DK1981874T3 - Aminophenylderivater som nye inhibitorer af histondeacetylase - Google Patents

Aminophenylderivater som nye inhibitorer af histondeacetylase

Info

Publication number
DK1981874T3
DK1981874T3 DK07703891T DK07703891T DK1981874T3 DK 1981874 T3 DK1981874 T3 DK 1981874T3 DK 07703891 T DK07703891 T DK 07703891T DK 07703891 T DK07703891 T DK 07703891T DK 1981874 T3 DK1981874 T3 DK 1981874T3
Authority
DK
Denmark
Prior art keywords
histone deacetylase
novel inhibitors
aminophenyl derivatives
aminophenyl
derivatives
Prior art date
Application number
DK07703891T
Other languages
Danish (da)
English (en)
Inventor
Patrick Rene Angibaud
Isabelle Noelle Constance Pilatte
Bruno Roux
Janine Arts
Original Assignee
Janssen Pharmactuica N V
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmactuica N V filed Critical Janssen Pharmactuica N V
Application granted granted Critical
Publication of DK1981874T3 publication Critical patent/DK1981874T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
DK07703891T 2006-01-19 2007-01-16 Aminophenylderivater som nye inhibitorer af histondeacetylase DK1981874T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06100584 2006-01-19
PCT/EP2007/050376 WO2007082878A1 (fr) 2006-01-19 2007-01-16 Dérivés d'aminophényle en tant que nouveaux inibiteurs d'histone désacétylase

Publications (1)

Publication Number Publication Date
DK1981874T3 true DK1981874T3 (da) 2009-09-28

Family

ID=36579211

Family Applications (1)

Application Number Title Priority Date Filing Date
DK07703891T DK1981874T3 (da) 2006-01-19 2007-01-16 Aminophenylderivater som nye inhibitorer af histondeacetylase

Country Status (19)

Country Link
US (1) US8119650B2 (fr)
EP (1) EP1981874B1 (fr)
JP (1) JP5225104B2 (fr)
CN (1) CN101370804B (fr)
AT (1) ATE432272T1 (fr)
AU (1) AU2007206946B2 (fr)
CA (1) CA2631876C (fr)
CY (1) CY1109331T1 (fr)
DE (1) DE602007001190D1 (fr)
DK (1) DK1981874T3 (fr)
ES (1) ES2327972T3 (fr)
HK (1) HK1128283A1 (fr)
HR (1) HRP20090459T1 (fr)
ME (1) ME01060B (fr)
PL (1) PL1981874T3 (fr)
PT (1) PT1981874E (fr)
RS (1) RS51191B (fr)
SI (1) SI1981874T1 (fr)
WO (1) WO2007082878A1 (fr)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100519527C (zh) * 2002-03-13 2009-07-29 詹森药业有限公司 组织蛋白去乙酰酶抑制剂
AU2003209727B2 (en) 2002-03-13 2008-10-16 Janssen Pharmaceutica N.V. Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
JP4674045B2 (ja) * 2002-03-13 2011-04-20 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ヒストンデアセチラーゼの新規な阻害剤としてのピペラジニル−、ピペリジニル−およびモルホリニル−誘導体
DE60321548D1 (de) * 2002-03-13 2008-07-24 Janssen Pharmaceutica Nv Carbonylamino- derivativate als neue inhibitoren von histone deacetylase
PL1781639T3 (pl) 2004-07-28 2012-07-31 Janssen Pharmaceutica Nv Podstawione pochodne indolilo-alkiloaminowe jako nowe inhibitory deacetylazy histonowej
RS51189B (sr) * 2004-07-28 2010-10-31 Janssen Pharmaceutica N.V. Supstituisani derivati propenil piperazina kao novi inhibitori histonske deacetilaze
AU2006248938B2 (en) 2005-05-18 2011-09-29 Janssen Pharmaceutica N.V. Substituted aminopropenyl piperidine or morpholine derivatives as novel inhibitors of histone deacetylase
ATE509920T1 (de) * 2005-10-27 2011-06-15 Janssen Pharmaceutica Nv Quadratsäurederivate als inhibitoren von histondeacetylase
WO2007082878A1 (fr) 2006-01-19 2007-07-26 Janssen Pharmaceutica N.V. Dérivés d'aminophényle en tant que nouveaux inibiteurs d'histone désacétylase
EP1979327A1 (fr) 2006-01-19 2008-10-15 Janssen Pharmaceutica, N.V. Dérivés de pyridine et de pyrimidine en tant qu'inhibiteurs d'histone désacétylase
EP1979326B1 (fr) 2006-01-19 2012-10-03 Janssen Pharmaceutica N.V. Dérivés de pyridine et de pyrimidine en tant qu'inhibiteurs d'histone désacétylase
DK1979328T3 (da) * 2006-01-19 2013-03-25 Janssen Pharmaceutica Nv Pyridin- og pyrimidinderivater i deres egenskab af histondeacetylasehæmmere
US7834025B2 (en) * 2006-01-19 2010-11-16 Janssen Pharmaceutica N.V. Substituted indolyl-alkyl-amino-derivatives as inhibitors of histone deacetylase
DK2274301T3 (da) 2008-03-27 2013-01-02 Janssen Pharmaceutica Nv Azabicyclohexylsubstituerede indolylalkylaminoderivater som hidtil ukendte inhibitorer af histondeacetylase
BRPI0915720A2 (pt) * 2008-06-12 2015-08-04 Janssen Pharmaceutica Nv Moduladores de diaminopiridina, pirimidina, e piridazina do receptor de histamina h4
US9265734B2 (en) 2008-09-03 2016-02-23 Biomarin Pharmaceutical Inc. Compositions including 6-aminohexanoic acid derivatives as HDAC inhibitors
US8957066B2 (en) 2011-02-28 2015-02-17 Biomarin Pharmaceutical Inc. Histone deacetylase inhibitors
US10059723B2 (en) 2011-02-28 2018-08-28 Biomarin Pharmaceutical Inc. Histone deacetylase inhibitors
US9540395B2 (en) 2011-02-28 2017-01-10 Biomarin Pharmaceutical Inc. Histone deacetylase inhibitors
DK2683371T3 (da) 2011-03-09 2021-01-18 Cereno Scient Ab Forbindelser og fremgangsmåder til forbedring af forringet endogen fibrinolyse ved anvendelse af histondeacetylasehæmmere
AU2014228344C1 (en) 2013-03-15 2019-02-07 Biomarin Pharmaceutical Inc. HDAC inhibitors
DE102015106979B4 (de) * 2015-05-05 2023-01-12 Infineon Technologies Austria Ag Halbleiterwafer und Verfahren zum Herstellen von Halbleitervorrichtungen in einem Halbleiterwafer
WO2023044364A1 (fr) 2021-09-15 2023-03-23 Enko Chem, Inc. Inhibiteurs de protoporphyrinogène oxydase

