DK174995B1 - Substitueret 3-propenylcephem-derivat, fremgangsmåde til fremstilling deraf, farmaceutisk præparat indeholdende en sådan forbindelse og anvendelse af en sådan forbindelse til fremstilling af et præparat til behandling af sygdomme forårsaget af bakterier - Google Patents

Substitueret 3-propenylcephem-derivat, fremgangsmåde til fremstilling deraf, farmaceutisk præparat indeholdende en sådan forbindelse og anvendelse af en sådan forbindelse til fremstilling af et præparat til behandling af sygdomme forårsaget af bakterier Download PDF

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Publication number
DK174995B1
DK174995B1 DK198705313A DK531387A DK174995B1 DK 174995 B1 DK174995 B1 DK 174995B1 DK 198705313 A DK198705313 A DK 198705313A DK 531387 A DK531387 A DK 531387A DK 174995 B1 DK174995 B1 DK 174995B1
Authority
DK
Denmark
Prior art keywords
alkyl
substituted lower
salts
compound
amino
Prior art date
Application number
DK198705313A
Other languages
Danish (da)
English (en)
Other versions
DK531387A (da
DK531387D0 (da
Inventor
Hiroshi Yamauchi
Isao Sugiyama
Seiichiro Nomoto
Takashi Kamiya
Yoshimasa Machida
Shigeto Negi
Takaharu Nakamura
Yuuki Komatu
Yasunobu Kai
Toshihiko Naito
Kyosuke Kitoh
Kanemasa Katsu
Original Assignee
Eisai Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai Co Ltd filed Critical Eisai Co Ltd
Publication of DK531387D0 publication Critical patent/DK531387D0/da
Publication of DK531387A publication Critical patent/DK531387A/da
Application granted granted Critical
Publication of DK174995B1 publication Critical patent/DK174995B1/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK198705313A 1986-10-13 1987-10-12 Substitueret 3-propenylcephem-derivat, fremgangsmåde til fremstilling deraf, farmaceutisk præparat indeholdende en sådan forbindelse og anvendelse af en sådan forbindelse til fremstilling af et præparat til behandling af sygdomme forårsaget af bakterier DK174995B1 (da)

Applications Claiming Priority (12)

Application Number Priority Date Filing Date Title
JP24148086 1986-10-13
JP24148086 1986-10-13
JP26279986 1986-11-06
JP26279986 1986-11-06
JP29257486 1986-12-10
JP29257486 1986-12-10
JP2186687 1987-02-03
JP2186687 1987-02-03
JP21923087 1987-09-03
JP21923087 1987-09-03
JP22214787 1987-09-07
JP22214787 1987-09-07

Publications (3)

Publication Number Publication Date
DK531387D0 DK531387D0 (da) 1987-10-12
DK531387A DK531387A (da) 1988-04-14
DK174995B1 true DK174995B1 (da) 2004-04-13

Family

ID=27549011

Family Applications (1)

Application Number Title Priority Date Filing Date
DK198705313A DK174995B1 (da) 1986-10-13 1987-10-12 Substitueret 3-propenylcephem-derivat, fremgangsmåde til fremstilling deraf, farmaceutisk præparat indeholdende en sådan forbindelse og anvendelse af en sådan forbindelse til fremstilling af et præparat til behandling af sygdomme forårsaget af bakterier

Country Status (14)

Country Link
US (4) US4921850A (fr)
EP (1) EP0264091B1 (fr)
CN (1) CN1020104C (fr)
CA (1) CA1290748C (fr)
DE (1) DE3776620D1 (fr)
DK (1) DK174995B1 (fr)
ES (1) ES2039223T3 (fr)
FI (1) FI89169C (fr)
GR (1) GR3003841T3 (fr)
HU (1) HU207088B (fr)
IL (1) IL84128A (fr)
NO (1) NO170021C (fr)
NZ (1) NZ222116A (fr)
PT (1) PT85906B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5373000A (en) * 1985-12-26 1994-12-13 Eisai Co., Ltd. 7Beta-(thiadiazolyl)-2-iminoacetamido-3cephem compounds
CA1339738C (fr) * 1988-03-16 1998-03-17 Takashi Kamiya Methode de preparation de derives de cephemes; produits intermediaires utiles a cette fin
CS273349B2 (en) * 1988-03-31 1991-03-12 Hoffmann La Roche Method of cephalosporin's new derivatives production
DK0421297T3 (da) * 1989-09-30 1994-01-17 Eisai Co Ltd Injicerbare præparater indeholdende cephalosporin som lægemiddel og anvendelse deraf
FR2663332B1 (fr) * 1990-06-15 1997-11-07 Roussel Uclaf Nouvelles cephalosporines comportant en position 3 un radical propenyle substitue par un ammonium quaternaire, leur procede de preparation, leur application comme medicaments, les compositions les renfermant et les nouveaux intermediaires obtenus.
US5126336A (en) * 1990-08-23 1992-06-30 Bristol-Myers Squibb Company Antibiotic c-3 catechol-substituted cephalosporin compounds, compositions and method of use thereof
AT396108B (de) * 1991-08-21 1993-06-25 Biochemie Gmbh Neues verfahren und neue zwischenprodukte zur herstellung von 7-aminocephalosporansaeurederivaten
US5523400A (en) * 1993-04-16 1996-06-04 Hoffmann-La Roche Inc. Cephalosporin antibiotics
JPH07173168A (ja) * 1993-07-14 1995-07-11 Sumitomo Chem Co Ltd セフェム系化合物、その製法、およびそれのセフェム系抗生物質製造への利用
US6265394B1 (en) 1997-07-31 2001-07-24 Bristol-Myers Squibb Company Bis quaternary MRSA cephem derivatives
US7160537B2 (en) * 2003-12-15 2007-01-09 Siemens Medical Solutions Usa, Inc. Method for preparing radiolabeled thymidine having low chromophoric byproducts
JP2011514364A (ja) * 2008-03-21 2011-05-06 クロリオン ファーマ，インコーポレーテッド 置換されたピロリジン及びピペリジン化合物、その誘導体、並びに疼痛を治療するための方法
CN114315872A (zh) * 2021-12-25 2022-04-12 海南海灵化学制药有限公司 一种盐酸头孢唑兰中间体的制备方法

