sammensætning, der omfatter forbindelsen med formel I, på planterne eller på voksestedet derfor, og hvor afgrøderne af nytteplanter er hvede, byg, ris, majs, raps, sukkerroe, sukkerrør, sojabønne, bomuld, solsikke eller j ordnød.
18. Fremgangsmåde ifølge krav 17, hvor afgrøderne af nytteplanter er hvede eller byg.
19. Blanding med en forbindelse med formel I ifølge et hvilket som helst af kravene 1 til 8 i kombination med et yderligere herbicid, hvor blandingen med forbindelsen med formel I er udvalgt blandt: forbindelse med formel I + acetochlor, forbindelse med formel I + acifluorfen, forbindelse med formel I + acifluorfen-natrium, forbindelse med formel I + aclonifen, forbindelse med formel I + acrolein, forbindelse med formel I + alachlor, forbindelse med formel I + alloxydim, forbindelse med formel I + allylalkohol, forbindelse med formel I + ametryn, forbindelse med formel I + amicarbazon, forbindelse med formel I + amidosulfuron, forbindelse med formel I + aminopyralid, forbindelse med formel I + amitrol, forbindelse med formel I + ammoniumsulfamat, forbindelse med formel I + anilofos, forbindelse med formel I + asulam, forbindelse med formel I + atraton, forbindelse med formel I + atrazin, forbindelse med formel I + azimsulfuron, forbindelse med formel I + BCPC, forbindelse med formel I + beflubutamid, forbindelse med formel I + benazolin, forbindelse med formel I + benfluralin, forbindelse med formel I + benfuresat, forbindelse med formel I + bensulfuron, forbindelse med formel I + bensulfuron-methyl, forbindelse med formel I + bensulid, forbindelse med formel I + bentazon, forbindelse med formel I + benzfendizon, forbindelse med formel I + benzobicyclon, forbindelse med formel I + benzofenap, forbindelse med formel I + bifenox, forbindelse med formel I + bilanafos, forbindelse med formel I + bispyribac, forbindelse med formel I + bispyribac-natrium, forbindelse med formel I + borax, forbindelse med formel I + bromacil, forbindelse med formel I + bromobutid, forbindelse med formel I + bromoxynil, forbindelse med formel I + butachlor, forbindelse med formel I + butafenacil, forbindelse med formel I + butamifos, forbindelse med formel I + butralin, forbindelse med formel I + butroxydim, forbindelse med formel I + butylat, forbindelse med formel I + cacodylsyre, forbindelse med formel I + calciumchlorat, forbindelse med formel I + cafenstrol, forbindelse med formel I + carbetamid, forbindelse med formel I + carfentrazon, forbindelse med formel I + carfentrazon-ethyl, forbindelse med formel I + CDEA, forbindelse med formel I + CEPC, forbindelse med formel I + chlorflurenol, forbindelse med formel I + chlorflurenol-methyl, forbindelse med formel I + chloridazon, forbindelse med formel I + chlorimuron, forbindelse med formel I + chlorimuron-ethyl, forbindelse med formel I + chloreddikesyre, forbindelse med formel I + chlortoluron, forbindelse med formel I + chlorpropham, forbindelse med formel I + chlorsulfuron, forbindelse med formel I + chlorthal, forbindelse med formel I + chlorthal-dimethyl, forbindelse med formel I + cinidonethyl, forbindelse med formel I + cinmethylin, forbindelse med formel I + cinosulfuron, forbindelse med formel I + cisanilid, forbindelse med formel I + clethodim, forbindelse med formel I + clodinafop, forbindelse med formel I + clodinafop-propargyl, forbindelse med formel I + clomazon, forbindelse med formel I + clomeprop, forbindelse med formel I + clopyralid, forbindelse med formel I + cloransulam, forbindelse med formel I + cloransulam-methyl, forbindelse med formel I + CMA, forbindelse med formel I + 4-CPB, forbindelse med formel I + CPMF, forbindelse med formel I + 4-CPP, forbindelse med formel I + CPPC, forbindelse med formel I + cresol, forbindelse med formel I + cumyluron, forbindelse med formel I + cyanamid, forbindelse med formel I + cyanazin, forbindelse med formel I + cycloat, forbindelse med formel I + cyclosulfamuron, forbindelse med formel I + cycloxydim, forbindelse med formel I + cyhalofop, forbindelse med formel I + cyhalofop-butyl, forbindelse med formel I + 2.4- D, forbindelse med formel