Family Cites Families (76)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE637271A (fr) * 1963-04-04 1900-01-01
US3459731A (en) * 1966-12-16 1969-08-05 Corn Products Co Cyclodextrin polyethers and their production
US3966743A (en) * 1968-07-23 1976-06-29 Boehringer Mannheim G.M.B.H. Ortho fused cycloalkano-4-quinolone-3-carboxylic acid derivatives
US4049811A (en) * 1968-07-23 1977-09-20 Boehringer Mannheim G.M.B.H. Compositions using cycloalkano-quinolone derivatives and their method of use
GB1345872A (en) 1970-09-03 1974-02-06 Wyeth John & Brother Ltd Amino-and acylamino-pyridine and hydropyridine derivatives
DE2939292A1 (de) * 1979-09-28 1981-04-09 Boehringer Mannheim Gmbh, 6800 Mannheim N-phenoxyalkylpiperidin-derivate, verfahrenn zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
PH17194A (en) * 1980-03-06 1984-06-19 Otsuka Pharma Co Ltd Novel carbostyril derivatives,and pharmaceutical composition containing the same
CA1183847A (fr) 1981-10-01 1985-03-12 Georges Van Daele N-(3-hydroxy-4-piperidinyl)benzamide; derives
US4734418A (en) 1984-12-14 1988-03-29 Mitsui Petrochemical Industries, Ltd. Quinazoline compounds and antihypertensives
HU206337B (en) * 1988-12-29 1992-10-28 Mitsui Petrochemical Ind Process for producing pyrimidine derivatives and pharmaceutical compositions
JP2664238B2 (ja) * 1989-03-01 1997-10-15 日清製粉株式会社 ニコチン酸またはそのエステル誘導体
US5342846A (en) * 1990-12-05 1994-08-30 Synphar Laboratories, Inc. 7-substituted-6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid compounds and 7-(substituted triazolyl pyrrolidin-1-yl) 4-oxoquinoline-3-carboxylic acid derivatives useful as antibacterial agents
DE4228792A1 (de) 1992-08-29 1994-03-03 Hoechst Ag Pyridylaminopiperidine, Verfahren zu ihrer Herstellung, sie enthaltende Mittel und deren Verwendung als Fungizide
US5338738A (en) * 1993-04-19 1994-08-16 Bristol-Myers Squibb Company Cerebral function enhancers: acyclic amide derivatives of pyrimidinylpiperidines
FR2722788B1 (fr) * 1994-07-20 1996-10-04 Pf Medicament Nouvelles piperazides derivees d'aryl piperazine, leurs procedes de preparation, leur utilisation a titre de medicament et les compositions pharmaceutiques les comprenant
US6083903A (en) * 1994-10-28 2000-07-04 Leukosite, Inc. Boronic ester and acid compounds, synthesis and uses
ES2104509B1 (es) 1995-06-13 1998-07-01 Ferrer Int Nuevos compuestos derivados de 2-(3,4-disustituido-1-piperazinil)-5-fluoropirimidina.
US5952349A (en) * 1996-07-10 1999-09-14 Schering Corporation Muscarinic antagonists for treating memory loss
EP0827742A1 (fr) 1996-09-04 1998-03-11 Vrije Universiteit Brussel Utilisation des inhibiteurs de l'histone déacétylase pour le traitement de la fibrose ou de la cirrhose
EA004049B1 (ru) 1998-11-10 2003-12-25 Янссен Фармацевтика Н.В. Пиримидины, ингибирующие репликацию вич
DK1041068T3 (da) * 1999-04-01 2004-05-10 Pfizer Prod Inc Compounds for treating and preventing diabetic complications
US6518283B1 (en) * 1999-05-28 2003-02-11 Celltech R&D Limited Squaric acid derivatives
GB9918035D0 (en) * 1999-07-30 1999-09-29 Novartis Ag Organic compounds
