DK1506171T3 - Fremstillinger af et sulfinylacetamid - Google Patents

Fremstillinger af et sulfinylacetamid

Info

Publication number
DK1506171T3
DK1506171T3 DK03729108T DK03729108T DK1506171T3 DK 1506171 T3 DK1506171 T3 DK 1506171T3 DK 03729108 T DK03729108 T DK 03729108T DK 03729108 T DK03729108 T DK 03729108T DK 1506171 T3 DK1506171 T3 DK 1506171T3
Authority
DK
Denmark
Prior art keywords
preparations
sulfinyl acetamide
sulfinyl
acetamide
Prior art date
Application number
DK03729108T
Other languages
Danish (da)
English (en)
Inventor
Denis Largeau
Gilles Oddon
Original Assignee
Cephalon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cephalon Inc filed Critical Cephalon Inc
Application granted granted Critical
Publication of DK1506171T3 publication Critical patent/DK1506171T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00Preparation of sulfones; Preparation of sulfoxides
    • C07C315/02Preparation of sulfones; Preparation of sulfoxides by formation of sulfone or sulfoxide groups by oxidation of sulfides, or by formation of sulfone groups by oxidation of sulfoxides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/095Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A61K31/10Sulfides; Sulfoxides; Sulfones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK03729108T 2002-05-23 2003-05-23 Fremstillinger af et sulfinylacetamid DK1506171T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38317302P 2002-05-23 2002-05-23
US10/443,327 US6875893B2 (en) 2002-05-23 2003-05-22 Preparations of a sulfinyl acetamide
PCT/US2003/016379 WO2003099774A1 (fr) 2002-05-23 2003-05-23 Preparations d'un acetamide de sulfinyle

Publications (1)

Publication Number Publication Date
DK1506171T3 true DK1506171T3 (da) 2009-01-19

Family

ID=29586987

Family Applications (1)

Application Number Title Priority Date Filing Date
DK03729108T DK1506171T3 (da) 2002-05-23 2003-05-23 Fremstillinger af et sulfinylacetamid

Country Status (29)

Country Link
US (2) US6875893B2 (fr)
EP (1) EP1506171B1 (fr)
JP (1) JP4351627B2 (fr)
KR (1) KR100984571B1 (fr)
CN (1) CN100379721C (fr)
AR (1) AR039857A1 (fr)
AT (1) ATE414058T1 (fr)
BR (1) BR0311242A (fr)
CA (1) CA2486533C (fr)
CY (1) CY1108747T1 (fr)
DE (1) DE60324671D1 (fr)
DK (1) DK1506171T3 (fr)
EA (1) EA007561B1 (fr)
EG (1) EG23693A (fr)
ES (1) ES2316755T3 (fr)
HK (1) HK1072596A1 (fr)
IL (2) IL165095A0 (fr)
IS (1) IS2650B (fr)
MX (1) MXPA04011459A (fr)
MY (1) MY129141A (fr)
NO (1) NO329559B1 (fr)
NZ (1) NZ536747A (fr)
PL (1) PL211695B1 (fr)
PT (1) PT1506171E (fr)
SI (1) SI1506171T1 (fr)
TW (1) TWI317733B (fr)
UA (1) UA79790C2 (fr)
WO (1) WO2003099774A1 (fr)
ZA (1) ZA200409400B (fr)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2416792C (fr) * 2000-07-27 2010-02-09 Teva Pharmaceutical Industries Ltd. Modafinil cristallin et pur et procede de preparation associe
US6875893B2 (en) * 2002-05-23 2005-04-05 Cephalon, Inc. Preparations of a sulfinyl acetamide
US6992219B2 (en) * 2002-08-09 2006-01-31 Cephalon France Modafinil polymorphic forms
FR2849029B1 (fr) * 2002-12-20 2005-03-18 Lafon Labor Procede de preparation et formes cristallines des enantiomeres optiques du modafinil.
MXPA05008088A (es) * 2003-02-24 2005-09-21 Mallinckrodt Inc Proceso mejorado para preparar benzhidril tioacetamida.
US20040253308A1 (en) * 2003-04-29 2004-12-16 Barr Laboratories, Inc. Surface-treated modafinil particles
US7368591B2 (en) 2003-09-19 2008-05-06 Cephalon France Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation
SI1678129T1 (sl) * 2003-10-23 2009-10-31 Mallinckrodt Inc Izboljĺ an proces za pripravo benzhidril tioacetamida
US20060086667A1 (en) * 2004-09-13 2006-04-27 Cephalon, Inc., U.S. Corporation Methods for the separation of enantiomeric sulfinylacetamides
DK1737889T3 (da) 2004-10-19 2011-01-03 Lonza Ag Fremgangsmåde til fastfase-peptidsyntese
AU2006272874B2 (en) * 2005-07-21 2010-03-11 Neurohealing Pharmaceuticals, Inc. Rapid onset and short term modafinil compositions and methods of use thereof
WO2007027328A2 (fr) * 2005-07-28 2007-03-08 University Of Iowa Research Foundation Sulfoxydation et amidation microbienne d'acides benzhydrylsulfanylcarboxyliques et utilisations de celles-ci
EP1805204A2 (fr) * 2005-09-14 2007-07-11 Novetide Ltd. Procédé destiné à la production de bivalirudine
AU2006325144A1 (en) * 2005-12-09 2007-06-21 Mallinckrodt Inc. Processes for the preparation of modafinil and analogs thereof
CN100343228C (zh) * 2006-02-17 2007-10-17 中国科学院上海有机化学研究所 高对映体选择性制备 2-二苯甲基亚磺酰基-乙酰胺单一对映体的方法
JP2009508880A (ja) * 2006-02-21 2009-03-05 テバ ファーマシューティカル インダストリーズ リミティド アルモダフィニルの新規な結晶形とその調製方法
US20080031939A1 (en) * 2006-03-01 2008-02-07 Viviana Braude Process for the preparation of armodafinil
GB0604233D0 (en) * 2006-03-02 2006-04-12 Syngenta Participations Ag Process
JP2009543803A (ja) * 2006-07-12 2009-12-10 エラン・ファルマ・インターナショナル・リミテッド モダフィニルのナノ粒子製剤
US7884135B2 (en) * 2006-08-14 2011-02-08 Neurohealing Pharmaceuticals, Inc. Modafinil-based treatment for premature ejaculation
US7960586B2 (en) * 2007-08-16 2011-06-14 Teva Pharmaceutical Industries Ltd. Purification of armodafinil
US20100036164A1 (en) * 2008-08-06 2010-02-11 Srinivas Areveli Preparation of armodafinil form i
CN102976985A (zh) * 2011-09-07 2013-03-20 大连大学 一锅法合成二苯甲基亚磺酰基乙酰胺及其类似物的方法
CN105992734A (zh) * 2014-02-06 2016-10-05 比勒鲁迪克斯那斯公司 由可拉伸的纸构成的直立袋