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE439312B (sv) * 1977-03-25 1985-06-10 Roussel Uclaf Sett att framstella nya oximderivat av 3-acetoximetyl-7-aminotiazolylacetamido cefalosporansyra
FR2494280A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouveaux derives de la cephalosporine et leur preparation
US4408515A (en) * 1981-07-13 1983-10-11 Sciuto Michael N Stringed instrument conversion kit employing combined bridge/tuning mechanism
US4406899A (en) * 1982-03-04 1983-09-27 Bristol-Myers Company Cephalosporins
US4457929A (en) * 1982-03-29 1984-07-03 Bristol-Myers Company 3-Quaternary ammonium methyl)-substituted cephalosporin derivatives
DE3247613A1 (de) * 1982-12-23 1984-07-05 Hoechst Ag, 6230 Frankfurt Cephalosporinderivate und verfahren zu ihrer herstellung
US4486586A (en) * 1983-02-10 1984-12-04 Bristol-Myers Company Cephalosporin derivatives
US4525473A (en) * 1983-03-30 1985-06-25 Bristol-Myers Company Cephalosporins
ZA847825B (en) * 1983-10-08 1985-05-29 Hoechst Ag Caphalosporin derivatives and processes for their preparations
GB8406231D0 (en) * 1984-03-09 1984-04-11 Fujisawa Pharmaceutical Co Cephem compounds
JPS60197693A (ja) * 1984-03-19 1985-10-07 Eisai Co Ltd ３−（キヌクリジニウム）メチル−３−セフエム誘導体
JPS60197692A (ja) * 1984-03-19 1985-10-07 Eisai Co Ltd ７−アミノチアゾリルアセトアミドセフエム誘導体
US4751295A (en) * 1984-04-09 1988-06-14 Bristol-Myers Company Cephalosporin derivatives
CA1276929C (fr) * 1984-04-09 1990-11-27 Masahisa Oka Agents antibacteriens de cephalosporine
DK500285A (da) * 1984-11-02 1986-05-03 Glaxo Group Ltd Cephalosporinantibiotika
US4761410A (en) * 1985-01-14 1988-08-02 Fujisawa Pharmaceutical Co., Ltd. Cephem Compounds
GB2177691A (en) * 1985-07-18 1987-01-28 Glaxo Group Ltd Cephalosporin antibiotics

Also Published As

Publication number Publication date
HUT47119A (en) 1989-01-30
CN87107610A (zh) 1988-06-01
NO874255D0 (no) 1987-10-12
US5006649A (en) 1991-04-09
NO874255L (no) 1988-04-14
NZ222116A (en) 1990-08-28
EP0264091A2 (fr) 1988-04-20
US5066812A (en) 1991-11-19
HU207088B (en) 1993-03-01
DK531387A (da) 1988-04-14
FI89169C (fi) 1993-08-25
PT85906B (pt) 1990-08-31
NO170021C (no) 1992-09-02
DK531387D0 (da) 1987-10-12
PT85906A (en) 1987-11-01
US5089491A (en) 1992-02-18
FI874492A (fi) 1988-04-14
FI89169B (fi) 1993-05-14
CN1020104C (zh) 1993-03-17
CA1290748C (fr) 1991-10-15
ES2039223T3 (es) 1993-09-16
IL84128A0 (en) 1988-03-31
US4921850A (en) 1990-05-01
EP0264091B1 (fr) 1992-02-05
DE3776620D1 (de) 1992-03-19
EP0264091A3 (en) 1989-12-27
IL84128A (en) 1992-12-01
GR3003841T3 (fr) 1993-03-16
NO170021B (no) 1992-05-25
FI874492A0 (fi) 1987-10-12

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