US6608052B2 (en) * 2000-02-16 2003-08-19 Boehringer Ingelheim Pharmaceuticals, Inc. Compounds useful as anti-inflammatory agents
DE10130374A1 (de) * 2001-06-23 2003-01-02 Boehringer Ingelheim Pharma Substituierte N-Acyl-anilinderivate, deren Herstellung und deren Verwendung als Arzneimittel
US6897220B2 (en) 2001-09-14 2005-05-24 Methylgene, Inc. Inhibitors of histone deacetylase
GB0127929D0 (en) * 2001-11-21 2002-01-16 Celltech R&D Ltd Chemical compounds
GB0229931D0 (en) 2002-12-21 2003-01-29 Astrazeneca Ab Therapeutic agents
WO2003066579A2 (fr) 2002-02-07 2003-08-14 Axys Pharmaceuticals Nouveaux hydroxamates bicycliques servant d'inhibiteurs de histone desacetylase
DE60321548D1 (de) * 2002-03-13 2008-07-24 Janssen Pharmaceutica Nv Carbonylamino- derivativate als neue inhibitoren von histone deacetylase
EP1485378B1 (fr) 2002-03-13 2008-06-18 Janssen Pharmaceutica N.V. Derives piperazinyl-, piperidinyl- et morpholinyl- utilises en tant que nouveaux inhibiteurs d'histone deacetylase
CN100519527C (zh) 2002-03-13 2009-07-29 詹森药业有限公司 组织蛋白去乙酰酶抑制剂
JP4674045B2 (ja) * 2002-03-13 2011-04-20 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ヒストンデアセチラーゼの新規な阻害剤としてのピペラジニル−、ピペリジニル−およびモルホリニル−誘導体
AU2003209727B2 (en) 2002-03-13 2008-10-16 Janssen Pharmaceutica N.V. Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
BR0307575A (pt) * 2002-03-13 2004-12-21 Janssen Pharmaceutica Nv Derivados de sulfonila como inibidores de histona desacetilase
US6897307B2 (en) * 2002-03-28 2005-05-24 Novartis Ag Process for preparing 2,6-diaminopurine derivatives
NZ536116A (en) 2002-04-03 2007-01-26 Topotarget Uk Ltd Carbamic acid compounds comprising a piperazine linkage as HDAC inhibitors
TWI319387B (en) 2002-04-05 2010-01-11 Astrazeneca Ab Benzamide derivatives
GB0209715D0 (en) 2002-04-27 2002-06-05 Astrazeneca Ab Chemical compounds
DE10233412A1 (de) 2002-07-23 2004-02-12 4Sc Ag Neue Verbindungen als Histondeacetylase-Inhibitoren
PL374970A1 (en) 2002-08-02 2005-11-14 Argenta Discovery Limited Substituted thienyl-hydroxamic acids as histone deacetylase inhibitors
ITMI20030025A1 (it) 2003-01-10 2004-07-11 Italfarmaco Spa Derivati dell'acido idrossammico ad attivita' antinfiammatoria.
TW200418806A (en) 2003-01-13 2004-10-01 Fujisawa Pharmaceutical Co HDAC inhibitor
JP4612621B2 (ja) 2003-01-17 2011-01-12 トポターゲット ユーケー リミテッド Hdac阻害剤としてのエステル又はケトン結合を含むカルバミン酸化合物
TW200424174A (en) 2003-02-06 2004-11-16 Hoffmann La Roche New TP diamide
AU2003900608A0 (en) 2003-02-11 2003-02-27 Fujisawa Pharmaceutical Co., Ltd. Hdac inhibitor
US7244751B2 (en) 2003-02-14 2007-07-17 Shenzhen Chipscreen Biosciences Ltd. Histone deacetylase inhibitors of novel benzamide derivatives with potent differentiation and anti-proliferation activity
US7375228B2 (en) 2003-03-17 2008-05-20 Takeda San Diego, Inc. Histone deacetylase inhibitors
TW200424187A (en) 2003-04-04 2004-11-16 Hoffmann La Roche New oxime derivatives and their use as pharmaceutically active agents
NZ542445A (en) 2003-04-07 2008-03-28 Pharmacyclics Inc Hydroxamates as therapeutic agents
ATE553092T1 (de) 2003-07-30 2012-04-15 Kyowa Hakko Kirin Co Ltd Indazolderivate
KR101127201B1 (ko) 2003-09-22 2012-04-12 에스*바이오 피티이 리미티드 벤즈이미다졸 유도체와 그의 제조방법 및 약학적 적용
