FR2776660B1 - Diazepino-indoles de phosphodiesterases iv - Google Patents
Diazepino-indoles de phosphodiesterases ivInfo
- Publication number
- FR2776660B1 FR2776660B1 FR9803851A FR9803851A FR2776660B1 FR 2776660 B1 FR2776660 B1 FR 2776660B1 FR 9803851 A FR9803851 A FR 9803851A FR 9803851 A FR9803851 A FR 9803851A FR 2776660 B1 FR2776660 B1 FR 2776660B1
- Authority
- FR
- France
- Prior art keywords
- diazepino
- phosphodiesterases
- indoles
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/06—Peri-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9803851A FR2776660B1 (fr) | 1998-03-27 | 1998-03-27 | Diazepino-indoles de phosphodiesterases iv |
ZA9902322A ZA992322B (en) | 1998-03-27 | 1999-03-25 | Phosphodiesterase iv-inhibiting diazepinoindoles. |
AU37063/99A AU3706399A (en) | 1998-03-27 | 1999-03-26 | Phosphodiesterase iv-inhibiting diazepinoindoles |
US09/556,000 US6365585B1 (en) | 1998-03-27 | 1999-03-26 | Phosphodiesterase IV-inhibiting diazepinoindoles |
PCT/EP1999/002336 WO1999050270A1 (fr) | 1998-03-27 | 1999-03-26 | Diazepinoindoles inhibant la phosphodiesterase iv |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9803851A FR2776660B1 (fr) | 1998-03-27 | 1998-03-27 | Diazepino-indoles de phosphodiesterases iv |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2776660A1 FR2776660A1 (fr) | 1999-10-01 |
FR2776660B1 true FR2776660B1 (fr) | 2000-05-12 |
Family
ID=9524601
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR9803851A Expired - Fee Related FR2776660B1 (fr) | 1998-03-27 | 1998-03-27 | Diazepino-indoles de phosphodiesterases iv |
Country Status (5)
Country | Link |
---|---|
US (1) | US6365585B1 (fr) |
AU (1) | AU3706399A (fr) |
FR (1) | FR2776660B1 (fr) |
WO (1) | WO1999050270A1 (fr) |
ZA (1) | ZA992322B (fr) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1188438A1 (fr) * | 2000-09-15 | 2002-03-20 | Warner-Lambert Company | Compositions pharmaceutiques pour la prévention ou le traitement de maladies associées à un excès de production de l' IL-12 |
EP1199074A1 (fr) * | 2000-09-15 | 2002-04-24 | Warner-Lambert Company | Composition pharmaceutique pour la prévention ou le traitement de maladies associées à un excès de production d' IL-12 |
US6872382B1 (en) | 2001-05-21 | 2005-03-29 | Alcon, Inc. | Use of selective PDE IV inhibitors to treat dry eye disorders |
EP1484345A1 (fr) | 2003-06-06 | 2004-12-08 | Borealis Technology Oy | Procédé de préparation de polypropylène au moyen d'un catalyseur Ziegler-Natta |
EP1526135A1 (fr) * | 2003-10-24 | 2005-04-27 | Warner-Lambert Company LLC | Azabenzodiazepines utiles comme inhibiteurs de pde4 |
CA2620333A1 (fr) | 2005-08-26 | 2007-03-01 | Braincells, Inc. | Neurogenese par modulation du recepteur muscarinique |
EP2258358A3 (fr) | 2005-08-26 | 2011-09-07 | Braincells, Inc. | Neurogenèse avec un inhibiteur de l'acetylcholinestérase |
EP1940389A2 (fr) | 2005-10-21 | 2008-07-09 | Braincells, Inc. | Modulation de la neurogenese par inhibition de la pde |
CA2625210A1 (fr) | 2005-10-31 | 2007-05-10 | Braincells, Inc. | Modulation de la neurogenese dont la mediation est assuree par recepteur gaba |
US20100216734A1 (en) | 2006-03-08 | 2010-08-26 | Braincells, Inc. | Modulation of neurogenesis by nootropic agents |
MX2008014320A (es) | 2006-05-09 | 2009-03-25 | Braincells Inc | Neurogenesis mediada por el receptor de 5-hidroxitriptamina. |
AU2007249399A1 (en) | 2006-05-09 | 2007-11-22 | Braincells, Inc. | Neurogenesis by modulating angiotensin |
MX2009002496A (es) | 2006-09-08 | 2009-07-10 | Braincells Inc | Combinaciones que contienen un derivado de 4-acilaminopiridina. |
US20100184806A1 (en) | 2006-09-19 | 2010-07-22 | Braincells, Inc. | Modulation of neurogenesis by ppar agents |
US20100216805A1 (en) | 2009-02-25 | 2010-08-26 | Braincells, Inc. | Modulation of neurogenesis using d-cycloserine combinations |
EP2804603A1 (fr) | 2012-01-10 | 2014-11-26 | President and Fellows of Harvard College | Composés promoteurs de réplication des cellules bêta et leurs procédés d'utilisation |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2630440B1 (fr) * | 1988-04-25 | 1991-09-20 | Jouveinal Sa | Benzodiazepines, leur procede et intermediaires de preparation et leurs applications en therapeutique |
IL91361A (en) * | 1988-09-09 | 1994-10-07 | Fujisawa Pharmaceutical Co | Benzodiazepinone compounds [4,1] connected via positions 1 and 9 and carrying two transducers, processes for their preparation and pharmaceutical preparations containing them |
WO1996006617A1 (fr) * | 1994-08-30 | 1996-03-07 | Fujisawa Pharmaceutical Co., Ltd. | Preparation de liposomes |
FR2725719B1 (fr) * | 1994-10-14 | 1996-12-06 | Jouveinal Inst Rech | Diazepino-indoles inhibiteurs de phosphodiesterases iv |
-
1998
- 1998-03-27 FR FR9803851A patent/FR2776660B1/fr not_active Expired - Fee Related
-
1999
- 1999-03-25 ZA ZA9902322A patent/ZA992322B/xx unknown
- 1999-03-26 WO PCT/EP1999/002336 patent/WO1999050270A1/fr active Application Filing
- 1999-03-26 US US09/556,000 patent/US6365585B1/en not_active Expired - Fee Related
- 1999-03-26 AU AU37063/99A patent/AU3706399A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
WO1999050270A1 (fr) | 1999-10-07 |
ZA992322B (en) | 1999-09-20 |
AU3706399A (en) | 1999-10-18 |
US6365585B1 (en) | 2002-04-02 |
FR2776660A1 (fr) | 1999-10-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |
Effective date: 20071130 |