DK1802620T3 - Fremgangsmåde til enantioselektiv fremstilling af sulfoxidderivater - Google Patents
Fremgangsmåde til enantioselektiv fremstilling af sulfoxidderivaterInfo
- Publication number
- DK1802620T3 DK1802620T3 DK05804208T DK05804208T DK1802620T3 DK 1802620 T3 DK1802620 T3 DK 1802620T3 DK 05804208 T DK05804208 T DK 05804208T DK 05804208 T DK05804208 T DK 05804208T DK 1802620 T3 DK1802620 T3 DK 1802620T3
- Authority
- DK
- Denmark
- Prior art keywords
- enantioselective
- useful
- pyridinyl ring
- enantioselective preparation
- sulfoxide derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C07C315/02—Preparation of sulfones; Preparation of sulfoxides by formation of sulfone or sulfoxide groups by oxidation of sulfides, or by formation of sulfone groups by oxidation of sulfoxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/32—Sulfur atoms
- C07D213/34—Sulfur atoms to which a second hetero atom is attached
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nutrition Science (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Catalysts (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0410483A FR2876101B1 (fr) | 2004-10-05 | 2004-10-05 | Procede de preparation enantioselective de derives de sulfoxydes |
| PCT/FR2005/002447 WO2006037894A1 (fr) | 2004-10-05 | 2005-10-05 | Procede de preparation enantioselective de derives de sulfoxydes. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1802620T3 true DK1802620T3 (da) | 2009-04-06 |
Family
ID=34949706
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK05804208T DK1802620T3 (da) | 2004-10-05 | 2005-10-05 | Fremgangsmåde til enantioselektiv fremstilling af sulfoxidderivater |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US7528251B2 (da) |
| EP (1) | EP1802620B1 (da) |
| JP (1) | JP5213444B2 (da) |
| KR (1) | KR101258744B1 (da) |
| CN (1) | CN101035787B (da) |
| AT (1) | ATE417848T1 (da) |
| AU (1) | AU2005291156B2 (da) |
| BR (1) | BRPI0516465A (da) |
| CA (1) | CA2580446C (da) |
| DE (1) | DE602005011840D1 (da) |
| DK (1) | DK1802620T3 (da) |
| ES (1) | ES2319804T3 (da) |
| FR (1) | FR2876101B1 (da) |
| IL (1) | IL181831A (da) |
| MX (1) | MX2007003953A (da) |
| NO (1) | NO20071524L (da) |
| NZ (1) | NZ553841A (da) |
| PL (1) | PL1802620T3 (da) |
| RU (1) | RU2380357C2 (da) |
| WO (1) | WO2006037894A1 (da) |
| ZA (1) | ZA200702273B (da) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101012141B (zh) * | 2007-02-02 | 2012-05-23 | 沈阳药科大学 | 手性亚砜类化合物的制备方法 |
| FR2925899B1 (fr) * | 2007-12-27 | 2012-12-21 | Sidem Pharma Sa | Procede de preparation enantioselective de sulfoxydes. |
| MX2012000583A (es) | 2009-07-16 | 2012-02-13 | Bayer Cropscience Ag | Procedimiento para la preparacion de derivados de 3-triazolil-sulfoxido quirales. |
| RU2448954C1 (ru) * | 2010-10-18 | 2012-04-27 | Учреждение Российской академии наук Институт катализа им. Г.К. Борескова Сибирского отделения РАН | Способ получения сульфоксидов |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE504459C2 (sv) * | 1994-07-15 | 1997-02-17 | Astra Ab | Förfarande för framställning av substituerade sulfoxider |
| AR030284A1 (es) | 2000-06-08 | 2003-08-20 | Merck & Co Inc | Proceso para la sintesis de (2r, 2-alfa-r,3a) -2-[1-(3,5-bis(trifluorometil) fenil) etoxi]-3-(4-fluorofenil)-1,4-oxazina; dicho compuesto y sus formas polimorficas |