PL1673349T3 (pl) 2003-09-22 2010-11-30 Mei Pharma Inc Pochodne benzimidazolu: wytwarzanie i zastosowania farmaceutyczne
WO2005030704A1 (fr) 2003-09-24 2005-04-07 Methylgene, Inc. Inhibiteurs d'histone deacetylase
MXPA06004735A (es) 2003-10-27 2006-12-14 S Bio Pte Ltd Hidroxamatos conectados a acilurea y a sulfonilurea.
US20070167499A1 (en) 2003-10-27 2007-07-19 A*Bio Pte Ltd. Biaryl linked hydroxamates: preparation and pharmaceutical applications
GB0402496D0 (en) 2004-02-04 2004-03-10 Argenta Discovery Ltd Novel compounds
US20050197336A1 (en) * 2004-03-08 2005-09-08 Miikana Therapeutics Corporation Inhibitors of histone deacetylase
WO2005092899A1 (fr) 2004-03-26 2005-10-06 Methylgene Inc. Inhibiteurs d'histone désacétylase
RS51189B (sr) * 2004-07-28 2010-10-31 Janssen Pharmaceutica N.V. Supstituisani derivati propenil piperazina kao novi inhibitori histonske deacetilaze
PL1781639T3 (pl) 2004-07-28 2012-07-31 Janssen Pharmaceutica Nv Podstawione pochodne indolilo-alkiloaminowe jako nowe inhibitory deacetylazy histonowej
WO2006010749A2 (fr) 2004-07-28 2006-02-02 Janssen Pharmaceutica N.V. Derives de piperazine de propenyle substituee comme nouveaux inhibiteurs de l'histone deacetylase
AU2006248938B2 (en) 2005-05-18 2011-09-29 Janssen Pharmaceutica N.V. Substituted aminopropenyl piperidine or morpholine derivatives as novel inhibitors of histone deacetylase
WO2006136553A1 (fr) 2005-06-23 2006-12-28 Janssen Pharmaceutica N.V. Dérivés d'imidazolinone et d'hydantoïne en tant que nouveaux inhibiteurs de l’histone désacétylase
JP5345388B2 (ja) * 2005-06-30 2013-11-20 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 環式アニリノ−ピリジノトリアジン
WO2007016532A2 (fr) 2005-08-02 2007-02-08 Novartis Ag Mutations et polymorphismes de hdac4
ATE509920T1 (de) * 2005-10-27 2011-06-15 Janssen Pharmaceutica Nv Quadratsäurederivate als inhibitoren von histondeacetylase
WO2007082878A1 (fr) 2006-01-19 2007-07-26 Janssen Pharmaceutica N.V. Dérivés d'aminophényle en tant que nouveaux inibiteurs d'histone désacétylase
EP1979326B1 (fr) * 2006-01-19 2012-10-03 Janssen Pharmaceutica N.V. Dérivés de pyridine et de pyrimidine en tant qu'inhibiteurs d'histone désacétylase
DK1979328T3 (da) * 2006-01-19 2013-03-25 Janssen Pharmaceutica Nv Pyridin- og pyrimidinderivater i deres egenskab af histondeacetylasehæmmere
EP1981871B1 (fr) 2006-01-19 2011-12-28 Janssen Pharmaceutica N.V. Dérivés d'hétérocyclylalkyle en tant que nouveaux inhibiteurs d'histone désacétylase
EP1979327A1 (fr) * 2006-01-19 2008-10-15 Janssen Pharmaceutica, N.V. Dérivés de pyridine et de pyrimidine en tant qu'inhibiteurs d'histone désacétylase
US7834025B2 (en) * 2006-01-19 2010-11-16 Janssen Pharmaceutica N.V. Substituted indolyl-alkyl-amino-derivatives as inhibitors of histone deacetylase
AU2007296259A1 (en) * 2006-09-15 2008-03-20 Janssen Pharmaceutica Nv Combinations of class-I specific histone deacetylase inhibitors with proteasome inhibitors
EP2234883B1 (fr) * 2007-12-14 2017-08-02 Urban Aeronautics Ltd. Véhicule vtol et procédé de fonctionnement
GB0901749D0 (en) 2009-02-03 2009-03-11 Oxford Nanopore Tech Ltd Adaptor method