I + 3,4-DA, forbindelse med formel I + daimuron, forbindelse med formel I + dalapon, forbindelse med formel I + dazomet, forbindelse med formel I + 2.4- DB, forbindelse med formel I + 3,4-DB, forbindelse med formel I + 2,4-DEB, forbindelse med formel I + desmedipham, forbindelse med formel I + dicamba, forbindelse med formel I + dichlobenil, forbindelse med formel I + ortho-dichlorbenzen, forbindelse med formel I + para-dichlorbenzen, forbindelse med formel I + dichlorprop, forbindelse med formel I + dichlorprop-P, forbindelse med formel I + diclofop, forbindelse med formel I + diclofop-methyl, forbindelse med formel I + diclosulam, forbindelse med formel I + difenzoquat, forbindelse med formel I + difenzoquat-metilsulfat, forbindelse med formel I + diflufenican, forbindelse med formel I + diflufenzopyr, forbindelse med formel I + dimefuron, forbindelse med formel I + dimepiperat, forbindelse med formel I + dimethachlor, forbindelse med formel I + dimethametryn, forbindelse med formel I + dimethenamid, forbindelse med formel I + dimethenamid-P, forbindelse med formel I + dimethipin, forbindelse med formel I + dimethylarsinsyre, forbindelse med formel I + dinitramin, forbindelse med formel I + dinoterb, forbindelse med formel I + diphenamid, forbindelse med formel I + diquat, forbindelse med formel I + diquat-dibromid, forbindelse med formel I + dithiopyr, forbindelse med formel I + diuron, forbindelse med formel I + DNOC, forbindelse med formel I + 3,4-DP, forbindelse med formel I + DSMA, forbindelse med formel I + EBEP, forbindelse med formel I + endothal, forbindelse med formel I + EPTC, forbindelse med formel I + esprocarb, forbindelse med formel I + ethalfluralin, forbindelse med formel I + ethametsulfuron, forbindelse med formel I + ethametsulfuron-methyl, forbindelse med formel I + ethofumesat, forbindelse med formel I + ethoxyfen, forbindelse med formel I + ethoxysulfuron, forbindelse med formel I + etobenzanid, forbindelse med formel I + fenoxaprop-P, forbindelse med formel I + fenoxaprop-P-ethyl, forbindelse med formel I + fentrazamid, forbindelse med formel I + ferrosulfat, forbindelse med formel I + flamprop-M, forbindelse med formel I + flazasulfuron, forbindelse med formel I + florasulam, forbindelse med formel I + fluazifop, forbindelse med formel I + fluazifop-butyl, forbindelse med formel I + fluazifop-P, forbindelse med formel I + fluazifop-P-butyl, forbindelse med formel I + flucarbazon, forbindelse med formel I + flucarbazon-natrium, forbindelse med formel I + flucetosulfuron, forbindelse med formel I + fluchloralin, forbindelse med formel I + flufenacet, forbindelse med formel I + flufenpyr, forbindelse med formel I + flufenpyr-ethyl, forbindelse med formel I + flumetsulam, forbindelse med formel I + flumiclorac, forbindelse med formel I + flumiclorac-pentyl, forbindelse med formel I + flumioxazin, forbindelse med formel I + fluometuron, forbindelse med formel I + fluorglycofen, forbindelse med formel I + fluorglycofen-ethyl, forbindelse med formel I + flupropanat, forbindelse med formel I + flupyrsulfuron, forbindelse med formel I + flupyrsulfuron-methylnatrium, forbindelse med formel I + flurenol, forbindelse med formel I + fluridon, forbindelse med formel I + flurochloridon, forbindelse med formel I + fluroxypyr, forbindelse med formel I + flurtamon, forbindelse med formel I + fluthiacet, forbindelse med formel I + fluthiacet-methyl, forbindelse med formel I + fomesafen, forbindelse med formel I + foramsulfuron, forbindelse med formel I + fosamin, forbindelse med formel I + glufosinat, forbindelse med formel I + glufosinat-ammonium, forbindelse med formel I + glyphosat, forbindelse med formel I + halosulfuron, forbindelse med formel I + halosulfuron-methyl, forbindelse med formel I + haloxyfop, forbindelse med formel I + haloxyfop-P, forbindelse med formel I + HC-252, forbindelse med formel I + hexazinon, forbindelse med formel I + imazamethabenz, forbindelse med formel I + imazamethabenz-methyl, forbindelse med formel I + imazamox, forbindelse med formel I + imazapic, forbindelse med formel I + imazapyr, forbindelse