DK150604C - Analogifremgangsmaade til fremstilling af calciumoxaprozin - Google Patents
Analogifremgangsmaade til fremstilling af calciumoxaprozinInfo
- Publication number
- DK150604C DK150604C DK183582A DK183582A DK150604C DK 150604 C DK150604 C DK 150604C DK 183582 A DK183582 A DK 183582A DK 183582 A DK183582 A DK 183582A DK 150604 C DK150604 C DK 150604C
- Authority
- DK
- Denmark
- Prior art keywords
- oxaprozine
- preparing calcium
- analogy procedure
- oxaprozin
- calcium
- Prior art date
Links
- OFPXSFXSNFPTHF-UHFFFAOYSA-N oxaprozin Chemical compound O1C(CCC(=O)O)=NC(C=2C=CC=CC=2)=C1C1=CC=CC=C1 OFPXSFXSNFPTHF-UHFFFAOYSA-N 0.000 title abstract 4
- OYPRJOBELJOOCE-UHFFFAOYSA-N Calcium Chemical compound [Ca] OYPRJOBELJOOCE-UHFFFAOYSA-N 0.000 title abstract 3
- 229910052791 calcium Inorganic materials 0.000 title abstract 3
- 239000011575 calcium Substances 0.000 title abstract 3
- 229960002739 oxaprozin Drugs 0.000 abstract 3
- 229940121363 anti-inflammatory agent Drugs 0.000 abstract 1
- 239000002260 anti-inflammatory agent Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicinal Preparation (AREA)
- Plural Heterocyclic Compounds (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8113074 | 1981-04-28 | ||
| GB8113074 | 1981-04-28 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK183582A DK183582A (da) | 1982-10-29 |
| DK150604B DK150604B (da) | 1987-04-13 |
| DK150604C true DK150604C (da) | 1987-12-07 |
Family
ID=10521427
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK183582A DK150604C (da) | 1981-04-28 | 1982-04-23 | Analogifremgangsmaade til fremstilling af calciumoxaprozin |
Country Status (24)
| Country | Link |
|---|---|
| US (2) | US4465838A (cs) |
| EP (1) | EP0063884B1 (cs) |
| JP (1) | JPS57181072A (cs) |
| KR (1) | KR880000871B1 (cs) |
| AT (1) | ATE14015T1 (cs) |
| AU (1) | AU544975B2 (cs) |
| CA (1) | CA1169867A (cs) |
| CS (1) | CS236674B2 (cs) |
| DD (1) | DD202017A5 (cs) |
| DE (1) | DE3264400D1 (cs) |
| DK (1) | DK150604C (cs) |
| ES (1) | ES511730A0 (cs) |
| FI (1) | FI71314C (cs) |
| GR (1) | GR75913B (cs) |
| HU (1) | HU185276B (cs) |
| IE (1) | IE52909B1 (cs) |
| IL (1) | IL65443A (cs) |
| MY (1) | MY8700599A (cs) |
| NZ (1) | NZ200247A (cs) |
| PH (1) | PH18053A (cs) |
| PL (1) | PL136322B1 (cs) |
| PT (1) | PT74794B (cs) |
| ZA (1) | ZA822355B (cs) |
| ZW (1) | ZW7482A1 (cs) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5380738A (en) * | 1993-05-21 | 1995-01-10 | Monsanto Company | 2-substituted oxazoles further substituted by 4-fluorophenyl and 4-methylsulfonylphenyl as antiinflammatory agents |
| US6726928B2 (en) * | 1994-10-28 | 2004-04-27 | R.P. Scherer Technologies, Inc. | Process for preparing solid dosage forms for unpalatable pharmaceuticals |
| AU718030B2 (en) * | 1996-05-20 | 2000-04-06 | G.D. Searle & Co. | Potassium, sodium and tris oxaprozin salt pharmaceutical formulations |
| US7358254B2 (en) * | 2001-07-13 | 2008-04-15 | Bristol-Myers Squibb Company | Method for treating atherosclerosis employing an aP2 inhibitor and combination |
| PE20061303A1 (es) * | 2005-03-30 | 2006-12-07 | Astion Dev As | Composicion farmaceutica que comprende oxaprozina |
| AU2006228869A1 (en) * | 2005-03-30 | 2006-10-05 | Astion Pharma A/S | Oxaprozin or a closely related compound for the treatment of eczema |
| AU2009286319B2 (en) * | 2008-08-26 | 2013-05-16 | Dorf Ketal Chemicals (I) Private Limited | A new additive for inhibiting acid corrosion and method of using the new additive |
| KR20140065862A (ko) * | 2012-11-22 | 2014-05-30 | 에스케이케미칼주식회사 | 발포성 속붕해성 이매티닙 제제 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1206403A (en) * | 1966-12-15 | 1970-09-23 | Wyeth John & Brother Ltd | Oxazoles |
| GB1245087A (en) * | 1967-10-26 | 1971-09-02 | Wyeth John & Brother Ltd | Heterocyclic compounds |
| US3578671A (en) * | 1967-11-06 | 1971-05-11 | Wyeth John & Brother Ltd | Oxazoles |
-
1982
- 1982-03-31 IE IE766/82A patent/IE52909B1/en not_active IP Right Cessation
- 1982-04-05 CA CA000400464A patent/CA1169867A/en not_active Expired
- 1982-04-05 ZA ZA822355A patent/ZA822355B/xx unknown
- 1982-04-06 AU AU82378/82A patent/AU544975B2/en not_active Expired
- 1982-04-06 IL IL65443A patent/IL65443A/xx not_active IP Right Cessation
- 1982-04-06 NZ NZ200247A patent/NZ200247A/en unknown
- 1982-04-07 EP EP82301839A patent/EP0063884B1/en not_active Expired
- 1982-04-07 AT AT82301839T patent/ATE14015T1/de not_active IP Right Cessation
- 1982-04-07 DE DE8282301839T patent/DE3264400D1/de not_active Expired
- 1982-04-09 GR GR67879A patent/GR75913B/el unknown
- 1982-04-15 FI FI821324A patent/FI71314C/fi not_active IP Right Cessation
- 1982-04-15 ZW ZW74/82A patent/ZW7482A1/xx unknown
- 1982-04-22 PH PH27171A patent/PH18053A/en unknown
- 1982-04-23 JP JP57069463A patent/JPS57181072A/ja active Granted
- 1982-04-23 DK DK183582A patent/DK150604C/da not_active IP Right Cessation
- 1982-04-26 KR KR8201829A patent/KR880000871B1/ko not_active Expired
- 1982-04-26 US US06/371,904 patent/US4465838A/en not_active Expired - Lifetime
- 1982-04-26 PL PL1982236145A patent/PL136322B1/pl unknown
- 1982-04-26 PT PT74794A patent/PT74794B/pt unknown
- 1982-04-27 DD DD82239350A patent/DD202017A5/de not_active IP Right Cessation
- 1982-04-27 ES ES511730A patent/ES511730A0/es active Granted
- 1982-04-27 HU HU821325A patent/HU185276B/hu unknown
- 1982-04-28 CS CS823052A patent/CS236674B2/cs unknown
-
1984
- 1984-07-11 US US06/629,704 patent/US4532253A/en not_active Expired - Lifetime
-
1987
- 1987-12-30 MY MY599/87A patent/MY8700599A/xx unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PUP | Patent expired |