DK172664B1 - Benzodiazepiner, mellemprodukter til deres fremstilling, medicinsk produkt indeholdende benzodiazepinerne samt deres anvend - Google Patents

Benzodiazepiner, mellemprodukter til deres fremstilling, medicinsk produkt indeholdende benzodiazepinerne samt deres anvend Download PDF

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Publication number
DK172664B1
DK172664B1 DK198901972A DK197289A DK172664B1 DK 172664 B1 DK172664 B1 DK 172664B1 DK 198901972 A DK198901972 A DK 198901972A DK 197289 A DK197289 A DK 197289A DK 172664 B1 DK172664 B1 DK 172664B1
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DK
Denmark
Prior art keywords
ppm
formula
proton
protons
phenyl
Prior art date
Application number
DK198901972A
Other languages
Danish (da)
English (en)
Other versions
DK197289D0 (da
DK197289A (da
Inventor
Jean-Louis Junien
Xavier Bernard Pascaud
Alain Pierre Calvet
Francois Joseph Roman
Yves Robert Pascal
Original Assignee
Jouveinal Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jouveinal Sa filed Critical Jouveinal Sa
Publication of DK197289D0 publication Critical patent/DK197289D0/da
Publication of DK197289A publication Critical patent/DK197289A/da
Application granted granted Critical
Publication of DK172664B1 publication Critical patent/DK172664B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Indole Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK198901972A 1988-04-25 1989-04-24 Benzodiazepiner, mellemprodukter til deres fremstilling, medicinsk produkt indeholdende benzodiazepinerne samt deres anvend DK172664B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8805443 1988-04-25
FR8805443A FR2630440B1 (fr) 1988-04-25 1988-04-25 Benzodiazepines, leur procede et intermediaires de preparation et leurs applications en therapeutique

Publications (3)

Publication Number Publication Date
DK197289D0 DK197289D0 (da) 1989-04-24
DK197289A DK197289A (da) 1989-10-26
DK172664B1 true DK172664B1 (da) 1999-05-10

Family

ID=9365634

Family Applications (1)

Application Number Title Priority Date Filing Date
DK198901972A DK172664B1 (da) 1988-04-25 1989-04-24 Benzodiazepiner, mellemprodukter til deres fremstilling, medicinsk produkt indeholdende benzodiazepinerne samt deres anvend

Country Status (19)

