FR2776660B1 - Diazepino-indoles de phosphodiesterases iv - Google Patents

Diazepino-indoles de phosphodiesterases iv

Info

Publication number
FR2776660B1
FR2776660B1 FR9803851A FR9803851A FR2776660B1 FR 2776660 B1 FR2776660 B1 FR 2776660B1 FR 9803851 A FR9803851 A FR 9803851A FR 9803851 A FR9803851 A FR 9803851A FR 2776660 B1 FR2776660 B1 FR 2776660B1
Authority
FR
France
Prior art keywords
diazepino
phosphodiesterases
indoles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9803851A
Other languages
English (en)
Other versions
FR2776660A1 (fr
Inventor
Henry Jacobelli
Larose Christine Julien
Sylvie Marc
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Parke Davis and Co
Original Assignee
Parke Davis and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Parke Davis and Co filed Critical Parke Davis and Co
Priority to FR9803851A priority Critical patent/FR2776660B1/fr
Priority to ZA9902322A priority patent/ZA992322B/xx
Priority to AU37063/99A priority patent/AU3706399A/en
Priority to US09/556,000 priority patent/US6365585B1/en
Priority to PCT/EP1999/002336 priority patent/WO1999050270A1/fr
Publication of FR2776660A1 publication Critical patent/FR2776660A1/fr
Application granted granted Critical
Publication of FR2776660B1 publication Critical patent/FR2776660B1/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR9803851A 1998-03-27 1998-03-27 Diazepino-indoles de phosphodiesterases iv Expired - Fee Related FR2776660B1 (fr)

Priority Applications (5)

Application Number Priority Date Filing Date Title
FR9803851A FR2776660B1 (fr) 1998-03-27 1998-03-27 Diazepino-indoles de phosphodiesterases iv
ZA9902322A ZA992322B (en) 1998-03-27 1999-03-25 Phosphodiesterase iv-inhibiting diazepinoindoles.
AU37063/99A AU3706399A (en) 1998-03-27 1999-03-26 Phosphodiesterase iv-inhibiting diazepinoindoles
US09/556,000 US6365585B1 (en) 1998-03-27 1999-03-26 Phosphodiesterase IV-inhibiting diazepinoindoles
PCT/EP1999/002336 WO1999050270A1 (fr) 1998-03-27 1999-03-26 Diazepinoindoles inhibant la phosphodiesterase iv

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9803851A FR2776660B1 (fr) 1998-03-27 1998-03-27 Diazepino-indoles de phosphodiesterases iv

Publications (2)

Publication Number Publication Date
FR2776660A1 FR2776660A1 (fr) 1999-10-01
FR2776660B1 true FR2776660B1 (fr) 2000-05-12

Family

ID=9524601

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9803851A Expired - Fee Related FR2776660B1 (fr) 1998-03-27 1998-03-27 Diazepino-indoles de phosphodiesterases iv

Country Status (5)

Country Link
US (1) US6365585B1 (fr)
AU (1) AU3706399A (fr)
FR (1) FR2776660B1 (fr)
WO (1) WO1999050270A1 (fr)
ZA (1) ZA992322B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1188438A1 (fr) * 2000-09-15 2002-03-20 Warner-Lambert Company Compositions pharmaceutiques pour la prévention ou le traitement de maladies associées à un excès de production de l' IL-12
EP1199074A1 (fr) * 2000-09-15 2002-04-24 Warner-Lambert Company Composition pharmaceutique pour la prévention ou le traitement de maladies associées à un excès de production d' IL-12
US6872382B1 (en) 2001-05-21 2005-03-29 Alcon, Inc. Use of selective PDE IV inhibitors to treat dry eye disorders
EP1484345A1 (fr) 2003-06-06 2004-12-08 Borealis Technology Oy Procédé de préparation de polypropylène au moyen d'un catalyseur Ziegler-Natta
EP1526135A1 (fr) * 2003-10-24 2005-04-27 Warner-Lambert Company LLC Azabenzodiazepines utiles comme inhibiteurs de pde4
CA2620333A1 (fr) 2005-08-26 2007-03-01 Braincells, Inc. Neurogenese par modulation du recepteur muscarinique
EP2258358A3 (fr) 2005-08-26 2011-09-07 Braincells, Inc. Neurogenèse avec un inhibiteur de l'acetylcholinestérase
EP1940389A2 (fr) 2005-10-21 2008-07-09 Braincells, Inc. Modulation de la neurogenese par inhibition de la pde
CA2625210A1 (fr) 2005-10-31 2007-05-10 Braincells, Inc. Modulation de la neurogenese dont la mediation est assuree par recepteur gaba
US20100216734A1 (en) 2006-03-08 2010-08-26 Braincells, Inc. Modulation of neurogenesis by nootropic agents
MX2008014320A (es) 2006-05-09 2009-03-25 Braincells Inc Neurogenesis mediada por el receptor de 5-hidroxitriptamina.
AU2007249399A1 (en) 2006-05-09 2007-11-22 Braincells, Inc. Neurogenesis by modulating angiotensin
MX2009002496A (es) 2006-09-08 2009-07-10 Braincells Inc Combinaciones que contienen un derivado de 4-acilaminopiridina.
US20100184806A1 (en) 2006-09-19 2010-07-22 Braincells, Inc. Modulation of neurogenesis by ppar agents
US20100216805A1 (en) 2009-02-25 2010-08-26 Braincells, Inc. Modulation of neurogenesis using d-cycloserine combinations
EP2804603A1 (fr) 2012-01-10 2014-11-26 President and Fellows of Harvard College Composés promoteurs de réplication des cellules bêta et leurs procédés d'utilisation

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2630440B1 (fr) * 1988-04-25 1991-09-20 Jouveinal Sa Benzodiazepines, leur procede et intermediaires de preparation et leurs applications en therapeutique
IL91361A (en) * 1988-09-09 1994-10-07 Fujisawa Pharmaceutical Co Benzodiazepinone compounds [4,1] connected via positions 1 and 9 and carrying two transducers, processes for their preparation and pharmaceutical preparations containing them
WO1996006617A1 (fr) * 1994-08-30 1996-03-07 Fujisawa Pharmaceutical Co., Ltd. Preparation de liposomes
FR2725719B1 (fr) * 1994-10-14 1996-12-06 Jouveinal Inst Rech Diazepino-indoles inhibiteurs de phosphodiesterases iv

Also Published As

Publication number Publication date
WO1999050270A1 (fr) 1999-10-07
ZA992322B (en) 1999-09-20
AU3706399A (en) 1999-10-18
US6365585B1 (en) 2002-04-02
FR2776660A1 (fr) 1999-10-01

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Legal Events

Date Code Title Description
ST Notification of lapse

Effective date: 20071130