med formel I + imazaquin, forbindelse med formel I + imazethapyr, forbindelse med formel I + imazosulfuron, forbindelse med formel I + indanofan, forbindelse med formel I + iodmethan, forbindelse med formel I + iodsulfuron, forbindelse med formel I + iodsulfuron-methylnatrium, forbindelse med formel I + ioxynil, forbindelse med formel I + isoproturon, forbindelse med formel I + isouron, forbindelse med formel I + isoxaben, forbindelse med formel I + isoxachlortol, forbindelse med formel I + isoxaflutol, forbindelse med formel I + karbutilat, forbindelse med formel I + lactofen, forbindelse med formel I + lenacil, forbindelse med formel I + linuron, forbindelse med formel I + MAA, forbindelse med formel I + MAMA, forbindelse med formel I + MCPA, forbindelse med formel I + MCPA-thioethyl, forbindelse med formel I + MCPB, forbindelse med formel I + mecoprop, forbindelse med formel I + mecoprop-P, forbindelse med formel I + mefenacet, forbindelse med formel I + mefluidid, forbindelse med formel I + mesosulfuron, forbindelse med formel I + mesosulfuron-methyl, forbindelse med formel I + mesotrion, forbindelse med formel I + metam, forbindelse med formel I + metamifop, forbindelse med formel I + metamitron, forbindelse med formel I + metazachlor, forbindelse med formel I + methabenzthiazuron, forbindelse med formel I + methylarsonsyre, forbindelse med formel I + methyldymron, forbindelse med formel I + methylisothiocyanat, forbindelse med formel I + metobenzuron, forbindelse med formel I + metolachlor, forbindelse med formel I + S-metolachlor, forbindelse med formel I + metosulam, forbindelse med formel I + metoxuron, forbindelse med formel I + metribuzin, forbindelse med formel I + metsulfuron, forbindelse med formel I + metsulfuron-methyl, forbindelse med formel I + MK-616, forbindelse med formel I + molinat, forbindelse med formel I + monolinuron, forbindelse med formel I + MSMA, forbindelse med formel I + naproanilid, forbindelse med formel I + napropamid, forbindelse med formel I + naptalam, forbindelse med formel I + neburon, forbindelse med formel I + nicosulfuron, forbindelse med formel I + nonansyre, forbindelse med formel I + norflurazon, forbindelse med formel I + oleinsyre (fedtsyrer), forbindelse med formel I + orbencarb, forbindelse med formel I + orthosulfamuron, forbindelse med formel I + oryzalin, forbindelse med formel I + oxadiargyl, forbindelse med formel I + oxadiazon, forbindelse med formel I + oxasulfuron, forbindelse med formel I + oxaziclomefon, forbindelse med formel I + oxyfluorfen, forbindelse med formel I + paraquat, forbindelse med formel I + paraquat-dichlorid, forbindelse med formel I + pebulat, forbindelse med formel I + pendimethalin, forbindelse med formel I + penoxsulam, forbindelse med formel I + pentachlorphenol, forbindelse med formel I + pentanochlor, forbindelse med formel I + pentoxazon, forbindelse med formel I + pethoxamid, forbindelse med formel I + jordolier, forbindelse med formel I + phenmedipham, forbindelse med formel I + phenmedipham-ethyl, forbindelse med formel I + picloram, forbindelse med formel I + picolinafen, forbindelse med formel I + pinoxaden, forbindelse med formel I + piperophos, forbindelse med formel I + kaliumarsenit, forbindelse med formel I + kaliumazid, forbindelse med formel I + pretilachlor, forbindelse med formel I + primisulfuron, forbindelse med formel I + primisulfuron-methyl, forbindelse med formel I + prodiamin, forbindelse med formel I + profluazol, forbindelse med formel I + profoxydim, forbindelse med formel I + prometon, forbindelse med formel I + prometryn, forbindelse med formel I + propachlor, forbindelse med formel I + propanil, forbindelse med formel I + propaquizafop, forbindelse med formel I + propazin, forbindelse med formel I + propham, forbindelse med formel I + propisochlor, forbindelse med formel I + propoxycarbazon, forbindelse med formel I + propoxycarbazon-natrium, forbindelse med formel I + propyzamid, forbindelse med formel I + prosulfocarb, forbindelse med formel I + prosulfuron, forbindelse med formel I + pyraclonil, forbindelse med formel I + pyraflufen, forbindelse med formel I + pyraflufen-ethyl, forbindelse med formel I + pyrazolynat, forbindelse med formel I + pyrazosulfuron, forbindelse med formel I + pyrazosulfuron-ethyl, forbindelse med formel I + pyrazoxyfen, forbindelse med formel I + pyribenzoxim, forbindelse med formel I + pyributicarb, forbindelse med formel I + pyridafol, forbindelse med formel I + pyridat, forbindelse med formel I + pyriftalid, forbindelse med formel I + pyriminobac, forbindelse med formel I + pyriminobac-methyl, forbindelse med formel I + pyrimisulfan, forbindelse med formel I + pyrithiobac, forbindelse med formel I + pyrithiobac-natrium, forbindelse med formel I + quinclorac, forbindelse med formel I + quinmerac, forbindelse med formel I + quinoclamin, forbindelse med formel I + quizalofop, forbindelse med formel I + quizalofop-P, forbindelse med formel I + rimsulfuron, forbindelse med formel I + sethoxydim, forbindelse med formel I + siduron, forbindelse med formel I + simazin, forbindelse med formel I + simetryn, forbindelse med formel I + SMA, forbindelse med formel I + natriumarsenit, forbindelse med formel I + natriumazid, forbindelse med formel I + natriumchlorat, forbindelse med formel I + sulcotrion, forbindelse med formel I + sulfentrazon, forbindelse med formel I + sulfometuron, forbindelse med formel I + sulfometuron-methyl, forbindelse med formel I + sulfosat, forbindelse med formel I + sulfosulfuron, forbindelse med formel I + svovlsyre, forbindelse med formel I + tjæreolier, forbindelse med formel I + 2,3,6-TBA, forbindelse med formel I + TCA, forbindelse med formel I + TCA-natrium, forbindelse med formel I + tebuthiuron, forbindelse med formel I + tepraloxydim, forbindelse med formel I + terbacil, forbindelse med formel I + terbumeton, forbindelse med formel I + terbuthylazin, forbindelse med formel I + terbutryn, forbindelse med formel I + thenylchlor, forbindelse med formel I + thiazopyr, forbindelse med formel I + thifensulfuron, forbindelse med formel I + thifensulfuron-methyl, forbindelse med formel I + thiobencarb, forbindelse med formel I + tiocarbazil, forbindelse med formel I + topramezon, forbindelse med formel I + tralkoxydim, forbindelse med formel I + triallat, forbindelse med formel I + triasulfuron, forbindelse med formel I + triaziflam, forbindelse med formel I + tribenuron, forbindelse med formel I + tribenuron-methyl, forbindelse med formel I + tricamba, forbindelse med formel I + triclopyr, forbindelse med formel I + trietazin, forbindelse med formel I + trifloxysulfuron, forbindelse med formel I + trifloxysulfuron-natrium, forbindelse med formel I + trifluralin, forbindelse med formel I + triflusulfuron, forbindelse med formel I + triflusulfuron-methyl, forbindelse med formel I + trihydroxytriazin, forbindelse med formel I + tritosulfuron, forbindelse med formel I + [3-[2-chlor-4-fluor- 5-(1-methyl-6-trifluormethyl-2,4-dioxo-l,2,3,4-tetrahydropyrimidin-3-yl)phenoxy]-2- pyridyloxy]eddikesyreethylester, forbindelse med formel 1 + 4-[(4,5-dihydro-3-methoxy-4-methyl-5-oxo)-1H-1,2,4-triazol-l-ylcarbonylsulfamoyl]-5-methy1thiophen-3-carboxylsyre, forbindelse med formel I + BAY747, som har CAS (Chemical Abstracts Service)-referencenummer 335104-84-2, forbindelse med formel I + topramezon, forbindelse med formel 1+4-hydroxy-3-[[2-[(2-methoxyethoxy)methyl]-6-(trifluormethyl)-3-pyridinyl]carbonyl]-bicyclo[3.2.1]oct-3-en-2-on og forbindelse med formel I + 4-hydroxy-3-[[2-(3-methoxypropyl)-6-(difluormethyl)-3-pyridinyl]carbonyl]-bicyclo[3.2.1]oct-3-en-2-on; og hvor blandingspartneren til forbindelsen med formel I eventuelt foreligger i form af en ester eller et salt.
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CA2746961A1 (en) 2010-06-24
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PL2375898T3 (pl) 2016-01-29
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US20120065064A1 (en) 2012-03-15
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US8889595B2 (en) 2014-11-18
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AR074735A1 (es) 2011-02-09
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