Also Published As

Publication number Publication date
JP2009523760A (ja) 2009-06-25
PL1981874T3 (pl) 2009-10-30
EP1981874B1 (fr) 2009-05-27
CN101370804B (zh) 2013-05-29
JP5225104B2 (ja) 2013-07-03
SI1981874T1 (sl) 2009-10-31
EP1981874A1 (fr) 2008-10-22
ME01060B (me) 2012-10-20
PT1981874E (pt) 2009-09-02
CA2631876A1 (fr) 2007-07-26
US20090018152A1 (en) 2009-01-15
CN101370804A (zh) 2009-02-18
AU2007206946B2 (en) 2011-12-15
RS51191B (sr) 2010-10-31
CY1109331T1 (el) 2014-07-02
WO2007082878A1 (fr) 2007-07-26
US8119650B2 (en) 2012-02-21
ES2327972T3 (es) 2009-11-05
ATE432272T1 (de) 2009-06-15
CA2631876C (fr) 2014-05-27
DE602007001190D1 (de) 2009-07-09
HRP20090459T1 (hr) 2009-09-30
HK1128283A1 (en) 2009-10-23
AU2007206946A1 (en) 2007-07-26

Similar Documents

Publication Publication Date Title
DK1981874T3 (da) Aminophenylderivater som nye inhibitorer af histondeacetylase
DK1981871T3 (da) Heterocyclylalkylderivater som hidtil ukendte inhibitorer af histondeacetylase
DK1899325T3 (da) Imidazolinon- og hydantoinderivater som hidtil ukendte hæmmere af histondeacetylase
ECSP20027480A (es) Indolil alquil amino derivados sustituidos como nuevos inhibidores de la histona desacetilasa
DK1943232T3 (da) Kvadratsyrederivater som inhibitorer af histondeacetylase
DK2134691T3 (da) Quinolinonderivativer som parp- og tank-inhibitorer
TW200616998A (en) Substituted propenyl piperazine derivatives as novel inhibitors of histone deacetylase
UA86066C2 (ru) Производные замещенного пропенилпиперазина как ингибиторы гистондеацетилазы
TW200740761A (en) Histone deacetylase inhibitors
PL370991A1 (en) New inhibitors of histone deacetylase
MXPA04008796A (es) Derivados de carbonilamino como novedosos inhibidores de desacetilasa de histona.
PL370990A1 (en) Sulfonyl-derivatives as novel inhibitors of histone deacetylase
PL371036A1 (en) Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase
MXPA04007776A (es) Derivados de sulfonilamino como nuevos inhibidores de histona deacetilasa.
IL185275A0 (en) N-sulphonylpyrrole derivatives and pharmaceutical compositions containing the same
ATE547415T1 (de) Inhibitoren der wechselwirkung zwischen mdm2 und p53
EA201101334A1 (ru) Новые соединения бензотиадиазепина, способ их приготовления и фармацевтические композиции, содержащие их
ATE500222T1 (de) Benzamid- und heteroarenderivate als cetp- inhibitoren
ATE542812T1 (de) Substituierte indolylalkylaminoderivate als neue inhibitoren von histondeacetylase