Country Link
US (1) US4929614A (pt)
EP (1) EP0340064B1 (pt)
JP (1) JP2805634B2 (pt)
KR (1) KR0142328B1 (pt)
AT (1) ATE86995T1 (pt)
AU (1) AU618086B2 (pt)
CA (1) CA1340074C (pt)
DE (1) DE68905365T2 (pt)
DK (1) DK172664B1 (pt)
ES (1) ES2054045T3 (pt)
FI (1) FI91409C (pt)
FR (1) FR2630440B1 (pt)
HK (1) HK95496A (pt)
IE (1) IE62663B1 (pt)
IS (1) IS3454A7 (pt)
NO (1) NO169653C (pt)
NZ (1) NZ228650A (pt)
PT (1) PT90339B (pt)
ZA (1) ZA892682B (pt)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5248679A (en) * 1988-09-09 1993-09-28 Fujisawa Pharmaceutical Co., Ltd. Tricyclic compounds
IL91361A (en) * 1988-09-09 1994-10-07 Fujisawa Pharmaceutical Co Benzodiazepinone compounds [4,1] connected via positions 1 and 9 and carrying two transducers, processes for their preparation and pharmaceutical preparations containing them
PH26955A (en) * 1989-03-08 1992-12-03 Kali Chemie Pharma Gmbh Novel 1,7-fused 1H-indole-2-carboxylic acid N-(1,4-benzodiazepin-3-YL) amides
FR2652352A1 (fr) * 1989-09-28 1991-03-29 Jouveinal Sa Benzodiazepines, leur procede et intermediaires de preparation et leurs applications en therapeutique.
CA2032427A1 (en) * 1989-12-18 1991-06-19 Mark G. Bock Benzodiazepines analogs
GB9018601D0 (en) * 1990-08-24 1990-10-10 Fujisawa Pharmaceutical Co Tricyclic compounds
US5206238A (en) * 1990-11-13 1993-04-27 Merck & Co., Inc. Cholecystokinin antagonists
CA2056809A1 (en) * 1990-12-07 1992-06-08 Mark G. Bock Benzodiazepine analogs
AU6045994A (en) * 1993-03-03 1994-09-26 Fujisawa Pharmaceutical Co., Ltd. Optical isomerization inhibitor
ZA957201B (en) * 1994-08-30 1996-04-01 Fujisawa Pharmaceutical Co Liposome preparation
FR2725719B1 (fr) * 1994-10-14 1996-12-06 Jouveinal Inst Rech Diazepino-indoles inhibiteurs de phosphodiesterases iv
FR2776660B1 (fr) * 1998-03-27 2000-05-12 Parke Davis Diazepino-indoles de phosphodiesterases iv
HRP990246A2 (en) * 1998-08-07 2000-06-30 Du Pont Pharm Co Succinoylamino benzodiazepines as inhibitors of a beta protein production
NZ509241A (en) 1998-08-07 2003-08-29 Du Pont Pharm Co Succinoylamino lactams as inhibitors of alpha-beta protein production
US6890492B1 (en) * 1998-08-13 2005-05-10 Symyx Technologies, Inc. Parallel reactor with internal sensing and method of using same
CN1636011A (zh) 1998-12-24 2005-07-06 杜邦药品公司 作为Aβ蛋白产生抑制剂的琥珀酰氨基苯并二氮杂䓬
AU7997600A (en) * 1999-10-08 2001-04-23 Du Pont Pharmaceuticals Company Amino lactam sulfonamides as inhibitors of abeta protein production
WO2001060826A2 (en) * 2000-02-17 2001-08-23 Bristol-Myers Squibb Pharma Company SUCCINOYLAMINO CARBOCYCLES AND HETEROCYCLES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
BR0107532A (pt) 2000-04-03 2004-11-03 Bristol Myers Squibb Pharma Co Composto, uso do composto, método para o tratamento de disfunções neurológicas associadas com a produção de b-amilóide, método de inibição da atividade de y-secretase e composição farmacêutica
US6692708B2 (en) * 2001-04-05 2004-02-17 Symyx Technologies, Inc. Parallel reactor for sampling and conducting in situ flow-through reactions and a method of using same
KR101155335B1 (ko) * 2005-01-07 2012-06-11 엘지전자 주식회사 이동통신 단말기의 멀티미디어 메시지 동작방법

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1332410C (en) * 1984-06-26 1994-10-11 Roger M. Freidinger Benzodiazepine analogs
IL91361A (en) * 1988-09-09 1994-10-07 Fujisawa Pharmaceutical Co Benzodiazepinone compounds [4,1] connected via positions 1 and 9 and carrying two transducers, processes for their preparation and pharmaceutical preparations containing them
FR2652352A1 (fr) * 1989-09-28 1991-03-29 Jouveinal Sa Benzodiazepines, leur procede et intermediaires de preparation et leurs applications en therapeutique.

Also Published As

Publication number Publication date
DK197289D0 (da) 1989-04-24
KR0142328B1 (ko) 1998-06-01
FR2630440B1 (fr) 1991-09-20
FI91409C (fi) 1994-06-27
HK95496A (en) 1996-06-07
KR900016158A (ko) 1990-11-12
DE68905365T2 (de) 1993-10-14
ZA892682B (en) 1990-12-28
FI91409B (fi) 1994-03-15
IE62663B1 (en) 1995-02-22
NO169653C (no) 1992-07-22
US4929614A (en) 1990-05-29
JP2805634B2 (ja) 1998-09-30
FI891952A0 (fi) 1989-04-25
DE68905365D1 (de) 1993-04-22
IS3454A7 (is) 1989-10-26
NO891692L (no) 1989-10-26
ATE86995T1 (de) 1993-04-15
NZ228650A (en) 1990-12-21
AU618086B2 (en) 1991-12-12
NO891692D0 (no) 1989-04-24
EP0340064A1 (fr) 1989-11-02
FR2630440A1 (fr) 1989-10-27
JPH0215083A (ja) 1990-01-18
CA1340074C (en) 1998-10-06
PT90339B (pt) 1994-08-31
AU3302589A (en) 1989-10-26
ES2054045T3 (es) 1994-08-01
IE891067L (en) 1989-10-25
FI891952A (fi) 1989-10-26
NO169653B (no) 1992-04-13
EP0340064B1 (fr) 1993-03-17
DK197289A (da) 1989-10-26
PT90339A (pt) 1989-11-10

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