ZA992322B - Phosphodiesterase iv-inhibiting diazepinoindoles. - Google Patents

Phosphodiesterase iv-inhibiting diazepinoindoles.

Info

Publication number
ZA992322B
ZA992322B ZA9902322A ZA992322A ZA992322B ZA 992322 B ZA992322 B ZA 992322B ZA 9902322 A ZA9902322 A ZA 9902322A ZA 992322 A ZA992322 A ZA 992322A ZA 992322 B ZA992322 B ZA 992322B
Authority
ZA
South Africa
Prior art keywords
diazepinoindoles
phosphodiesterase
inhibiting
inhibiting diazepinoindoles
Prior art date
Application number
ZA9902322A
Other languages
English (en)
Inventor
Henri Jacobelli
Christine Julien-Larose
Sylvie Marc
Original Assignee
Parke Davis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Parke Davis filed Critical Parke Davis
Publication of ZA992322B publication Critical patent/ZA992322B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA9902322A 1998-03-27 1999-03-25 Phosphodiesterase iv-inhibiting diazepinoindoles. ZA992322B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9803851A FR2776660B1 (fr) 1998-03-27 1998-03-27 Diazepino-indoles de phosphodiesterases iv

Publications (1)

Publication Number Publication Date
ZA992322B true ZA992322B (en) 1999-09-20

Family

ID=9524601

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA9902322A ZA992322B (en) 1998-03-27 1999-03-25 Phosphodiesterase iv-inhibiting diazepinoindoles.

Country Status (5)

Country Link
US (1) US6365585B1 (fr)
AU (1) AU3706399A (fr)
FR (1) FR2776660B1 (fr)
WO (1) WO1999050270A1 (fr)
ZA (1) ZA992322B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1199074A1 (fr) * 2000-09-15 2002-04-24 Warner-Lambert Company Composition pharmaceutique pour la prévention ou le traitement de maladies associées à un excès de production d' IL-12
EP1188438A1 (fr) * 2000-09-15 2002-03-20 Warner-Lambert Company Compositions pharmaceutiques pour la prévention ou le traitement de maladies associées à un excès de production de l' IL-12
US6872382B1 (en) 2001-05-21 2005-03-29 Alcon, Inc. Use of selective PDE IV inhibitors to treat dry eye disorders
EP1484345A1 (fr) 2003-06-06 2004-12-08 Borealis Technology Oy Procédé de préparation de polypropylène au moyen d'un catalyseur Ziegler-Natta
EP1526135A1 (fr) * 2003-10-24 2005-04-27 Warner-Lambert Company LLC Azabenzodiazepines utiles comme inhibiteurs de pde4
EP2258358A3 (fr) 2005-08-26 2011-09-07 Braincells, Inc. Neurogenèse avec un inhibiteur de l'acetylcholinestérase
EP2275095A3 (fr) 2005-08-26 2011-08-17 Braincells, Inc. Neurogenese par modulation des recepteurs muscariniques
JP2009512711A (ja) 2005-10-21 2009-03-26 ブレインセルス,インコーポレイティド Pde阻害による神経新生の調節
CA2625210A1 (fr) 2005-10-31 2007-05-10 Braincells, Inc. Modulation de la neurogenese dont la mediation est assuree par recepteur gaba
US20100216734A1 (en) 2006-03-08 2010-08-26 Braincells, Inc. Modulation of neurogenesis by nootropic agents
AU2007249399A1 (en) 2006-05-09 2007-11-22 Braincells, Inc. Neurogenesis by modulating angiotensin
JP2009536667A (ja) 2006-05-09 2009-10-15 ブレインセルス,インコーポレイティド 5ht受容体介在性の神経新生
KR20090064418A (ko) 2006-09-08 2009-06-18 브레인셀즈 인코퍼레이션 4-아실아미노피리딘 유도체 포함 조합물
US20100184806A1 (en) 2006-09-19 2010-07-22 Braincells, Inc. Modulation of neurogenesis by ppar agents
WO2010099217A1 (fr) 2009-02-25 2010-09-02 Braincells, Inc. Modulation de neurogenèse à l'aide de combinaisons de d-cyclosérine
WO2013106547A1 (fr) 2012-01-10 2013-07-18 President And Fellows Of Harvard College Composés promoteurs de réplication des cellules bêta et leurs procédés d'utilisation

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2630440B1 (fr) * 1988-04-25 1991-09-20 Jouveinal Sa Benzodiazepines, leur procede et intermediaires de preparation et leurs applications en therapeutique
IL91361A (en) * 1988-09-09 1994-10-07 Fujisawa Pharmaceutical Co Benzodiazepinone compounds [4,1] connected via positions 1 and 9 and carrying two transducers, processes for their preparation and pharmaceutical preparations containing them
IL115089A0 (en) * 1994-08-30 1995-12-08 Fujisawa Pharmaceutical Co A liposome preparation containing a tricyclic compound and process for the preparation thereof
FR2725719B1 (fr) * 1994-10-14 1996-12-06 Jouveinal Inst Rech Diazepino-indoles inhibiteurs de phosphodiesterases iv

Also Published As

Publication number Publication date
FR2776660A1 (fr) 1999-10-01
AU3706399A (en) 1999-10-18
FR2776660B1 (fr) 2000-05-12
US6365585B1 (en) 2002-04-02
WO1999050270A1 (fr) 1999-10-07

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