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1520812A (en) * 1975-10-02 1978-08-09 Lafon Labor Benzhydrylsulphinyl derivatives
GB1584462A (en) * 1977-03-31 1981-02-11 Lafon Labor N-diaryl-malonamide and diarylmethyl-sulphinyl-acetamide derivatives and pharmaceutical compositions containing them
FR2593809B1 (fr) * 1986-01-31 1988-07-22 Lafon Labor Benzhydrylsulfinylacetamide, procede de preparation et utilisation en therapeutique
US20030187023A1 (en) * 2000-07-17 2003-10-02 Keiji Kubo Sulfone derivatives, process for their production and use thereof
CA2416792C (fr) 2000-07-27 2010-02-09 Teva Pharmaceutical Industries Ltd. Modafinil cristallin et pur et procede de preparation associe
IL143106A (en) 2001-05-13 2005-11-20 Chemagis Ltd Process for the preparation of diphenylmethylthioacetamide
US6875893B2 (en) * 2002-05-23 2005-04-05 Cephalon, Inc. Preparations of a sulfinyl acetamide
DE10245546B3 (de) * 2002-09-30 2004-05-13 Infineon Technologies Ag Pseudostatische Speicherschaltung
JP3838972B2 (ja) * 2002-12-25 2006-10-25 Necエレクトロニクス株式会社 周波数検出回路及びデータ処理装置

Also Published As

Publication number Publication date
KR100984571B1 (ko) 2010-09-30
IS7523A (is) 2004-11-09
IS2650B (is) 2010-08-15
EA200401551A1 (ru) 2005-04-28
EP1506171B1 (fr) 2008-11-12
US20050171209A1 (en) 2005-08-04
JP2005527623A (ja) 2005-09-15
NZ536747A (en) 2006-11-30
JP4351627B2 (ja) 2009-10-28
ZA200409400B (en) 2005-12-28
PL211695B1 (pl) 2012-06-29
KR20050016421A (ko) 2005-02-21
EG23693A (en) 2007-05-15
CA2486533C (fr) 2011-01-04
PL373792A1 (en) 2005-09-19
WO2003099774A1 (fr) 2003-12-04
MY129141A (en) 2007-03-30
US7057069B2 (en) 2006-06-06
UA79790C2 (en) 2007-07-25
NO329559B1 (no) 2010-11-15
BR0311242A (pt) 2005-03-15
AR039857A1 (es) 2005-03-02
IL165095A (en) 2010-11-30
EA007561B1 (ru) 2006-12-29
ATE414058T1 (de) 2008-11-15
NO20044916L (no) 2004-12-16
ES2316755T3 (es) 2009-04-16
CN1656064A (zh) 2005-08-17
MXPA04011459A (es) 2005-02-14
HK1072596A1 (en) 2005-09-02
AU2003233668A1 (en) 2003-12-12
US6875893B2 (en) 2005-04-05
TWI317733B (en) 2009-12-01
DE60324671D1 (de) 2008-12-24
PT1506171E (pt) 2009-01-02
CA2486533A1 (fr) 2003-12-04
EP1506171A1 (fr) 2005-02-16
SI1506171T1 (sl) 2009-06-30
US20040002547A1 (en) 2004-01-01
CN100379721C (zh) 2008-04-09
CY1108747T1 (el) 2014-04-09
IL165095A0 (en) 2005-12-18
TW200406196A (en) 2004-05-01

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