| WO2003089408A2 (en) * | 2002-04-22 | 2003-10-30 | Sun Pharmaceutical Industries Limited | Optically active substituted pyridinylmethyl-sulphinyl-benzimidazole and salts |
| CN1453278A (zh) * | 2002-04-23 | 2003-11-05 | 中国人民解放军军事医学科学院放射医学研究所 | 一种拉唑类化合物及其制备方法与应用 |
| FR2848555B1 (fr) * | 2002-12-16 | 2006-07-28 | Negma Gild | Enantiomere(-)du tenatoprazole et son application en therapeutique |
| KR20130066701A (ko) * | 2003-02-24 | 2013-06-20 | 미쓰비시 타나베 파마 코퍼레이션 | 테나토프라졸의 거울상 이성질체 및 치료를 위한 그 용도 |
-
2004
- 2004-10-05 FR FR0410483A patent/FR2876101B1/fr not_active Expired - Fee Related
-
2005
- 2005-10-05 MX MX2007003953A patent/MX2007003953A/es active IP Right Grant
- 2005-10-05 DK DK05804208T patent/DK1802620T3/da active
- 2005-10-05 KR KR1020077008091A patent/KR101258744B1/ko not_active IP Right Cessation
- 2005-10-05 WO PCT/FR2005/002447 patent/WO2006037894A1/fr active Application Filing
- 2005-10-05 PL PL05804208T patent/PL1802620T3/pl unknown
- 2005-10-05 NZ NZ553841A patent/NZ553841A/en not_active IP Right Cessation
- 2005-10-05 BR BRPI0516465-6A patent/BRPI0516465A/pt not_active IP Right Cessation
- 2005-10-05 EP EP05804208A patent/EP1802620B1/fr not_active Not-in-force
- 2005-10-05 AT AT05804208T patent/ATE417848T1/de active
- 2005-10-05 CA CA2580446A patent/CA2580446C/fr not_active Expired - Fee Related
- 2005-10-05 AU AU2005291156A patent/AU2005291156B2/en not_active Ceased
- 2005-10-05 JP JP2007535193A patent/JP5213444B2/ja not_active Expired - Fee Related
- 2005-10-05 ES ES05804208T patent/ES2319804T3/es active Active
- 2005-10-05 US US11/663,647 patent/US7528251B2/en not_active Expired - Fee Related
- 2005-10-05 CN CN2005800338604A patent/CN101035787B/zh not_active Expired - Fee Related
- 2005-10-05 DE DE602005011840T patent/DE602005011840D1/de active Active
- 2005-10-05 RU RU2007116816/04A patent/RU2380357C2/ru not_active IP Right Cessation
-
2007
- 2007-03-08 IL IL181831A patent/IL181831A/en not_active IP Right Cessation
- 2007-03-19 ZA ZA200702273A patent/ZA200702273B/en unknown
- 2007-03-23 NO NO20071524A patent/NO20071524L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| IL181831A (en) | 2011-04-28 |
| JP5213444B2 (ja) | 2013-06-19 |
| RU2380357C2 (ru) | 2010-01-27 |
| US7528251B2 (en) | 2009-05-05 |
| ES2319804T3 (es) | 2009-05-12 |
| IL181831A0 (en) | 2007-07-04 |
| NO20071524L (no) | 2007-04-27 |
| MX2007003953A (es) | 2007-06-14 |
| WO2006037894A1 (fr) | 2006-04-13 |
| CN101035787A (zh) | 2007-09-12 |
| NZ553841A (en) | 2010-09-30 |
| CA2580446C (fr) | 2013-05-21 |
| AU2005291156A1 (en) | 2006-04-13 |
| ATE417848T1 (de) | 2009-01-15 |
| EP1802620A1 (fr) | 2007-07-04 |
| CA2580446A1 (fr) | 2006-04-13 |
| FR2876101B1 (fr) | 2007-03-02 |
| ZA200702273B (en) | 2008-06-25 |
| CN101035787B (zh) | 2013-03-27 |
| JP2008515860A (ja) | 2008-05-15 |
| BRPI0516465A (pt) | 2008-09-09 |
| US20070299261A1 (en) | 2007-12-27 |
| AU2005291156B2 (en) | 2011-12-22 |
| FR2876101A1 (fr) | 2006-04-07 |
| RU2007116816A (ru) | 2008-11-20 |
| DE602005011840D1 (de) | 2009-01-29 |
| EP1802620B1 (fr) | 2008-12-17 |
| PL1802620T3 (pl) | 2009-07-31 |
| KR20070102660A (ko) | 2007-10-19 |
| KR101258744B1 (ko) | 2013-04-29 |
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